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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2-fluorophenyl)methyl]-3-[(2S)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O4S
5-[(2-fluorophenyl)methyl]-3-[(2S)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— 5-[(4-chlorophenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O4S
5-[(4-chlorophenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-3-(4-benzylpiperazine-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H27N3O3S
(11R)-3-(4-benzylpiperazine-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O4S
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O4S
5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-benzyl-3-[(2R)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C27H26N2O4S
5-benzyl-3-[(2R)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— 5-ethyl-6,11,11-trioxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O4S
5-ethyl-6,11,11-trioxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H34N2O4S
N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H28N2O4S
N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl (3R)-1-(5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carbonyl)piperidine-3-carboxylate —— C24H26N2O6S
ethyl (3R)-1-(5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carbonyl)piperidine-3-carboxylate
—— 5-ethyl-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H31N3O4S
5-ethyl-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H26N2O5S
(11S)-5-benzyl-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-[2-(3,4-diethoxyphenyl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H30N2O5S
(11R)-N-[2-(3,4-diethoxyphenyl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H29N3O3S
(11S)-5-ethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-N-(2-morpholin-4-ylethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C22H25N3O4S
(11S)-5-ethyl-N-(2-morpholin-4-ylethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-chlorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O4S
5-[(4-chlorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C23H26N2O4S
3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-[2-(4-benzylpiperazin-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H32N4O3S
(11S)-N-[2-(4-benzylpiperazin-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O3S
(11R)-5-benzyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H34N2O4S
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H28N2O4S
N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-methylphenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O4S
3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-methylphenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— N-(furan-2-ylmethyl)-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C22H18N2O3S
N-(furan-2-ylmethyl)-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-fluorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O4S
5-[(4-fluorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O4S
3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-ethyl-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11S)-5-ethyl-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C23H26N2O3S
(11R)-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— ethyl (3S)-1-(5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carbonyl)piperidine-3-carboxylate —— C24H26N2O6S
ethyl (3S)-1-(5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carbonyl)piperidine-3-carboxylate
—— 5-ethyl-6,11,11-trioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C24H22N2O4S
5-ethyl-6,11,11-trioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2O3S
(11S)-5-ethyl-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(4-benzylpiperidine-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H28N2O3S
(11R)-3-(4-benzylpiperidine-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H33N3O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(2-cyanoethyl)-5-[(4-fluorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H20FN3O3S
(11R)-N-(2-cyanoethyl)-5-[(4-fluorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-propan-2-ylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-propan-2-ylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O4S
(11R)-5-[(4-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-methylphenyl)methyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H33N3O4S
5-[(3-methylphenyl)methyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28N2O5S
5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H29N3O3S
(11S)-5-benzyl-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 10-allyl-N-[2-(4-chlorophenyl)ethyl]-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C25H21ClN2O2S
10-allyl-N-[2-(4-chlorophenyl)ethyl]-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O4S
(11S)-5-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[2-(dimethylamino)ethyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H29N3O3S
(11R)-N-[2-(dimethylamino)ethyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[2-(azepan-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H29N3O3S
(11S)-N-[2-(azepan-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O4S
5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-fluorophenyl)methyl]-6,11,11-trioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O4S
5-[(2-fluorophenyl)methyl]-6,11,11-trioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-benzyl-3-[(2S)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C27H26N2O4S
5-benzyl-3-[(2S)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H32N2O4S
(11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-(2,2-dimethoxyethyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C20H22N2O5S
(11S)-N-(2,2-dimethoxyethyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[3-[butyl(methyl)amino]propyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H37N3O3S
(11S)-N-[3-[butyl(methyl)amino]propyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide