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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1S)-1-phenylethyl]acetamide —— C22H19N3O2S
2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1S)-1-phenylethyl]acetamide
—— N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C23H28N4O2S
N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— 2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1R)-1-phenylethyl]acetamide —— C22H19N3O2S
2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1R)-1-phenylethyl]acetamide
—— 2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C24H23N3O2S
2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— 4-[(Z)-(4,4-dimethyl-3,3a-dihydro-2H-cyclopenta[c][1,5]benzothiazepin-1-ylidene)methyl]-N,N-dimethylaniline —— C23H26N2S
4-[(Z)-(4,4-dimethyl-3,3a-dihydro-2H-cyclopenta[c][1,5]benzothiazepin-1-ylidene)methyl]-N,N-dimethylaniline
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C22H21N3O3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-pyrazol-1-ylbenzoate —— C22H21N3O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-pyrazol-1-ylbenzoate
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27FN2O4S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27FN2O4S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(4-fluorophenyl)imidazole-4-carboxylate —— C22H20FN3O3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(4-fluorophenyl)imidazole-4-carboxylate
—— (3R)-1-(4-methylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide —— C28H27N3O3S
(3R)-1-(4-methylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide
—— (3R)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)-1-phenylpyrrolidine-3-carboxamide —— C27H25N3O3S
(3R)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)-1-phenylpyrrolidine-3-carboxamide
—— N-[(2S)-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]propan-2-yl]benzamide —— C26H25N3O3S
N-[(2S)-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]propan-2-yl]benzamide
—— (3R)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-5-oxo-1-phenylpyrrolidine-3-carboxamide —— C27H25N3O4S
(3R)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-5-oxo-1-phenylpyrrolidine-3-carboxamide
—— 1-[7-[(3S)-3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C26H33N3O3S2
1-[7-[(3S)-3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— ethyl 4-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]piperidine-1-carboxylate —— C18H25N3O5S2
ethyl 4-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]piperidine-1-carboxylate
—— (3S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H14ClF3N2O3S2
(3S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(2,4-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(3R)-N-(2,4-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(2,5-dimethylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3S)-N-(2,5-dimethylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 5-[4-ethyl-3-[[(3R)-3-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]phenyl]-3-methyl-1,2-oxazole —— C22H24N2O3S2
5-[4-ethyl-3-[[(3R)-3-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]phenyl]-3-methyl-1,2-oxazole
—— ethyl 4-[[(3S)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]piperidine-1-carboxylate —— C18H25N3O5S2
ethyl 4-[[(3S)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]piperidine-1-carboxylate
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]urea —— C23H28N4O2S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]urea
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[[(2S)-oxolan-2-yl]methyl]urea —— C21H23N3O3S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[[(2S)-oxolan-2-yl]methyl]urea
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[[(2R)-oxolan-2-yl]methyl]urea —— C21H23N3O3S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[[(2R)-oxolan-2-yl]methyl]urea
—— (11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O4S
(11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O4S
(11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H28N2O3S
(11S)-5-benzyl-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(3-chlorophenyl)methyl]-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O4S
(11R)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-(3-methoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O4S
(11R)-5-[(3-chlorophenyl)methyl]-N-(3-methoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-(4-fluorophenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H18ClFN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-(4-fluorophenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H19ClN2O3S2
(11R)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27ClN2O4S
(11S)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-3-(1,3-dihydroisoindole-2-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H21ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-3-(1,3-dihydroisoindole-2-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-butyl-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11R)-N-butyl-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-benzyl-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11S)-N-benzyl-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-(3-ethoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25ClN2O4S
(11R)-5-[(3-chlorophenyl)methyl]-N-(3-ethoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N,N-diethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N,N-diethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl (3R)-1-[5-[(2-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate —— C30H30N2O4S
ethyl (3R)-1-[5-[(2-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate
—— (11S)-5-[(3-chlorophenyl)methyl]-N-(2,2-dimethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O5S
(11S)-5-[(3-chlorophenyl)methyl]-N-(2,2-dimethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C26H23ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(3-chlorophenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28ClN3O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C26H23ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one