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—— ethyl 2-[(2S,3Z)-2-(4-ethoxyphenyl)-3-[hydroxy-(4-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H26N2O6S
ethyl 2-[(2S,3Z)-2-(4-ethoxyphenyl)-3-[hydroxy-(4-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Ethyl 5-cyano-2-methyl-6-[2-[methyl-[(2-methylphenyl)methyl]amino]-2-oxoethyl]sulfanylpyridine-3-carboxylate —— C21H23N3O3S
Ethyl 5-cyano-2-methyl-6-[2-[methyl-[(2-methylphenyl)methyl]amino]-2-oxoethyl]sulfanylpyridine-3-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2S)-2-(2-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H27N3O6
ethyl 4-[(Z)-hydroxy-[(2S)-2-(2-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-(2-pyridin-2-ylbenzimidazol-1-yl)-3-[[(1S,4R)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate —— C31H30N4O5
ethyl 4-(2-pyridin-2-ylbenzimidazol-1-yl)-3-[[(1S,4R)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carbonyl]amino]benzoate
—— Ethyl 5-cyano-2-methyl-6-[2-oxo-2-(2-oxopyrrolidin-1-yl)ethyl]sulfanylpyridine-3-carboxylate —— C16H17N3O4S
Ethyl 5-cyano-2-methyl-6-[2-oxo-2-(2-oxopyrrolidin-1-yl)ethyl]sulfanylpyridine-3-carboxylate
—— ethyl (2R)-2-[[(2S)-butan-2-yl]amino]nonanoate —— C15H31NO2
ethyl (2R)-2-[[(2S)-butan-2-yl]amino]nonanoate
—— ethyl 4-[(Z)-[(2S)-2-(4-tert-butylphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O5
ethyl 4-[(Z)-[(2S)-2-(4-tert-butylphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[2-[5-(3-fluorophenyl)tetrazol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C18H18FN5O3
ethyl 4-[2-[5-(3-fluorophenyl)tetrazol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 5-cyano-6-[2-(2-fluorophenoxy)ethylsulfanyl]-2-methylpyridine-3-carboxylate —— C18H17FN2O3S
Ethyl 5-cyano-6-[2-(2-fluorophenoxy)ethylsulfanyl]-2-methylpyridine-3-carboxylate
—— Ethyl 5-cyano-6-[2-[(2-methoxyphenyl)methylamino]-2-oxoethyl]sulfanyl-2-methylpyridine-3-carboxylate —— C20H21N3O4S
Ethyl 5-cyano-6-[2-[(2-methoxyphenyl)methylamino]-2-oxoethyl]sulfanyl-2-methylpyridine-3-carboxylate
—— Ethyl 6-[2-(3-chloro-4-fluoroanilino)-2-oxoethyl]sulfanyl-5-cyano-2-methylpyridine-3-carboxylate —— C18H15ClFN3O3S
Ethyl 6-[2-(3-chloro-4-fluoroanilino)-2-oxoethyl]sulfanyl-5-cyano-2-methylpyridine-3-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(4-tert-butylphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H37N3O5
ethyl 4-[(Z)-[(2R)-2-(4-tert-butylphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-(3-ethoxypropyl)-N-[2-[(4R)-4-(4-methylphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide —— C30H33N3O5S
(E)-N-(3-ethoxypropyl)-N-[2-[(4R)-4-(4-methylphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide
—— ethyl 4-[(Z)-hydroxy-[(2R)-2-(2-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H35N3O7
ethyl 4-[(Z)-hydroxy-[(2R)-2-(2-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2R)-2-(2-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H27N3O6
ethyl 4-[(Z)-hydroxy-[(2R)-2-(2-methoxyphenyl)-4,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (3S)-1-[2-(3,4-dimethylphenyl)-3,5-dioxo-4-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-triazine-6-carbonyl]piperidine-3-carboxylate —— C28H29F3N4O5
ethyl (3S)-1-[2-(3,4-dimethylphenyl)-3,5-dioxo-4-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-triazine-6-carbonyl]piperidine-3-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2S)-2-(2-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H35N3O7
ethyl 4-[(Z)-hydroxy-[(2S)-2-(2-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— Ethyl 3-[2-(4-chlorophenyl)sulfanylethyl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxylate —— C18H17ClN2O3S2
Ethyl 3-[2-(4-chlorophenyl)sulfanylethyl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl (E)-3-[2-(N-acetyl-3,4-dimethylanilino)-1,3-thiazol-4-yl]-2-cyanoprop-2-enoate —— C19H19N3O3S
ethyl (E)-3-[2-(N-acetyl-3,4-dimethylanilino)-1,3-thiazol-4-yl]-2-cyanoprop-2-enoate
—— ethyl (E)-2-cyano-3-[2-(difluoromethoxy)naphthalen-1-yl]prop-2-enoate —— C17H13F2NO3
ethyl (E)-2-cyano-3-[2-(difluoromethoxy)naphthalen-1-yl]prop-2-enoate
—— ethyl (E)-3-[3-chloro-4-(difluoromethoxy)-5-methoxyphenyl]-2-cyanoprop-2-enoate —— C14H12ClF2NO4
ethyl (E)-3-[3-chloro-4-(difluoromethoxy)-5-methoxyphenyl]-2-cyanoprop-2-enoate
—— ethyl (E)-2-cyano-3-(2-phenylmethoxyphenyl)prop-2-enoate —— C19H17NO3
ethyl (E)-2-cyano-3-(2-phenylmethoxyphenyl)prop-2-enoate
—— (E)-N-(3-ethoxypropyl)-N-[2-[(4S)-4-(4-methylphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide —— C30H33N3O5S
(E)-N-(3-ethoxypropyl)-N-[2-[(4S)-4-(4-methylphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide
—— ethyl (E)-2-cyano-3-(3-ethoxy-4-phenylmethoxyphenyl)prop-2-enoate —— C21H21NO4
ethyl (E)-2-cyano-3-(3-ethoxy-4-phenylmethoxyphenyl)prop-2-enoate
—— [(E)-3-phenylprop-2-enyl] 5-(dimethylsulfamoyl)-2-(2-hydroxyethylamino)benzoate —— C20H24N2O5S
[(E)-3-phenylprop-2-enyl] 5-(dimethylsulfamoyl)-2-(2-hydroxyethylamino)benzoate
—— ethyl (3R)-1-[2-(3,4-dimethylphenyl)-3,5-dioxo-4-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-triazine-6-carbonyl]piperidine-3-carboxylate —— C28H29F3N4O5
ethyl (3R)-1-[2-(3,4-dimethylphenyl)-3,5-dioxo-4-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-triazine-6-carbonyl]piperidine-3-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(3,4-dimethoxyphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H32N4O7
ethyl 4-[(Z)-[(2S)-2-(3,4-dimethoxyphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (1S,5S)-3-[[(2R)-butan-2-yl]amino]-8-methyl-8-azabicyclo[3.2.1]octane-3-carboxylate —— C15H28N2O2
ethyl (1S,5S)-3-[[(2R)-butan-2-yl]amino]-8-methyl-8-azabicyclo[3.2.1]octane-3-carboxylate
—— ethyl 6-benzyl-2-[[(2R)-2-(3,4,5-trimethoxybenzoyl)oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H34N2O8S
ethyl 6-benzyl-2-[[(2R)-2-(3,4,5-trimethoxybenzoyl)oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2,4-dimethyl-5-[(2S)-2-[2-(2-oxopyridin-1-yl)acetyl]oxypropanoyl]-1H-pyrrole-3-carboxylate —— C19H22N2O6
ethyl 2,4-dimethyl-5-[(2S)-2-[2-(2-oxopyridin-1-yl)acetyl]oxypropanoyl]-1H-pyrrole-3-carboxylate
—— ethyl 4-[(Z)-hydroxy-[(2S)-2-(4-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H35N3O7
ethyl 4-[(Z)-hydroxy-[(2S)-2-(4-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl (2R)-2-[[(2R)-butan-2-yl]amino]nonanoate —— C15H31NO2
ethyl (2R)-2-[[(2R)-butan-2-yl]amino]nonanoate
—— ethyl (2S)-2-[[(2R)-butan-2-yl]amino]nonanoate —— C15H31NO2
ethyl (2S)-2-[[(2R)-butan-2-yl]amino]nonanoate
—— ethyl 4-[(Z)-hydroxy-[(2R)-2-(4-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H35N3O7
ethyl 4-[(Z)-hydroxy-[(2R)-2-(4-methoxyphenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(3,4-dimethoxyphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H32N4O7
ethyl 4-[(Z)-[(2R)-2-(3,4-dimethoxyphenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-N-tert-butyl-N-[2-[(4R)-4-(4-methoxyphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide —— C29H31N3O5S
(E)-N-tert-butyl-N-[2-[(4R)-4-(4-methoxyphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide
—— ethyl 6-benzyl-2-[[(2S)-2-(3,4,5-trimethoxybenzoyl)oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H34N2O8S
ethyl 6-benzyl-2-[[(2S)-2-(3,4,5-trimethoxybenzoyl)oxypropanoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl (2S)-2-[[(2S)-butan-2-yl]amino]nonanoate —— C15H31NO2
ethyl (2S)-2-[[(2S)-butan-2-yl]amino]nonanoate
—— ethyl (1S,5S)-3-[[(2S)-butan-2-yl]amino]-8-methyl-8-azabicyclo[3.2.1]octane-3-carboxylate —— C15H28N2O2
ethyl (1S,5S)-3-[[(2S)-butan-2-yl]amino]-8-methyl-8-azabicyclo[3.2.1]octane-3-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(3-bromophenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H30BrN3O5
ethyl 4-[(Z)-[(2R)-2-(3-bromophenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 2-[[(2R)-2-(2,6-dimethoxybenzoyl)oxy-2-phenylacetyl]amino]-4-phenylthiophene-3-carboxylate —— C30H27NO7S
ethyl 2-[[(2R)-2-(2,6-dimethoxybenzoyl)oxy-2-phenylacetyl]amino]-4-phenylthiophene-3-carboxylate
—— (E)-N-tert-butyl-N-[2-[(4S)-4-(4-methoxyphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide —— C29H31N3O5S
(E)-N-tert-butyl-N-[2-[(4S)-4-(4-methoxyphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-(4-nitrophenyl)prop-2-enamide
—— ethyl 2-[[(2S)-2-(2,6-dimethoxybenzoyl)oxy-2-phenylacetyl]amino]-4-phenylthiophene-3-carboxylate —— C30H27NO7S
ethyl 2-[[(2S)-2-(2,6-dimethoxybenzoyl)oxy-2-phenylacetyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(2,3-dimethoxyphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O7
ethyl 4-[(Z)-[(2R)-2-(2,3-dimethoxyphenyl)-1-[2-(dimethylamino)ethyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(2,5-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H35N3O7
ethyl 4-[(Z)-[(2S)-2-(2,5-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(2,5-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H35N3O7
ethyl 4-[(Z)-[(2R)-2-(2,5-dimethoxyphenyl)-1-[3-(dimethylamino)propyl]-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[(2R,3E)-3-[hydroxy-(4-nitrophenyl)methylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]benzoate —— C27H22N2O8
ethyl 4-[(2R,3E)-3-[hydroxy-(4-nitrophenyl)methylidene]-2-(4-methoxyphenyl)-4,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl (3S)-1-[4-[6-[2-(4-methoxyphenoxy)acetyl]-3-oxo-1,4-benzoxazin-4-yl]butanoyl]piperidine-3-carboxylate —— C29H34N2O8
ethyl (3S)-1-[4-[6-[2-(4-methoxyphenoxy)acetyl]-3-oxo-1,4-benzoxazin-4-yl]butanoyl]piperidine-3-carboxylate
—— ethyl 7-[(1S)-6-methoxy-1-(4-phenylmethoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-7-oxoheptanoate —— C34H38N2O5
ethyl 7-[(1S)-6-methoxy-1-(4-phenylmethoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-7-oxoheptanoate
—— ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-2-(4-methoxycarbonylphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H33N3O7
ethyl 4-[(Z)-[(2S)-1-[3-(dimethylamino)propyl]-2-(4-methoxycarbonylphenyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate