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—— ethyl 5-[2-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C29H35FN4O4S
ethyl 5-[2-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 4-(furan-2-yl)-2-[[2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl]amino]thiophene-3-carboxylate —— C17H16N2O4S3
Ethyl 4-(furan-2-yl)-2-[[2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl]amino]thiophene-3-carboxylate
—— ethyl (6R)-2-[[2-[[3-[(2R)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H35N3O4S3
ethyl (6R)-2-[[2-[[3-[(2R)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 4-[[(1R,5R)-8-[4-(thiophen-2-ylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C28H29NO4S2
ethyl 4-[[(1R,5R)-8-[4-(thiophen-2-ylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl (3S)-1-[2-[3-[benzyl-(2,4-dichlorobenzoyl)amino]phenyl]acetyl]piperidine-3-carboxylate —— C30H30Cl2N2O4
ethyl (3S)-1-[2-[3-[benzyl-(2,4-dichlorobenzoyl)amino]phenyl]acetyl]piperidine-3-carboxylate
—— Ethyl 2-amino-5-(methylcarbamoyl)-4-[(4-methyl-1,3-thiazol-2-yl)sulfanylmethyl]thiophene-3-carboxylate —— C14H17N3O3S3
Ethyl 2-amino-5-(methylcarbamoyl)-4-[(4-methyl-1,3-thiazol-2-yl)sulfanylmethyl]thiophene-3-carboxylate
—— ethyl 4-[[(1S,5S)-8-[4-[(2-fluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C30H30FNO4S
ethyl 4-[[(1S,5S)-8-[4-[(2-fluorophenyl)sulfanylmethyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl (3R)-1-[2-[3-[benzyl-(2,4-dichlorobenzoyl)amino]phenyl]acetyl]piperidine-3-carboxylate —— C30H30Cl2N2O4
ethyl (3R)-1-[2-[3-[benzyl-(2,4-dichlorobenzoyl)amino]phenyl]acetyl]piperidine-3-carboxylate
—— ethyl (4S)-1-[[4-[2-(2,4-dichlorophenyl)ethylcarbamoyl]phenyl]methyl]-6-methyl-4-(4-methylphenyl)-2-oxo-3,4-dihydropyridine-5-carboxylate —— C32H32Cl2N2O4
ethyl (4S)-1-[[4-[2-(2,4-dichlorophenyl)ethylcarbamoyl]phenyl]methyl]-6-methyl-4-(4-methylphenyl)-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (6S)-2-[[2-[[3-[(2R)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H35N3O4S3
ethyl (6S)-2-[[2-[[3-[(2R)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 3-[2-(2-benzylanilino)-2-oxoethoxy]benzoate —— C24H23NO4
Ethyl 3-[2-(2-benzylanilino)-2-oxoethoxy]benzoate
—— Ethyl 3-[2-(4-cyanoanilino)-2-oxoethoxy]benzoate —— C18H16N2O4
Ethyl 3-[2-(4-cyanoanilino)-2-oxoethoxy]benzoate
—— ethyl (4R)-6-methyl-2-oxo-4-(3-phenoxyphenyl)-1-[[5-[[(1S)-1-phenylethyl]carbamoyl]furan-2-yl]methyl]-3,4-dihydropyridine-5-carboxylate —— C35H34N2O6
ethyl (4R)-6-methyl-2-oxo-4-(3-phenoxyphenyl)-1-[[5-[[(1S)-1-phenylethyl]carbamoyl]furan-2-yl]methyl]-3,4-dihydropyridine-5-carboxylate
—— ethyl 1-[2-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-4-carboxylate —— C28H37FN4O4S
ethyl 1-[2-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-4-carboxylate
—— ethyl 3-[(2R)-1-oxo-1-(4-sulfamoylanilino)propan-2-yl]oxybenzoate —— C18H20N2O6S
ethyl 3-[(2R)-1-oxo-1-(4-sulfamoylanilino)propan-2-yl]oxybenzoate
—— Ethyl 3-[2-[(4-chlorophenyl)methylamino]-2-oxoethoxy]benzoate —— C18H18ClNO4
Ethyl 3-[2-[(4-chlorophenyl)methylamino]-2-oxoethoxy]benzoate
—— ethyl (2S)-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]-2-phenylacetate —— C17H16N2O4S
ethyl (2S)-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]-2-phenylacetate
—— ethyl 2-[[5-(4-tert-butylphenyl)-4-[(2S)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C31H41N5O3S2
ethyl 2-[[5-(4-tert-butylphenyl)-4-[(2S)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 5-methyl-4-[(2S)-2-methylbutyl]-2-[[2-(1,3,4-thiadiazol-2-ylsulfanyl)acetyl]amino]thiophene-3-carboxylate —— C17H23N3O3S3
ethyl 5-methyl-4-[(2S)-2-methylbutyl]-2-[[2-(1,3,4-thiadiazol-2-ylsulfanyl)acetyl]amino]thiophene-3-carboxylate
—— Ethyl 4-[2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]piperazine-1-carboxylate —— C16H20N4O5S
Ethyl 4-[2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]piperazine-1-carboxylate
—— ethyl (6S)-2-[[2-[[3-[(2S)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H35N3O4S3
ethyl (6S)-2-[[2-[[3-[(2S)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 1-[2-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-4-carboxylate —— C28H37FN4O4S
ethyl 1-[2-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-4-carboxylate
—— Ethyl 3-[2-(2,3-dihydroindol-1-yl)-2-oxoethoxy]benzoate —— C19H19NO4
Ethyl 3-[2-(2,3-dihydroindol-1-yl)-2-oxoethoxy]benzoate
—— ethyl 1-[2-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-4-carboxylate —— C28H37FN4O4S
ethyl 1-[2-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]piperidine-4-carboxylate
—— Ethyl 2-amino-5-(methylcarbamoyl)-4-(1,3,4-thiadiazol-2-ylsulfanylmethyl)thiophene-3-carboxylate —— C12H14N4O3S3
Ethyl 2-amino-5-(methylcarbamoyl)-4-(1,3,4-thiadiazol-2-ylsulfanylmethyl)thiophene-3-carboxylate
—— ethyl 5-[2-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C29H35FN4O4S
ethyl 5-[2-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 3-[2-(4,5-dimethyl-2-nitroanilino)-2-oxoethoxy]benzoate —— C19H20N2O6
Ethyl 3-[2-(4,5-dimethyl-2-nitroanilino)-2-oxoethoxy]benzoate
—— ethyl 2-[[5-(4-tert-butylphenyl)-4-[(2R)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C31H41N5O3S2
ethyl 2-[[5-(4-tert-butylphenyl)-4-[(2R)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— Ethyl 3-[2-[4-(difluoromethylsulfanyl)anilino]-2-oxoethoxy]benzoate —— C18H17F2NO4S
Ethyl 3-[2-[4-(difluoromethylsulfanyl)anilino]-2-oxoethoxy]benzoate
—— ethyl 5-[2-[[5-(4-tert-butylphenyl)-4-[(2S)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C31H44N4O3S
ethyl 5-[2-[[5-(4-tert-butylphenyl)-4-[(2S)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (3R)-1-[2-(2-fluorophenyl)-3,5-dioxo-4-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-triazine-6-carbonyl]piperidine-3-carboxylate —— C26H24F4N4O5
ethyl (3R)-1-[2-(2-fluorophenyl)-3,5-dioxo-4-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-triazine-6-carbonyl]piperidine-3-carboxylate
—— ethyl 3-[(2S)-1-(3-acetylanilino)-1-oxopropan-2-yl]oxybenzoate —— C20H21NO5
ethyl 3-[(2S)-1-(3-acetylanilino)-1-oxopropan-2-yl]oxybenzoate
—— Ethyl 3-[2-oxo-2-[[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]amino]ethoxy]benzoate —— C19H17F3N2O5
Ethyl 3-[2-oxo-2-[[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]amino]ethoxy]benzoate
—— Ethyl 3-[2-[3-(dimethylsulfamoyl)anilino]-2-oxoethoxy]benzoate —— C19H22N2O6S
Ethyl 3-[2-[3-(dimethylsulfamoyl)anilino]-2-oxoethoxy]benzoate
—— Ethyl 3-[2-(2,6-dichloro-3-methylanilino)-2-oxoethoxy]benzoate —— C18H17Cl2NO4
Ethyl 3-[2-(2,6-dichloro-3-methylanilino)-2-oxoethoxy]benzoate
—— Ethyl 3-[2-[(2-chlorophenyl)methylamino]-2-oxoethoxy]benzoate —— C18H18ClNO4
Ethyl 3-[2-[(2-chlorophenyl)methylamino]-2-oxoethoxy]benzoate
—— Ethyl 3-[2-oxo-2-[4-(trifluoromethoxy)anilino]ethoxy]benzoate —— C18H16F3NO5
Ethyl 3-[2-oxo-2-[4-(trifluoromethoxy)anilino]ethoxy]benzoate
—— ethyl 5-[2-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C29H35FN4O4S
ethyl 5-[2-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 3-[2-[(2-fluorophenyl)carbamoylamino]-2-oxoethoxy]benzoate —— C18H17FN2O5
Ethyl 3-[2-[(2-fluorophenyl)carbamoylamino]-2-oxoethoxy]benzoate
—— Ethyl 3-[2-(2-methyl-6-propan-2-ylanilino)-2-oxoethoxy]benzoate —— C21H25NO4
Ethyl 3-[2-(2-methyl-6-propan-2-ylanilino)-2-oxoethoxy]benzoate
—— ethyl 4-[[(6R)-6-[(4-butoxyphenyl)carbamoyl]-3-[(4-chlorophenyl)methyl]-4-oxo-1,3-thiazinan-2-ylidene]amino]benzoate —— C31H32ClN3O5S
ethyl 4-[[(6R)-6-[(4-butoxyphenyl)carbamoyl]-3-[(4-chlorophenyl)methyl]-4-oxo-1,3-thiazinan-2-ylidene]amino]benzoate
—— ethyl 5-[2-[[5-(4-tert-butylphenyl)-4-[(2R)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C31H44N4O3S
ethyl 5-[2-[[5-(4-tert-butylphenyl)-4-[(2R)-2-methylheptyl]-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (6R)-2-[[2-[[3-[(2S)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H35N3O4S3
ethyl (6R)-2-[[2-[[3-[(2S)-butan-2-yl]-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 3-[2-(4-fluoroanilino)-2-oxoethoxy]benzoate —— C17H16FNO4
Ethyl 3-[2-(4-fluoroanilino)-2-oxoethoxy]benzoate
—— ethyl (4S)-4-ethyl-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C13H18N4O3S2
ethyl (4S)-4-ethyl-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[[(1R,5R)-8-[4-(1,3-thiazol-2-ylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C27H28N2O4S2
ethyl 4-[[(1R,5R)-8-[4-(1,3-thiazol-2-ylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— Ethyl 3-[2-(3-acetylanilino)-2-oxoethoxy]benzoate —— C19H19NO5
Ethyl 3-[2-(3-acetylanilino)-2-oxoethoxy]benzoate
—— ethyl 3-[(2R)-1-(2,5-dichloroanilino)-1-oxopropan-2-yl]oxybenzoate —— C18H17Cl2NO4
ethyl 3-[(2R)-1-(2,5-dichloroanilino)-1-oxopropan-2-yl]oxybenzoate
—— ethyl 4-[[(1S,5S)-8-[4-(1,3-thiazol-2-ylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate —— C27H28N2O4S2
ethyl 4-[[(1S,5S)-8-[4-(1,3-thiazol-2-ylsulfanylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzoate
—— ethyl 3-[(2S)-1-oxo-1-(4-sulfamoylanilino)propan-2-yl]oxybenzoate —— C18H20N2O6S
ethyl 3-[(2S)-1-oxo-1-(4-sulfamoylanilino)propan-2-yl]oxybenzoate