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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 2-[[2-[(Z)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate —— C23H26ClN3O7S2
ethyl 2-[[2-[(Z)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate
—— ethyl (4S)-1-[[3-(benzhydrylcarbamoyl)phenyl]methyl]-6-methyl-4-(4-methylphenyl)-2-oxo-3,4-dihydropyridine-5-carboxylate —— C37H36N2O4
ethyl (4S)-1-[[3-(benzhydrylcarbamoyl)phenyl]methyl]-6-methyl-4-(4-methylphenyl)-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (E)-3-[[4-[4-(2-acetamidoethyl)phenyl]-1,3-thiazol-2-yl]amino]-2-cyanoprop-2-enoate —— C19H20N4O3S
ethyl (E)-3-[[4-[4-(2-acetamidoethyl)phenyl]-1,3-thiazol-2-yl]amino]-2-cyanoprop-2-enoate
—— ethyl (E)-2-cyano-3-[(4-pyridin-3-yl-1,3-thiazol-2-yl)amino]prop-2-enoate —— C14H12N4O2S
ethyl (E)-2-cyano-3-[(4-pyridin-3-yl-1,3-thiazol-2-yl)amino]prop-2-enoate
—— ethyl (1R,9S,13Z,16R)-13-(furan-3-ylmethylidene)-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C21H18N2O5S
ethyl (1R,9S,13Z,16R)-13-(furan-3-ylmethylidene)-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— ethyl (4R)-1-[[5-(benzhydrylcarbamoyl)furan-2-yl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate —— C34H32N2O5
ethyl (4R)-1-[[5-(benzhydrylcarbamoyl)furan-2-yl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate
—— ethyl (4S)-4-(3,4-dichlorophenyl)-1-[[4-[(2-fluorophenyl)carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C29H25Cl2FN2O4
ethyl (4S)-4-(3,4-dichlorophenyl)-1-[[4-[(2-fluorophenyl)carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (4S)-1-[[3-[benzyl(2-phenylethyl)carbamoyl]phenyl]methyl]-4-(2-chlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C38H37ClN2O4
ethyl (4S)-1-[[3-[benzyl(2-phenylethyl)carbamoyl]phenyl]methyl]-4-(2-chlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— (E)-N-methyl-3-(3-nitrophenyl)-N-[(1S)-1-(3-nitrophenyl)ethyl]prop-2-enamide —— C18H17N3O5
(E)-N-methyl-3-(3-nitrophenyl)-N-[(1S)-1-(3-nitrophenyl)ethyl]prop-2-enamide
—— ethyl (4R)-1-[[3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate —— C34H37N3O5
ethyl (4R)-1-[[3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate
—— ethyl (4S)-4-(4-chlorophenyl)-1-[[4-[[(1R)-1,2-diphenylethyl]carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C37H35ClN2O4
ethyl (4S)-4-(4-chlorophenyl)-1-[[4-[[(1R)-1,2-diphenylethyl]carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (4S)-1-[[3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate —— C34H37N3O5
ethyl (4S)-1-[[3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]prop-2-enamide —— C19H20N2O4
(E)-3-(4-methoxyphenyl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]prop-2-enamide
—— ethyl (4R)-1-[[4-[2-(2,4-dichlorophenyl)ethylcarbamoyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate —— C31H30Cl2N2O4
ethyl (4R)-1-[[4-[2-(2,4-dichlorophenyl)ethylcarbamoyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-1-[[4-[[(1R)-1,2-diphenylethyl]carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C37H35ClN2O4
ethyl (4R)-4-(4-chlorophenyl)-1-[[4-[[(1R)-1,2-diphenylethyl]carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— (E)-1-[4-methoxy-3-(methoxymethyl)phenyl]-3-(4-morpholin-4-ylphenyl)prop-2-en-1-one —— C22H25NO4
(E)-1-[4-methoxy-3-(methoxymethyl)phenyl]-3-(4-morpholin-4-ylphenyl)prop-2-en-1-one
—— (E)-N-benzyl-4-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide —— C31H31N5O3S
(E)-N-benzyl-4-[[5-(4-tert-butylphenyl)-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide
—— ethyl (4R)-4-(4-chlorophenyl)-1-[[4-[[(1S)-1,2-diphenylethyl]carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C37H35ClN2O4
ethyl (4R)-4-(4-chlorophenyl)-1-[[4-[[(1S)-1,2-diphenylethyl]carbamoyl]phenyl]methyl]-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (4R)-4-(3,4-dichlorophenyl)-6-methyl-1-[[3-[(4-methylphenyl)carbamoyl]phenyl]methyl]-2-oxo-3,4-dihydropyridine-5-carboxylate —— C30H28Cl2N2O4
ethyl (4R)-4-(3,4-dichlorophenyl)-6-methyl-1-[[3-[(4-methylphenyl)carbamoyl]phenyl]methyl]-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (4S)-1-[[4-[benzyl(2-phenylethyl)carbamoyl]phenyl]methyl]-4-(2-fluorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C38H37FN2O4
ethyl (4S)-1-[[4-[benzyl(2-phenylethyl)carbamoyl]phenyl]methyl]-4-(2-fluorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (4S)-1-[[4-[2-(2,4-dichlorophenyl)ethylcarbamoyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate —— C31H30Cl2N2O4
ethyl (4S)-1-[[4-[2-(2,4-dichlorophenyl)ethylcarbamoyl]phenyl]methyl]-6-methyl-2-oxo-4-phenyl-3,4-dihydropyridine-5-carboxylate
—— (E)-3-(2-chlorophenyl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]prop-2-enamide —— C18H17ClN2O3
(E)-3-(2-chlorophenyl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]prop-2-enamide
—— (E)-N-benzyl-4-[[4-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide —— C27H22ClN5O3S
(E)-N-benzyl-4-[[4-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-2-cyano-3-hydroxybut-2-enamide
—— ethyl (4S)-4-(3,4-dichlorophenyl)-6-methyl-1-[[3-[(4-methylphenyl)carbamoyl]phenyl]methyl]-2-oxo-3,4-dihydropyridine-5-carboxylate —— C30H28Cl2N2O4
ethyl (4S)-4-(3,4-dichlorophenyl)-6-methyl-1-[[3-[(4-methylphenyl)carbamoyl]phenyl]methyl]-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (4R)-1-[[4-[benzyl(2-phenylethyl)carbamoyl]phenyl]methyl]-4-(3-chlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C38H37ClN2O4
ethyl (4R)-1-[[4-[benzyl(2-phenylethyl)carbamoyl]phenyl]methyl]-4-(3-chlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (3S)-1-[4-(4-benzylpiperidin-1-yl)-2-(4-methoxyphenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate —— C32H38N4O4
ethyl (3S)-1-[4-(4-benzylpiperidin-1-yl)-2-(4-methoxyphenyl)pyrimidine-5-carbonyl]piperidine-3-carboxylate
—— (E)-N-[[2-[(dimethylamino)methyl]phenyl]methyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide —— C24H26N2O2
(E)-N-[[2-[(dimethylamino)methyl]phenyl]methyl]-3-(6-methoxynaphthalen-2-yl)prop-2-enamide
—— Ethyl 4-methyl-2-[[3-(2-oxopyrrolidin-1-yl)phenoxy]methyl]quinoline-3-carboxylate —— C24H24N2O4
Ethyl 4-methyl-2-[[3-(2-oxopyrrolidin-1-yl)phenoxy]methyl]quinoline-3-carboxylate
—— (E)-2-cyano-N-cyclopropyl-3-[4-(difluoromethoxy)-3-methoxyphenyl]prop-2-enamide —— C15H14F2N2O3
(E)-2-cyano-N-cyclopropyl-3-[4-(difluoromethoxy)-3-methoxyphenyl]prop-2-enamide
—— (E)-3-(2-bromophenyl)-N-[[2-[(dimethylamino)methyl]phenyl]methyl]prop-2-enamide —— C19H21BrN2O
(E)-3-(2-bromophenyl)-N-[[2-[(dimethylamino)methyl]phenyl]methyl]prop-2-enamide
—— (E)-3-(4-morpholin-4-ylphenyl)-2-(4-phenyl-1,3-thiazol-2-yl)prop-2-enenitrile —— C22H19N3OS
(E)-3-(4-morpholin-4-ylphenyl)-2-(4-phenyl-1,3-thiazol-2-yl)prop-2-enenitrile
—— ethyl 2-[[2-[(Z)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate —— C23H26ClN3O7S2
ethyl 2-[[2-[(Z)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate
—— ethyl (6R)-4-[[(3R)-4-(benzenesulfonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H31F3N4O5S
ethyl (6R)-4-[[(3R)-4-(benzenesulfonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[2-[(3S)-3-(2,4-dimethoxyphenyl)-5-(3,4-dimethoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C29H37N3O7
ethyl (3S)-1-[2-[(3S)-3-(2,4-dimethoxyphenyl)-5-(3,4-dimethoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[2-(4-oxo-3,5-diphenylthieno[2,3-d]pyrimidin-2-yl)sulfanylacetyl]piperidine-3-carboxylate —— C28H27N3O4S2
ethyl (3S)-1-[2-(4-oxo-3,5-diphenylthieno[2,3-d]pyrimidin-2-yl)sulfanylacetyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H36F3N5O3S
ethyl (3R)-1-[3-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-(4-oxo-3,5-diphenylthieno[2,3-d]pyrimidin-2-yl)sulfanylacetyl]piperidine-3-carboxylate —— C28H27N3O4S2
ethyl (3R)-1-[2-(4-oxo-3,5-diphenylthieno[2,3-d]pyrimidin-2-yl)sulfanylacetyl]piperidine-3-carboxylate
—— (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-(5-fluoro-2-methylphenyl)prop-2-enamide —— C19H17ClFNO3
(E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-(5-fluoro-2-methylphenyl)prop-2-enamide
—— ethyl (6S)-4-methyl-6-(3-nitrophenyl)-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H23N3O5S
ethyl (6S)-4-methyl-6-(3-nitrophenyl)-3-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[[(3R)-4-(benzenesulfonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C27H31F3N4O5S
ethyl (6S)-4-[[(3R)-4-(benzenesulfonyl)-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxo-6-[2-(trifluoromethyl)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 4,5-dimethyl-2-[[2-[3-(2-oxopyrrolidin-1-yl)phenoxy]acetyl]amino]thiophene-3-carboxylate —— C21H24N2O5S
Ethyl 4,5-dimethyl-2-[[2-[3-(2-oxopyrrolidin-1-yl)phenoxy]acetyl]amino]thiophene-3-carboxylate
—— ethyl (4S)-6-[[(3-chlorophenyl)methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24ClN3O3
ethyl (4S)-6-[[(3-chlorophenyl)methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2R)-2-[[(2R)-butan-2-yl]-[2-[(5-methylfuran-2-yl)methyl-(2-phenylethyl)amino]-2-oxoethyl]amino]propanoate —— C25H36N2O4
ethyl (2R)-2-[[(2R)-butan-2-yl]-[2-[(5-methylfuran-2-yl)methyl-(2-phenylethyl)amino]-2-oxoethyl]amino]propanoate
—— ethyl 4-[[butyl-[2-[(4S)-4-(4-chlorophenyl)-4H-pyrrolo[1,2-a]quinoxalin-5-yl]-2-oxoethyl]carbamoyl]amino]benzoate —— C33H33ClN4O4
ethyl 4-[[butyl-[2-[(4S)-4-(4-chlorophenyl)-4H-pyrrolo[1,2-a]quinoxalin-5-yl]-2-oxoethyl]carbamoyl]amino]benzoate
—— (E)-1-(4-Fluoro-phenyl)-3-(3-hydroxy-4-methoxy-phenyl)-propenone —— C16H13FO3
(E)-1-(4-Fluoro-phenyl)-3-(3-hydroxy-4-methoxy-phenyl)-propenone
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-(5-prop-2-enylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide —— C13H10ClN5OS3
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-(5-prop-2-enylsulfanyl-1,3,4-thiadiazol-2-yl)prop-2-enamide
—— Ethyl 4-[4-(4-fluorophenyl)piperazin-1-yl]sulfonylbenzoate —— C19H21FN2O4S
Ethyl 4-[4-(4-fluorophenyl)piperazin-1-yl]sulfonylbenzoate
—— (E)-2-cyano-3-(4-hydroxy-3,5-dimethylphenyl)-N-propan-2-ylprop-2-enamide —— C15H18N2O2
(E)-2-cyano-3-(4-hydroxy-3,5-dimethylphenyl)-N-propan-2-ylprop-2-enamide
—— (E)-N-(2-methyl-5-piperidin-1-ylsulfonylphenyl)-2-phenylethenesulfonamide —— C20H24N2O4S2
(E)-N-(2-methyl-5-piperidin-1-ylsulfonylphenyl)-2-phenylethenesulfonamide
—— Ethyl 4-[[2-(4-pyrimidin-2-ylpiperazin-1-yl)acetyl]amino]butanoate —— C16H25N5O3
Ethyl 4-[[2-(4-pyrimidin-2-ylpiperazin-1-yl)acetyl]amino]butanoate