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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 6-[[4-[(1S,5R)-3-(2-chloro-5-methylphenoxy)-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl]methylsulfanyl]-5-cyano-2-methylpyridine-3-carboxylate —— C32H32ClN3O4S
ethyl 6-[[4-[(1S,5R)-3-(2-chloro-5-methylphenoxy)-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl]methylsulfanyl]-5-cyano-2-methylpyridine-3-carboxylate
—— ethyl 4-[[(1S,5S)-8-[4-[(2,3,5,6-tetrafluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H27F4NO4S
ethyl 4-[[(1S,5S)-8-[4-[(2,3,5,6-tetrafluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[(Z)-hydroxy-[(2R)-2-(4-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H27N3O6
ethyl 4-[(Z)-hydroxy-[(2R)-2-(4-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— Ethyl 5-amino-4-cyano-3-[(2-ethoxy-2-oxoethyl)sulfanylmethyl]thiophene-2-carboxylate —— C13H16N2O4S2
Ethyl 5-amino-4-cyano-3-[(2-ethoxy-2-oxoethyl)sulfanylmethyl]thiophene-2-carboxylate
—— ethyl 2-[2-[(4S)-4-methyl-2-oxo-3,4-dihydro-1H-1,5-benzodiazepin-5-yl]-2-oxoethyl]sulfanylacetate —— C16H20N2O4S
ethyl 2-[2-[(4S)-4-methyl-2-oxo-3,4-dihydro-1H-1,5-benzodiazepin-5-yl]-2-oxoethyl]sulfanylacetate
—— ethyl 4-[[(1R,5R)-8-[4-[(4-chlorophenyl)methylsulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C31H32ClNO4S
ethyl 4-[[(1R,5R)-8-[4-[(4-chlorophenyl)methylsulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(4-benzylpiperidin-1-yl)methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C36H42N2O4
ethyl 4-[[(1R,5R)-8-[4-[(4-benzylpiperidin-1-yl)methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(2,4-dimethylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C32H35NO4S
ethyl 4-[[(1R,5R)-8-[4-[(2,4-dimethylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl N-[(2'R,3'R,6'S,7'R)-1'-bromospiro[1,3-dioxolane-2,9'-pentacyclo[4.3.0.02,5.03,8.04,7]nonane]-4'-yl]carbamate —— C14H16BrNO4
ethyl N-[(2'R,3'R,6'S,7'R)-1'-bromospiro[1,3-dioxolane-2,9'-pentacyclo[4.3.0.02,5.03,8.04,7]nonane]-4'-yl]carbamate
—— ethyl 5,5,7,7-tetramethyl-2-[[2-[(1R,2S)-2-methylcyclopropanecarbonyl]oxyacetyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C21H30N2O5S
ethyl 5,5,7,7-tetramethyl-2-[[2-[(1R,2S)-2-methylcyclopropanecarbonyl]oxyacetyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-2-(5-methylfuran-2-yl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H31N3O6
ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-2-(5-methylfuran-2-yl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-phenyl-2-[[(2R)-2-phenyl-2-[3-(3,4,5-trimethoxyphenyl)propanoyloxy]acetyl]amino]thiophene-3-carboxylate —— C33H33NO8S
ethyl 4-phenyl-2-[[(2R)-2-phenyl-2-[3-(3,4,5-trimethoxyphenyl)propanoyloxy]acetyl]amino]thiophene-3-carboxylate
—— ethyl 1-[4-(4-chlorobutanoylamino)-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]phenyl]piperidine-4-carboxylate —— C28H36ClN3O5S
ethyl 1-[4-(4-chlorobutanoylamino)-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]phenyl]piperidine-4-carboxylate
—— ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-(4-propan-2-ylphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O5
ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-(4-propan-2-ylphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2S)-2-(4-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H27N3O6
ethyl 4-[(Z)-hydroxy-[(2S)-2-(4-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-phenyl-2-[[(2S)-2-phenyl-2-[3-(3,4,5-trimethoxyphenyl)propanoyloxy]acetyl]amino]thiophene-3-carboxylate —— C33H33NO8S
ethyl 4-phenyl-2-[[(2S)-2-phenyl-2-[3-(3,4,5-trimethoxyphenyl)propanoyloxy]acetyl]amino]thiophene-3-carboxylate
—— ethyl 2-[(2S,3Z)-3-[(4-fluorophenyl)-hydroxymethylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H21FN2O6S
ethyl 2-[(2S,3Z)-3-[(4-fluorophenyl)-hydroxymethylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3R)-1-[2-[[(1S)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate —— C31H37N3O6S
ethyl (3R)-1-[2-[[(1S)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate
—— ethyl 4-[[(1S,5R)-8-[4-[(5-methoxy-1,3-benzothiazol-2-yl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C32H32N2O5S2
ethyl 4-[[(1S,5R)-8-[4-[(5-methoxy-1,3-benzothiazol-2-yl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1S,5S)-8-[4-[(5-methoxy-1,3-benzothiazol-2-yl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C32H32N2O5S2
ethyl 4-[[(1S,5S)-8-[4-[(5-methoxy-1,3-benzothiazol-2-yl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate —— C31H38N4O6S
ethyl 4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate
—— ethyl 2-[(2R,3Z)-3-[(4-fluorophenyl)-hydroxymethylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H21FN2O6S
ethyl 2-[(2R,3Z)-3-[(4-fluorophenyl)-hydroxymethylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O6
ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate —— C31H38N4O6S
ethyl 4-[4-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate
—— ethyl (3S)-1-[2-[[(1S)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate —— C31H37N3O6S
ethyl (3S)-1-[2-[[(1S)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate
—— ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-(4-propan-2-ylphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O5
ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-(4-propan-2-ylphenyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[[(1R,5R)-8-[4-[(5-methoxy-1,3-benzothiazol-2-yl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C32H32N2O5S2
ethyl 4-[[(1R,5R)-8-[4-[(5-methoxy-1,3-benzothiazol-2-yl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]prop-2-enamide —— C20H24N2O2
(E)-3-(1,3-benzoxazol-2-yl)-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]prop-2-enamide
—— ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O6
ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (3S)-1-[(2R)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate —— C36H38N4O6
ethyl (3S)-1-[(2R)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(2,3-dimethoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C29H37N3O8
ethyl 4-[(Z)-[(2S)-2-(2,3-dimethoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2S)-1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-pyridin-3-ylpyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H32N4O6
ethyl 4-[(Z)-hydroxy-[(2S)-1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-pyridin-3-ylpyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (3S)-1-[(2S)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate —— C36H38N4O6
ethyl (3S)-1-[(2S)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate
—— ethyl 2-[(2S,3Z)-2-(3,4-dichlorophenyl)-3-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H22Cl2N2O6S
ethyl 2-[(2S,3Z)-2-(3,4-dichlorophenyl)-3-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3R)-1-[(2S)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate —— C36H38N4O6
ethyl (3R)-1-[(2S)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate
—— ethyl 1-[3-[(5-benzyl-4-oxo-7,8-dihydro-6H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)-[(2S)-butan-2-yl]amino]propanoyl]piperidine-4-carboxylate —— C30H41N5O5
ethyl 1-[3-[(5-benzyl-4-oxo-7,8-dihydro-6H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)-[(2S)-butan-2-yl]amino]propanoyl]piperidine-4-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(2,3-dimethoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C29H37N3O8
ethyl 4-[(Z)-[(2R)-2-(2,3-dimethoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (4S)-6-[(3-chloro-4-fluorophenoxy)methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H18ClFN2O4
ethyl (4S)-6-[(3-chloro-4-fluorophenoxy)methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[(2R,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H22N2O7S
ethyl 2-[(2R,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(2S,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C24H22N2O7S
ethyl 2-[(2S,3Z)-2-(furan-2-yl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— (E)-3-[4-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]phenyl]prop-2-enoic acid —— C14H13NO4
(E)-3-[4-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]phenyl]prop-2-enoic acid
—— ethyl (3R)-1-[(2R)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate —— C36H38N4O6
ethyl (3R)-1-[(2R)-2-[(4S)-1-methyl-2,5-dioxo-4-(3-phenoxyphenyl)-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate
—— ethyl 4,5-dimethyl-2-[[2-[2-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzoyl]oxyacetyl]amino]thiophene-3-carboxylate —— C22H21F3N2O6S
ethyl 4,5-dimethyl-2-[[2-[2-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzoyl]oxyacetyl]amino]thiophene-3-carboxylate
—— ethyl 2-[(2R,3Z)-2-(3,4-dichlorophenyl)-3-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C26H22Cl2N2O6S
ethyl 2-[(2R,3Z)-2-(3,4-dichlorophenyl)-3-[hydroxy-(4-methoxy-2-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 4-thiophen-2-yl-2-[[2-[2-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzoyl]oxyacetyl]amino]thiophene-3-carboxylate —— C24H19F3N2O6S2
ethyl 4-thiophen-2-yl-2-[[2-[2-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzoyl]oxyacetyl]amino]thiophene-3-carboxylate
—— ethyl 4-(2-methylpropyl)-2-[[2-[2-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzoyl]oxyacetyl]amino]thiophene-3-carboxylate —— C24H25F3N2O6S
ethyl 4-(2-methylpropyl)-2-[[2-[2-[[(Z)-4,4,4-trifluoro-3-oxobut-1-enyl]amino]benzoyl]oxyacetyl]amino]thiophene-3-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2R)-1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-pyridin-3-ylpyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H32N4O6
ethyl 4-[(Z)-hydroxy-[(2R)-1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-pyridin-3-ylpyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-(4-methylphenyl)-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide —— C18H21NOS
(E)-3-(4-methylphenyl)-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide
—— ethyl N-[4-[2-(3-fluorophenyl)ethylcarbamoyl]phenyl]carbamate —— C18H19FN2O3
ethyl N-[4-[2-(3-fluorophenyl)ethylcarbamoyl]phenyl]carbamate
—— ethyl (3S)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3S)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate