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—— ethyl 4-[methyl-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]benzoate —— C20H23NO4S
ethyl 4-[methyl-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]sulfamoyl]benzoate
—— (E)-3-(3,4-dichlorophenyl)-N-[3-(hydroxymethyl)phenyl]prop-2-enamide —— C16H13Cl2NO2
(E)-3-(3,4-dichlorophenyl)-N-[3-(hydroxymethyl)phenyl]prop-2-enamide
—— (E)-3-(5-bromo-2-methoxyphenyl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]prop-2-enamide —— C15H19BrN2O3
(E)-3-(5-bromo-2-methoxyphenyl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]prop-2-enamide
—— (E)-3-(5-methylthiophen-2-yl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]prop-2-enamide —— C13H18N2O2S
(E)-3-(5-methylthiophen-2-yl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]prop-2-enamide
—— (E)-N-[3-(hydroxymethyl)phenyl]-3-(2-methoxyphenyl)prop-2-enamide —— C17H17NO3
(E)-N-[3-(hydroxymethyl)phenyl]-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-N-[(2S)-3-methylbutan-2-yl]-3-(4-methylphenyl)prop-2-enamide —— C15H21NO
(E)-N-[(2S)-3-methylbutan-2-yl]-3-(4-methylphenyl)prop-2-enamide
—— (E)-2-cyano-3-(2,5-dimethyl-1-propylpyrrol-3-yl)-N-(2-methyl-3-nitrophenyl)prop-2-enamide —— C20H22N4O3
(E)-2-cyano-3-(2,5-dimethyl-1-propylpyrrol-3-yl)-N-(2-methyl-3-nitrophenyl)prop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-phenylpropyl]prop-2-enamide —— C20H21NO3
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-phenylpropyl]prop-2-enamide
—— ethyl (3R)-1-[(2S)-2-hydroxy-3-(3-nitrophenoxy)propyl]piperidine-3-carboxylate —— C17H24N2O6
ethyl (3R)-1-[(2S)-2-hydroxy-3-(3-nitrophenoxy)propyl]piperidine-3-carboxylate
—— (E)-3-(3-methoxy-4-prop-2-enoxyphenyl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]prop-2-enamide —— C18H24N2O4
(E)-3-(3-methoxy-4-prop-2-enoxyphenyl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]prop-2-enamide
—— (E)-3-[4-(azepan-1-ylsulfonyl)phenyl]-N-[3-(hydroxymethyl)phenyl]prop-2-enamide —— C22H26N2O4S
(E)-3-[4-(azepan-1-ylsulfonyl)phenyl]-N-[3-(hydroxymethyl)phenyl]prop-2-enamide
—— (E)-3-(3-chloro-4-fluorophenyl)-N-[3-(hydroxymethyl)phenyl]prop-2-enamide —— C16H13ClFNO2
(E)-3-(3-chloro-4-fluorophenyl)-N-[3-(hydroxymethyl)phenyl]prop-2-enamide
—— (E)-N-[3-(hydroxymethyl)phenyl]-3-(4-methylphenyl)prop-2-enamide —— C17H17NO2
(E)-N-[3-(hydroxymethyl)phenyl]-3-(4-methylphenyl)prop-2-enamide
—— (E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-benzyl-N-[(2S)-butan-2-yl]prop-2-enamide —— C25H26FN3O2S
(E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-benzyl-N-[(2S)-butan-2-yl]prop-2-enamide
—— (E)-3-[4-chloro-3-(trifluoromethyl)phenyl]-N-[3-(hydroxymethyl)phenyl]prop-2-enamide —— C17H13ClF3NO2
(E)-3-[4-chloro-3-(trifluoromethyl)phenyl]-N-[3-(hydroxymethyl)phenyl]prop-2-enamide
—— (E)-N-[(2S)-1-[4-[(5-bromothiophen-2-yl)methyl]piperazin-1-yl]-1-oxopropan-2-yl]-3-phenylprop-2-enamide —— C21H24BrN3O2S
(E)-N-[(2S)-1-[4-[(5-bromothiophen-2-yl)methyl]piperazin-1-yl]-1-oxopropan-2-yl]-3-phenylprop-2-enamide
—— (E)-N-[2-oxo-2-(propan-2-ylamino)ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide —— C22H23N5O2
(E)-N-[2-oxo-2-(propan-2-ylamino)ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide
—— ethyl 5-[[2-([1]benzofuro[3,2-d]pyrimidin-4-yl)hydrazinyl]methylidene]-2,4-dimethylpyrrole-3-carboxylate —— C20H19N5O3
ethyl 5-[[2-([1]benzofuro[3,2-d]pyrimidin-4-yl)hydrazinyl]methylidene]-2,4-dimethylpyrrole-3-carboxylate
—— (E)-N-[3-(hydroxymethyl)phenyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C19H21NO5
(E)-N-[3-(hydroxymethyl)phenyl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-benzyl-N-[(2S)-butan-2-yl]-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]prop-2-enamide —— C27H32N2O4
(E)-N-benzyl-N-[(2S)-butan-2-yl]-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]prop-2-enamide
—— ethyl 1-[(2R)-1-oxo-1-(4-piperidin-1-ylanilino)propan-2-yl]piperidin-1-ium-4-carboxylate —— C22H34N3O3+
ethyl 1-[(2R)-1-oxo-1-(4-piperidin-1-ylanilino)propan-2-yl]piperidin-1-ium-4-carboxylate
—— ethyl (3S)-1-[(2S)-2-hydroxy-3-(3-nitrophenoxy)propyl]piperidine-3-carboxylate —— C17H24N2O6
ethyl (3S)-1-[(2S)-2-hydroxy-3-(3-nitrophenoxy)propyl]piperidine-3-carboxylate
—— (E)-N-cyclopropyl-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(4-methoxyphenyl)methyl]prop-2-enamide —— C23H25NO5
(E)-N-cyclopropyl-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(4-methoxyphenyl)methyl]prop-2-enamide
—— (E)-N-[2-oxo-2-(propan-2-ylamino)ethyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C15H17F3N2O2
(E)-N-[2-oxo-2-(propan-2-ylamino)ethyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— ethyl 4-[(1S,2R,5S,6R,7S)-2-(cyclohexylcarbamoyl)-6-[(3,4-dichlorophenyl)carbamoyl]-7-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]piperidine-1-carboxylate —— C31H38Cl2N4O6
ethyl 4-[(1S,2R,5S,6R,7S)-2-(cyclohexylcarbamoyl)-6-[(3,4-dichlorophenyl)carbamoyl]-7-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]piperidine-1-carboxylate
—— (E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-thiophen-2-ylprop-2-en-1-one —— C18H20N2O3S2
(E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-thiophen-2-ylprop-2-en-1-one
—— (E)-N-benzyl-N-[(2R)-butan-2-yl]-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]prop-2-enamide —— C27H32N2O4
(E)-N-benzyl-N-[(2R)-butan-2-yl]-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]prop-2-enamide
—— ethyl 4-[(1R,2R,5R,6R,7S)-2-(cyclohexylcarbamoyl)-6-[(3,4-dichlorophenyl)carbamoyl]-7-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]piperidine-1-carboxylate —— C31H38Cl2N4O6
ethyl 4-[(1R,2R,5R,6R,7S)-2-(cyclohexylcarbamoyl)-6-[(3,4-dichlorophenyl)carbamoyl]-7-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]piperidine-1-carboxylate
—— ethyl 4-[(1R,2R,5S,6R,7S)-2-(cyclohexylcarbamoyl)-6-[(3,4-dichlorophenyl)carbamoyl]-7-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]piperidine-1-carboxylate —— C31H38Cl2N4O6
ethyl 4-[(1R,2R,5S,6R,7S)-2-(cyclohexylcarbamoyl)-6-[(3,4-dichlorophenyl)carbamoyl]-7-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]piperidine-1-carboxylate
—— ethyl 4-[(2R)-3-[(4-chlorophenyl)methyl-methylamino]-2-hydroxypropoxy]benzoate —— C20H24ClNO4
ethyl 4-[(2R)-3-[(4-chlorophenyl)methyl-methylamino]-2-hydroxypropoxy]benzoate
—— (E)-3-(2-bromophenyl)-N-cyclopropyl-N-[(4-methoxyphenyl)methyl]prop-2-enamide —— C20H20BrNO2
(E)-3-(2-bromophenyl)-N-cyclopropyl-N-[(4-methoxyphenyl)methyl]prop-2-enamide
—— ethyl 4-[(2R)-2-hydroxy-3-[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]propoxy]benzoate —— C21H24F3NO4
ethyl 4-[(2R)-2-hydroxy-3-[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]propoxy]benzoate
—— (E)-N-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-propylprop-2-enamide —— C26H28ClN3O4
(E)-N-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-propylprop-2-enamide
—— (E)-N-[(2R)-1-[4-[(5-bromothiophen-2-yl)methyl]piperazin-1-yl]-1-oxopropan-2-yl]-3-phenylprop-2-enamide —— C21H24BrN3O2S
(E)-N-[(2R)-1-[4-[(5-bromothiophen-2-yl)methyl]piperazin-1-yl]-1-oxopropan-2-yl]-3-phenylprop-2-enamide
—— (E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-(4-methylsulfanylphenyl)prop-2-en-1-one —— C21H24N2O3S2
(E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-(4-methylsulfanylphenyl)prop-2-en-1-one
—— ethyl 4-[(2S)-2-hydroxy-3-[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]propoxy]benzoate —— C21H24F3NO4
ethyl 4-[(2S)-2-hydroxy-3-[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]propoxy]benzoate
—— (E)-N-cyclopropyl-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[(4-methoxyphenyl)methyl]prop-2-enamide —— C25H29NO4
(E)-N-cyclopropyl-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[(4-methoxyphenyl)methyl]prop-2-enamide
—— (E)-N-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-propylprop-2-enamide —— C26H28ClN3O4
(E)-N-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-propylprop-2-enamide
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]prop-2-enamide —— C21H19F4NO5
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]prop-2-enamide
—— ethyl 4-[(3S)-2,5-dioxo-3-(4-sulfamoylanilino)pyrrolidin-1-yl]benzoate —— C19H19N3O6S
ethyl 4-[(3S)-2,5-dioxo-3-(4-sulfamoylanilino)pyrrolidin-1-yl]benzoate
—— ethyl 1-[(2S)-1-oxo-1-(4-piperidin-1-ylanilino)propan-2-yl]piperidine-4-carboxylate —— C22H33N3O3
ethyl 1-[(2S)-1-oxo-1-(4-piperidin-1-ylanilino)propan-2-yl]piperidine-4-carboxylate
—— (E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-(4-methoxyphenyl)prop-2-en-1-one —— C21H24N2O4S
(E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-(4-methoxyphenyl)prop-2-en-1-one
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-cyclopropyl-N-[(4-methoxyphenyl)methyl]prop-2-enamide —— C22H22ClNO4
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-cyclopropyl-N-[(4-methoxyphenyl)methyl]prop-2-enamide
—— (E)-N-cyclopropyl-3-(2-fluorophenyl)-N-[(4-methoxyphenyl)methyl]prop-2-enamide —— C20H20FNO2
(E)-N-cyclopropyl-3-(2-fluorophenyl)-N-[(4-methoxyphenyl)methyl]prop-2-enamide
—— (E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-(3-methylphenyl)prop-2-en-1-one —— C21H24N2O3S
(E)-1-(4-benzylsulfonylpiperazin-1-yl)-3-(3-methylphenyl)prop-2-en-1-one
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]prop-2-en-1-one —— C19H17F4NO3S
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-1-[(2S)-2-thiophen-2-ylpyrrolidin-1-yl]prop-2-en-1-one
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C28H32N4O2
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C25H30F2N2O4
(E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[[4-(dimethylamino)phenyl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl 4-[(1S,9R,13S)-13-(dimethylcarbamoyl)-6-methoxy-9-methyl-11-sulfanylidene-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-10-yl]benzoate —— C24H27N3O5S
ethyl 4-[(1S,9R,13S)-13-(dimethylcarbamoyl)-6-methoxy-9-methyl-11-sulfanylidene-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-10-yl]benzoate
—— ethyl (4R)-6-[[(5-bromothiophen-2-yl)methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H22BrN3O3S
ethyl (4R)-6-[[(5-bromothiophen-2-yl)methyl-methylamino]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate