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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (5R)-5-(3,5-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(3,5-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2R)-4-[[5-methyl-4-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C20H22N4O3S2
ethyl (2R)-4-[[5-methyl-4-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (2R)-2-(4-methyl-1,3-thiazol-2-yl)-4-naphthalen-2-ylsulfanyl-3-oxobutanoate —— C20H19NO3S2
ethyl (2R)-2-(4-methyl-1,3-thiazol-2-yl)-4-naphthalen-2-ylsulfanyl-3-oxobutanoate
—— ethyl (2S)-4-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C19H19ClN4O3S2
ethyl (2S)-4-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxo-4-([1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-ylsulfanyl)butanoate —— C18H16N4O3S3
ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxo-4-([1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-ylsulfanyl)butanoate
—— ethyl (2R)-4-[[4-methyl-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C18H20N4O4S2
ethyl (2R)-4-[[4-methyl-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (3R)-1-[3-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C31H36ClN5O3S
ethyl (3R)-1-[3-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-4-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-3-oxobutanoate —— C13H16N4O3S2
ethyl (2S)-2-(4-methyl-1,3-thiazol-2-yl)-4-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-3-oxobutanoate
—— ethyl (2R)-4-[[4-methyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C20H22N4O3S2
ethyl (2R)-4-[[4-methyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl 4-[[(1R,5R)-8-[4-[[methyl(pentyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H40N2O4
ethyl 4-[[(1R,5R)-8-[4-[[methyl(pentyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl (3S)-1-[3-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C31H36ClN5O3S
ethyl (3S)-1-[3-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (2S)-4-[[4-methyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C20H22N4O3S2
ethyl (2S)-4-[[4-methyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (2Z)-2-[(2E)-2-(2-amino-1-cyano-2-oxoethylidene)-3-(4-bromophenyl)-4-oxo-1,3-thiazolidin-5-ylidene]acetate —— C16H12BrN3O4S
ethyl (2Z)-2-[(2E)-2-(2-amino-1-cyano-2-oxoethylidene)-3-(4-bromophenyl)-4-oxo-1,3-thiazolidin-5-ylidene]acetate
—— ethyl (2S)-4-[[5-methyl-4-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C20H22N4O3S2
ethyl (2S)-4-[[5-methyl-4-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (2S)-4-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C18H20N4O4S2
ethyl (2S)-4-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (5R)-5-(3,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(3,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2R)-1-[2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-2-carboxylate —— C18H21ClN4O3S
ethyl (2R)-1-[2-[[4-(3-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-2-carboxylate
—— ethyl (5S)-5-(3,5-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(3,5-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3R)-1-[4-[(4-bromobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32BrN3O5S
ethyl (3R)-1-[4-[(4-bromobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (5S)-5-(3,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(3,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(3,5-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(3,5-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl-[2-(2-methoxyanilino)-2-oxoethyl]-[[4-(phenylcarbamoyl)phenyl]methyl]azanium —— C25H28N3O3+
Ethyl-[2-(2-methoxyanilino)-2-oxoethyl]-[[4-(phenylcarbamoyl)phenyl]methyl]azanium
—— ethyl (2R)-4-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C18H20N4O4S2
ethyl (2R)-4-[[4-ethyl-5-(furan-2-yl)-1,2,4-triazol-3-yl]sulfanyl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (5S)-5-(3,5-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(3,5-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-phenylprop-2-enamide —— C24H28N2O3S
(E)-N-[4-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-phenylprop-2-enamide
—— ethyl (E)-2-cyano-3-(2-phenylhydrazinyl)prop-2-enoate —— C12H13N3O2
ethyl (E)-2-cyano-3-(2-phenylhydrazinyl)prop-2-enoate
—— (E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(4-chlorophenyl)prop-2-enamide —— C24H27ClN2O3S
(E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(4-chlorophenyl)prop-2-enamide
—— ethyl (3R)-1-[4-[(2-fluorobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32FN3O5S
ethyl (3R)-1-[4-[(2-fluorobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— (E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-phenylprop-2-enamide —— C24H28N2O3S
(E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-phenylprop-2-enamide
—— (E)-3-anilino-N-(3-chlorophenyl)-2-cyanoprop-2-enamide —— C16H12ClN3O
(E)-3-anilino-N-(3-chlorophenyl)-2-cyanoprop-2-enamide
—— ethyl (3S)-1-[4-[(2-fluorobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32FN3O5S
ethyl (3S)-1-[4-[(2-fluorobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[(4-bromobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32BrN3O5S
ethyl (3S)-1-[4-[(4-bromobenzoyl)amino]-2-[[(1S)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— (E)-N-[4-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(3-chlorophenyl)prop-2-enamide —— C24H27ClN2O3S
(E)-N-[4-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(3-chlorophenyl)prop-2-enamide
—— (E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(3-chlorophenyl)prop-2-enamide —— C24H27ClN2O3S
(E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(3-chlorophenyl)prop-2-enamide
—— (E)-N-(3-chlorophenyl)-2-cyano-3-(2,5-dichloroanilino)prop-2-enamide —— C16H10Cl3N3O
(E)-N-(3-chlorophenyl)-2-cyano-3-(2,5-dichloroanilino)prop-2-enamide
—— (E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide —— C26H32N2O5S
(E)-N-[4-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[4-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(4-chlorophenyl)prop-2-enamide —— C24H27ClN2O3S
(E)-N-[4-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(4-chlorophenyl)prop-2-enamide
—— (E)-3-(3-chloro-2-methylanilino)-N-(3-chlorophenyl)-2-cyanoprop-2-enamide —— C17H13Cl2N3O
(E)-3-(3-chloro-2-methylanilino)-N-(3-chlorophenyl)-2-cyanoprop-2-enamide
—— (E)-3-(3-bromoanilino)-N-(3-chlorophenyl)-2-cyanoprop-2-enamide —— C16H11BrClN3O
(E)-3-(3-bromoanilino)-N-(3-chlorophenyl)-2-cyanoprop-2-enamide
—— Ethyl 4-[4-[(2-methoxyphenyl)methyl]piperazin-4-ium-1-yl]sulfonylbenzoate —— C21H27N2O5S+
Ethyl 4-[4-[(2-methoxyphenyl)methyl]piperazin-4-ium-1-yl]sulfonylbenzoate
—— (E)-3-(4-acetylanilino)-N-(3-chlorophenyl)-2-cyanoprop-2-enamide —— C18H14ClN3O2
(E)-3-(4-acetylanilino)-N-(3-chlorophenyl)-2-cyanoprop-2-enamide
—— ethyl 4-[4-[(1R)-1-phenylethyl]piperazin-1-yl]sulfonylbenzoate —— C21H26N2O4S
ethyl 4-[4-[(1R)-1-phenylethyl]piperazin-1-yl]sulfonylbenzoate
—— ethyl (3S)-1-[2-[2-[[2-[(2,4-dichlorobenzoyl)-(2-methylpropyl)amino]acetyl]amino]-1,3-thiazol-4-yl]acetyl]piperidine-3-carboxylate —— C26H32Cl2N4O5S
ethyl (3S)-1-[2-[2-[[2-[(2,4-dichlorobenzoyl)-(2-methylpropyl)amino]acetyl]amino]-1,3-thiazol-4-yl]acetyl]piperidine-3-carboxylate
—— ethyl N-[2-[[2-(4-cyano-2-methoxyphenoxy)acetyl]-ethylamino]acetyl]carbamate —— C17H21N3O6
ethyl N-[2-[[2-(4-cyano-2-methoxyphenoxy)acetyl]-ethylamino]acetyl]carbamate
—— (E)-N-(3-chlorophenyl)-2-cyano-3-(2,3-dichloroanilino)prop-2-enamide —— C16H10Cl3N3O
(E)-N-(3-chlorophenyl)-2-cyano-3-(2,3-dichloroanilino)prop-2-enamide
—— ethyl 4-[2-[[(1S)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl]piperazine-1-carboxylate —— C15H24N4O3
ethyl 4-[2-[[(1S)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl]piperazine-1-carboxylate
—— (E)-N-(3-chlorophenyl)-2-cyano-3-(4-cyanoanilino)prop-2-enamide —— C17H11ClN4O
(E)-N-(3-chlorophenyl)-2-cyano-3-(4-cyanoanilino)prop-2-enamide
—— (E)-N-(3-chlorophenyl)-2-cyano-3-(2,4-dichloroanilino)prop-2-enamide —— C16H10Cl3N3O
(E)-N-(3-chlorophenyl)-2-cyano-3-(2,4-dichloroanilino)prop-2-enamide
—— ethyl (3R)-1-[2-[2-[[2-[(2,4-dichlorobenzoyl)-(2-methylpropyl)amino]acetyl]amino]-1,3-thiazol-4-yl]acetyl]piperidine-3-carboxylate —— C26H32Cl2N4O5S
ethyl (3R)-1-[2-[2-[[2-[(2,4-dichlorobenzoyl)-(2-methylpropyl)amino]acetyl]amino]-1,3-thiazol-4-yl]acetyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[[4-(phenylcarbamoyl)phenyl]methyl]piperidine-3-carboxylate —— C22H26N2O3
ethyl (3S)-1-[[4-(phenylcarbamoyl)phenyl]methyl]piperidine-3-carboxylate