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—— ethyl 4-[(Z)-[(2R)-2-(3,4-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H35N3O7
ethyl 4-[(Z)-[(2R)-2-(3,4-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6S)-3-butyl-6-[3-[[(Z)-3-(4-nitrophenyl)prop-2-enoyl]amino]phenyl]-2-oxo-4-phenyl-1,6-dihydropyrimidine-5-carboxylate —— C32H32N4O6
ethyl (6S)-3-butyl-6-[3-[[(Z)-3-(4-nitrophenyl)prop-2-enoyl]amino]phenyl]-2-oxo-4-phenyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(3,4-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H35N3O7
ethyl 4-[(Z)-[(2S)-2-(3,4-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6R)-6-[4-[[(Z)-3-(4-nitrophenyl)prop-2-enoyl]amino]phenyl]-2-oxo-4-phenyl-3-propyl-1,6-dihydropyrimidine-5-carboxylate —— C31H30N4O6
ethyl (6R)-6-[4-[[(Z)-3-(4-nitrophenyl)prop-2-enoyl]amino]phenyl]-2-oxo-4-phenyl-3-propyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2R)-2-(5-methylfuran-2-yl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O7
ethyl 4-[(Z)-hydroxy-[(2R)-2-(5-methylfuran-2-yl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 5-[(2R)-2-[[2-(3-methoxyanilino)-2-oxoethyl]-methylamino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H29N3O5
ethyl 5-[(2R)-2-[[2-(3-methoxyanilino)-2-oxoethyl]-methylamino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 5-[(2S)-2-[[2-(3-methoxyanilino)-2-oxoethyl]-methylamino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H29N3O5
ethyl 5-[(2S)-2-[[2-(3-methoxyanilino)-2-oxoethyl]-methylamino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2S)-2-(5-methylfuran-2-yl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O7
ethyl 4-[(Z)-hydroxy-[(2S)-2-(5-methylfuran-2-yl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-phenylpyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H31N3O5
ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-phenylpyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (6R)-2-oxo-4-phenyl-3-propyl-6-[3-[[4-(trifluoromethyl)benzoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C30H28F3N3O4
ethyl (6R)-2-oxo-4-phenyl-3-propyl-6-[3-[[4-(trifluoromethyl)benzoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[[[(1S)-1-[7-chloro-3-(4-methylphenyl)-4-oxoquinazolin-2-yl]ethyl]-pentylcarbamoyl]amino]benzoate —— C32H35ClN4O4
ethyl 4-[[[(1S)-1-[7-chloro-3-(4-methylphenyl)-4-oxoquinazolin-2-yl]ethyl]-pentylcarbamoyl]amino]benzoate
—— ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-phenylpyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H31N3O5
ethyl 4-[(Z)-[(2R)-1-[3-(dimethylamino)propyl]-4,5-dioxo-2-phenylpyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2S)-1-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H28FN3O5
ethyl 4-[(Z)-[(2S)-1-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-(1-butyl-2,5-dimethylpyrrol-3-yl)-2-cyano-N-(3-cyanophenyl)prop-2-enamide —— C21H22N4O
(E)-3-(1-butyl-2,5-dimethylpyrrol-3-yl)-2-cyano-N-(3-cyanophenyl)prop-2-enamide
—— ethyl (6S)-2-oxo-4-phenyl-3-propyl-6-[3-[[4-(trifluoromethyl)benzoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C30H28F3N3O4
ethyl (6S)-2-oxo-4-phenyl-3-propyl-6-[3-[[4-(trifluoromethyl)benzoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— (E)-N-[(1S)-1-(1-adamantyl)ethyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C21H31N3O
(E)-N-[(1S)-1-(1-adamantyl)ethyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— ethyl 4-[(Z)-[(2R)-2-(3-chlorophenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H30ClN3O5
ethyl 4-[(Z)-[(2R)-2-(3-chlorophenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-(3-cyanophenyl)-3-(2-methylphenyl)prop-2-enamide —— C17H14N2O
(E)-N-(3-cyanophenyl)-3-(2-methylphenyl)prop-2-enamide
—— (E)-N-cycloheptyl-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]prop-2-enamide —— C19H28N2O4S
(E)-N-cycloheptyl-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]prop-2-enamide
—— (E)-N-(3-cyanophenyl)-3-(3-methoxy-4-propoxyphenyl)prop-2-enamide —— C20H20N2O3
(E)-N-(3-cyanophenyl)-3-(3-methoxy-4-propoxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-(3-cyanophenyl)-3-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]prop-2-enamide —— C22H22N4O2
(E)-2-cyano-N-(3-cyanophenyl)-3-[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]prop-2-enamide
—— (E)-3-(4-bromophenyl)-N-(3-cyanophenyl)prop-2-enamide —— C16H11BrN2O
(E)-3-(4-bromophenyl)-N-(3-cyanophenyl)prop-2-enamide
—— (E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide —— C18H21N3O3S2
(E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide
—— (E)-N-(3-cyanophenyl)-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide —— C20H19N3O4S
(E)-N-(3-cyanophenyl)-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide
—— (E)-2-cyano-N-(3-cyanophenyl)-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]prop-2-enamide —— C21H22N4O
(E)-2-cyano-N-(3-cyanophenyl)-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]prop-2-enamide
—— (E)-N-(2-fluoro-4-methylphenyl)-3-(4-fluorophenyl)prop-2-enamide —— C16H13F2NO
(E)-N-(2-fluoro-4-methylphenyl)-3-(4-fluorophenyl)prop-2-enamide
—— ethyl 4-[(Z)-hydroxy-[(2R)-1-(3-imidazol-1-ylpropyl)-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H30N4O6
ethyl 4-[(Z)-hydroxy-[(2R)-1-(3-imidazol-1-ylpropyl)-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(4-tert-butylphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C30H36N4O5
ethyl 4-[(Z)-[(2R)-2-(4-tert-butylphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide —— C15H15N3O3S2
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide
—— ethyl 4-[(Z)-[(2R)-1-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H28FN3O5
ethyl 4-[(Z)-[(2R)-1-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-(4-methyl-3-morpholin-4-ylsulfonylphenyl)-3-phenylprop-2-enamide —— C20H22N2O4S
(E)-N-(4-methyl-3-morpholin-4-ylsulfonylphenyl)-3-phenylprop-2-enamide
—— ethyl 4-[[[(1R)-1-[7-chloro-3-(4-methylphenyl)-4-oxoquinazolin-2-yl]ethyl]-pentylcarbamoyl]amino]benzoate —— C32H35ClN4O4
ethyl 4-[[[(1R)-1-[7-chloro-3-(4-methylphenyl)-4-oxoquinazolin-2-yl]ethyl]-pentylcarbamoyl]amino]benzoate
—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-(2-methyl-6-propan-2-ylphenyl)prop-2-enamide —— C22H24N2O3
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-(2-methyl-6-propan-2-ylphenyl)prop-2-enamide
—— ethyl 4-[(Z)-[(2S)-2-(3-chlorophenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H30ClN3O5
ethyl 4-[(Z)-[(2S)-2-(3-chlorophenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C16H19N3O4S2
(E)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— Ethyl 2-[[2-(3-formylphenoxy)acetyl]amino]-5-propan-2-ylthiophene-3-carboxylate —— C19H21NO5S
Ethyl 2-[[2-(3-formylphenoxy)acetyl]amino]-5-propan-2-ylthiophene-3-carboxylate
—— (E)-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide —— C16H17N3O3S2
(E)-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide
—— ethyl 4-[(Z)-[(2S)-2-(4-tert-butylphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C30H36N4O5
ethyl 4-[(Z)-[(2S)-2-(4-tert-butylphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-(2,3-dichlorophenyl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide —— C13H11Cl2N3OS2
(E)-3-(2,3-dichlorophenyl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide
—— ethyl 4-[(Z)-[(2S)-2-(2-fluorophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H32FN3O6
ethyl 4-[(Z)-[(2S)-2-(2-fluorophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(2-fluorophenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H24FN3O5
ethyl 4-[(Z)-[(2R)-2-(2-fluorophenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— Ethyl 5-ethyl-2-[[2-(3-formylphenoxy)acetyl]amino]-4-methylthiophene-3-carboxylate —— C19H21NO5S
Ethyl 5-ethyl-2-[[2-(3-formylphenoxy)acetyl]amino]-4-methylthiophene-3-carboxylate
—— Ethyl 2-[[2-(1,3-benzodioxol-5-yloxy)acetyl]amino]-5-propan-2-ylthiophene-3-carboxylate —— C19H21NO6S
Ethyl 2-[[2-(1,3-benzodioxol-5-yloxy)acetyl]amino]-5-propan-2-ylthiophene-3-carboxylate
—— ethyl 1-[4-[(2-methoxybenzoyl)amino]-2-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]phenyl]piperidine-4-carboxylate —— C32H37N3O6S
ethyl 1-[4-[(2-methoxybenzoyl)amino]-2-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]phenyl]piperidine-4-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(2-fluorophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H32FN3O6
ethyl 4-[(Z)-[(2R)-2-(2-fluorophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enamide —— C17H19N3O3S2
(E)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enamide
—— ethyl 2-[(2S,3Z)-2-(2-fluorophenyl)-3-[hydroxy-(4-prop-2-enoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H23FN2O6S
ethyl 2-[(2S,3Z)-2-(2-fluorophenyl)-3-[hydroxy-(4-prop-2-enoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 1-[4-[(2-methoxybenzoyl)amino]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]phenyl]piperidine-4-carboxylate —— C32H37N3O6S
ethyl 1-[4-[(2-methoxybenzoyl)amino]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]phenyl]piperidine-4-carboxylate
—— ethyl 2-[(4Z,5R)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-thiophen-2-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H24N2O6S2
ethyl 2-[(4Z,5R)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-thiophen-2-ylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide —— C16H18ClN3O3S2
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-(5-ethylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide