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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (3R)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3R)-1-[2-[6-[1-(2,5-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— ethyl 4-[(Z)-[(2R)-2-(2-fluorophenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H27FN4O5
ethyl 4-[(Z)-[(2R)-2-(2-fluorophenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 2-[(4Z,5S)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H26N2O6S
ethyl 2-[(4Z,5S)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3S)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3S)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— (E)-N-[2-(3-fluorophenyl)ethyl]-3-(4-methoxyphenyl)prop-2-enamide —— C18H18FNO2
(E)-N-[2-(3-fluorophenyl)ethyl]-3-(4-methoxyphenyl)prop-2-enamide
—— ethyl (3S)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3S)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— ethyl 4-[(Z)-[(2S)-2-(2-fluorophenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H27FN4O5
ethyl 4-[(Z)-[(2S)-2-(2-fluorophenyl)-1-(3-imidazol-1-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 2-[(2R,3Z)-2-(2,5-dimethoxyphenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O8S
ethyl 2-[(2R,3Z)-2-(2,5-dimethoxyphenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(4Z,5R)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H26N2O6S
ethyl 2-[(4Z,5R)-4-[hydroxy-(4-propoxyphenyl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (3R)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3R)-1-[2-[6-[1-(2,4-dimethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— (E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-[2-(3-fluorophenyl)ethyl]prop-2-enamide —— C20H23FN2O4S
(E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-[2-(3-fluorophenyl)ethyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-(3-fluorophenyl)ethyl]prop-2-enamide —— C18H16FNO3
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-(3-fluorophenyl)ethyl]prop-2-enamide
—— (E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(1R)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide —— C18H18ClNO3S
(E)-3-(7-chloro-1,3-benzodioxol-5-yl)-N-[(1R)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide
—— (E)-3-(2-ethyl-1-benzofuran-3-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide —— C24H24N4O2
(E)-3-(2-ethyl-1-benzofuran-3-yl)-N-methyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide
—— (E)-N-[(1R)-1-(1,3-benzothiazol-2-yl)ethyl]-3-(3,5-dimethoxyphenyl)-N-methylprop-2-enamide —— C21H22N2O3S
(E)-N-[(1R)-1-(1,3-benzothiazol-2-yl)ethyl]-3-(3,5-dimethoxyphenyl)-N-methylprop-2-enamide
—— ethyl 2-[(2S,3Z)-2-(2,5-dimethoxyphenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O8S
ethyl 2-[(2S,3Z)-2-(2,5-dimethoxyphenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— (E)-3-(5-bromothiophen-2-yl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide —— C15H15BrN2O2S
(E)-3-(5-bromothiophen-2-yl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide
—— (E)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-(5-methylthiophen-2-yl)prop-2-enamide —— C16H18N2O2S
(E)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-(5-methylthiophen-2-yl)prop-2-enamide
—— ethyl (6R)-2-[[(2R)-2-(4-methoxy-3-nitrobenzoyl)oxy-2-phenylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28N2O8S
ethyl (6R)-2-[[(2R)-2-(4-methoxy-3-nitrobenzoyl)oxy-2-phenylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 4-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylamino]-4-oxobutanoate —— C14H20N2O4
ethyl 4-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylamino]-4-oxobutanoate
—— Ethyl 4-[4-[2-(4-fluoroanilino)-2-oxoethyl]piperazin-4-ium-1-yl]-4-oxobutanoate —— C18H25FN3O4+
Ethyl 4-[4-[2-(4-fluoroanilino)-2-oxoethyl]piperazin-4-ium-1-yl]-4-oxobutanoate
—— (E)-N-(2-benzylsulfanylethyl)-3-(5-nitrofuran-2-yl)prop-2-enamide —— C16H16N2O4S
(E)-N-(2-benzylsulfanylethyl)-3-(5-nitrofuran-2-yl)prop-2-enamide
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-N-[(2-methoxy-5-methylphenyl)methyl]-N-methylprop-2-enamide —— C24H26ClN3O2
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-N-[(2-methoxy-5-methylphenyl)methyl]-N-methylprop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide —— C19H21NO3S
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide —— C19H22N2O4
(E)-3-(3,4-dimethoxyphenyl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide
—— ethyl 4-[5-cyano-1,4-dimethyl-3-[(E)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-6-oxopyridin-2-yl]piperazine-1-carboxylate —— C27H29N5O4S2
ethyl 4-[5-cyano-1,4-dimethyl-3-[(E)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-6-oxopyridin-2-yl]piperazine-1-carboxylate
—— ethyl 3-[[2-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-5-phenylthiophene-2-carboxylate —— C24H27NO5S
ethyl 3-[[2-[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-5-phenylthiophene-2-carboxylate
—— ethyl (6S)-2-[[(2S)-2-(4-methoxy-3-nitrobenzoyl)oxy-2-phenylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28N2O8S
ethyl (6S)-2-[[(2S)-2-(4-methoxy-3-nitrobenzoyl)oxy-2-phenylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (4S)-6-[[2-[(5-bromothiophen-2-yl)sulfonylamino]benzoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H20BrN3O7S2
ethyl (4S)-6-[[2-[(5-bromothiophen-2-yl)sulfonylamino]benzoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 5-phenyl-2-[[(2R)-2-(4-pyrrolidin-1-ylsulfonylbenzoyl)oxypropanoyl]amino]thiophene-3-carboxylate —— C27H28N2O7S2
ethyl 5-phenyl-2-[[(2R)-2-(4-pyrrolidin-1-ylsulfonylbenzoyl)oxypropanoyl]amino]thiophene-3-carboxylate
—— (E)-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-3-phenylsulfanylprop-2-enamide —— C19H18N2O2S
(E)-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-3-phenylsulfanylprop-2-enamide
—— ethyl-[(4-ethyl-5-sulfanylidene-1,2,4-triazol-1-yl)methyl]-[(4-oxo-3H-quinazolin-2-yl)methyl]azanium —— C16H21N6OS+
ethyl-[(4-ethyl-5-sulfanylidene-1,2,4-triazol-1-yl)methyl]-[(4-oxo-3H-quinazolin-2-yl)methyl]azanium
—— ethyl 2-[3-[[ethyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]methyl]-2-sulfanylidene-1,3-thiazol-4-yl]acetate —— C19H22N4O3S2
ethyl 2-[3-[[ethyl-[(4-oxo-3H-quinazolin-2-yl)methyl]amino]methyl]-2-sulfanylidene-1,3-thiazol-4-yl]acetate
—— (E)-N-[(1R)-1-(1-benzofuran-2-yl)ethyl]-3-(3,5-dimethoxyphenyl)prop-2-enamide —— C21H21NO4
(E)-N-[(1R)-1-(1-benzofuran-2-yl)ethyl]-3-(3,5-dimethoxyphenyl)prop-2-enamide
—— (E)-3-(4-bromophenyl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide —— C17H17BrN2O2
(E)-3-(4-bromophenyl)-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]prop-2-enamide
—— (E)-N-[(1S)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methyl-3-(5-nitrofuran-2-yl)prop-2-enamide —— C17H15N3O4S
(E)-N-[(1S)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methyl-3-(5-nitrofuran-2-yl)prop-2-enamide
—— ethyl 3-[[2-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-5-phenylthiophene-2-carboxylate —— C24H27NO5S
ethyl 3-[[2-[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]amino]-5-phenylthiophene-2-carboxylate
—— ethyl 4-[[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]carbamoyl]piperidine-1-carboxylate —— C19H30N2O3
ethyl 4-[[(1S,2R,6S,7R,8S)-8-tricyclo[5.2.1.02,6]decanyl]carbamoyl]piperidine-1-carboxylate
—— ethyl (3R)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C29H33N5O4S
ethyl (3R)-1-[2-[6-[1-(2-ethylphenyl)-5-methylpyrazol-3-yl]-7-methyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— (E)-N-[(1S)-1-(1,3-benzothiazol-2-yl)ethyl]-3-(3,5-dimethoxyphenyl)-N-methylprop-2-enamide —— C21H22N2O3S
(E)-N-[(1S)-1-(1,3-benzothiazol-2-yl)ethyl]-3-(3,5-dimethoxyphenyl)-N-methylprop-2-enamide
—— ethyl (4R)-6-[[2-[(5-bromothiophen-2-yl)sulfonylamino]benzoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H20BrN3O7S2
ethyl (4R)-6-[[2-[(5-bromothiophen-2-yl)sulfonylamino]benzoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-3-phenylsulfanylprop-2-enamide —— C21H23NO3S
(E)-N-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-3-phenylsulfanylprop-2-enamide
—— (E)-3-(2-ethoxyphenyl)-N-[(1R)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide —— C19H23NO2S
(E)-3-(2-ethoxyphenyl)-N-[(1R)-2-methyl-1-thiophen-2-ylpropyl]prop-2-enamide
—— ethyl (6R)-6-methyl-2-[[(2S)-2-[3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]oxypropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C32H42N2O7S2
ethyl (6R)-6-methyl-2-[[(2S)-2-[3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]sulfonyl]benzoyl]oxypropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(1S)-1-(1-benzofuran-2-yl)ethyl]-3-phenylsulfanylprop-2-enamide —— C19H17NO2S
(E)-N-[(1S)-1-(1-benzofuran-2-yl)ethyl]-3-phenylsulfanylprop-2-enamide
—— Ethyl 4-[4-(2,5-dimethoxyphenyl)sulfonylpiperazin-1-yl]-4-oxobutanoate —— C18H26N2O7S
Ethyl 4-[4-(2,5-dimethoxyphenyl)sulfonylpiperazin-1-yl]-4-oxobutanoate
—— (E)-N-(1,3-benzothiazol-2-ylmethyl)-3-(1-benzyltriazol-4-yl)-N-methylprop-2-enamide —— C21H19N5OS
(E)-N-(1,3-benzothiazol-2-ylmethyl)-3-(1-benzyltriazol-4-yl)-N-methylprop-2-enamide
—— ethyl (3aS)-4-butyl-2-methyl-3,3a-dihydroimidazo[1,2-a]benzimidazole-1-carboxylate —— C17H23N3O2
ethyl (3aS)-4-butyl-2-methyl-3,3a-dihydroimidazo[1,2-a]benzimidazole-1-carboxylate
—— (E)-N-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C24H25N3O3
(E)-N-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl 5-phenyl-2-[[(2S)-2-(4-pyrrolidin-1-ylsulfonylbenzoyl)oxypropanoyl]amino]thiophene-3-carboxylate —— C27H28N2O7S2
ethyl 5-phenyl-2-[[(2S)-2-(4-pyrrolidin-1-ylsulfonylbenzoyl)oxypropanoyl]amino]thiophene-3-carboxylate