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—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide —— C19H18F4N2O4
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide
—— (E)-N-[2-(4-chlorophenoxy)ethyl]-3-(3,5-dimethoxyphenyl)prop-2-enamide —— C19H20ClNO4
(E)-N-[2-(4-chlorophenoxy)ethyl]-3-(3,5-dimethoxyphenyl)prop-2-enamide
—— (E)-N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(5-nitrofuran-2-yl)prop-2-enamide —— C16H13N3O4S
(E)-N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(5-nitrofuran-2-yl)prop-2-enamide
—— ethyl (6R)-2-[[2-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H31NO5S
ethyl (6R)-2-[[2-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[4-(diethylsulfamoyl)benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate —— C27H30N2O7S2
ethyl 2-[[(2R)-2-[4-(diethylsulfamoyl)benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate
—— ethyl (6S)-2-[[(2R)-2-(4-methoxy-3-nitrobenzoyl)oxy-2-phenylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28N2O8S
ethyl (6S)-2-[[(2R)-2-(4-methoxy-3-nitrobenzoyl)oxy-2-phenylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (6R)-2-[[(2S)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H31FN2O7S2
ethyl (6R)-2-[[(2S)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-(4-imidazol-1-ylphenyl)prop-2-enamide —— C20H20N4O2
(E)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-(4-imidazol-1-ylphenyl)prop-2-enamide
—— ethyl 2-[[(2S)-2-[4-(diethylsulfamoyl)benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate —— C27H30N2O7S2
ethyl 2-[[(2S)-2-[4-(diethylsulfamoyl)benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-3-(3-bromophenyl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide —— C17H17BrN2O2
(E)-3-(3-bromophenyl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide
—— ethyl (6S)-2-[[(2S)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H31FN2O7S2
ethyl (6S)-2-[[(2S)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (6S)-2-[[(2R)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H31FN2O7S2
ethyl (6S)-2-[[(2R)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(3-chlorophenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H24ClN3O5
ethyl 4-[(Z)-[(2R)-2-(3-chlorophenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (2Z)-2-[3-[2-[4-(5-chloro-2-methylphenyl)piperazin-1-ium-1-yl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C20H27ClN3O3S+
ethyl (2Z)-2-[3-[2-[4-(5-chloro-2-methylphenyl)piperazin-1-ium-1-yl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 2-[(2S,3Z)-2-(4-tert-butylphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C36H36N2O6S
ethyl 2-[(2S,3Z)-2-(4-tert-butylphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 4-[[2-(3,4-dihydro-2H-quinolin-1-yl)acetyl]amino]piperidine-1-carboxylate —— C19H27N3O3
ethyl 4-[[2-(3,4-dihydro-2H-quinolin-1-yl)acetyl]amino]piperidine-1-carboxylate
—— ethyl 2-[(2R,3Z)-2-(4-tert-butylphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C36H36N2O6S
ethyl 2-[(2R,3Z)-2-(4-tert-butylphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 5-(2,4-dichlorophenyl)-3-[[2-[(Z)-3-(3-nitrophenyl)prop-2-enoyl]oxyacetyl]amino]thiophene-2-carboxylate —— C24H18Cl2N2O7S
ethyl 5-(2,4-dichlorophenyl)-3-[[2-[(Z)-3-(3-nitrophenyl)prop-2-enoyl]oxyacetyl]amino]thiophene-2-carboxylate
—— ethyl (6R)-2-[[2-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H31NO5S
ethyl (6R)-2-[[2-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (4S)-4-(furan-2-yl)-2-oxo-6-[(4-phenylpiperazin-1-ium-1-yl)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H27N4O4+
ethyl (4S)-4-(furan-2-yl)-2-oxo-6-[(4-phenylpiperazin-1-ium-1-yl)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (6R)-2-[[(2R)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28F2N2O7S2
ethyl (6R)-2-[[(2R)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (4R)-4-(furan-2-yl)-6-[(N-methylanilino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H21N3O4
ethyl (4R)-4-(furan-2-yl)-6-[(N-methylanilino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (6R)-2-[[(2R)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H31FN2O7S2
ethyl (6R)-2-[[(2R)-2-[2-[(4-fluoro-2-methylphenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (2Z)-2-[3-[2-[4-(2-hydroxyphenyl)piperazin-1-yl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C19H25N3O4S
ethyl (2Z)-2-[3-[2-[4-(2-hydroxyphenyl)piperazin-1-yl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (6R)-2-[[(2S)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28F2N2O7S2
ethyl (6R)-2-[[(2S)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 5-[(2S)-3-(furan-2-ylmethyl)-4-oxo-1,2-dihydroquinazolin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H23N3O4
ethyl 5-[(2S)-3-(furan-2-ylmethyl)-4-oxo-1,2-dihydroquinazolin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (2Z)-2-[3-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C19H24ClN3O3S
ethyl (2Z)-2-[3-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 2-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-ethylamino]acetate —— C15H25NO3
ethyl 2-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-ethylamino]acetate
—— ethyl 4-[(3R)-3-(1-benzylindol-3-yl)-3-(3-phenoxyphenyl)propanoyl]piperazine-1-carboxylate —— C37H37N3O4
ethyl 4-[(3R)-3-(1-benzylindol-3-yl)-3-(3-phenoxyphenyl)propanoyl]piperazine-1-carboxylate
—— Ethyl 2-[2-[2-oxo-2-[4-(2-oxopyrrolidin-1-yl)anilino]ethyl]sulfanyl-1,3-thiazol-4-yl]acetate —— C19H21N3O4S2
Ethyl 2-[2-[2-oxo-2-[4-(2-oxopyrrolidin-1-yl)anilino]ethyl]sulfanyl-1,3-thiazol-4-yl]acetate
—— ethyl 4-[(2R,3Z)-2-(4-bromophenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]benzoate —— C26H20BrNO5
ethyl 4-[(2R,3Z)-2-(4-bromophenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]benzoate
—— Ethyl 2-[2-[(4,6-diamino-1,3,5-triazin-2-yl)methylsulfanyl]-1,3-thiazol-4-yl]acetate —— C11H14N6O2S2
Ethyl 2-[2-[(4,6-diamino-1,3,5-triazin-2-yl)methylsulfanyl]-1,3-thiazol-4-yl]acetate
—— ethyl (3S)-1-[2-[[(3-methoxyphenyl)methyl-[[3-(trifluoromethyl)phenyl]methyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate —— C29H32F3N3O5
ethyl (3S)-1-[2-[[(3-methoxyphenyl)methyl-[[3-(trifluoromethyl)phenyl]methyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[[(3-methoxyphenyl)methyl-[[3-(trifluoromethyl)phenyl]methyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate —— C29H32F3N3O5
ethyl (3R)-1-[2-[[(3-methoxyphenyl)methyl-[[3-(trifluoromethyl)phenyl]methyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
—— ethyl 2-[(2S,3Z)-2-(3-bromophenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H19BrN2O5S
ethyl 2-[(2S,3Z)-2-(3-bromophenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(2S,3Z)-3-[hydroxy-(4-methoxyphenyl)methylidene]-2-(2-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H24N2O7S
ethyl 2-[(2S,3Z)-3-[hydroxy-(4-methoxyphenyl)methylidene]-2-(2-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 4-[(Z)-[(2S)-1-[2-(dimethylamino)ethyl]-2-(3-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H28FN3O5
ethyl 4-[(Z)-[(2S)-1-[2-(dimethylamino)ethyl]-2-(3-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3-[[(5R,7R)-3-acetamidoadamantane-1-carbonyl]oxymethyl]-1-benzofuran-2-carboxylate —— C25H29NO6
ethyl 3-[[(5R,7R)-3-acetamidoadamantane-1-carbonyl]oxymethyl]-1-benzofuran-2-carboxylate
—— ethyl 4-[(Z)-[(2R)-1-[2-(dimethylamino)ethyl]-2-(3-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H28FN3O5
ethyl 4-[(Z)-[(2R)-1-[2-(dimethylamino)ethyl]-2-(3-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(3-chlorophenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H24ClN3O5
ethyl 4-[(Z)-[(2S)-2-(3-chlorophenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (3R)-1-[2-[4-[2-[3-(trifluoromethyl)anilino]-1,3-thiazole-4-carbonyl]piperazin-1-yl]acetyl]piperidine-3-carboxylate —— C25H30F3N5O4S
ethyl (3R)-1-[2-[4-[2-[3-(trifluoromethyl)anilino]-1,3-thiazole-4-carbonyl]piperazin-1-yl]acetyl]piperidine-3-carboxylate
—— ethyl (6S)-2-[[(2S)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28F2N2O7S2
ethyl (6S)-2-[[(2S)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (6S)-2-[[(2R)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28F2N2O7S2
ethyl (6S)-2-[[(2R)-2-[3-[(3,4-difluorophenyl)sulfonylamino]benzoyl]oxypropanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 5-(4-methoxyphenyl)-3-[[(1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]thiophene-2-carboxylate —— C24H27NO5S
ethyl 5-(4-methoxyphenyl)-3-[[(1R,5R)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]thiophene-2-carboxylate
—— ethyl 2-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-ethylamino]acetate —— C15H25NO3
ethyl 2-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]-ethylamino]acetate
—— ethyl 4-[(2S,3Z)-3-[(4-chlorophenyl)-hydroxymethylidene]-2-(3-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]benzoate —— C26H19ClN2O7
ethyl 4-[(2S,3Z)-3-[(4-chlorophenyl)-hydroxymethylidene]-2-(3-nitrophenyl)-4,5-dioxopyrrolidin-1-yl]benzoate
—— Ethyl 4-acetyl-2-[[2-(4-cyclohexylbutanoyloxy)acetyl]amino]-5-methylfuran-3-carboxylate —— C22H31NO7
Ethyl 4-acetyl-2-[[2-(4-cyclohexylbutanoyloxy)acetyl]amino]-5-methylfuran-3-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(3-bromophenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H27BrN4O5
ethyl 4-[(Z)-[(2S)-2-(3-bromophenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(2S,3Z)-2-(4-bromophenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]benzoate —— C26H20BrNO5
ethyl 4-[(2S,3Z)-2-(4-bromophenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl 4-[(Z)-[(2S)-4,5-dioxo-1-(pyridin-3-ylmethyl)-2-(3,4,5-trimethoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C29H31N3O8
ethyl 4-[(Z)-[(2S)-4,5-dioxo-1-(pyridin-3-ylmethyl)-2-(3,4,5-trimethoxyphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate