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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2S)-oxolan-2-yl]methyl 5-[(2,5-dimethylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C28H27NO4S
[(2S)-oxolan-2-yl]methyl 5-[(2,5-dimethylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— N-(furan-2-ylmethyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C22H27N3O5S2
N-(furan-2-ylmethyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— [(2R)-oxolan-2-yl]methyl 5-[(2-chloro-4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H21ClFNO4S
[(2R)-oxolan-2-yl]methyl 5-[(2-chloro-4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— ethyl (3R)-3-(4-methylphenyl)-3-[(4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl)sulfonylamino]propanoate —— C21H24N2O5S2
ethyl (3R)-3-(4-methylphenyl)-3-[(4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl)sulfonylamino]propanoate
—— (3R)-N-(furan-2-ylmethyl)-3-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O4S2
(3R)-N-(furan-2-ylmethyl)-3-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(2-ethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O4S2
(2S)-N-[(2-ethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[3-(N-ethylanilino)propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O3S2
(3R)-N-[3-(N-ethylanilino)propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-[(3R)-3-(azepan-1-yl)butyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H29N3O3S2
N-[(3R)-3-(azepan-1-yl)butyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2R)-2-ethyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H20N2O3S3
7-[[(2R)-2-ethyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-3-methyl-4-oxo-N-[[1-(2-thiophen-2-ylethyl)piperidin-4-yl]methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O3S3
(3S)-3-methyl-4-oxo-N-[[1-(2-thiophen-2-ylethyl)piperidin-4-yl]methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[(2-ethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O4S2
(3S)-N-[(2-ethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(furan-2-ylmethyl)-3-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O4S2
(3S)-N-(furan-2-ylmethyl)-3-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[3-(furan-2-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O4S2
(2S)-N-[3-(furan-2-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[3-(furan-2-yl)propyl]-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H22N2O4S2
(2S)-N-[3-(furan-2-yl)propyl]-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-(4-sulfamoylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O5S3
(3S)-3-methyl-4-oxo-N-(4-sulfamoylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3-methoxypropyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C14H20N2O4S2
(3S)-N-(3-methoxypropyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-benzyl-2-methyl-4-oxo-N-propan-2-yl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O3S2
(2S)-N-benzyl-2-methyl-4-oxo-N-propan-2-yl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-ethyl-N-(4-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O4S2
(3R)-N-ethyl-N-(4-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-butyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H24N2O3S3
(3R)-N-butyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-2-methyl-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S3
(2S)-2-methyl-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(2-fluorophenyl)-2-methyl-4-oxo-N-propyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H21FN2O3S2
(2R)-N-(2-fluorophenyl)-2-methyl-4-oxo-N-propyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(3-cyanophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15N3O3S2
(3R)-N-(3-cyanophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-7-[4-[cyclohexyl(methyl)amino]piperidin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C22H33N3O3S2
(3S)-7-[4-[cyclohexyl(methyl)amino]piperidin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-N-[(2,5-dimethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O5S2
(3S)-N-[(2,5-dimethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(2-ethyl-6-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(2S)-N-(2-ethyl-6-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-cyclopentyl-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(3S)-N-cyclopentyl-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(4-cyanophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15N3O3S2
(2R)-N-(4-cyanophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— methyl 3-[N-[[(3S)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C20H22N2O5S2
methyl 3-[N-[[(3S)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— (2S)-N-(3-chloro-4-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17ClN2O3S2
(2S)-N-(3-chloro-4-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-N-[(3-methylphenyl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3R)-3-methyl-N-[(3-methylphenyl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(2-chlorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H15ClN2O3S2
(2R)-N-(2-chlorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[(3,4-dimethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O5S2
(3R)-N-[(3,4-dimethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2R)-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C18H18N2O4S2
7-[[(2R)-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-2-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C15H16N2O3S3
(2S)-2-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-[3-(pyrrolidin-1-ylmethyl)phenyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H25N3O3S2
(3S)-3-methyl-4-oxo-N-[3-(pyrrolidin-1-ylmethyl)phenyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(1,3-benzodioxol-5-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H16N2O5S2
(2S)-N-(1,3-benzodioxol-5-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[(4-fluorophenyl)methyl]-3-methyl-4-oxo-N-(pyridin-3-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C23H22FN3O3S2
(3R)-N-[(4-fluorophenyl)methyl]-3-methyl-4-oxo-N-(pyridin-3-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-[4-(trifluoromethoxy)phenyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15F3N2O4S2
(3S)-3-methyl-4-oxo-N-[4-(trifluoromethoxy)phenyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-5-acetyl-2-methyl-N-(2,4,6-trimethylphenyl)-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H26N2O3S2
(2S)-5-acetyl-2-methyl-N-(2,4,6-trimethylphenyl)-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[(2,5-dimethylphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(3R)-N-[(2,5-dimethylphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N,2-dimethyl-4-oxo-N-[(1-phenylpyrazol-4-yl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H22N4O3S2
(2R)-N,2-dimethyl-4-oxo-N-[(1-phenylpyrazol-4-yl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(2,5-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(3S)-N-(2,5-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(2,3-dimethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(2S)-N-(2,3-dimethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(4-bromo-3-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17BrN2O3S2
(2R)-N-(4-bromo-3-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-7-(4-piperidin-1-ylpiperidin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H29N3O3S2
(3S)-3-methyl-7-(4-piperidin-1-ylpiperidin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-N-cyclohexyl-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H24N2O3S2
(2R)-N-cyclohexyl-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(3,4-dimethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(2R)-N-(3,4-dimethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-7-[[3-[(4-fluorophenyl)methyl]-1,3-diazinan-1-yl]sulfonyl]-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C21H24FN3O3S2
(3S)-7-[[3-[(4-fluorophenyl)methyl]-1,3-diazinan-1-yl]sulfonyl]-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-2-methyl-7-[(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C21H22N2O3S2
(2S)-2-methyl-7-[(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-N-(1,3-benzodioxol-5-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H18N2O5S2
(3S)-N-(1,3-benzodioxol-5-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide