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—— ethyl (2R)-4-[5-(4-chlorophenyl)tetrazol-2-yl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C17H16ClN5O3S
ethyl (2R)-4-[5-(4-chlorophenyl)tetrazol-2-yl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (4S)-4-methyl-6-[[(7R)-7-(2-methylbutan-2-yl)-4-oxo-3-propyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H38N4O4S2
ethyl (4S)-4-methyl-6-[[(7R)-7-(2-methylbutan-2-yl)-4-oxo-3-propyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2S)-4-[5-(4-chlorophenyl)tetrazol-2-yl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate —— C17H16ClN5O3S
ethyl (2S)-4-[5-(4-chlorophenyl)tetrazol-2-yl]-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanoate
—— ethyl (6R)-2-[[2-[butyl-(4-ethoxyphenyl)sulfonylamino]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H36N2O6S2
ethyl (6R)-2-[[2-[butyl-(4-ethoxyphenyl)sulfonylamino]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (5R)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
ethyl (5R)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(3-nitrophenyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]prop-2-enamide —— C19H22N2O3
(E)-3-(3-nitrophenyl)-N-[(1S,2R,6S,7R,8R)-8-tricyclo[5.2.1.02,6]decanyl]prop-2-enamide
—— ethyl (6S)-2-[[2-[butyl-(4-ethoxyphenyl)sulfonylamino]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H36N2O6S2
ethyl (6S)-2-[[2-[butyl-(4-ethoxyphenyl)sulfonylamino]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
ethyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
ethyl (5S)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
ethyl (5S)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[2-[2-(3,4-dimethoxyphenyl)ethyl-(thiophen-2-ylmethyl)amino]-2-oxoethyl]-3-(4-nitrophenyl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C31H35N3O7S
(E)-N-[2-[2-(3,4-dimethoxyphenyl)ethyl-(thiophen-2-ylmethyl)amino]-2-oxoethyl]-3-(4-nitrophenyl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl (5R)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
ethyl (5R)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H34N4O4S
ethyl (5S)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2,4-dimethyl-5-[(2R)-2-[(2S)-5-oxopyrrolidine-2-carbonyl]oxypropanoyl]-1H-pyrrole-3-carboxylate —— C17H22N2O6
ethyl 2,4-dimethyl-5-[(2R)-2-[(2S)-5-oxopyrrolidine-2-carbonyl]oxypropanoyl]-1H-pyrrole-3-carboxylate
—— (E)-3-(3-methoxyphenyl)-N-[(1R)-1-(4-methoxyphenyl)propyl]prop-2-enamide —— C20H23NO3
(E)-3-(3-methoxyphenyl)-N-[(1R)-1-(4-methoxyphenyl)propyl]prop-2-enamide
—— ethyl (5R)-5-(2-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N4O4S
ethyl (5R)-5-(2-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(3-nitrophenyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]prop-2-enamide —— C19H22N2O3
(E)-3-(3-nitrophenyl)-N-[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]prop-2-enamide
—— ethyl (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O4S
ethyl (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(3-methoxyphenyl)-N-[4-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)-1,3-thiazol-2-yl]prop-2-enamide —— C22H19N3O3S
(E)-3-(3-methoxyphenyl)-N-[4-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)-1,3-thiazol-2-yl]prop-2-enamide
—— ethyl (5R)-5-(4-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N4O4S
ethyl (5R)-5-(4-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-(2-adamantyl)-3-(4-methylphenyl)prop-2-enamide —— C20H25NO
(E)-N-(2-adamantyl)-3-(4-methylphenyl)prop-2-enamide
—— ethyl (5S)-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H34N4O4S
ethyl (5S)-3-[2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[(4aS,5S)-3-[(4-chlorophenyl)methyl]-8-nitro-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinoline-5-carbonyl]piperazine-1-carboxylate —— C27H32ClN5O5
ethyl 4-[(4aS,5S)-3-[(4-chlorophenyl)methyl]-8-nitro-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinoline-5-carbonyl]piperazine-1-carboxylate
—— (E)-3-(furan-2-yl)-N-[4-(2-oxo-1,3-dihydroindol-5-yl)-1,3-thiazol-2-yl]prop-2-enamide —— C18H13N3O3S
(E)-3-(furan-2-yl)-N-[4-(2-oxo-1,3-dihydroindol-5-yl)-1,3-thiazol-2-yl]prop-2-enamide
—— ethyl (5S)-5-(4-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N4O4S
ethyl (5S)-5-(4-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)-1,3-thiazol-2-yl]-3-phenylprop-2-enamide —— C21H17N3O2S
(E)-N-[4-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)-1,3-thiazol-2-yl]-3-phenylprop-2-enamide
—— ethyl (5S)-5-(3,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(3,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2,5-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,5-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3R)-1-[4-[[4-(4-ethylpiperazin-1-yl)-6-phenylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H39N5O3S
ethyl (3R)-1-[4-[[4-(4-ethylpiperazin-1-yl)-6-phenylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (5S)-5-(2,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl oxo[(5-{[3-(trifluoromethyl)benzyl]sulfanyl}-1,3,4-thiadiazol-2-yl)amino]acetate —— C14H12F3N3O3S2
Ethyl oxo[(5-{[3-(trifluoromethyl)benzyl]sulfanyl}-1,3,4-thiadiazol-2-yl)amino]acetate
—— ethyl (5R)-5-(2,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,5-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2R,4E)-4-hydroxyimino-7,8-dimethoxy-2,3-dihydro-1H-naphthalene-2-carboxylate —— C15H19NO5
ethyl (2R,4E)-4-hydroxyimino-7,8-dimethoxy-2,3-dihydro-1H-naphthalene-2-carboxylate
—— ethyl (5S)-5-(2,4-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,4-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2,4-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,4-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H30N4O4S
ethyl (5R)-5-(2-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2,5-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,5-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(3,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(3,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N4O4S
ethyl (5S)-5-(2-methoxyphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2,4-dimethyl-5-[(2R)-2-(4-methyl-3-nitrobenzoyl)oxypropanoyl]-1H-pyrrole-3-carboxylate —— C20H22N2O7
ethyl 2,4-dimethyl-5-[(2R)-2-(4-methyl-3-nitrobenzoyl)oxypropanoyl]-1H-pyrrole-3-carboxylate
—— (E)-3-(4-fluorophenyl)-N-[(1S)-1-(4-methoxyphenyl)propyl]prop-2-enamide —— C19H20FNO2
(E)-3-(4-fluorophenyl)-N-[(1S)-1-(4-methoxyphenyl)propyl]prop-2-enamide
—— ethyl (5R)-5-(3,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(3,4-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(3,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(3,4-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2S,4E)-4-hydroxyimino-7,8-dimethoxy-2,3-dihydro-1H-naphthalene-2-carboxylate —— C15H19NO5
ethyl (2S,4E)-4-hydroxyimino-7,8-dimethoxy-2,3-dihydro-1H-naphthalene-2-carboxylate
—— ethyl 4-[(4aS,5R)-3-[(4-chlorophenyl)methyl]-8-nitro-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinoline-5-carbonyl]piperazine-1-carboxylate —— C27H32ClN5O5
ethyl 4-[(4aS,5R)-3-[(4-chlorophenyl)methyl]-8-nitro-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinoline-5-carbonyl]piperazine-1-carboxylate
—— ethyl (5S)-5-(2-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H30N4O4S
ethyl (5S)-5-(2-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate