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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11R)-5-[(4-chlorophenyl)methyl]-N-cyclohexyl-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-N-cyclohexyl-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28ClN3O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H25FN2O3S
(11S)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-(2,2-dimethoxyethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23FN2O5S
(11S)-N-(2,2-dimethoxyethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11S)-N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[(2S)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11R)-N-[(2S)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N,N-diethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N,N-diethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[3-(diethylamino)propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H30FN3O3S
(11R)-N-[3-(diethylamino)propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(2,2-dimethoxyethyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O5S
(11R)-N-(2,2-dimethoxyethyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-cyclopentyl-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23FN2O3S
(11R)-N-cyclopentyl-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-methylphenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C27H26N2O3S
(11S)-5-[(2-methylphenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-3-[(2S)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-3-[(2S)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-chlorophenyl)methyl]-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-cyclooctyl-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
(11R)-N-cyclooctyl-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-butyl-5-[(4-chlorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25ClN2O3S
(11R)-N-butyl-5-[(4-chlorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-(2,2-diethoxyethyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27FN2O5S
(11S)-N-(2,2-diethoxyethyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H25FN2O5S
(11S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H30N2O4S
(11S)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26N2O4S
(11R)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(2-methoxyphenyl)methyl]-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H26N2O4S
(11S)-N-[(2-methoxyphenyl)methyl]-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24ClN3O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(2,2-diethoxyethyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27FN2O5S
(11R)-N-(2,2-diethoxyethyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-butyl-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11S)-N-butyl-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-(3-methoxypropyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O4S
(11S)-N-(3-methoxypropyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-benzyl-5-[(2-fluorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11S)-N-benzyl-5-[(2-fluorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H22N2O3S2
(11S)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(2-methylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O3S
(11S)-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(2-methylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23FN2O4S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-cyclopropyl-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H19FN2O3S
(11S)-N-cyclopropyl-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-cycloheptyl-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O3S
(11R)-N-cycloheptyl-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-cyclopentyl-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide —— C19H18N2O2S
N-cyclopentyl-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-methoxyphenyl)methyl]-6-oxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C30H26N2O3S
5-[(3-methoxyphenyl)methyl]-6-oxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[[4-(trifluoromethyl)phenyl]methyl]benzo[b][1,4]benzothiazepin-6-one —— C29H27F3N2O2S
3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[[4-(trifluoromethyl)phenyl]methyl]benzo[b][1,4]benzothiazepin-6-one
—— N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O2S2
N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O2S2
N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-methoxyphenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30N2O3S
5-[(3-methoxyphenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[[4-(trifluoromethyl)phenyl]methyl]benzo[b][1,4]benzothiazepin-6-one —— C29H27F3N2O2S
3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[[4-(trifluoromethyl)phenyl]methyl]benzo[b][1,4]benzothiazepin-6-one
—— 2-(2-Fluorophenyl)-4-(thiophen-2-yl)-2,3-dihydro-1,5-benzothiazepine —— C19H14FNS2
2-(2-Fluorophenyl)-4-(thiophen-2-yl)-2,3-dihydro-1,5-benzothiazepine
—— 2-(2,4-Dichlorophenyl)-4-(thiophen-2-yl)-2,3-dihydrobenzo[b][1,4]thiazepine —— C19H13Cl2NS2
2-(2,4-Dichlorophenyl)-4-(thiophen-2-yl)-2,3-dihydrobenzo[b][1,4]thiazepine
—— 2-[2-(Difluoromethoxy)phenyl]-4-(thiophen-2-yl)-2,3-dihydro-1,5-benzothiazepine —— C20H15F2NOS2
2-[2-(Difluoromethoxy)phenyl]-4-(thiophen-2-yl)-2,3-dihydro-1,5-benzothiazepine