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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (3R)-3-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)piperidine-1-carboxylate —— C18H24N2O3S
ethyl (3R)-3-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)piperidine-1-carboxylate
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-naphthalen-1-yloxyethanone —— C22H21NO2S
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-naphthalen-1-yloxyethanone
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(trifluoromethyl)benzoate —— C20H18F3NO3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(trifluoromethyl)benzoate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2R)-oxolan-2-yl]acetate —— C18H23NO4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2R)-oxolan-2-yl]acetate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2R)-oxolan-2-yl]acetate —— C18H23NO4S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2R)-oxolan-2-yl]acetate
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(2-nitrophenoxy)ethanone —— C18H18N2O4S
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(2-nitrophenoxy)ethanone
—— 2-(2,4-dichlorophenoxy)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H17Cl2NO2S
2-(2,4-dichlorophenoxy)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(2-nitrophenoxy)ethanone —— C18H18N2O4S
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(2-nitrophenoxy)ethanone
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[(5-thiophen-2-yl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone —— C18H18N4OS3
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[(5-thiophen-2-yl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanone
—— (3R)-5-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C20H20N4O2S
(3R)-5-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— (3S)-5-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C21H22N4O2S
(3S)-5-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— (3S)-5-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C21H22N4O2S
(3S)-5-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— (3R)-5-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C21H22N4O2S
(3R)-5-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— (3R)-5-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C21H22N4O2S
(3R)-5-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— (3S)-5-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C20H20N4O2S
(3S)-5-(3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl)-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-3-(furan-2-yl)prop-2-enoate —— C19H19NO4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-3-(furan-2-yl)prop-2-enoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-3-(furan-2-yl)prop-2-enoate —— C19H19NO4S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-3-(furan-2-yl)prop-2-enoate
—— 1-O-ethyl 4-O-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-but-2-enedioate —— C18H21NO5S
1-O-ethyl 4-O-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-but-2-enedioate
—— 6-(furan-2-yl)-3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1H-pyridin-2-one —— C20H18N2O3S
6-(furan-2-yl)-3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-1H-pyridin-2-one
—— [2-(naphthalen-1-ylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C22H18N2O4S
[2-(naphthalen-1-ylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(1-cyanocyclohexyl)-methylamino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H23N3O4S
[2-[(1-cyanocyclohexyl)-methylamino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (2-oxo-2-piperidin-1-ylethyl) 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C17H20N2O4S
(2-oxo-2-piperidin-1-ylethyl) 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(2-methyl-6-propan-2-ylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C22H24N2O4S
[2-(2-methyl-6-propan-2-ylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (2-ethoxyphenyl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H19NO4S
(2-ethoxyphenyl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(1R)-1-(2-chlorophenyl)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H16ClNO3S
[(1R)-1-(2-chlorophenyl)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (3-phenyl-1,2,4-oxadiazol-5-yl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H15N3O4S
(3-phenyl-1,2,4-oxadiazol-5-yl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(1,3-benzodioxol-5-ylmethylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H18N2O6S
[2-(1,3-benzodioxol-5-ylmethylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(azepan-1-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H22N2O4S
[2-(azepan-1-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(3-cyanoanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H15N3O4S
[2-(3-cyanoanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(2,6-dimethylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H20N2O4S
[2-(2,6-dimethylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H15FN2O3S2
[2-(4-fluorophenyl)-1,3-thiazol-4-yl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (4-methylsulfanylphenyl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H17NO3S2
(4-methylsulfanylphenyl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H22N2O5S
[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(5-chlorothiophen-2-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C16H12ClNO4S2
[2-(5-chlorothiophen-2-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(4-ethylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H20N2O4S
[2-(4-ethylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(2-methylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H18N2O4S
[2-(2-methylanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(4-methylpiperidin-1-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H22N2O4S
[2-(4-methylpiperidin-1-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-oxo-2-[[(2S)-4-phenylbutan-2-yl]amino]ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C22H24N2O4S
[2-oxo-2-[[(2S)-4-phenylbutan-2-yl]amino]ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(3-chloroanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H15ClN2O4S
[2-(3-chloroanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H22N2O4S
[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(4-fluoroanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H15FN2O4S
[2-(4-fluoroanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H24N2O4S
[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-oxo-2-(2,3,4-trifluoroanilino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H13F3N2O4S
[2-oxo-2-(2,3,4-trifluoroanilino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[2-[(2R)-butan-2-yl]anilino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C22H24N2O4S
[2-[2-[(2R)-butan-2-yl]anilino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(cyclopentylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C17H20N2O4S
[2-(cyclopentylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(cyclohexylmethylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H24N2O4S
[2-(cyclohexylmethylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (4,5-dimethoxy-2-methylphenyl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H21NO5S
(4,5-dimethoxy-2-methylphenyl)methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(3-methoxyanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H18N2O5S
[2-(3-methoxyanilino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C17H20N2O5S
[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(1-cyanocyclohexyl)amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H21N3O4S
[2-[(1-cyanocyclohexyl)amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate