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—— ethyl 2-[benzyl-[2-[[4-[(1S,2R)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C30H34N6O3S2
ethyl 2-[benzyl-[2-[[4-[(1S,2R)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3S)-1-[2-[[(3-phenoxyphenyl)methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate —— C34H37N3O5
ethyl (3S)-1-[2-[[(3-phenoxyphenyl)methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
—— ethyl 4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate —— C31H38N4O6S
ethyl 4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1S)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate
—— ethyl 4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate —— C31H38N4O6S
ethyl 4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]-3-[[(1R)-1-phenylethyl]sulfamoyl]anilino]-4-oxobutanoate
—— ethyl 2-[benzyl-[2-[[4-[(1S,2S)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C30H34N6O3S2
ethyl 2-[benzyl-[2-[[4-[(1S,2S)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3R)-1-[2-[[(3-phenoxyphenyl)methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate —— C34H37N3O5
ethyl (3R)-1-[2-[[(3-phenoxyphenyl)methyl-[(1S)-1-phenylethyl]amino]methyl]-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
—— ethyl 4-[[(E)-[1-[(4-fluorophenyl)methyl]-2,2,4-trioxothieno[3,2-c]thiazin-3-ylidene]methyl]amino]benzoate —— C23H19FN2O5S2
ethyl 4-[[(E)-[1-[(4-fluorophenyl)methyl]-2,2,4-trioxothieno[3,2-c]thiazin-3-ylidene]methyl]amino]benzoate
—— ethyl 2-[benzyl-[2-[[4-[(1R,2R)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C30H34N6O3S2
ethyl 2-[benzyl-[2-[[4-[(1R,2R)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[benzyl-[2-[[4-[(1R,2S)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C30H34N6O3S2
ethyl 2-[benzyl-[2-[[4-[(1R,2S)-2-methylcyclohexyl]-5-pyridin-3-yl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 4-[[(E)-[1-[(4-methylphenyl)methyl]-2,2,4-trioxothieno[3,2-c]thiazin-3-ylidene]methyl]amino]benzoate —— C24H22N2O5S2
ethyl 4-[[(E)-[1-[(4-methylphenyl)methyl]-2,2,4-trioxothieno[3,2-c]thiazin-3-ylidene]methyl]amino]benzoate
—— ethyl (5S)-3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H32N4O4S
ethyl (5S)-3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-cyano-3-[4-(dimethylamino)-3-nitrophenyl]-N-(4-methoxyphenyl)prop-2-enamide —— C19H18N4O4
(E)-2-cyano-3-[4-(dimethylamino)-3-nitrophenyl]-N-(4-methoxyphenyl)prop-2-enamide
—— ethyl (5R)-3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H32N4O4S
ethyl (5R)-3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[(1R,2S,6R,7R)-10-[bis(4-methoxyphenyl)methylidene]-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate —— C33H29NO6
ethyl 2-[(1R,2S,6R,7R)-10-[bis(4-methoxyphenyl)methylidene]-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate
—— ethyl 1-[2-[(E)-3-(1-benzylpyrazol-4-yl)prop-2-enoyl]oxyacetyl]piperidine-4-carboxylate —— C23H27N3O5
ethyl 1-[2-[(E)-3-(1-benzylpyrazol-4-yl)prop-2-enoyl]oxyacetyl]piperidine-4-carboxylate
—— ethyl 2-[(1R,2R,6R,7R)-10-[bis(4-methoxyphenyl)methylidene]-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate —— C33H29NO6
ethyl 2-[(1R,2R,6R,7R)-10-[bis(4-methoxyphenyl)methylidene]-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate
—— ethyl 5-[[(1R,2S,4S)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C19H19NO3S
ethyl 5-[[(1R,2S,4S)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— ethyl 2-[(1R,2S,6S,7R)-10-[bis(4-methoxyphenyl)methylidene]-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate —— C33H29NO6
ethyl 2-[(1R,2S,6S,7R)-10-[bis(4-methoxyphenyl)methylidene]-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]benzoate
—— (E)-N-benzyl-2-cyano-3-hydroxy-4-[1-(2-methylpropyl)benzimidazol-2-yl]sulfanylbut-2-enamide —— C23H24N4O2S
(E)-N-benzyl-2-cyano-3-hydroxy-4-[1-(2-methylpropyl)benzimidazol-2-yl]sulfanylbut-2-enamide
—— ethyl (1R,5S,6R)-3-(4-bromophenyl)-1-(4-chlorophenyl)-2,4-dioxo-3-azabicyclo[3.1.0]hexane-6-carboxylate —— C20H15BrClNO4
ethyl (1R,5S,6R)-3-(4-bromophenyl)-1-(4-chlorophenyl)-2,4-dioxo-3-azabicyclo[3.1.0]hexane-6-carboxylate
—— ethyl 5-[[(1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C21H23NO4S
ethyl 5-[[(1S,5S)-9-oxobicyclo[3.3.1]nonane-3-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— ethyl 5-[[(1R,2R,4S)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C19H19NO3S
ethyl 5-[[(1R,2R,4S)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— ethyl 5-[2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylacetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H18FN5O3S
ethyl 5-[2-[1-(3-fluorophenyl)tetrazol-5-yl]sulfanylacetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 6-benzyl-2-[[(2S)-2-[1-(2-methoxyethyl)benzimidazol-2-yl]sulfanylpropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H34N4O4S2
ethyl 6-benzyl-2-[[(2S)-2-[1-(2-methoxyethyl)benzimidazol-2-yl]sulfanylpropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 6-benzyl-2-[[(2R)-2-[1-(2-methoxyethyl)benzimidazol-2-yl]sulfanylpropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H34N4O4S2
ethyl 6-benzyl-2-[[(2R)-2-[1-(2-methoxyethyl)benzimidazol-2-yl]sulfanylpropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 1-[2-[(4E)-1-(5-chloro-2-methoxyphenyl)-4-[(3-methylthiophen-2-yl)methylidene]-5-oxoimidazol-2-yl]sulfanylacetyl]piperidine-4-carboxylate —— C26H28ClN3O5S2
ethyl 1-[2-[(4E)-1-(5-chloro-2-methoxyphenyl)-4-[(3-methylthiophen-2-yl)methylidene]-5-oxoimidazol-2-yl]sulfanylacetyl]piperidine-4-carboxylate
—— ethyl 4-methyl-2-[[(E)-3-(5-nitrofuran-2-yl)prop-2-enoyl]oxymethyl]quinoline-3-carboxylate —— C21H18N2O7
ethyl 4-methyl-2-[[(E)-3-(5-nitrofuran-2-yl)prop-2-enoyl]oxymethyl]quinoline-3-carboxylate
—— (E)-2-cyano-N,3-bis(2,4-difluorophenyl)prop-2-enamide —— C16H8F4N2O
(E)-2-cyano-N,3-bis(2,4-difluorophenyl)prop-2-enamide
—— (E)-2-cyano-N-(2,4-difluorophenyl)-3-(2,4-dimethylphenyl)prop-2-enamide —— C18H14F2N2O
(E)-2-cyano-N-(2,4-difluorophenyl)-3-(2,4-dimethylphenyl)prop-2-enamide
—— (E)-2-cyano-N-(4-methoxyphenyl)-3-(3-phenylmethoxyphenyl)prop-2-enamide —— C24H20N2O3
(E)-2-cyano-N-(4-methoxyphenyl)-3-(3-phenylmethoxyphenyl)prop-2-enamide
—— ethyl 5-[(E)-2-cyano-3-(5-methylfuran-2-yl)prop-2-enoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H18N2O4
ethyl 5-[(E)-2-cyano-3-(5-methylfuran-2-yl)prop-2-enoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-N-[4-[(2S)-butan-2-yl]phenyl]-2-cyano-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C18H19N3OS
(E)-N-[4-[(2S)-butan-2-yl]phenyl]-2-cyano-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-N-[4-[(2S)-butan-2-yl]phenyl]-2-cyano-3-(4,5-dimethoxy-2-nitrophenyl)prop-2-enamide —— C22H23N3O5
(E)-N-[4-[(2S)-butan-2-yl]phenyl]-2-cyano-3-(4,5-dimethoxy-2-nitrophenyl)prop-2-enamide
—— (E)-3-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-2-cyano-N-(4-methoxyphenyl)prop-2-enamide —— C20H14ClN3O2S
(E)-3-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-2-cyano-N-(4-methoxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-[3-methoxy-4-(2-methylpropoxy)phenyl]-N-(4-methoxyphenyl)prop-2-enamide —— C22H24N2O4
(E)-2-cyano-3-[3-methoxy-4-(2-methylpropoxy)phenyl]-N-(4-methoxyphenyl)prop-2-enamide
—— ethyl 2,5-dimethyl-4-[2-[(E)-3-(5-nitrofuran-2-yl)prop-2-enoyl]oxyacetyl]-1H-pyrrole-3-carboxylate —— C18H18N2O8
ethyl 2,5-dimethyl-4-[2-[(E)-3-(5-nitrofuran-2-yl)prop-2-enoyl]oxyacetyl]-1H-pyrrole-3-carboxylate
—— (E)-2-cyano-N-(4-methoxyphenyl)-3-(4-methoxy-3-propoxyphenyl)prop-2-enamide —— C21H22N2O4
(E)-2-cyano-N-(4-methoxyphenyl)-3-(4-methoxy-3-propoxyphenyl)prop-2-enamide
—— ethyl 4-[[2-[benzyl-[[1-[(3-methoxyphenyl)methyl]pyrrol-2-yl]methyl]amino]-2-oxoethyl]-[(2R)-butan-2-yl]amino]-4-oxobutanoate —— C32H41N3O5
ethyl 4-[[2-[benzyl-[[1-[(3-methoxyphenyl)methyl]pyrrol-2-yl]methyl]amino]-2-oxoethyl]-[(2R)-butan-2-yl]amino]-4-oxobutanoate
—— (E)-2-cyano-N-(2,4-difluorophenyl)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-enamide —— C21H18F2N2O3
(E)-2-cyano-N-(2,4-difluorophenyl)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-enamide
—— ethyl 4-[[2-[benzyl-[[1-[(3-methoxyphenyl)methyl]pyrrol-2-yl]methyl]amino]-2-oxoethyl]-[(2S)-butan-2-yl]amino]-4-oxobutanoate —— C32H41N3O5
ethyl 4-[[2-[benzyl-[[1-[(3-methoxyphenyl)methyl]pyrrol-2-yl]methyl]amino]-2-oxoethyl]-[(2S)-butan-2-yl]amino]-4-oxobutanoate
—— ethyl 6-benzyl-2-[[(2S)-2-[2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H31N3O6S2
ethyl 6-benzyl-2-[[(2S)-2-[2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 6-benzyl-2-[[(2S)-2-[2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H31N3O6S2
ethyl 6-benzyl-2-[[(2S)-2-[2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 6-benzyl-2-[[(2R)-2-[2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H31N3O6S2
ethyl 6-benzyl-2-[[(2R)-2-[2-[(2R)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 6-benzyl-2-[[(2R)-2-[2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H31N3O6S2
ethyl 6-benzyl-2-[[(2R)-2-[2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetyl]oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— (E)-3-[4-(azepan-1-yl)phenyl]-2-cyano-N-(2,4-difluorophenyl)prop-2-enamide —— C22H21F2N3O
(E)-3-[4-(azepan-1-yl)phenyl]-2-cyano-N-(2,4-difluorophenyl)prop-2-enamide
—— (E)-2-cyano-N-(2,4-difluorophenyl)-3-(3-fluorophenyl)prop-2-enamide —— C16H9F3N2O
(E)-2-cyano-N-(2,4-difluorophenyl)-3-(3-fluorophenyl)prop-2-enamide
—— ethyl (6S)-6-[4-[[3,5-bis(trifluoromethyl)benzoyl]amino]phenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C24H21F6N3O3S
ethyl (6S)-6-[4-[[3,5-bis(trifluoromethyl)benzoyl]amino]phenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-cyano-3-[4-(diethylamino)phenyl]-N-(2,4-difluorophenyl)prop-2-enamide —— C20H19F2N3O
(E)-2-cyano-3-[4-(diethylamino)phenyl]-N-(2,4-difluorophenyl)prop-2-enamide
—— (E)-2-cyano-N-(2,4-difluorophenyl)-3-(3-methylphenyl)prop-2-enamide —— C17H12F2N2O
(E)-2-cyano-N-(2,4-difluorophenyl)-3-(3-methylphenyl)prop-2-enamide
—— (E)-2-cyano-3-(2,4-dimethylphenyl)-N-(3-piperidin-1-ylsulfonylphenyl)prop-2-enamide —— C23H25N3O3S
(E)-2-cyano-3-(2,4-dimethylphenyl)-N-(3-piperidin-1-ylsulfonylphenyl)prop-2-enamide