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—— (E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide —— C22H29N3O4S
(E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide
—— ethyl (2E,5S)-2-[[1-[(2-chlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H32ClN3O3S
ethyl (2E,5S)-2-[[1-[(2-chlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 6,6-dioxo-2-[[(4S)-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C20H20N2O6S2
ethyl 6,6-dioxo-2-[[(4S)-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— ethyl (2E,5R)-2-[(3,5-dibromo-4-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H16Br2N2O4S2
ethyl (2E,5R)-2-[(3,5-dibromo-4-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-butyl-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C23H30ClN3O3S
(E)-N-butyl-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— ethyl 5-[butyl-[(3R)-1,1-dioxothiolan-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H28N2O5S
ethyl 5-[butyl-[(3R)-1,1-dioxothiolan-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[4-[(2-cyanophenyl)methoxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H27N3O7S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[4-[(2-cyanophenyl)methoxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2,4-dimethoxyphenyl)-2-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O7S
ethyl (2E,5S)-5-(2,4-dimethoxyphenyl)-2-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-2-[(4-methoxy-2-methylphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H28N2O6S
ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-2-[(4-methoxy-2-methylphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-phenyl-2-(thiophen-2-ylmethylidene)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24N2O4S2
ethyl (2E,5R)-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-phenyl-2-(thiophen-2-ylmethylidene)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C24H29N5O2S
(E)-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl 3,5-dimethyl-4-[[4-(methylcarbamoyl)phenyl]carbamoyl]-1H-pyrrole-2-carboxylate —— C18H21N3O4
ethyl 3,5-dimethyl-4-[[4-(methylcarbamoyl)phenyl]carbamoyl]-1H-pyrrole-2-carboxylate
—— (E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]prop-2-enamide —— C25H27N3O3
(E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]prop-2-enamide
—— ethyl (4R)-4-(4-bromo-5-methylthiophen-2-yl)-2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydroquinoline-3-carboxylate —— C20H24BrNO3S
ethyl (4R)-4-(4-bromo-5-methylthiophen-2-yl)-2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydroquinoline-3-carboxylate
—— ethyl 4-[5-[(Z)-2-cyano-3-[[5-[(2,5-dichlorophenyl)methyl]-1,3-thiazol-2-yl]amino]-3-oxoprop-1-enyl]furan-2-yl]benzoate —— C27H19Cl2N3O4S
ethyl 4-[5-[(Z)-2-cyano-3-[[5-[(2,5-dichlorophenyl)methyl]-1,3-thiazol-2-yl]amino]-3-oxoprop-1-enyl]furan-2-yl]benzoate
—— ethyl (2E,5R)-2-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-5-(2,5-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H25BrN2O7S
ethyl (2E,5R)-2-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-5-(2,5-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[(5-bromo-2-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H17BrN2O4S2
ethyl (2E,5S)-2-[(5-bromo-2-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-(2-ethylanilino)-2-oxoethyl]-N-methylprop-2-enamide —— C22H24N2O4
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-(2-ethylanilino)-2-oxoethyl]-N-methylprop-2-enamide
—— (E)-3-[4-methoxy-3-(methylsulfamoyl)phenyl]-N-[4-(4-methoxyphenyl)-5-methyl-1,3-thiazol-2-yl]prop-2-enamide —— C22H23N3O5S2
(E)-3-[4-methoxy-3-(methylsulfamoyl)phenyl]-N-[4-(4-methoxyphenyl)-5-methyl-1,3-thiazol-2-yl]prop-2-enamide
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide —— C21H23ClN2O4
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C19H23F4NO5S
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-butyl-N-[(3S)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (E)-N-[4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide —— C22H29N3O4S
(E)-N-[4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide —— C19H23F4NO5S
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-N-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]prop-2-enamide
—— (E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C24H29N5O2S
(E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl 6,6-dioxo-2-[[(4R)-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C20H20N2O6S2
ethyl 6,6-dioxo-2-[[(4R)-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]amino]-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— (E)-3-(5-bromo-2-fluorophenyl)-N-[2-(2-ethylanilino)-2-oxoethyl]-N-methylprop-2-enamide —— C20H20BrFN2O2
(E)-3-(5-bromo-2-fluorophenyl)-N-[2-(2-ethylanilino)-2-oxoethyl]-N-methylprop-2-enamide
—— ethyl (2E)-2-[(5Z)-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C25H32N2O7S
ethyl (2E)-2-[(5Z)-3-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— (E)-3-(3-bromophenyl)-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide —— C19H19BrN2O2
(E)-3-(3-bromophenyl)-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-(2-ethylanilino)-2-oxoethyl]-3-(4-methylphenyl)prop-2-enamide —— C20H22N2O2
(E)-N-[2-(2-ethylanilino)-2-oxoethyl]-3-(4-methylphenyl)prop-2-enamide
—— ethyl (2E)-2-[(5Z)-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C25H32N2O7S
ethyl (2E)-2-[(5Z)-3-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— (E)-N-[2-(4-bromo-2-methylanilino)-2-oxoethyl]-3-(2-fluorophenyl)-N-methylprop-2-enamide —— C19H18BrFN2O2
(E)-N-[2-(4-bromo-2-methylanilino)-2-oxoethyl]-3-(2-fluorophenyl)-N-methylprop-2-enamide
—— ethyl 6-[(5Z)-5-[(5Z)-3-ethyl-5-[(2E)-2-(3-ethyl-1,3-benzothiazol-2-ylidene)ethylidene]-4-oxo-1,3-thiazolidin-2-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate —— C27H31N3O4S4
ethyl 6-[(5Z)-5-[(5Z)-3-ethyl-5-[(2E)-2-(3-ethyl-1,3-benzothiazol-2-ylidene)ethylidene]-4-oxo-1,3-thiazolidin-2-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoate
—— (E)-N-[(3R)-1,1-dioxothiolan-3-yl]-3-[5-(4-fluorophenyl)thiophen-2-yl]-N',N'-dimethylprop-2-enehydrazide —— C19H21FN2O3S2
(E)-N-[(3R)-1,1-dioxothiolan-3-yl]-3-[5-(4-fluorophenyl)thiophen-2-yl]-N',N'-dimethylprop-2-enehydrazide
—— (E)-1-[4-[4-[(2S)-butan-2-yl]phenyl]sulfonylpiperazin-1-yl]but-2-en-1-one —— C18H26N2O3S
(E)-1-[4-[4-[(2S)-butan-2-yl]phenyl]sulfonylpiperazin-1-yl]but-2-en-1-one
—— (E)-3-(4-chlorophenyl)-1-[4-[5-(trifluoromethyl)pyridin-1-ium-2-yl]piperazin-1-yl]prop-2-en-1-one —— C19H18ClF3N3O+
(E)-3-(4-chlorophenyl)-1-[4-[5-(trifluoromethyl)pyridin-1-ium-2-yl]piperazin-1-yl]prop-2-en-1-one
—— (E)-N-[5-[(2S)-2-methylpiperidine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]-3-phenylprop-2-enamide —— C33H36N4O3
(E)-N-[5-[(2S)-2-methylpiperidine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]-3-phenylprop-2-enamide
—— (E)-N-[5-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]-3-phenylprop-2-enamide —— C39H41N5O3
(E)-N-[5-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]phenyl]-3-phenylprop-2-enamide
—— (E)-3-(4-nitrophenyl)-1-[4-[5-(trifluoromethyl)pyridin-1-ium-2-yl]piperazin-1-yl]prop-2-en-1-one —— C19H18F3N4O3+
(E)-3-(4-nitrophenyl)-1-[4-[5-(trifluoromethyl)pyridin-1-ium-2-yl]piperazin-1-yl]prop-2-en-1-one
—— (E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-[5-(4-fluorophenyl)thiophen-2-yl]-N',N'-dimethylprop-2-enehydrazide —— C19H21FN2O3S2
(E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-[5-(4-fluorophenyl)thiophen-2-yl]-N',N'-dimethylprop-2-enehydrazide
—— ethyl 2-[[(2S)-2,3-dihydro-1-benzothiophene-2-carbonyl]oxymethyl]-4-methylquinoline-3-carboxylate —— C23H21NO4S
ethyl 2-[[(2S)-2,3-dihydro-1-benzothiophene-2-carbonyl]oxymethyl]-4-methylquinoline-3-carboxylate
—— ethyl 3-oxo-3-[[(1S,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propanoate —— C15H25NO3
ethyl 3-oxo-3-[[(1S,2S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]amino]propanoate
—— (E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]prop-2-enamide —— C25H27N3O3
(E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-(1-phenylpyrazol-4-yl)ethyl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-1-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]prop-2-en-1-one —— C21H22F3N3O3
(E)-3-(3,4-dimethoxyphenyl)-1-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(2-nitrophenyl)-1-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]prop-2-en-1-one —— C19H17F3N4O3
(E)-3-(2-nitrophenyl)-1-[4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(4-fluorophenyl)-N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]prop-2-enamide —— C21H22F2N2O2
(E)-3-(4-fluorophenyl)-N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]prop-2-enamide
—— (E)-3-(2,4-dimethoxyphenyl)-1-[4-[5-(trifluoromethyl)pyridin-1-ium-2-yl]piperazin-1-yl]prop-2-en-1-one —— C21H23F3N3O3+
(E)-3-(2,4-dimethoxyphenyl)-1-[4-[5-(trifluoromethyl)pyridin-1-ium-2-yl]piperazin-1-yl]prop-2-en-1-one
—— (E)-N-[3-[2-(cyclopentylcarbamothioyl)hydrazinyl]-3-oxopropyl]-3-(4-methoxyphenyl)prop-2-enamide —— C19H26N4O3S
(E)-N-[3-[2-(cyclopentylcarbamothioyl)hydrazinyl]-3-oxopropyl]-3-(4-methoxyphenyl)prop-2-enamide
—— ethyl (3R)-1-(5-aminofuran-2-carbonyl)piperidine-3-carboxylate —— C13H18N2O4
ethyl (3R)-1-(5-aminofuran-2-carbonyl)piperidine-3-carboxylate
—— (E)-N-[(2S)-1-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)prop-2-enamide —— C25H28N4O3
(E)-N-[(2S)-1-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)prop-2-enamide
—— (E)-N-[(2R)-1-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)prop-2-enamide —— C25H28N4O3
(E)-N-[(2R)-1-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)prop-2-enamide