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—— Ethyl 4-acetyl-2-[[2-(4-benzylpiperidin-1-ium-1-yl)acetyl]amino]-5-methylfuran-3-carboxylate —— C24H31N2O5+
Ethyl 4-acetyl-2-[[2-(4-benzylpiperidin-1-ium-1-yl)acetyl]amino]-5-methylfuran-3-carboxylate
—— (E)-3-[5-(dimethylamino)furan-2-yl]-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoic acid —— C14H18N4O3S
(E)-3-[5-(dimethylamino)furan-2-yl]-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoic acid
—— (E)-3-[3-bromo-4-(dimethylamino)phenyl]-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoate —— C16H18BrN4O2S-
(E)-3-[3-bromo-4-(dimethylamino)phenyl]-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoate
—— (E)-2-[[5-(3,5-dimethoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-3-pyridin-3-ylprop-2-enoic acid —— C18H15N3O5S
(E)-2-[[5-(3,5-dimethoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-3-pyridin-3-ylprop-2-enoic acid
—— (E)-3-(4-propan-2-ylphenyl)-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoate —— C17H20N3O2S-
(E)-3-(4-propan-2-ylphenyl)-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoate
—— (E)-2-[[5-(3,5-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(2-hydroxyphenyl)prop-2-enoic acid —— C19H17N3O5S
(E)-2-[[5-(3,5-dimethoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]-3-(2-hydroxyphenyl)prop-2-enoic acid
—— (E)-3-(5-bromofuran-2-yl)-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoic acid —— C12H12BrN3O3S
(E)-3-(5-bromofuran-2-yl)-2-[(5-propyl-1H-1,2,4-triazol-3-yl)sulfanyl]prop-2-enoic acid
—— ethyl 4-[2-[4-(4-hydroxyphenyl)piperazin-1-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C21H27N3O4
ethyl 4-[2-[4-(4-hydroxyphenyl)piperazin-1-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 4-cyano-5-(2,3-dihydrobenzo[b][1,4]dioxine-2-carboxamido)-3-methylthiophene-2-carboxylate —— C18H16N2O5S
Ethyl 4-cyano-5-(2,3-dihydrobenzo[b][1,4]dioxine-2-carboxamido)-3-methylthiophene-2-carboxylate
—— ethyl 1-[(2R)-2-[4-(4-hydroxyphenyl)piperazin-1-yl]propanoyl]piperidine-4-carboxylate —— C21H31N3O4
ethyl 1-[(2R)-2-[4-(4-hydroxyphenyl)piperazin-1-yl]propanoyl]piperidine-4-carboxylate
—— (E)-3-[2-[(1S,5S)-2,4-dioxo-3-azabicyclo[3.1.0]hexan-3-yl]-1,3-thiazol-5-yl]prop-2-enoic acid —— C11H8N2O4S
(E)-3-[2-[(1S,5S)-2,4-dioxo-3-azabicyclo[3.1.0]hexan-3-yl]-1,3-thiazol-5-yl]prop-2-enoic acid
—— ethyl 4-carbamoyl-2-methyl-5-[[2-[(3R)-3-methylpiperidin-1-yl]acetyl]amino]furan-3-carboxylate —— C17H25N3O5
ethyl 4-carbamoyl-2-methyl-5-[[2-[(3R)-3-methylpiperidin-1-yl]acetyl]amino]furan-3-carboxylate
—— Ethyl 4-[(2-morpholin-4-ylacetyl)amino]piperidine-1-carboxylate —— C14H25N3O4
Ethyl 4-[(2-morpholin-4-ylacetyl)amino]piperidine-1-carboxylate
—— Ethyl 2-[[2-(4-acetylpiperazin-1-yl)acetyl]amino]-5-ethylthiophene-3-carboxylate —— C17H25N3O4S
Ethyl 2-[[2-(4-acetylpiperazin-1-yl)acetyl]amino]-5-ethylthiophene-3-carboxylate
—— Ethyl 2-[(4-fluorophenyl)methyl-(2-morpholin-4-ylacetyl)amino]-4-methyl-1,3-thiazole-5-carboxylate —— C20H24FN3O4S
Ethyl 2-[(4-fluorophenyl)methyl-(2-morpholin-4-ylacetyl)amino]-4-methyl-1,3-thiazole-5-carboxylate
—— Ethyl 4-acetyl-2-[[2-[benzyl(methyl)amino]acetyl]amino]-5-methylfuran-3-carboxylate —— C20H24N2O5
Ethyl 4-acetyl-2-[[2-[benzyl(methyl)amino]acetyl]amino]-5-methylfuran-3-carboxylate
—— Ethyl 2-[(2-piperidin-1-ium-1-ylacetyl)amino]-6-propan-2-yl-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-6-ium-3-carboxylate —— C20H33N3O3S+2
Ethyl 2-[(2-piperidin-1-ium-1-ylacetyl)amino]-6-propan-2-yl-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-6-ium-3-carboxylate
—— (E)-2-(4-aminobenzoyl)-3-(3-hydroxyphenyl)prop-2-enenitrile —— C16H12N2O2
(E)-2-(4-aminobenzoyl)-3-(3-hydroxyphenyl)prop-2-enenitrile
—— ethyl (4R)-6-(azepan-1-ylmethyl)-4-(furan-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H25N3O4
ethyl (4R)-6-(azepan-1-ylmethyl)-4-(furan-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H30N4O4S
ethyl (5R)-3-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(3-bromo-4-hydroxyphenyl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H23BrN2O6S
ethyl (2E,5R)-2-[(3-bromo-4-hydroxyphenyl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[2-[(2-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5R)-2-[[2-[(2-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 6-[(2S)-2-(2,4-dichlorophenoxy)propanoyl]imino-2-oxo-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxylate —— C26H24Cl2N4O5
ethyl 6-[(2S)-2-(2,4-dichlorophenoxy)propanoyl]imino-2-oxo-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24Cl2N2O6S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[[5-(4-methyl-2-nitrophenyl)furan-2-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H27N3O8S
ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[[5-(4-methyl-2-nitrophenyl)furan-2-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H23BrN2O7S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 6-[(2R)-2-(2,4-dichlorophenoxy)propanoyl]imino-2-oxo-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxylate —— C26H24Cl2N4O5
ethyl 6-[(2R)-2-(2,4-dichlorophenoxy)propanoyl]imino-2-oxo-7-propyl-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(2-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25ClN2O6S
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(2-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[5-(4-bromophenyl)furan-2-yl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H25BrN2O6S
ethyl (2E,5R)-2-[[5-(4-bromophenyl)furan-2-yl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25ClN2O6S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24Cl2N2O6S
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5S)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[(3-bromo-4-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H19BrN2O6S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[(3-bromo-4-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34ClN3O5S
ethyl (2E,5R)-2-[[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-5-(1,3-benzothiazol-2-yl)-6-(5-bromothiophen-2-yl)hex-5-enoic acid —— C17H14BrNO2S2
(E)-5-(1,3-benzothiazol-2-yl)-6-(5-bromothiophen-2-yl)hex-5-enoic acid
—— ethyl (2E,5S)-2-[[2-[(2-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5S)-2-[[2-[(2-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 5-cyano-6-[(2-cyanophenyl)methylsulfanyl]-2-methylpyridine-3-carboxylate —— C18H15N3O2S
Ethyl 5-cyano-6-[(2-cyanophenyl)methylsulfanyl]-2-methylpyridine-3-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24Cl2N2O6S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24Cl2N2O6S
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[5-(4-bromophenyl)furan-2-yl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H25BrN2O6S
ethyl (2E,5S)-2-[[5-(4-bromophenyl)furan-2-yl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5R)-2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25ClN2O6S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(2-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25ClN2O6S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-[(2-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34ClN3O5S
ethyl (2E,5R)-2-[[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-5-[4-(dimethylamino)phenyl]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[4-[(2-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5S)-2-[[4-[(2-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[[5-(4-methyl-2-nitrophenyl)furan-2-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H27N3O8S
ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[[5-(4-methyl-2-nitrophenyl)furan-2-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5R)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25ClN2O6S
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 5-cyano-2-methyl-6-[2-oxo-2-[[(2R)-1-oxo-1-(propylamino)propan-2-yl]amino]ethyl]sulfanylpyridine-3-carboxylate —— C18H24N4O4S
ethyl 5-cyano-2-methyl-6-[2-oxo-2-[[(2R)-1-oxo-1-(propylamino)propan-2-yl]amino]ethyl]sulfanylpyridine-3-carboxylate
—— ethyl (2E,5R)-5-(4-chlorophenyl)-2-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H29ClN2O5S
ethyl (2E,5R)-5-(4-chlorophenyl)-2-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate