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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-(2,5-dichlorophenyl)sulfonyl-3,4-dihydro-2H-1,5-benzothiazepine —— C15H13Cl2NO2S2
5-(2,5-dichlorophenyl)sulfonyl-3,4-dihydro-2H-1,5-benzothiazepine
—— (E)-3-(1,3-benzoxazol-2-yl)-1-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)prop-2-en-1-one —— C19H16N2O2S
(E)-3-(1,3-benzoxazol-2-yl)-1-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)prop-2-en-1-one
—— 2-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C24H31N3O2S
2-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C24H31N3O2S
2-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(5-thiophen-3-yltetrazol-2-yl)ethanone —— C17H17N5OS2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(5-thiophen-3-yltetrazol-2-yl)ethanone
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(5-thiophen-3-yltetrazol-2-yl)ethanone —— C17H17N5OS2
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(5-thiophen-3-yltetrazol-2-yl)ethanone
—— 2-(1-cyclohexyl-4,5-dimethylimidazol-2-yl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C23H31N3OS2
2-(1-cyclohexyl-4,5-dimethylimidazol-2-yl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[(3-fluoro-4-methoxyphenyl)methyl-methylamino]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H25FN2O2S
2-[(3-fluoro-4-methoxyphenyl)methyl-methylamino]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[(3-fluoro-4-methoxyphenyl)methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H25FN2O2S
2-[(3-fluoro-4-methoxyphenyl)methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C16H16ClN3OS
(5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C16H16ClN3OS
(5-chloro-2-methylpyrimidin-4-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [2-oxo-2-(2-phenylsulfanylethylamino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H20N2O4S2
[2-oxo-2-(2-phenylsulfanylethylamino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(1S)-1-(5-phenyl-1,3,4-oxadiazol-2-yl)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H17N3O4S
[(1S)-1-(5-phenyl-1,3,4-oxadiazol-2-yl)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(3S)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H15N3O4S2
[(3S)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-oxo-2-(2-thiophen-2-ylethylamino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H18N2O4S2
[2-oxo-2-(2-thiophen-2-ylethylamino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(2R)-1-(2-benzoylhydrazinyl)-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H19N3O5S
[(2R)-1-(2-benzoylhydrazinyl)-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— 2-(3,4-difluorophenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H17F2NOS2
2-(3,4-difluorophenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[4-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylmethyl)-1,3-thiazol-2-yl]-N-(4-methylphenyl)acetamide —— C22H23N3OS2
2-[4-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylmethyl)-1,3-thiazol-2-yl]-N-(4-methylphenyl)acetamide
—— (6S)-6-(4-methoxyphenyl)-6,10-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol —— C19H17NO2S
(6S)-6-(4-methoxyphenyl)-6,10-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol
—— (6R)-6-(4-methoxyphenyl)-6,10-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol —— C19H17NO2S
(6R)-6-(4-methoxyphenyl)-6,10-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol
—— 5-bromo-6-methyl-3-[(2R)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]pyran-2,4-dione —— C21H16BrNO3S
5-bromo-6-methyl-3-[(2R)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]pyran-2,4-dione
—— 5-bromo-6-methyl-3-[(2S)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]pyran-2,4-dione —— C21H16BrNO3S
5-bromo-6-methyl-3-[(2S)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]pyran-2,4-dione
—— [(2S)-1-[[(3R)-1,1-dioxothiolan-3-yl]amino]-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C17H20N2O6S2
[(2S)-1-[[(3R)-1,1-dioxothiolan-3-yl]amino]-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-ethyl-2,5-dimethylpyrrole-3-carboxylate —— C21H26N2O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-ethyl-2,5-dimethylpyrrole-3-carboxylate
—— ethyl N-[2-[ethyl-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]amino]acetyl]carbamate —— C19H27N3O4S
ethyl N-[2-[ethyl-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]amino]acetyl]carbamate
—— ethyl N-[2-[ethyl-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]amino]acetyl]carbamate —— C19H27N3O4S
ethyl N-[2-[ethyl-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]amino]acetyl]carbamate
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(1,5-diphenyl-1,2,4-triazol-3-yl)methanone —— C24H20N4OS
3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(1,5-diphenyl-1,2,4-triazol-3-yl)methanone
—— 2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H24N2OS
2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(2-ethoxypyridin-3-yl)methanone —— C17H18N2O2S
3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(2-ethoxypyridin-3-yl)methanone
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(2,5-dimethylfuran-3-yl)methanone —— C16H17NO2S
3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(2,5-dimethylfuran-3-yl)methanone
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl(pyridin-4-yl)methanone —— C15H14N2OS
3,4-dihydro-2H-1,5-benzothiazepin-5-yl(pyridin-4-yl)methanone
—— 2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)ethanone —— C19H19NO3S
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)ethanone
—— (5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)methanone —— C18H16ClNO3S
(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)methanone
—— 2-(2,5-difluorophenyl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H17F2NOS2
2-(2,5-difluorophenyl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-(2,5-difluorophenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H17F2NOS2
2-(2,5-difluorophenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,5-dimethylfuran-3-carboxylate —— C19H21NO4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,5-dimethylfuran-3-carboxylate
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(2-phenyltriazol-4-yl)methanone —— C18H16N4OS
3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(2-phenyltriazol-4-yl)methanone
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone —— C17H17N5OS
3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone
—— 4-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)-2-phenylphthalazin-1-one —— C24H19N3O2S
4-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)-2-phenylphthalazin-1-one
—— 1-[4-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylsulfonyl)phenyl]pyrrolidin-2-one —— C19H20N2O3S2
1-[4-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylsulfonyl)phenyl]pyrrolidin-2-one
—— 3-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylsulfonyl)-4-methylbenzoic acid —— C17H17NO4S2
3-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylsulfonyl)-4-methylbenzoic acid
—— 4-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylsulfonyl)benzenesulfonamide —— C15H16N2O4S3
4-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylsulfonyl)benzenesulfonamide
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,3-dihydro-1,4-benzodioxine-6-carboxylate —— C21H21NO5S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,3-dihydro-1,4-benzodioxine-6-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-oxo-1H-pyridine-3-carboxylate —— C18H18N2O4S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-oxo-1H-pyridine-3-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-methylsulfanylpyridine-3-carboxylate —— C19H20N2O3S2
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-methylsulfanylpyridine-3-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-oxochromene-3-carboxylate —— C22H19NO5S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-oxochromene-3-carboxylate
—— 2-(N-methylanilino)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H22N2OS
2-(N-methylanilino)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [(1S)-2-(cyclopropylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C21H20N2O4S
[(1S)-2-(cyclopropylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(1S)-2-(diethylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C22H24N2O4S
[(1S)-2-(diethylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H20N4O4S
[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate