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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 4-[[(1R,5R)-8-[4-[(4-tert-butylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C34H39NO4S
ethyl 4-[[(1R,5R)-8-[4-[(4-tert-butylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(2-methylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C31H33NO4S
ethyl 4-[[(1R,5R)-8-[4-[(2-methylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(3,5-dimethylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C32H35NO4S
ethyl 4-[[(1R,5R)-8-[4-[(3,5-dimethylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— (E)-N-(3,4-dimethylphenyl)-2-phenylethenesulfonamide —— C16H17NO2S
(E)-N-(3,4-dimethylphenyl)-2-phenylethenesulfonamide
—— ethyl 4-[[(1S,5S)-8-[4-[(4-methylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C31H33NO4S
ethyl 4-[[(1S,5S)-8-[4-[(4-methylphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(E)-2-(4-chlorophenyl)ethenyl]sulfonylamino]benzoate —— C17H16ClNO4S
ethyl 4-[[(E)-2-(4-chlorophenyl)ethenyl]sulfonylamino]benzoate
—— (E)-N-(2-methyl-5-nitrophenyl)-2-phenylethenesulfonamide —— C15H14N2O4S
(E)-N-(2-methyl-5-nitrophenyl)-2-phenylethenesulfonamide
—— Ethyl 4-[(5-acetamido-2-methoxyphenyl)sulfamoyl]benzoate —— C18H20N2O6S
Ethyl 4-[(5-acetamido-2-methoxyphenyl)sulfamoyl]benzoate
—— (E)-N-[4-(2,5-dimethoxyphenyl)-1,3-thiazol-2-yl]-2-phenylethenesulfonamide —— C19H18N2O4S2
(E)-N-[4-(2,5-dimethoxyphenyl)-1,3-thiazol-2-yl]-2-phenylethenesulfonamide
—— ethyl 5-chloro-2-[[2-[4-[[(2S)-oxolan-2-yl]methoxy]benzoyl]oxyacetyl]amino]-4-phenylthiophene-3-carboxylate —— C27H26ClNO7S
ethyl 5-chloro-2-[[2-[4-[[(2S)-oxolan-2-yl]methoxy]benzoyl]oxyacetyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl (3S)-1-[(2R)-2-[(4S)-4-(2,4-dichlorophenyl)-1-ethyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]propanoyl]piperidine-3-carboxylate —— C25H30Cl2N4O5
ethyl (3S)-1-[(2R)-2-[(4S)-4-(2,4-dichlorophenyl)-1-ethyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]propanoyl]piperidine-3-carboxylate
—— ethyl 2-[(1S)-1-[(4-fluorophenyl)methylsulfanyl]ethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C19H19FN2O3S2
ethyl 2-[(1S)-1-[(4-fluorophenyl)methylsulfanyl]ethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl (E)-2-cyano-3-[2-[(4-ethoxyphenyl)sulfonylamino]anilino]prop-2-enoate —— C20H21N3O5S
ethyl (E)-2-cyano-3-[2-[(4-ethoxyphenyl)sulfonylamino]anilino]prop-2-enoate
—— ethyl 2-[(1S)-1-[2-(2-methoxyethylamino)-2-oxoethyl]sulfanylethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C17H23N3O5S2
ethyl 2-[(1S)-1-[2-(2-methoxyethylamino)-2-oxoethyl]sulfanylethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl (E)-3-[2-(benzenesulfonamido)anilino]-2-cyanoprop-2-enoate —— C18H17N3O4S
ethyl (E)-3-[2-(benzenesulfonamido)anilino]-2-cyanoprop-2-enoate
—— ethyl (3S)-1-[(2R)-2-[(4S)-4-(4-chlorophenyl)-1-methyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate —— C30H33ClN4O5
ethyl (3S)-1-[(2R)-2-[(4S)-4-(4-chlorophenyl)-1-methyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-phenylpropanoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[(2S)-2-[(4S)-4-(2,4-dichlorophenyl)-1-ethyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]propanoyl]piperidine-3-carboxylate —— C25H30Cl2N4O5
ethyl (3S)-1-[(2S)-2-[(4S)-4-(2,4-dichlorophenyl)-1-ethyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]propanoyl]piperidine-3-carboxylate
—— ethyl 5-methyl-4-oxo-2-[(1R)-1-[2-oxo-2-[[(2R)-pentan-2-yl]amino]ethyl]sulfanylethyl]-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C19H27N3O4S2
ethyl 5-methyl-4-oxo-2-[(1R)-1-[2-oxo-2-[[(2R)-pentan-2-yl]amino]ethyl]sulfanylethyl]-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 5-methyl-2-[(1R)-1-[(4-methylphenyl)methylsulfanyl]ethyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C20H22N2O3S2
ethyl 5-methyl-2-[(1R)-1-[(4-methylphenyl)methylsulfanyl]ethyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 4-[[(1S,5S)-8-[4-[(3,4-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1S,5S)-8-[4-[(3,4-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl (3R)-1-[(4-oxo-3H-[1]benzofuro[3,2-d]pyrimidin-2-yl)methyl]piperidine-3-carboxylate —— C19H21N3O4
ethyl (3R)-1-[(4-oxo-3H-[1]benzofuro[3,2-d]pyrimidin-2-yl)methyl]piperidine-3-carboxylate
—— ethyl (5R)-5-(2,3-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,3-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[2-[2-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]oxyacetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate —— C23H26N2O7S
ethyl 2-[[2-[2-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]oxyacetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate
—— ethyl 2-[2-[2-[(3R)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,3-thiazol-4-yl]acetate —— C29H27N3O4S2
ethyl 2-[2-[2-[(3R)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,3-thiazol-4-yl]acetate
—— ethyl 5-chloro-2-[[2-[4-[[(2R)-oxolan-2-yl]methoxy]benzoyl]oxyacetyl]amino]-4-phenylthiophene-3-carboxylate —— C27H26ClNO7S
ethyl 5-chloro-2-[[2-[4-[[(2R)-oxolan-2-yl]methoxy]benzoyl]oxyacetyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl (1'S,2'R,3S,3'aR)-2-oxo-2'-(4-pentylbenzoyl)spiro[1H-indole-3,3'-2,3a-dihydro-1H-pyrrolo[1,2-a]quinoline]-1'-carboxylate —— C34H34N2O4
ethyl (1'S,2'R,3S,3'aR)-2-oxo-2'-(4-pentylbenzoyl)spiro[1H-indole-3,3'-2,3a-dihydro-1H-pyrrolo[1,2-a]quinoline]-1'-carboxylate
—— ethyl 4-[[(1R,5S)-8-[4-[(2,3-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1R,5S)-8-[4-[(2,3-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(2,5-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1R,5R)-8-[4-[(2,5-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(2,3-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1R,5R)-8-[4-[(2,3-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1S,5S)-8-[4-(phenylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H31NO4S
ethyl 4-[[(1S,5S)-8-[4-(phenylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetate —— C17H17N3O5
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetate
—— ethyl (3S)-1-[(2S)-2-[(4R)-4-(2,4-dichlorophenyl)-1-ethyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]propanoyl]piperidine-3-carboxylate —— C25H30Cl2N4O5
ethyl (3S)-1-[(2S)-2-[(4R)-4-(2,4-dichlorophenyl)-1-ethyl-2,5-dioxo-4,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-6-yl]propanoyl]piperidine-3-carboxylate
—— ethyl (5R)-5-(2,3-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5R)-5-(2,3-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(1S,5S)-8-[4-[(2-methoxyphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C31H33NO5S
ethyl 4-[[(1S,5S)-8-[4-[(2-methoxyphenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5S)-8-[4-[(3,4-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1R,5S)-8-[4-[(3,4-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1S,5S)-8-[4-[(3-fluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H30FNO4S
ethyl 4-[[(1S,5S)-8-[4-[(3-fluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 2-[2-[2-[(3S)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,3-thiazol-4-yl]acetate —— C29H27N3O4S2
ethyl 2-[2-[2-[(3S)-3-(4-methoxyphenyl)-5-naphthalen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1,3-thiazol-4-yl]acetate
—— ethyl (5S)-5-(2,3-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,3-dimethoxyphenyl)-3-[2-(4-ethoxycarbonylpiperidin-1-yl)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(1R,5R)-8-[4-[(3-fluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H30FNO4S
ethyl 4-[[(1R,5R)-8-[4-[(3-fluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetate —— C17H17N3O5
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetate
—— ethyl 4-[[(1R,5R)-8-[4-[[bis(3-methylbutyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C34H48N2O4
ethyl 4-[[(1R,5R)-8-[4-[[bis(3-methylbutyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 2-[[2-[2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]oxyacetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate —— C23H26N2O7S
ethyl 2-[[2-[2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]oxyacetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate
—— ethyl 4-[[(1S,5S)-8-[4-[(2,3-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1S,5S)-8-[4-[(2,3-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl (5S)-5-(2,3-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,3-dimethoxyphenyl)-3-[2-[(3S)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(1R,5S)-8-[4-[[bis(3-methylbutyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C34H48N2O4
ethyl 4-[[(1R,5S)-8-[4-[[bis(3-methylbutyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1S,5S)-8-[4-[(2,5-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1S,5S)-8-[4-[(2,5-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1R,5R)-8-[4-[(3,4-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H29Cl2NO4S
ethyl 4-[[(1R,5R)-8-[4-[(3,4-dichlorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 4-[[(1S,5S)-8-[4-[[bis(3-methylbutyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C34H48N2O4
ethyl 4-[[(1S,5S)-8-[4-[[bis(3-methylbutyl)amino]methyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl (5S)-5-(2,3-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H37N3O7S
ethyl (5S)-5-(2,3-dimethoxyphenyl)-3-[2-[(3R)-3-ethoxycarbonylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(1R,5R)-8-[4-(phenylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H31NO4S
ethyl 4-[[(1R,5R)-8-[4-(phenylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate