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—— (6R,7S)-7-[[2-[4-chloro-3-(difluoromethyl)-5-methylpyrazol-1-yl]acetyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C18H17ClF2N6O4S3
(6R,7S)-7-[[2-[4-chloro-3-(difluoromethyl)-5-methylpyrazol-1-yl]acetyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-O-ethyl 8-O-propan-2-yl 5-amino-7-(2-fluorophenyl)-2-[(2-fluorophenyl)methylidene]-3-oxo-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate —— C27H24F2N2O5S
6-O-ethyl 8-O-propan-2-yl 5-amino-7-(2-fluorophenyl)-2-[(2-fluorophenyl)methylidene]-3-oxo-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate
—— (6R,7S)-7-[[2-[4-chloro-3-(difluoromethyl)-5-methylpyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17ClF2N8O4S2
(6R,7S)-7-[[2-[4-chloro-3-(difluoromethyl)-5-methylpyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7S)-7-[[2-[5-cyclopropyl-3-(difluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H20F2N8O4S2
(6S,7S)-7-[[2-[5-cyclopropyl-3-(difluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7R)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-[[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C18H17F3N6O4S3
(6S,7R)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-[[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7R)-7-[[2-[4-chloro-3-(difluoromethyl)-5-methylpyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17ClF2N8O4S2
(6S,7R)-7-[[2-[4-chloro-3-(difluoromethyl)-5-methylpyrazol-1-yl]acetyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7S)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17F3N8O4S2
(6S,7S)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R)-2-(3,5-dichloro-4-hydroxyphenyl)imino-3-ethyl-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C20H19Cl2N3O4S
(6R)-2-(3,5-dichloro-4-hydroxyphenyl)imino-3-ethyl-N-(4-methoxyphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-Benzyl-2,5-dimethyl-7-(4-methylpiperidin-1-yl)-3-phenylpyrazolo[1,5-a]pyrimidine —— C27H30N4
6-Benzyl-2,5-dimethyl-7-(4-methylpiperidin-1-yl)-3-phenylpyrazolo[1,5-a]pyrimidine
—— (6R,7R)-7-[[2-[5-cyclopropyl-3-(difluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H20F2N6O4S3
(6R,7R)-7-[[2-[5-cyclopropyl-3-(difluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7S)-7-[[(2R)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)butanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H23ClN6O4S3
(6S,7S)-7-[[(2R)-2-(4-chloro-3,5-dimethylpyrazol-1-yl)butanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S)-N-(3,5-dichlorophenyl)-2-(4-methoxyphenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamide —— C19H17Cl2N3O3S
(6S)-N-(3,5-dichlorophenyl)-2-(4-methoxyphenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-3-prop-2-enyl-1,3-thiazinane-6-carboxamide —— C22H22FN3O3S
(6R)-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-3-prop-2-enyl-1,3-thiazinane-6-carboxamide
—— 6-Chloro-2-(1-oxo-1-phenylpropan-2-yl)isoquinolin-1-one —— C18H14ClNO2
6-Chloro-2-(1-oxo-1-phenylpropan-2-yl)isoquinolin-1-one
—— (6R)-N-(4-bromophenyl)-2-(4-fluorophenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamide —— C18H15BrFN3O2S
(6R)-N-(4-bromophenyl)-2-(4-fluorophenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-3-benzyl-N-(3-chlorophenyl)-2-(4-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C24H19ClFN3O2S
(6R)-3-benzyl-N-(3-chlorophenyl)-2-(4-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-3-prop-2-enyl-1,3-thiazinane-6-carboxamide —— C22H22FN3O3S
(6S)-N-(4-ethoxyphenyl)-2-(2-fluorophenyl)imino-4-oxo-3-prop-2-enyl-1,3-thiazinane-6-carboxamide
—— (6R)-N-(3,5-dichlorophenyl)-2-(4-methoxyphenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamide —— C19H17Cl2N3O3S
(6R)-N-(3,5-dichlorophenyl)-2-(4-methoxyphenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S,7R)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H17F3N8O4S2
(6S,7R)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-bromo-N-[(6S)-3-carbamoyl-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-(3-methylphenyl)quinoline-4-carboxamide —— C31H32BrN3O2S
6-bromo-N-[(6S)-3-carbamoyl-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-(3-methylphenyl)quinoline-4-carboxamide
—— (6S,7S)-7-[[2-[5-cyclopropyl-3-(difluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C20H20F2N6O4S3
(6S,7S)-7-[[2-[5-cyclopropyl-3-(difluoromethyl)pyrazol-1-yl]acetyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S)-N-(3,5-dichlorophenyl)-3-methyl-4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide —— C19H14Cl2F3N3O2S
(6S)-N-(3,5-dichlorophenyl)-3-methyl-4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide
—— 6-ethyl-6-methyl-2-(propylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine-4-thiol —— C15H20N2OS3
6-ethyl-6-methyl-2-(propylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidine-4-thiol
—— (6R)-2-(3,5-dichloro-4-hydroxyphenyl)imino-3-ethyl-N-(3-methylphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C20H19Cl2N3O3S
(6R)-2-(3,5-dichloro-4-hydroxyphenyl)imino-3-ethyl-N-(3-methylphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(3,5-dichlorophenyl)-3-methyl-4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide —— C19H14Cl2F3N3O2S
(6R)-N-(3,5-dichlorophenyl)-3-methyl-4-oxo-2-[3-(trifluoromethyl)phenyl]imino-1,3-thiazinane-6-carboxamide
—— (6S)-3-benzyl-N-(3-chlorophenyl)-2-(4-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C24H19ClFN3O2S
(6S)-3-benzyl-N-(3-chlorophenyl)-2-(4-fluorophenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-3-[2-(4-chlorophenyl)ethyl]-N-methyl-4-oxo-2-phenylimino-1,3-thiazinane-6-carboxamide —— C20H20ClN3O2S
(6S)-3-[2-(4-chlorophenyl)ethyl]-N-methyl-4-oxo-2-phenylimino-1,3-thiazinane-6-carboxamide
—— 6-Amino-4-(2-propoxyphenyl)-3-(4-propoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C25H26N4O3
6-Amino-4-(2-propoxyphenyl)-3-(4-propoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-[[1-(2-Fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H24FN5OS
6-[[1-(2-Fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(1,3-benzodioxol-5-yl)-3-(furan-2-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C15H10N4O3S
6-(1,3-benzodioxol-5-yl)-3-(furan-2-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— 6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C26H28N6O3
6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-imino-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C27H30N6O3
6-imino-11-methyl-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1R)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C26H28N6O3
6-imino-7-(2-morpholin-4-ylethyl)-2-oxo-N-[(1R)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-[(5E)-5-[[(1R)-cyclohex-3-en-1-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C16H21NO3S2
6-[(5E)-5-[[(1R)-cyclohex-3-en-1-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-[(5E)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C19H19NO4S2
6-[(5E)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-Amino-4-{2-[(2-chlorobenzyl)oxy]-4-methoxyphenyl}-3-methyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H19ClN4O3
6-Amino-4-{2-[(2-chlorobenzyl)oxy]-4-methoxyphenyl}-3-methyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-[[1-(2,5-Dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H30N6O2S
6-[[1-(2,5-Dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-2-[5-(4-ethoxyphenyl)-3-(4-methylphenyl)-4,5-dihydro-1H-pyrazol-1-yl]-4-phenylquinazoline —— C32H27ClN4O
6-chloro-2-[5-(4-ethoxyphenyl)-3-(4-methylphenyl)-4,5-dihydro-1H-pyrazol-1-yl]-4-phenylquinazoline
—— (6S)-4-amino-6-tert-butyl-3-phenacylsulfanyl-1,6-dihydro-1,2,4-triazin-5-one —— C15H20N4O2S
(6S)-4-amino-6-tert-butyl-3-phenacylsulfanyl-1,6-dihydro-1,2,4-triazin-5-one
—— (6R)-4-amino-6-tert-butyl-3-phenacylsulfanyl-1,6-dihydro-1,2,4-triazin-5-one —— C15H20N4O2S
(6R)-4-amino-6-tert-butyl-3-phenacylsulfanyl-1,6-dihydro-1,2,4-triazin-5-one
—— 6-(Azepan-1-yl)-1,4-dimethyl-2-oxo-5-[(4-oxo-3-propyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile —— C21H26N4O2S2
6-(Azepan-1-yl)-1,4-dimethyl-2-oxo-5-[(4-oxo-3-propyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile
—— 6-ethyl-N-(3-methoxypropyl)-6-methyl-2-(methylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidin-4-amine —— C17H25N3O2S2
6-ethyl-N-(3-methoxypropyl)-6-methyl-2-(methylsulfanyl)-5,8-dihydro-6H-pyrano[4',3':4,5]thieno[2,3-d]pyrimidin-4-amine
—— 6-(2-Chlorophenyl)-4-[4-(2,4-dichlorophenoxy)phenyl]-8-methyl-9-[(3-phenoxyphenyl)methyl]-1-thia-4,6,7-triazaspiro[4.4]non-7-en-3-one —— C37H28Cl3N3O3S
6-(2-Chlorophenyl)-4-[4-(2,4-dichlorophenoxy)phenyl]-8-methyl-9-[(3-phenoxyphenyl)methyl]-1-thia-4,6,7-triazaspiro[4.4]non-7-en-3-one
—— (6R)-2-[4-(3,5-dimethyl-4-nitropyrazol-1-yl)butanoylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H25N5O4S
(6R)-2-[4-(3,5-dimethyl-4-nitropyrazol-1-yl)butanoylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(4-chlorophenyl)methylsulfanyl]-5-cyano-N-(2-methoxyphenyl)-2-methyl-4-thiophen-2-yl-1,4-dihydropyridine-3-carboxamide —— C26H22ClN3O2S2
6-[(4-chlorophenyl)methylsulfanyl]-5-cyano-N-(2-methoxyphenyl)-2-methyl-4-thiophen-2-yl-1,4-dihydropyridine-3-carboxamide
—— 6-Bromo-1-cyclohexyl-4-[(dimethylazaniumyl)methyl]-3-ethoxycarbonyl-2-(phenylsulfanylmethyl)indol-5-olate —— C27H33BrN2O3S
6-Bromo-1-cyclohexyl-4-[(dimethylazaniumyl)methyl]-3-ethoxycarbonyl-2-(phenylsulfanylmethyl)indol-5-olate
—— 6-methyl-N-(pyridin-3-ylmethyl)-2-[1-(2-thiophen-3-ylsulfanylacetyl)piperidin-4-yl]pyridine-3-carboxamide —— C24H26N4O2S2
6-methyl-N-(pyridin-3-ylmethyl)-2-[1-(2-thiophen-3-ylsulfanylacetyl)piperidin-4-yl]pyridine-3-carboxamide
—— 6-[4-(4-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]-N-methyl-5-nitro-N-(2-phenylethyl)pyrimidin-4-amine —— C24H24ClN5O2
6-[4-(4-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]-N-methyl-5-nitro-N-(2-phenylethyl)pyrimidin-4-amine
—— 6-hydroxy-3-phenyl-5-(1,2,3,4-tetrahydroisoquinolin-1-yl)-2-thioxo-2,3-dihydropyrimidin-4(1H)-one —— C19H17N3O2S
6-hydroxy-3-phenyl-5-(1,2,3,4-tetrahydroisoquinolin-1-yl)-2-thioxo-2,3-dihydropyrimidin-4(1H)-one
—— 6-[[1-[(2-Fluorophenyl)methyl]indol-3-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H24FN5OS
6-[[1-[(2-Fluorophenyl)methyl]indol-3-yl]methylidene]-5-imino-2-pentan-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one