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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[5-[[5-(2-Sulfamoylphenyl)-2,3-dihydroindol-1-yl]methyl]-3-(trifluoromethyl)pyrazol-1-yl]benzenecarboximidamide —— C26H23F3N6O2S
3-[5-[[5-(2-Sulfamoylphenyl)-2,3-dihydroindol-1-yl]methyl]-3-(trifluoromethyl)pyrazol-1-yl]benzenecarboximidamide
—— 2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-methylsulfinyl-5-[3-(2,4,6-trimethylphenyl)-1,2,4-triaza-3-boranuidacyclopenta-3,5-dien-5-yl]-1H-pyrazol-2-ium-3-amine —— C21H20BCl2F3N6OS
2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-methylsulfinyl-5-[3-(2,4,6-trimethylphenyl)-1,2,4-triaza-3-boranuidacyclopenta-3,5-dien-5-yl]-1H-pyrazol-2-ium-3-amine
—— 4-tert-butyl-N-[3-(2-{[2-(hydroxymethyl)-5-pyrimidinyl]oxy}ethoxy)-1-methyl-4-(4-methylphenyl)-1H-pyrazol-5-yl]benzenesulfonamide —— C28H33N5O5S
4-tert-butyl-N-[3-(2-{[2-(hydroxymethyl)-5-pyrimidinyl]oxy}ethoxy)-1-methyl-4-(4-methylphenyl)-1H-pyrazol-5-yl]benzenesulfonamide
—— N-[5-[2-[5-(hydroxymethyl)pyrimidin-2-yl]oxyethoxy]-2-methyl-4-(4-methylphenyl)pyrazol-3-yl]-5-propan-2-ylpyridine-2-sulfonamide —— C26H30N6O5S
N-[5-[2-[5-(hydroxymethyl)pyrimidin-2-yl]oxyethoxy]-2-methyl-4-(4-methylphenyl)pyrazol-3-yl]-5-propan-2-ylpyridine-2-sulfonamide
—— N-[(2-hydroxy-2-phenyl)ethyl]-3-{[(1S,2R)-2-(4,5-diphenyloxazol-2-yl)-1-cyclopentyl]methyl}benzamide 262595-40-4 C36H34N2O3
N-[(2-hydroxy-2-phenyl)ethyl]-3-{[(1S,2R)-2-(4,5-diphenyloxazol-2-yl)-1-cyclopentyl]methyl}benzamide
—— 4-[({4-[-(3-fluorophenyl)-6-(trifluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]phenyl}sulfonyl)amino]-4-oxobutanoic acid 267235-74-5 C24H17F4N3O5S
4-[({4-[-(3-fluorophenyl)-6-(trifluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]phenyl}sulfonyl)amino]-4-oxobutanoic acid
—— 1-[(2-Methyl-1,3-benzothiazol-5-yl)oxy]-3-[4-[[2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]methyl]piperazin-1-yl]propan-2-ol —— C26H27F3N4O3S
1-[(2-Methyl-1,3-benzothiazol-5-yl)oxy]-3-[4-[[2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]methyl]piperazin-1-yl]propan-2-ol
—— (2S)-2-[(4-methoxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]propanoic acid —— C30H30N2O7
(2S)-2-[(4-methoxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]propanoic acid
—— Ethyl 3-[1-[2-[(4-carbamimidoylanilino)methyl]-1-methylbenzimidazol-5-yl]-5-phenylpyrazol-3-yl]propanoate —— C30H31N7O2
Ethyl 3-[1-[2-[(4-carbamimidoylanilino)methyl]-1-methylbenzimidazol-5-yl]-5-phenylpyrazol-3-yl]propanoate
—— 3-[3-Methyl-5-[[3-oxo-7-(2-sulfamoylphenyl)-1,4-benzoxazin-4-yl]methyl]pyrazol-1-yl]benzenecarboximidamide —— C26H24N6O4S
3-[3-Methyl-5-[[3-oxo-7-(2-sulfamoylphenyl)-1,4-benzoxazin-4-yl]methyl]pyrazol-1-yl]benzenecarboximidamide
—— 8-[5-[2-[(dimethylamino)methyl]azetidin-1-yl]sulfonyl-2-propoxyphenyl]-6-ethyl-1H-[1,2,4]triazolo[3,4-f]purin-5-one —— C23H30N8O4S
8-[5-[2-[(dimethylamino)methyl]azetidin-1-yl]sulfonyl-2-propoxyphenyl]-6-ethyl-1H-[1,2,4]triazolo[3,4-f]purin-5-one
—— 3-(2,6-Difluoro-4-methyl-benzyloxy)-5-(3-{4-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-butyl}-ureido)-isothiazole-4-carboxylic Acid Amide —— C23H32F2N6O4S
3-(2,6-Difluoro-4-methyl-benzyloxy)-5-(3-{4-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-butyl}-ureido)-isothiazole-4-carboxylic Acid Amide
—— 3-[5-Methyl-3-[3-oxo-7-(2-sulfamoylphenyl)-1,4-benzoxazine-4-carbonyl]pyrazol-1-yl]benzenecarboximidamide —— C26H22N6O5S
3-[5-Methyl-3-[3-oxo-7-(2-sulfamoylphenyl)-1,4-benzoxazine-4-carbonyl]pyrazol-1-yl]benzenecarboximidamide
—— N-[[1-(2,4-dichlorophenyl)-7-methoxy-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]adamantan-2-amine —— C28H29Cl2N3OS
N-[[1-(2,4-dichlorophenyl)-7-methoxy-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]adamantan-2-amine
—— 6-(1-Benzyl-3,5-diphenylpyrazol-4-yl)-2-[(4-methoxyphenyl)methyl]pyridazin-3-one —— C34H28N4O2
6-(1-Benzyl-3,5-diphenylpyrazol-4-yl)-2-[(4-methoxyphenyl)methyl]pyridazin-3-one
—— 2-[[4-(2-cyclopropylethoxy)phenyl]sulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]-N-hydroxyacetamide;hydrochloride —— C22H26ClN5O5S
2-[[4-(2-cyclopropylethoxy)phenyl]sulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]-N-hydroxyacetamide;hydrochloride
—— N'-[3-(2,6-dichloro-4-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(1,2,3,4-tetrahydronaphthalen-2-yl)ethane-1,2-diamine —— C27H29Cl2N5O
N'-[3-(2,6-dichloro-4-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(1,2,3,4-tetrahydronaphthalen-2-yl)ethane-1,2-diamine
—— 4-(5-(4-methoxyphenyl)pyrazol-3-yloxy)-6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)quinazoline —— C27H32N6O4
4-(5-(4-methoxyphenyl)pyrazol-3-yloxy)-6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)quinazoline
—— ethyl 2-butyl-5-chloro-1-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]imidazole-4-carboxylate —— C26H27ClN6O2
ethyl 2-butyl-5-chloro-1-[(1S)-5-[2-(2H-tetrazol-5-yl)phenyl]-2,3-dihydro-1H-inden-1-yl]imidazole-4-carboxylate
—— 4-[3-methyl-2-[3-(methylamino)propyl]-5-[3-(trifluoromethyl)phenyl]imidazol-4-yl]-N-[(1S)-1-phenylethyl]pyridin-2-amine —— C28H30F3N5
4-[3-methyl-2-[3-(methylamino)propyl]-5-[3-(trifluoromethyl)phenyl]imidazol-4-yl]-N-[(1S)-1-phenylethyl]pyridin-2-amine
—— 3-(6-aminohexyl)-1-(1H-indol-3-ylmethyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1,3-diazinan-4-one —— C28H32N6OS
3-(6-aminohexyl)-1-(1H-indol-3-ylmethyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1,3-diazinan-4-one
—— 2-[(3-Hydroxyphenoxy)carbonyl-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid —— C28H26N2O7
2-[(3-Hydroxyphenoxy)carbonyl-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid
—— 2-[1-[[2-[3-(Aminomethyl)phenyl]-5-methylpyrazol-3-yl]methyl]-2-methylbenzimidazol-5-yl]benzenesulfonamide —— C26H26N6O2S
2-[1-[[2-[3-(Aminomethyl)phenyl]-5-methylpyrazol-3-yl]methyl]-2-methylbenzimidazol-5-yl]benzenesulfonamide
—— 3-[1-(Dimethylsulfamoyl)-4,5-dihydroimidazol-2-yl]-4-[4-[2-[3-(methylamino)pyridin-2-yl]ethoxy]phenyl]butanoic acid —— C23H31N5O5S
3-[1-(Dimethylsulfamoyl)-4,5-dihydroimidazol-2-yl]-4-[4-[2-[3-(methylamino)pyridin-2-yl]ethoxy]phenyl]butanoic acid
—— Ethyl 2-[1,5-bis(4-methoxyphenyl)-3-[(3-methylanilino)methyl]pyrazol-4-yl]acetate —— C29H31N3O4
Ethyl 2-[1,5-bis(4-methoxyphenyl)-3-[(3-methylanilino)methyl]pyrazol-4-yl]acetate
—— 1-[3-[5-(4-chlorophenyl)-4-pyridin-4-yl-imidazol-2-yl]-2,4,6-trimethylbenzyl]-4-methylpiperazine —— C29H32ClN5
1-[3-[5-(4-chlorophenyl)-4-pyridin-4-yl-imidazol-2-yl]-2,4,6-trimethylbenzyl]-4-methylpiperazine
—— 2-[1-[2-[(4-Carbamimidoylanilino)methyl]-1-methylbenzimidazol-5-yl]-5-phenylpyrazol-3-yl]acetic acid —— C27H25N7O2
2-[1-[2-[(4-Carbamimidoylanilino)methyl]-1-methylbenzimidazol-5-yl]-5-phenylpyrazol-3-yl]acetic acid
—— 1-benzyl-3-[6-methyl-2,5-bis(methylsulfanyl)pyridin-3-yl]-1-[[3-(1H-pyrazol-5-yl)phenyl]methyl]urea —— C26H27N5OS2
1-benzyl-3-[6-methyl-2,5-bis(methylsulfanyl)pyridin-3-yl]-1-[[3-(1H-pyrazol-5-yl)phenyl]methyl]urea
—— 2-cyclopentyl-N-[(1S)-2-hydroxy-1-phenylethyl]-2-[4-[(2-phenylimidazol-1-yl)methyl]phenyl]acetamide —— C31H33N3O2
2-cyclopentyl-N-[(1S)-2-hydroxy-1-phenylethyl]-2-[4-[(2-phenylimidazol-1-yl)methyl]phenyl]acetamide
—— CP547632 —— C20H24ClF2N5O3S
CP547632
—— 1-(3-imidazol-1-ylphenyl)cyclobutan-1-amine —— C13H15N3
1-(3-imidazol-1-ylphenyl)cyclobutan-1-amine
—— N-[5-(3-chlorophenyl)-1H-pyrazol-3-yl]-1-methylsulfonylspiro[2H-indole-3,4'-piperidine]-1'-carboxamide —— C23H24ClN5O3S
N-[5-(3-chlorophenyl)-1H-pyrazol-3-yl]-1-methylsulfonylspiro[2H-indole-3,4'-piperidine]-1'-carboxamide
—— N-[2-(4-(benzoxazol-2-yl)benzyloxy)ethyl]-2-[3-(4-methylphenyl)prop-2-ynyloxy]ethanamine hydrochloride —— C28H28N2O3*ClH
N-[2-(4-(benzoxazol-2-yl)benzyloxy)ethyl]-2-[3-(4-methylphenyl)prop-2-ynyloxy]ethanamine hydrochloride
—— (4Z)-4-[[5-ethoxy-2-(3-methylphenyl)-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid —— C22H20N4O6S
(4Z)-4-[[5-ethoxy-2-(3-methylphenyl)-3-oxo-1H-pyrazol-4-yl]hydrazinylidene]-3-oxonaphthalene-1-sulfonic acid
—— 5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-trichloromethylthiopyrazole 120067-91-6 C12H4Cl5F3N4S
5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-trichloromethylthiopyrazole
—— 6-[4-(5,6-dihydro-4H-pyrimidin-1-yl)-phenyl]-1-(4-methoxy-phenyl)-3-trifluoromethyl-1,4,5,6-tetrahydro-pyrazolo[3,4-c]pyridin-7-one —— C24H22F3N5O2
6-[4-(5,6-dihydro-4H-pyrimidin-1-yl)-phenyl]-1-(4-methoxy-phenyl)-3-trifluoromethyl-1,4,5,6-tetrahydro-pyrazolo[3,4-c]pyridin-7-one
—— N-[4-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3,5-difluorobenzenesulfonamide —— C17H9F8N3O2S
N-[4-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3,5-difluorobenzenesulfonamide
—— 3-(3-aminopropyl)-1-[2-(1H-indol-3-yl)ethyl]-5-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-sulfanylideneimidazolidin-4-one —— C26H28N6OS
3-(3-aminopropyl)-1-[2-(1H-indol-3-yl)ethyl]-5-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-sulfanylideneimidazolidin-4-one
—— 3-(4-aminobutyl)-1-(1H-indol-3-ylmethyl)-5-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-sulfanylideneimidazolidin-4-one —— C26H28N6OS
3-(4-aminobutyl)-1-(1H-indol-3-ylmethyl)-5-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-sulfanylideneimidazolidin-4-one
—— N'-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfanyl)pyrazol-3-yl]-N,N-dimethylmethanimidamide —— C15H9Cl2F6N5S
N'-[5-cyano-2-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-(trifluoromethylsulfanyl)pyrazol-3-yl]-N,N-dimethylmethanimidamide
—— 3-[[4-[5-(4-Bromophenyl)tetrazol-2-yl]phenyl]sulfonylamino]propanoic acid —— C16H14BrN5O4S
3-[[4-[5-(4-Bromophenyl)tetrazol-2-yl]phenyl]sulfonylamino]propanoic acid
—— 3-[(4-Chloro-2,6-difluorophenyl)methoxy]-5-[2-(1-methylpyrrolidin-2-yl)ethylcarbamoylamino]-1,2-thiazole-4-carboxamide —— C19H22ClF2N5O3S
3-[(4-Chloro-2,6-difluorophenyl)methoxy]-5-[2-(1-methylpyrrolidin-2-yl)ethylcarbamoylamino]-1,2-thiazole-4-carboxamide
—— 1-(2,4-Dimethyl-1,3-thiazol-5-yl)-3-[(6-nitropyridin-2-yl)amino]-3-phenyl-2-pyridin-2-ylpropan-1-ol —— C24H23N5O3S
1-(2,4-Dimethyl-1,3-thiazol-5-yl)-3-[(6-nitropyridin-2-yl)amino]-3-phenyl-2-pyridin-2-ylpropan-1-ol
—— 3-(6-aminohexyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1-(thiophen-3-ylmethyl)-1,3-diazinan-4-one —— C24H29N5OS2
3-(6-aminohexyl)-6-(5-phenyl-1H-imidazol-2-yl)-2-sulfanylidene-1-(thiophen-3-ylmethyl)-1,3-diazinan-4-one
—— 1-(2,4,6-trichlorophenyl)-3-(methylthio)-6-(3-hydroxybenzyl)pyrazolo[3,4-d]pyrimidin-4-one —— C19H13Cl3N4O2S
1-(2,4,6-trichlorophenyl)-3-(methylthio)-6-(3-hydroxybenzyl)pyrazolo[3,4-d]pyrimidin-4-one
—— N-[[7-chloro-1-(2,4-dichlorophenyl)-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]pyrrolidin-1-amine —— C21H19Cl3N4S
N-[[7-chloro-1-(2,4-dichlorophenyl)-5H-isothiochromeno[4,3-c]pyrazol-3-yl]methyl]pyrrolidin-1-amine
—— 2-(4-Fluorophenyl)-1-(2-cyclopentylamino-4-pyrimidinyl)-5-(4-piperidinyl)imidazo[4,5-b]pyridine 337902-58-6 C26H28FN7
2-(4-Fluorophenyl)-1-(2-cyclopentylamino-4-pyrimidinyl)-5-(4-piperidinyl)imidazo[4,5-b]pyridine
—— 2-[[5-[4-[(2-Butylbenzimidazol-1-yl)methyl]phenyl]tetrazol-2-yl]methyl]benzoic acid —— C27H26N6O2
2-[[5-[4-[(2-Butylbenzimidazol-1-yl)methyl]phenyl]tetrazol-2-yl]methyl]benzoic acid
—— 2-[[5-[3-Methoxy-4-[[methyl(2-methylpropoxycarbonyl)amino]methyl]phenyl]tetrazol-2-yl]methyl]benzoic acid —— C23H27N5O5
2-[[5-[3-Methoxy-4-[[methyl(2-methylpropoxycarbonyl)amino]methyl]phenyl]tetrazol-2-yl]methyl]benzoic acid
—— 6-chloro-3-(4-fluorophenyl)-2-(4-methylsulfonylphenyl)-9H-pyrazolo[5,1-b][1,3]benzoxazine —— C23H16ClFN2O3S
6-chloro-3-(4-fluorophenyl)-2-(4-methylsulfonylphenyl)-9H-pyrazolo[5,1-b][1,3]benzoxazine