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—— (E,1S,4R)-1,7,7-trimethyl-N-[(E)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]bicyclo[2.2.1]heptan-2-imine —— C18H21N3O4
(E,1S,4R)-1,7,7-trimethyl-N-[(E)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]bicyclo[2.2.1]heptan-2-imine
—— (E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H29FN4O
(E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— (E,1S,4R)-1,7,7-trimethyl-N-[(E)-[4-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-3-nitrophenyl]methylideneamino]bicyclo[2.2.1]heptan-2-imine —— C20H24N6O2S
(E,1S,4R)-1,7,7-trimethyl-N-[(E)-[4-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-3-nitrophenyl]methylideneamino]bicyclo[2.2.1]heptan-2-imine
—— (E)-N-[2-[(5E)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-3-quinolin-8-ylprop-2-enamide —— C24H18FN3O3S
(E)-N-[2-[(5E)-5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-3-quinolin-8-ylprop-2-enamide
—— (E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine —— C27H29FN4O
(E,1R,4S)-N-[(E)-[5-(4-fluorophenoxy)-3-methyl-1-phenylpyrazol-4-yl]methylideneamino]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-imine
—— (E,1S,4R)-1,7,7-trimethyl-N-[(E)-(4-nitrophenyl)methylideneamino]bicyclo[2.2.1]heptan-2-imine —— C17H21N3O2
(E,1S,4R)-1,7,7-trimethyl-N-[(E)-(4-nitrophenyl)methylideneamino]bicyclo[2.2.1]heptan-2-imine
—— ethyl N-[2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetyl]carbamate —— C17H21N3O3S
ethyl N-[2-[1-(4-propan-2-ylphenyl)imidazol-2-yl]sulfanylacetyl]carbamate
—— (E)-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C24H29N3O4
(E)-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]prop-2-enamide —— C21H18F7NO4
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]prop-2-enamide —— C22H22F5NO4
(E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[[4-(2,2,2-trifluoroethoxymethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(3-chloro-4-methylphenyl)-N-[3-(dimethylsulfamoyl)phenyl]prop-2-enamide —— C18H19ClN2O3S
(E)-3-(3-chloro-4-methylphenyl)-N-[3-(dimethylsulfamoyl)phenyl]prop-2-enamide
—— (E)-4-[[(3R)-1-(4-bromophenyl)-2,5-dioxopyrrolidin-3-yl]-[2-(3,4-dimethoxyphenyl)ethyl]amino]-4-oxobut-2-enoate —— C24H22BrN2O7-
(E)-4-[[(3R)-1-(4-bromophenyl)-2,5-dioxopyrrolidin-3-yl]-[2-(3,4-dimethoxyphenyl)ethyl]amino]-4-oxobut-2-enoate
—— ethyl (4R)-4-ethyl-6-[[4-(5-methylthiophen-2-yl)-4-oxobutanoyl]oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O6S
ethyl (4R)-4-ethyl-6-[[4-(5-methylthiophen-2-yl)-4-oxobutanoyl]oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-benzyl-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-propan-2-ylprop-2-enamide —— C20H20ClN3O
(E)-N-benzyl-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-propan-2-ylprop-2-enamide
—— (E)-2-(1,3-benzoxazol-2-yl)-3-(4-methyl-2-nitroanilino)prop-2-enal —— C17H13N3O4
(E)-2-(1,3-benzoxazol-2-yl)-3-(4-methyl-2-nitroanilino)prop-2-enal
—— (E)-1-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]-3-[4-(trifluoromethylsulfanyl)phenyl]prop-2-en-1-one —— C19H23F3N2O2S
(E)-1-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]-3-[4-(trifluoromethylsulfanyl)phenyl]prop-2-en-1-one
—— (E)-1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]-3-[4-(trifluoromethylsulfanyl)phenyl]prop-2-en-1-one —— C19H23F3N2O2S
(E)-1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]-3-[4-(trifluoromethylsulfanyl)phenyl]prop-2-en-1-one
—— ethyl 5-[(2S)-2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H24N2O6
ethyl 5-[(2S)-2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (2Z,5S)-5-(3,4-dimethoxyphenyl)-2-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H30N4O7S
ethyl (2Z,5S)-5-(3,4-dimethoxyphenyl)-2-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H22BrClN2O5S
ethyl (2E,5R)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E)-2-[(5E)-5-[(4-cyanophenyl)methylidene]-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C23H25N3O4S
ethyl (2E)-2-[(5E)-5-[(4-cyanophenyl)methylidene]-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (4S)-2-amino-1-(4-bromophenyl)-4-(4-bromothiophen-2-yl)-7,7-dimethyl-5-oxo-6,8-dihydro-4H-quinoline-3-carboxylate —— C24H24Br2N2O3S
ethyl (4S)-2-amino-1-(4-bromophenyl)-4-(4-bromothiophen-2-yl)-7,7-dimethyl-5-oxo-6,8-dihydro-4H-quinoline-3-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)-2-methylpropyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C25H26N4O2S
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)-2-methylpropyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl (2Z,5R)-5-(3,4-dimethoxyphenyl)-2-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H30N4O7S
ethyl (2Z,5R)-5-(3,4-dimethoxyphenyl)-2-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27BrN2O7S
ethyl (2E,5S)-2-[(3-bromo-4,5-dimethoxyphenyl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-(diethylamino)-2-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H39N3O5S
ethyl (2Z,5S)-2-[[4-(diethylamino)-2-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[3-bromo-5-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H31BrN2O6S
ethyl (2E,5S)-2-[[3-bromo-5-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[3-bromo-4-(dimethylamino)phenyl]methylidene]-5-(3-bromo-4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H25Br2N3O4S
ethyl (2Z,5S)-2-[[3-bromo-4-(dimethylamino)phenyl]methylidene]-5-(3-bromo-4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H23BrN2O7S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[(2-bromo-4,5-dimethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H30N2O7S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[3-methoxy-4-(naphthalen-1-ylmethoxy)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C21H22N2O6
ethyl 4-[2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (5R)-4-(3-chlorophenyl)-4'-(4-methylphenyl)-2'-phenylspiro[1,3,4-thiadiazole-5,1'-phthalazine]-2-carboxylate —— C31H25ClN4O2S
ethyl (5R)-4-(3-chlorophenyl)-4'-(4-methylphenyl)-2'-phenylspiro[1,3,4-thiadiazole-5,1'-phthalazine]-2-carboxylate
—— ethyl 5-[2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C21H22N2O6
ethyl 5-[2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (4S)-6-amino-5-cyano-2-[(3-cyano-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-2-yl)sulfanylmethyl]-4-(4-methylsulfanylphenyl)-4H-pyran-3-carboxylate —— C28H28N4O3S2
ethyl (4S)-6-amino-5-cyano-2-[(3-cyano-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-2-yl)sulfanylmethyl]-4-(4-methylsulfanylphenyl)-4H-pyran-3-carboxylate
—— ethyl (4S)-4-(4-bromophenyl)-5-cyano-2-methyl-6-(thiophen-2-ylmethylsulfanyl)-3,4-dihydropyridine-3-carboxylate —— C21H19BrN2O2S2
ethyl (4S)-4-(4-bromophenyl)-5-cyano-2-methyl-6-(thiophen-2-ylmethylsulfanyl)-3,4-dihydropyridine-3-carboxylate
—— ethyl (4R)-6-amino-5-cyano-2-[(3-cyano-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-2-yl)sulfanylmethyl]-4-(4-methylsulfanylphenyl)-4H-pyran-3-carboxylate —— C28H28N4O3S2
ethyl (4R)-6-amino-5-cyano-2-[(3-cyano-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-2-yl)sulfanylmethyl]-4-(4-methylsulfanylphenyl)-4H-pyran-3-carboxylate
—— ethyl N-[3-(1,3-benzothiazol-2-yl)phenyl]carbamate —— C16H14N2O2S
ethyl N-[3-(1,3-benzothiazol-2-yl)phenyl]carbamate
—— ethyl (4-cyano-3-chlorophenyl)carbamate —— C10H9ClN2O2
ethyl (4-cyano-3-chlorophenyl)carbamate
—— Ethyl [4-[(3-nitrobenzoyl)amino]phenyl] carbonate —— C16H14N2O6
Ethyl [4-[(3-nitrobenzoyl)amino]phenyl] carbonate
—— ethyl (4S)-6-amino-4-(4-chlorophenyl)-5-cyano-2-[(3-cyano-4-thiophen-2-yl-5,6,7,8-tetrahydroquinolin-2-yl)sulfanylmethyl]-4H-pyran-3-carboxylate —— C30H25ClN4O3S2
ethyl (4S)-6-amino-4-(4-chlorophenyl)-5-cyano-2-[(3-cyano-4-thiophen-2-yl-5,6,7,8-tetrahydroquinolin-2-yl)sulfanylmethyl]-4H-pyran-3-carboxylate
—— Ethyl 2-[[2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]acetyl]amino]benzoate —— C21H20N2O6
Ethyl 2-[[2-[3-(1,3-benzoxazol-2-yl)propanoyloxy]acetyl]amino]benzoate
—— ethyl (4R)-6-[[(3,4-dimethoxyphenyl)methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H27N3O5
ethyl (4R)-6-[[(3,4-dimethoxyphenyl)methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— Ethyl 4-[[2-[(3-fluorophenyl)methyl-methylamino]acetyl]amino]benzoate —— C19H21FN2O3
Ethyl 4-[[2-[(3-fluorophenyl)methyl-methylamino]acetyl]amino]benzoate
—— (E)-3-[2-(difluoromethoxy)phenyl]-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-ethylprop-2-enamide —— C21H21F2NO4
(E)-3-[2-(difluoromethoxy)phenyl]-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-ethylprop-2-enamide
—— ethyl (4R)-6-[[[4-(difluoromethoxy)-3-methoxyphenyl]methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H25F2N3O5
ethyl (4R)-6-[[[4-(difluoromethoxy)-3-methoxyphenyl]methyl-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2R)-2-cyano-4-(3,4-dimethoxyphenyl)-3-oxobutanoate —— C15H17NO5
ethyl (2R)-2-cyano-4-(3,4-dimethoxyphenyl)-3-oxobutanoate
—— (E)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-ethyl-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C24H26N2O4
(E)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-ethyl-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide —— C21H21N3O2S
(E)-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]-N-[(1R)-1-pyridin-2-ylethyl]prop-2-enamide
—— (E)-N-[(2R)-2-phenylbutyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide —— C22H21N5O
(E)-N-[(2R)-2-phenylbutyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide
—— (E)-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]-N-[(1S)-1-pyridin-2-ylethyl]prop-2-enamide —— C21H21N3O2S
(E)-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]-N-[(1S)-1-pyridin-2-ylethyl]prop-2-enamide