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—— 6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C26H30FN5O3S
6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-chloro-2-[5-(4-ethylphenyl)-3-(furan-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]-4-phenylquinazoline —— C29H23ClN4O
6-chloro-2-[5-(4-ethylphenyl)-3-(furan-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]-4-phenylquinazoline
—— 6-[(2,5-Dimethyl-1-phenylpyrrol-3-yl)methylidene]-2-hexyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H27N5OS
6-[(2,5-Dimethyl-1-phenylpyrrol-3-yl)methylidene]-2-hexyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-7-[4,6-bis(ethylamino)-1,3,5-triazin-2-yl]-6-hydroxy-6-(4-methoxyphenyl)-4,17-dithia-2,7,8-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),2,11(16)-trien-9-one —— C26H30N8O3S2
(6S)-7-[4,6-bis(ethylamino)-1,3,5-triazin-2-yl]-6-hydroxy-6-(4-methoxyphenyl)-4,17-dithia-2,7,8-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),2,11(16)-trien-9-one
—— 6-Hydroxy-5-[(4-hydroxy-1,3-dimethyl-2,6-dioxopyrimidin-5-yl)-pyridin-3-ylmethyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H19N5O6
6-Hydroxy-5-[(4-hydroxy-1,3-dimethyl-2,6-dioxopyrimidin-5-yl)-pyridin-3-ylmethyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-3-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C22H24FN3O2S
6-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-3-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— 6-[(2S)-2-ethylpiperidine-1-carbonyl]-5-methyl-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C23H32N4O3S
6-[(2S)-2-ethylpiperidine-1-carbonyl]-5-methyl-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C26H30ClN5O3S
6-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 6-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C26H30ClN5O3S
6-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— (6R)-7-[4,6-bis(ethylamino)-1,3,5-triazin-2-yl]-6-hydroxy-6-(4-methoxyphenyl)-4,17-dithia-2,7,8-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),2,11(16)-trien-9-one —— C26H30N8O3S2
(6R)-7-[4,6-bis(ethylamino)-1,3,5-triazin-2-yl]-6-hydroxy-6-(4-methoxyphenyl)-4,17-dithia-2,7,8-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),2,11(16)-trien-9-one
—— 6-[[8-[2-(3-Methoxyphenyl)acetyl]-2,8-diazaspiro[4.5]decan-2-yl]methyl]-2-methylsulfanylpyridine-3-carbonitrile —— C25H30N4O2S
6-[[8-[2-(3-Methoxyphenyl)acetyl]-2,8-diazaspiro[4.5]decan-2-yl]methyl]-2-methylsulfanylpyridine-3-carbonitrile
—— 6-chloro-N-(2,6-dimethoxypyridin-3-yl)-N-methylsulfonylpyridine-2-carboxamide —— C14H14ClN3O5S
6-chloro-N-(2,6-dimethoxypyridin-3-yl)-N-methylsulfonylpyridine-2-carboxamide
—— 6-Iodo-2-[(1-methyl-2-oxoindol-3-ylidene)methyl]-3-(3-methylphenyl)quinazolin-4-one —— C25H18IN3O2
6-Iodo-2-[(1-methyl-2-oxoindol-3-ylidene)methyl]-3-(3-methylphenyl)quinazolin-4-one
—— (6R)-N-(2,4-dimethoxyphenyl)-2-[(2,3-dimethoxyphenyl)methylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C27H32N2O5S
(6R)-N-(2,4-dimethoxyphenyl)-2-[(2,3-dimethoxyphenyl)methylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-(5-Bromo-2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-5-carbaldehyde —— C13H9BrN2O2S
6-(5-Bromo-2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-5-carbaldehyde
—— 6-(dibutylsulfamoyl)-2-oxo-N-[(1R)-1-phenylethyl]-1H-quinoline-4-carboxamide —— C26H33N3O4S
6-(dibutylsulfamoyl)-2-oxo-N-[(1R)-1-phenylethyl]-1H-quinoline-4-carboxamide
—— (6S)-2-[(2,3-dimethoxyphenyl)methylamino]-N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H30N2O4S
(6S)-2-[(2,3-dimethoxyphenyl)methylamino]-N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[[1-(3,5-Dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-methylphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H25N5OS
6-[[1-(3,5-Dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-methylphenyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-methyl-N-[4-(2-phenylethenyl)phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H23NOS
6-methyl-N-[4-(2-phenylethenyl)phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(2S)-2-ethylpiperidine-1-carbonyl]-3-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C22H24FN3O2S
6-[(2S)-2-ethylpiperidine-1-carbonyl]-3-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— 6-[(2R)-2-ethylpiperidine-1-carbonyl]-3-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-one —— C22H24FN3O2S
6-[(2R)-2-ethylpiperidine-1-carbonyl]-3-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidin-4-one
—— (6R)-N-(2-methoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H26N2O3S
(6R)-N-(2-methoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-(4-methoxyphenyl)-9-(4-methylphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H30N2O3
6-(4-methoxyphenyl)-9-(4-methylphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-N-(2,5-dimethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H34N2O6S
(6R)-N-(2,5-dimethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-(2-methoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C27H32N2O5S
(6R)-N-(2-methoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(4-ethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H34N2O5S
(6S)-N-(4-ethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-(2-ethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H34N2O5S
(6R)-N-(2-ethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-(2,4-dimethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H34N2O6S
(6R)-N-(2,4-dimethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(2-methoxyphenyl)-6-methyl-2-(pyridin-4-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H25N3O2S
(6S)-N-(2-methoxyphenyl)-6-methyl-2-(pyridin-4-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-(2,4-dimethoxyphenyl)-6-methyl-2-(thiophen-2-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H26N2O3S2
(6R)-N-(2,4-dimethoxyphenyl)-6-methyl-2-(thiophen-2-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(2,4-dimethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H34N2O6S
(6S)-N-(2,4-dimethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(2-ethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H34N2O5S
(6S)-N-(2-ethoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-ethyl-4-(ethylsulfanyl)-6-methyl-2-(propylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine —— C17H24N2OS3
6-ethyl-4-(ethylsulfanyl)-6-methyl-2-(propylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine
—— (6R)-N-(2-methoxyphenyl)-6-methyl-2-(pyridin-4-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H25N3O2S
(6R)-N-(2-methoxyphenyl)-6-methyl-2-(pyridin-4-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-Chloro-9-[(4-chlorophenyl)methyl]-3,4-dimethyl-8,10-dihydropyrano[2,3-f][1,3]benzoxazin-2-one —— C20H17Cl2NO3
6-Chloro-9-[(4-chlorophenyl)methyl]-3,4-dimethyl-8,10-dihydropyrano[2,3-f][1,3]benzoxazin-2-one
—— 6-[1,4-Diazepan-1-yl-(3,4-dimethoxyphenyl)methyl]isoquinoline —— C23H27N3O2
6-[1,4-Diazepan-1-yl-(3,4-dimethoxyphenyl)methyl]isoquinoline
—— 6-(1,4-Dioxa-8-azaspiro[4.5]decane-8-carbonyl)-2-(2-methylphenyl)-4,5-dihydropyridazin-3-one —— C19H23N3O4
6-(1,4-Dioxa-8-azaspiro[4.5]decane-8-carbonyl)-2-(2-methylphenyl)-4,5-dihydropyridazin-3-one
—— (6S,7R)-7-[[(2R)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H21ClN6O4S3
(6S,7R)-7-[[(2R)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S)-N-(4-ethoxyphenyl)-6-methyl-2-(thiophen-2-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H26N2O2S2
(6S)-N-(4-ethoxyphenyl)-6-methyl-2-(thiophen-2-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-(4-Ethylsulfonylphenyl)imidazo[2,1-b][1,3]thiazole-5-carbaldehyde —— C14H12N2O3S2
6-(4-Ethylsulfonylphenyl)imidazo[2,1-b][1,3]thiazole-5-carbaldehyde
—— (6R)-N-(4-ethoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H28N2O3S
(6R)-N-(4-ethoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(2,4-dimethoxyphenyl)-2-[(2,3-dimethoxyphenyl)methylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C27H32N2O5S
(6S)-N-(2,4-dimethoxyphenyl)-2-[(2,3-dimethoxyphenyl)methylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-(4-ethoxyphenyl)-6-methyl-2-(thiophen-2-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H26N2O2S2
(6R)-N-(4-ethoxyphenyl)-6-methyl-2-(thiophen-2-ylmethylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(4-ethoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H28N2O3S
(6S)-N-(4-ethoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-N-(2-methoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C27H32N2O5S
(6S)-N-(2-methoxyphenyl)-6-methyl-2-[(2,3,4-trimethoxyphenyl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-(4-methoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H26N2O3S
(6R)-N-(4-methoxyphenyl)-6-methyl-2-[(5-methylfuran-2-yl)methylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-2-[(2,3-dimethoxyphenyl)methylamino]-N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H30N2O4S
(6R)-2-[(2,3-dimethoxyphenyl)methylamino]-N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S,7S)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-[3-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H19F3N6O4S3
(6S,7S)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-[3-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,7S)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-[3-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H19F3N6O4S3
(6R,7S)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-[3-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7R)-7-[[2-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H19F3N8O4S2
(6S,7R)-7-[[2-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid