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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20ClN3O3S
(11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide —— C26H25N3O4S
N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide
—— 8-bromo-6-ethyl-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C21H21BrN2O2S
8-bromo-6-ethyl-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O2S
N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2-chlorophenyl)methyl]-2-[(2S)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]acetamide —— C24H21ClN2O4S
N-[(2-chlorophenyl)methyl]-2-[(2S)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]acetamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2-[(2S)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide —— C22H24N2O5S
N-[[(2S)-oxolan-2-yl]methyl]-2-[(2S)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide
—— 2-[(2R)-2-(3,4-dimethoxyphenyl)-1,1,4-trioxo-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]-N-(4-methylphenyl)acetamide —— C26H26N2O6S
2-[(2R)-2-(3,4-dimethoxyphenyl)-1,1,4-trioxo-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]-N-(4-methylphenyl)acetamide
—— 2-[(2S)-2-(3,4-dimethoxyphenyl)-1,1,4-trioxo-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]-N-(4-methylphenyl)acetamide —— C26H26N2O6S
2-[(2S)-2-(3,4-dimethoxyphenyl)-1,1,4-trioxo-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]-N-(4-methylphenyl)acetamide
—— N-(2-ethoxyphenyl)-2-[(2S)-2-methyl-1,1,4-trioxo-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide —— C20H22N2O5S
N-(2-ethoxyphenyl)-2-[(2S)-2-methyl-1,1,4-trioxo-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide
—— (2R)-1,1-dioxo-2-phenyl-5-propyl-2,3-dihydro-1λ6,5-benzothiazepin-4-one —— C18H19NO3S
(2R)-1,1-dioxo-2-phenyl-5-propyl-2,3-dihydro-1λ6,5-benzothiazepin-4-one
—— N-[[(2R)-oxolan-2-yl]methyl]-2-[(2R)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide —— C22H24N2O5S
N-[[(2R)-oxolan-2-yl]methyl]-2-[(2R)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide
—— N-(2-ethoxyphenyl)-2-[(2R)-2-methyl-1,1,4-trioxo-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide —— C20H22N2O5S
N-(2-ethoxyphenyl)-2-[(2R)-2-methyl-1,1,4-trioxo-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-[(2S)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide —— C22H24N2O5S
N-[[(2R)-oxolan-2-yl]methyl]-2-[(2S)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2-[(2R)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide —— C22H24N2O5S
N-[[(2S)-oxolan-2-yl]methyl]-2-[(2R)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1λ6,5-benzothiazepin-5-yl]acetamide
—— N-[(2-chlorophenyl)methyl]-2-[(2R)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]acetamide —— C24H21ClN2O4S
N-[(2-chlorophenyl)methyl]-2-[(2R)-1,1,4-trioxo-2-phenyl-2,3-dihydro-1lambda6,5-benzothiazepin-5-yl]acetamide
—— (3S,5S)-N-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3,5-dimethylpiperidine-1-carboxamide —— C28H29N3O2S
(3S,5S)-N-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3,5-dimethylpiperidine-1-carboxamide
—— 1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2S)-butan-2-yl]urea —— C25H25N3O2S
1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2S)-butan-2-yl]urea
—— 1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2S)-2-phenylpropyl]urea —— C30H27N3O2S
1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2S)-2-phenylpropyl]urea
—— 1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2R)-2-phenylpropyl]urea —— C30H27N3O2S
1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2R)-2-phenylpropyl]urea
—— 5-[(2-fluorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O2S
5-[(2-fluorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chlorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O2S
5-[(2-chlorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chlorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O2S
5-[(2-chlorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-fluorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O2S
5-[(4-fluorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O2S
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O2S
N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20ClN3O3S
(11S)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl (3S)-1-[5-[(3-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate —— C29H27FN2O4S
ethyl (3S)-1-[5-[(3-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[(3-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate —— C29H27FN2O4S
ethyl (3R)-1-[5-[(3-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate
—— (11R)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20ClN3O3S
(11R)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-fluorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O2S
5-[(4-fluorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-(6-methylpyridin-2-yl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20ClN3O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-(6-methylpyridin-2-yl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O2S
5-[(3-chlorophenyl)methyl]-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O2S
5-[(3-chlorophenyl)methyl]-N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (6R,7S)-6-phenyl-6,7-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol —— C18H15NOS
(6R,7S)-6-phenyl-6,7-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol
—— (11R)-5-benzyl-N-[2-(cyclohexen-1-yl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H28N2O3S
(11R)-5-benzyl-N-[2-(cyclohexen-1-yl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (2R)-2-(2-chloro-5-nitrophenyl)-4-naphthalen-1-yl-2,3-dihydro-1,5-benzothiazepine —— C25H17ClN2O2S
(2R)-2-(2-chloro-5-nitrophenyl)-4-naphthalen-1-yl-2,3-dihydro-1,5-benzothiazepine
—— ethyl 5-[(2S)-1-(2-methoxyanilino)-1-oxobutan-2-yl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C27H26N2O5S
ethyl 5-[(2S)-1-(2-methoxyanilino)-1-oxobutan-2-yl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— [(2S)-oxolan-2-yl]methyl 5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22FNO6S
[(2S)-oxolan-2-yl]methyl 5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-3-(4-ethylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H31N3O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-3-(4-ethylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— ethyl (3R)-1-(5-benzyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carbonyl)piperidine-3-carboxylate —— C29H28N2O6S
ethyl (3R)-1-(5-benzyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carbonyl)piperidine-3-carboxylate
—— ethyl 4-[[(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate —— C29H28FN3O5S
ethyl 4-[[(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate
—— [(2S)-oxolan-2-yl]methyl 5-[(4-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C27H25NO6S
[(2S)-oxolan-2-yl]methyl 5-[(4-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C33H30FN3O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— [(2R)-oxolan-2-yl]methyl 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C28H27NO6S
[(2R)-oxolan-2-yl]methyl 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C32H30N2O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— [(2R)-oxolan-2-yl]methyl 5-[(4-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C27H25NO6S
[(2R)-oxolan-2-yl]methyl 5-[(4-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— (11R)-5-ethyl-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C26H24FN3O3S
(11R)-5-ethyl-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H24N2O4S
(11R)-5-[(2,5-dimethylphenyl)methyl]-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— [(2S)-oxolan-2-yl]methyl 5-[(4-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22FNO6S
[(2S)-oxolan-2-yl]methyl 5-[(4-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— (11S)-N-benzyl-5-[(4-chlorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23ClN2O3S
(11S)-N-benzyl-5-[(4-chlorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide