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—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methyl-N-[(1S)-1-phenylethyl]prop-2-enamide —— C22H25N3O2
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methyl-N-[(1S)-1-phenylethyl]prop-2-enamide
—— (E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[(2S)-2-phenylbutyl]prop-2-enamide —— C21H24N2O3
(E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[(2S)-2-phenylbutyl]prop-2-enamide
—— ethyl (2S)-2-cyano-4-(3,4-dimethoxyphenyl)-3-oxobutanoate —— C15H17NO5
ethyl (2S)-2-cyano-4-(3,4-dimethoxyphenyl)-3-oxobutanoate
—— ethyl 2-[[(3S)-3-acetamido-3-(4-chlorophenyl)propanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate —— C22H21ClN2O5S
ethyl 2-[[(3S)-3-acetamido-3-(4-chlorophenyl)propanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate
—— ethyl 2-[[(3R)-3-acetamido-3-(4-chlorophenyl)propanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate —— C22H21ClN2O5S
ethyl 2-[[(3R)-3-acetamido-3-(4-chlorophenyl)propanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate
—— ethyl 2-[[(3S)-3-acetamido-3-thiophen-2-ylpropanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate —— C20H20N2O5S2
ethyl 2-[[(3S)-3-acetamido-3-thiophen-2-ylpropanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate
—— (E)-3-[4-(2-oxopyrrolidin-1-yl)phenyl]-N-[(4-oxo-1H-quinazolin-2-yl)methyl]-N-propan-2-ylprop-2-enamide —— C25H26N4O3
(E)-3-[4-(2-oxopyrrolidin-1-yl)phenyl]-N-[(4-oxo-1H-quinazolin-2-yl)methyl]-N-propan-2-ylprop-2-enamide
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]prop-2-enamide —— C24H27N3O4
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]prop-2-enamide
—— Ethyl 1-[2-[2-[2-(cyclopropylamino)-2-oxoacetyl]hydrazinyl]-2-oxoethyl]-2,5-dimethylpyrrole-3-carboxylate —— C16H22N4O5
Ethyl 1-[2-[2-[2-(cyclopropylamino)-2-oxoacetyl]hydrazinyl]-2-oxoethyl]-2,5-dimethylpyrrole-3-carboxylate
—— ethyl 2-[[(3R)-3-acetamido-3-thiophen-2-ylpropanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate —— C20H20N2O5S2
ethyl 2-[[(3R)-3-acetamido-3-thiophen-2-ylpropanoyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate
—— ethyl (2E,5R)-2-[[3,5-dibromo-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25Br2FN2O5S
ethyl (2E,5R)-2-[[3,5-dibromo-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(2S)-2-(3-chlorophenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C19H20ClNO6S2
ethyl 2-[[(2S)-2-(3-chlorophenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl 3-[(2R,3R,12aR)-1,1-dicyano-2-phenyl-3,12a-dihydro-2H-naphtho[2,1-e]indolizine-3-carbonyl]benzoate —— C34H25N3O3
ethyl 3-[(2R,3R,12aR)-1,1-dicyano-2-phenyl-3,12a-dihydro-2H-naphtho[2,1-e]indolizine-3-carbonyl]benzoate
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[2-(4-ethoxyphenoxy)ethyl]prop-2-enamide —— C24H27N3O3
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[2-(4-ethoxyphenoxy)ethyl]prop-2-enamide
—— ethyl 2-[[(2R)-2-(3-chlorophenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C19H20ClNO6S2
ethyl 2-[[(2R)-2-(3-chlorophenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— (E)-1-[(4R)-4-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-en-1-one —— C22H22N2O2S2
(E)-1-[(4R)-4-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-en-1-one
—— (E)-N-[4-(1-methylimidazol-2-yl)sulfanylphenyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C24H22N4O2S2
(E)-N-[4-(1-methylimidazol-2-yl)sulfanylphenyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl (1R,2S,3R,7R)-9-benzoyl-3,10-dimethyl-4-oxo-8-oxa-5,6,9-triazatricyclo[5.2.2.02,5]undec-10-ene-6-carboxylate —— C19H21N3O5
ethyl (1R,2S,3R,7R)-9-benzoyl-3,10-dimethyl-4-oxo-8-oxa-5,6,9-triazatricyclo[5.2.2.02,5]undec-10-ene-6-carboxylate
—— ethyl 2-[[(2S)-2-(3-methylphenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C20H23NO6S2
ethyl 2-[[(2S)-2-(3-methylphenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— (E)-N-[2-(dimethylamino)-2-oxoethyl]-3-[1-[(4-methylphenyl)methyl]-3-phenylpyrazol-4-yl]prop-2-enamide —— C24H26N4O2
(E)-N-[2-(dimethylamino)-2-oxoethyl]-3-[1-[(4-methylphenyl)methyl]-3-phenylpyrazol-4-yl]prop-2-enamide
—— (E)-1-[(1R,5R)-6,6-dimethyl-2-bicyclo[3.1.1]hept-2-enyl]-N-piperidin-1-ylmethanimine —— C15H24N2
(E)-1-[(1R,5R)-6,6-dimethyl-2-bicyclo[3.1.1]hept-2-enyl]-N-piperidin-1-ylmethanimine
—— ethyl 2-[[(3S)-3-acetamido-3-phenylpropanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C21H24N2O6S2
ethyl 2-[[(3S)-3-acetamido-3-phenylpropanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl (2E,5R)-5-(4-fluorophenyl)-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H27FN4O5S
ethyl (2E,5R)-5-(4-fluorophenyl)-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(2S)-2-[3-[[(S)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate —— C25H25NO6S2
ethyl 2-[[(2S)-2-[3-[[(S)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate
—— ethyl 2-[[2-[(1S,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C21H22N2O7S2
ethyl 2-[[2-[(1S,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— (E)-N-[2-(dimethylamino)-2-oxoethyl]-3-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]prop-2-enamide —— C20H25N3O2
(E)-N-[2-(dimethylamino)-2-oxoethyl]-3-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]prop-2-enamide
—— ethyl 6,6-dioxo-2-[[4-[[(2S)-oxolan-2-yl]methoxy]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C22H25NO7S2
ethyl 6,6-dioxo-2-[[4-[[(2S)-oxolan-2-yl]methoxy]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl 2-[[2-[(1R,2S,6S,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C21H22N2O7S2
ethyl 2-[[2-[(1R,2S,6S,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl 2-[[(2S)-2-[3-[[(R)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate —— C25H25NO6S2
ethyl 2-[[(2S)-2-[3-[[(R)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[3-[[(S)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate —— C25H25NO6S2
ethyl 2-[[(2R)-2-[3-[[(S)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-3-[4-(diethylsulfamoyl)phenyl]-N-(6-piperidin-1-ylpyridin-3-yl)prop-2-enamide —— C23H30N4O3S
(E)-3-[4-(diethylsulfamoyl)phenyl]-N-(6-piperidin-1-ylpyridin-3-yl)prop-2-enamide
—— ethyl 2-[[2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C21H22N2O7S2
ethyl 2-[[2-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]acetyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— Ethyl 4-[[2-(2-cyanophenoxy)acetyl]hydrazinylidene]piperidine-1-carboxylate —— C17H20N4O4
Ethyl 4-[[2-(2-cyanophenoxy)acetyl]hydrazinylidene]piperidine-1-carboxylate
—— ethyl (2S)-4-(4-chlorophenoxy)-2-cyano-3-oxobutanoate —— C13H12ClNO4
ethyl (2S)-4-(4-chlorophenoxy)-2-cyano-3-oxobutanoate
—— ethyl (2E,5S)-5-(3-methoxyphenyl)-2-[[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H34N4O5S
ethyl (2E,5S)-5-(3-methoxyphenyl)-2-[[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[5-[(Z)-[[2-(2-cyanophenoxy)acetyl]hydrazinylidene]methyl]furan-2-yl]benzoate —— C23H19N3O5
ethyl 4-[5-[(Z)-[[2-(2-cyanophenoxy)acetyl]hydrazinylidene]methyl]furan-2-yl]benzoate
—— ethyl 2-[[(2R)-2-(3-methylphenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C20H23NO6S2
ethyl 2-[[(2R)-2-(3-methylphenoxy)propanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl 6,6-dioxo-2-[[4-[[(2R)-oxolan-2-yl]methoxy]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C22H25NO7S2
ethyl 6,6-dioxo-2-[[4-[[(2R)-oxolan-2-yl]methoxy]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl 2-[[(2R)-2-[3-[[(R)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate —— C25H25NO6S2
ethyl 2-[[(2R)-2-[3-[[(R)-methylsulfinyl]methyl]benzoyl]oxypropanoyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[4-(2-pyrrolidin-1-ylethyl)piperazin-1-yl]prop-2-en-1-one —— C24H33N5O
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[4-(2-pyrrolidin-1-ylethyl)piperazin-1-yl]prop-2-en-1-one
—— ethyl (2R)-5-(3-chlorophenyl)-2-cyano-3-oxopentanoate —— C14H14ClNO3
ethyl (2R)-5-(3-chlorophenyl)-2-cyano-3-oxopentanoate
—— ethyl (2R)-4-(2-chlorophenoxy)-2-cyano-3-oxobutanoate —— C13H12ClNO4
ethyl (2R)-4-(2-chlorophenoxy)-2-cyano-3-oxobutanoate
—— ethyl (3R)-3-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate —— C16H27NO3
ethyl (3R)-3-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate
—— [(E)-[(4R)-10,11-dimethoxy-5-(4-methylphenyl)sulfonyl-5-azatricyclo[6.3.1.04,12]dodeca-1(12),8,10-trien-2-ylidene]amino] 4-methylbenzenesulfonate —— C27H28N2O7S2
[(E)-[(4R)-10,11-dimethoxy-5-(4-methylphenyl)sulfonyl-5-azatricyclo[6.3.1.04,12]dodeca-1(12),8,10-trien-2-ylidene]amino] 4-methylbenzenesulfonate
—— (E)-N-[2-(dimethylamino)-2-oxoethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C18H22N4O2
(E)-N-[2-(dimethylamino)-2-oxoethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl (3S)-3-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate —— C16H27NO3
ethyl (3S)-3-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate
—— ethyl (3R)-3-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate —— C16H27NO3
ethyl (3R)-3-[[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate
—— (E)-N-[2-(dimethylamino)-2-oxoethyl]-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)prop-2-enamide —— C19H23N3O2
(E)-N-[2-(dimethylamino)-2-oxoethyl]-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)prop-2-enamide
—— (E)-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]prop-2-en-1-one —— C27H30N2O5
(E)-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]prop-2-en-1-one
—— ethyl (2Z,5S)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H26F3N3O8S
ethyl (2Z,5S)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate