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—— ethyl (4S)-6-[(2-chloro-4,6-dimethylpyridine-3-carbonyl)oxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22ClN3O5
ethyl (4S)-6-[(2-chloro-4,6-dimethylpyridine-3-carbonyl)oxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-(2-methoxy-5-sulfamoylphenyl)-2-methylpent-2-enamide —— C13H18N2O4S
(E)-N-(2-methoxy-5-sulfamoylphenyl)-2-methylpent-2-enamide
—— (E,2R)-2-cyano-5-naphthalen-1-yl-3-oxo-N-[[(2R)-oxolan-2-yl]methyl]pent-4-enamide —— C21H20N2O3
(E,2R)-2-cyano-5-naphthalen-1-yl-3-oxo-N-[[(2R)-oxolan-2-yl]methyl]pent-4-enamide
—— ethyl (2Z,5R)-2-[[4-bromo-5-(dimethylamino)furan-2-yl]methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H21BrClN3O4S
ethyl (2Z,5R)-2-[[4-bromo-5-(dimethylamino)furan-2-yl]methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-methyl-N-(4-methyl-3-sulfamoylphenyl)pent-2-enamide —— C13H18N2O3S
(E)-2-methyl-N-(4-methyl-3-sulfamoylphenyl)pent-2-enamide
—— ethyl (2Z,5R)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H28BrN3O7S
ethyl (2Z,5R)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26BrN3O6S
ethyl (2Z,5S)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-cyano-N-[4-[[(E)-2-cyano-3-(5-methylfuran-2-yl)prop-2-enoyl]amino]phenyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C24H18N4O4
(E)-2-cyano-N-[4-[[(E)-2-cyano-3-(5-methylfuran-2-yl)prop-2-enoyl]amino]phenyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— ethyl (2S)-2-[7-[(1R,2R)-2-[(Z,3R)-3-hydroxyoct-1-enyl]-5-oxocyclopentyl]heptanoylamino]-3-(4-hydroxyphenyl)propanoate —— C31H47NO6
ethyl (2S)-2-[7-[(1R,2R)-2-[(Z,3R)-3-hydroxyoct-1-enyl]-5-oxocyclopentyl]heptanoylamino]-3-(4-hydroxyphenyl)propanoate
—— ethyl (2Z,5R)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H23BrClN3O5S
ethyl (2Z,5R)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(4-fluorophenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H25FN4O6S
ethyl (2E,5R)-5-(4-fluorophenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26BrN3O6S
ethyl (2Z,5S)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 3-[[4-(4-fluorophenyl)-4-oxobutanoyl]oxymethyl]-1-benzofuran-2-carboxylate —— C22H19FO6
Ethyl 3-[[4-(4-fluorophenyl)-4-oxobutanoyl]oxymethyl]-1-benzofuran-2-carboxylate
—— ethyl (2Z,5R)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26BrN3O6S
ethyl (2Z,5R)-2-[(4-bromo-5-morpholin-4-ylfuran-2-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-bromo-5-(dimethylamino)furan-2-yl]methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H21BrClN3O4S
ethyl (2Z,5S)-2-[[4-bromo-5-(dimethylamino)furan-2-yl]methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 3-[(2-thiophen-3-ylacetyl)oxymethyl]-1-benzofuran-2-carboxylate —— C18H16O5S
Ethyl 3-[(2-thiophen-3-ylacetyl)oxymethyl]-1-benzofuran-2-carboxylate
—— ethyl 4-[5-[(Z)-3-(4-chloro-3-nitroanilino)-2-cyano-3-oxoprop-1-enyl]furan-2-yl]benzoate —— C23H16ClN3O6
ethyl 4-[5-[(Z)-3-(4-chloro-3-nitroanilino)-2-cyano-3-oxoprop-1-enyl]furan-2-yl]benzoate
—— ethyl (2E,5S)-5-[4-(dimethylamino)phenyl]-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N5O6S
ethyl (2E,5S)-5-[4-(dimethylamino)phenyl]-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(2-methoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28N4O7S
ethyl (2E,5R)-5-(2-methoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3-methoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28N4O7S
ethyl (2E,5S)-5-(3-methoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(E)-3-(3-bromophenyl)-2-(furan-2-carbonylamino)prop-2-enoyl]amino]acetate —— C18H17BrN2O5
ethyl 2-[[(E)-3-(3-bromophenyl)-2-(furan-2-carbonylamino)prop-2-enoyl]amino]acetate
—— ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H30N4O8S
ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H30N4O8S
ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-3-methylphenyl]prop-2-enoic acid —— C16H19NO2
(E)-3-[4-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-3-methylphenyl]prop-2-enoic acid
—— ethyl (2E,5S)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24N4O6S2
ethyl (2E,5S)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (4S)-4-ethyl-6-[(2-fluoro-4-methoxybenzoyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H21FN2O6
ethyl (4S)-4-ethyl-6-[(2-fluoro-4-methoxybenzoyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2E,5R)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H30N4O8S
ethyl (2E,5R)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[3-ethoxy-4-(2-ethoxy-2-oxoethoxy)phenyl]methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H28N2O7S2
ethyl (2E,5S)-2-[[3-ethoxy-4-(2-ethoxy-2-oxoethoxy)phenyl]methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-[4-(dimethylamino)phenyl]-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N5O6S
ethyl (2E,5R)-5-[4-(dimethylamino)phenyl]-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(E)-3-(3-bromophenyl)-2-(furan-2-carbonylamino)prop-2-enoyl]amino]benzoate —— C23H19BrN2O5
ethyl 4-[[(E)-3-(3-bromophenyl)-2-(furan-2-carbonylamino)prop-2-enoyl]amino]benzoate
—— ethyl (2E,5S)-5-(4-fluorophenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H25FN4O6S
ethyl (2E,5S)-5-(4-fluorophenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H30N4O8S
ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24N4O6S2
ethyl (2E,5R)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(3-methoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28N4O7S
ethyl (2E,5R)-5-(3-methoxyphenyl)-7-methyl-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-(1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-3-phenylprop-2-enamide —— C19H14N2O3S
(E)-N-[4-(1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-3-phenylprop-2-enamide
—— ethyl 4-[5-[(Z)-3-(2-chloro-5-nitroanilino)-2-cyano-3-oxoprop-1-enyl]furan-2-yl]benzoate —— C23H16ClN3O6
ethyl 4-[5-[(Z)-3-(2-chloro-5-nitroanilino)-2-cyano-3-oxoprop-1-enyl]furan-2-yl]benzoate
—— ethyl (2E,5S)-5-[4-(dimethylamino)phenyl]-2-[[1-[(2-fluorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H31FN4O3S
ethyl (2E,5S)-5-[4-(dimethylamino)phenyl]-2-[[1-[(2-fluorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-[4-(dimethylamino)phenyl]-2-[[1-[(2-fluorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H31FN4O3S
ethyl (2E,5R)-5-[4-(dimethylamino)phenyl]-2-[[1-[(2-fluorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 4-[[[2-(3-fluorophenoxy)acetyl]amino]sulfamoyl]benzoate —— C17H17FN2O6S
Ethyl 4-[[[2-(3-fluorophenoxy)acetyl]amino]sulfamoyl]benzoate
—— (E)-N-[2-(2,3-dimethylanilino)-2-oxoethyl]-3-(4-fluorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C24H27FN2O3
(E)-N-[2-(2,3-dimethylanilino)-2-oxoethyl]-3-(4-fluorophenyl)-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-phenyl-1-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]prop-2-en-1-one —— C19H18F3N3O
(E)-3-phenyl-1-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]prop-2-en-1-one
—— Ethyl 2-[[2-[2-(thiophen-2-ylmethylsulfanyl)acetyl]oxyacetyl]amino]benzoate —— C18H19NO5S2
Ethyl 2-[[2-[2-(thiophen-2-ylmethylsulfanyl)acetyl]oxyacetyl]amino]benzoate
—— (E)-3-amino-4-[hydroxy(2-phenylethyl)phosphoryl]but-2-enoic acid —— C12H16NO4P
(E)-3-amino-4-[hydroxy(2-phenylethyl)phosphoryl]but-2-enoic acid
—— (E)-3-(3-chlorophenyl)-N-[2-(4-fluoroanilino)-2-oxoethyl]-N-methylprop-2-enamide —— C18H16ClFN2O2
(E)-3-(3-chlorophenyl)-N-[2-(4-fluoroanilino)-2-oxoethyl]-N-methylprop-2-enamide
—— (E,2R)-5-(3-fluorophenyl)-2-(2-methyl-1H-indole-3-carbonyl)-3-oxopent-4-enenitrile —— C21H15FN2O2
(E,2R)-5-(3-fluorophenyl)-2-(2-methyl-1H-indole-3-carbonyl)-3-oxopent-4-enenitrile
—— ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-2-[(3-methoxy-4-prop-2-enoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H30N2O7S
ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-2-[(3-methoxy-4-prop-2-enoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E,2S)-5-(3-fluorophenyl)-2-(2-methyl-1H-indole-3-carbonyl)-3-oxopent-4-enenitrile —— C21H15FN2O2
(E,2S)-5-(3-fluorophenyl)-2-(2-methyl-1H-indole-3-carbonyl)-3-oxopent-4-enenitrile
—— (E)-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methyl-3-thiophen-2-ylprop-2-enamide —— C17H17ClN2O3S
(E)-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methyl-3-thiophen-2-ylprop-2-enamide
—— ethyl 2-[2-bromo-4-[(E)-[1-(3,4-dimethylphenyl)-3,5-dioxopyrazolidin-4-ylidene]methyl]-6-ethoxyphenoxy]acetate —— C24H25BrN2O6
ethyl 2-[2-bromo-4-[(E)-[1-(3,4-dimethylphenyl)-3,5-dioxopyrazolidin-4-ylidene]methyl]-6-ethoxyphenoxy]acetate
—— ethyl 2-[5-bromo-4-[(E)-[1-(3-chlorophenyl)-3,5-dioxopyrazolidin-4-ylidene]methyl]-2-ethoxyphenoxy]acetate —— C22H20BrClN2O6
ethyl 2-[5-bromo-4-[(E)-[1-(3-chlorophenyl)-3,5-dioxopyrazolidin-4-ylidene]methyl]-2-ethoxyphenoxy]acetate