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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(2-methoxy-5-nitrophenoxy)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H20N2O5S
2-(2-methoxy-5-nitrophenoxy)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-(2-methoxy-5-nitrophenoxy)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H20N2O5S
2-(2-methoxy-5-nitrophenoxy)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[[1-(difluoromethyl)imidazol-2-yl]methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H22F2N4OS
2-[[1-(difluoromethyl)imidazol-2-yl]methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[[1-(difluoromethyl)imidazol-2-yl]methyl-methylamino]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H22F2N4OS
2-[[1-(difluoromethyl)imidazol-2-yl]methyl-methylamino]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-[(2R)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C21H18F3N3O2S
[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-[(2R)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 2-[2-[(2R)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C19H17F3N4O2S
2-[2-[(2R)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— [4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-[(2S)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C21H18F3N3O2S
[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-[(2S)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 1-[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]ethanone —— C21H28ClN3OS
1-[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]ethanone
—— 1-[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]ethanone —— C21H28ClN3OS
1-[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]ethanone
—— 3-ethyl-7-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1H-quinazoline-2,4-dione —— C21H21N3O3S
3-ethyl-7-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1H-quinazoline-2,4-dione
—— 3-ethyl-7-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1H-quinazoline-2,4-dione —— C21H21N3O3S
3-ethyl-7-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1H-quinazoline-2,4-dione
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-2-cyano-3-(furan-2-yl)prop-2-enoate —— C20H18N2O4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-2-cyano-3-(furan-2-yl)prop-2-enoate
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-(4-nitrophenoxy)propan-1-one —— C19H20N2O4S
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-(4-nitrophenoxy)propan-1-one
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-(4-nitrophenoxy)propan-1-one —— C19H20N2O4S
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-(4-nitrophenoxy)propan-1-one
—— 3-[3-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]phenyl]-1,3-oxazolidin-2-one —— C20H20N2O3S
3-[3-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]phenyl]-1,3-oxazolidin-2-one
—— 3-[3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]phenyl]-1,3-oxazolidin-2-one —— C20H20N2O3S
3-[3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]phenyl]-1,3-oxazolidin-2-one
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone —— C20H20N4OS2
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone —— C20H20N4OS2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone
—— 2-[(5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl)sulfanyl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H21N5OS2
2-[(5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl)sulfanyl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (3-bromothiophen-2-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C15H14BrNOS2
(3-bromothiophen-2-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 2-[(5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl)sulfanyl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H21N5OS2
2-[(5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidin-3-yl)sulfanyl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (3-bromothiophen-2-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C15H14BrNOS2
(3-bromothiophen-2-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(3,4-dimethylphenyl)acetate —— C22H25NO3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(3,4-dimethylphenyl)acetate
—— [(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]methanone —— C21H29N3O2S
[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]methanone
—— [(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]methanone —— C21H29N3O2S
[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]methanone
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone —— C21H21N3O2S2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone
—— (2R)-4-(4-bromophenyl)-2-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepine —— C22H18BrNOS
(2R)-4-(4-bromophenyl)-2-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepine
—— (2R)-2-(3-bromophenyl)-4-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepine —— C22H18BrNOS
(2R)-2-(3-bromophenyl)-4-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepine
—— (2S)-2-(3-bromophenyl)-4-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepine —— C22H18BrNOS
(2S)-2-(3-bromophenyl)-4-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazepine
—— 2-(4-chlorophenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H18ClNOS2
2-(4-chlorophenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-(4-chlorophenyl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H18ClNOS2
2-(4-chlorophenyl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-tert-butylbenzoate —— C23H27NO3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-tert-butylbenzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-tert-butylbenzoate —— C23H27NO3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-tert-butylbenzoate
—— 1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-5-nitropyridin-2-one —— C17H17N3O4S
1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-5-nitropyridin-2-one
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanyl)ethanone —— C18H18N4OS2
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanyl)ethanone
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanyl)ethanone —— C18H18N4OS2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanyl)ethanone
—— 2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C20H21N3OS3
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(1-methyl-4-piperidin-1-ylsulfonylpyrrol-2-yl)methanone —— C21H27N3O3S2
[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(1-methyl-4-piperidin-1-ylsulfonylpyrrol-2-yl)methanone
—— [(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(1-methyl-4-piperidin-1-ylsulfonylpyrrol-2-yl)methanone —— C21H27N3O3S2
[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(1-methyl-4-piperidin-1-ylsulfonylpyrrol-2-yl)methanone
—— 11-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-12-one —— C21H21N3O2S2
11-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-12-one
—— (4S)-1-(2,4-difluorophenyl)-4-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyrrolidin-2-one —— C21H20F2N2O2S
(4S)-1-(2,4-difluorophenyl)-4-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyrrolidin-2-one
—— (4S)-1-(2,4-difluorophenyl)-4-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyrrolidin-2-one —— C21H20F2N2O2S
(4S)-1-(2,4-difluorophenyl)-4-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyrrolidin-2-one
—— (4R)-1-(2,4-difluorophenyl)-4-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyrrolidin-2-one —— C21H20F2N2O2S
(4R)-1-(2,4-difluorophenyl)-4-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyrrolidin-2-one
—— 5-[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1-methylpyridin-2-one —— C17H17ClN2O2S
5-[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1-methylpyridin-2-one
—— 5-[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1-methylpyridin-2-one —— C17H17ClN2O2S
5-[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1-methylpyridin-2-one
—— 1-[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-methylsulfonylpropan-1-one —— C14H18ClNO3S2
1-[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-methylsulfonylpropan-1-one
—— 1-[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-methylsulfonylpropan-1-one —— C14H18ClNO3S2
1-[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-methylsulfonylpropan-1-one
—— [(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[(2S)-1,4-dioxan-2-yl]methanone —— C15H18ClNO3S
[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[(2S)-1,4-dioxan-2-yl]methanone
—— [(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[(2S)-1,4-dioxan-2-yl]methanone —— C15H18ClNO3S
[(2S)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[(2S)-1,4-dioxan-2-yl]methanone
—— [(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[(2R)-1,4-dioxan-2-yl]methanone —— C15H18ClNO3S
[(2R)-7-chloro-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[(2R)-1,4-dioxan-2-yl]methanone