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—— (E)-3-(4-methylphenyl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C22H26N2O
(E)-3-(4-methylphenyl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C24H27ClN2O3
(E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— ethyl 2-[[(2S)-2-methylbutanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate —— C15H21NO5S2
ethyl 2-[[(2S)-2-methylbutanoyl]amino]-6,6-dioxo-5,7-dihydro-4H-thieno[2,3-c]thiopyran-3-carboxylate
—— (E)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[(15R)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]prop-2-enamide —— C24H22N2OS
(E)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[(15R)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]prop-2-enamide
—— (E)-3-[1-[(2S)-3-(azepan-1-ium-1-yl)-2-hydroxypropyl]indol-3-yl]-1-(4-methoxyphenyl)prop-2-en-1-one —— C27H33N2O3+
(E)-3-[1-[(2S)-3-(azepan-1-ium-1-yl)-2-hydroxypropyl]indol-3-yl]-1-(4-methoxyphenyl)prop-2-en-1-one
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C24H30ClN2O3+
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— ethyl (4S,7R)-7-(4-chlorophenyl)-4-(4-fluorophenyl)-2-methyl-5-oxo-4,6,7,8-tetrahydro-3H-quinoline-3-carboxylate —— C25H23ClFNO3
ethyl (4S,7R)-7-(4-chlorophenyl)-4-(4-fluorophenyl)-2-methyl-5-oxo-4,6,7,8-tetrahydro-3H-quinoline-3-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C22H25N2O3+
(E)-3-(1,3-benzodioxol-5-yl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]prop-2-enamide —— C24H22N2OS
(E)-3-(2-methyl-1,3-thiazol-4-yl)-N-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]prop-2-enamide
—— (E)-3-[1-[(2R)-3-(azepan-1-yl)-2-hydroxypropyl]indol-3-yl]-1-(4-methoxyphenyl)prop-2-en-1-one —— C27H32N2O3
(E)-3-[1-[(2R)-3-(azepan-1-yl)-2-hydroxypropyl]indol-3-yl]-1-(4-methoxyphenyl)prop-2-en-1-one
—— ethyl (4R)-4-(furan-2-yl)-2-oxo-6-[[(E)-3-quinolin-8-ylprop-2-enoyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H21N3O6
ethyl (4R)-4-(furan-2-yl)-2-oxo-6-[[(E)-3-quinolin-8-ylprop-2-enoyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(2-methoxy-5-methylphenyl)-N-[4-(tetrazol-1-yl)phenyl]prop-2-enamide —— C18H17N5O2
(E)-3-(2-methoxy-5-methylphenyl)-N-[4-(tetrazol-1-yl)phenyl]prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C21H23FN2O
(E)-3-(4-fluorophenyl)-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— ethyl (3S)-1-[(2S)-3-[4-(cyanomethyl)phenoxy]-2-hydroxypropyl]piperidine-3-carboxylate —— C19H26N2O4
ethyl (3S)-1-[(2S)-3-[4-(cyanomethyl)phenoxy]-2-hydroxypropyl]piperidine-3-carboxylate
—— ethyl (4S)-4-[4-methoxy-3-(phenoxymethyl)phenyl]-2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydroquinoline-3-carboxylate —— C29H33NO5
ethyl (4S)-4-[4-methoxy-3-(phenoxymethyl)phenyl]-2,7,7-trimethyl-5-oxo-3,4,6,8-tetrahydroquinoline-3-carboxylate
—— (E)-3-(1,3-benzoxazol-2-yl)-4-(2-phenylmethoxyphenyl)but-3-enoate —— C24H18NO4-
(E)-3-(1,3-benzoxazol-2-yl)-4-(2-phenylmethoxyphenyl)but-3-enoate
—— ethyl 4-methyl-2-[[2-[(2R)-2-methylpiperidin-1-ium-1-yl]acetyl]amino]-5-phenylthiophene-3-carboxylate —— C22H29N2O3S+
ethyl 4-methyl-2-[[2-[(2R)-2-methylpiperidin-1-ium-1-yl]acetyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-3-(3-fluorophenyl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide —— C21H24FN2O+
(E)-3-(3-fluorophenyl)-N-[[4-(pyrrolidin-1-ium-1-ylmethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(3-chloro-4-fluorophenyl)-N-[2-(furan-2-ylmethylamino)-2-oxoethyl]-N-methylprop-2-enamide —— C17H16ClFN2O3
(E)-3-(3-chloro-4-fluorophenyl)-N-[2-(furan-2-ylmethylamino)-2-oxoethyl]-N-methylprop-2-enamide
—— (E)-3-(1,3-benzoxazol-2-yl)-4-(2-phenylmethoxyphenyl)but-3-enoic acid —— C24H19NO4
(E)-3-(1,3-benzoxazol-2-yl)-4-(2-phenylmethoxyphenyl)but-3-enoic acid
—— ethyl (2E,5R)-2-[(5-chloro-2-methoxyphenyl)methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H27ClN2O5S
ethyl (2E,5R)-2-[(5-chloro-2-methoxyphenyl)methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-(4-morpholin-4-ylphenyl)prop-2-enamide —— C22H23ClN2O4
(E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-(4-morpholin-4-ylphenyl)prop-2-enamide
—— ethyl 4-[(3S)-3-[(3-chlorophenyl)carbamothioyl-[2-(3,4-dimethoxyphenyl)ethyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate —— C30H30ClN3O6S
ethyl 4-[(3S)-3-[(3-chlorophenyl)carbamothioyl-[2-(3,4-dimethoxyphenyl)ethyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl (4R)-6-[3-(4-fluorophenyl)propanoyloxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H21FN2O5
ethyl (4R)-6-[3-(4-fluorophenyl)propanoyloxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2S,6R,8S,12R)-7-bromo-4,10-bis(4-ethoxyphenyl)-1,14-dimethyl-3,5,9,11-tetraoxo-4,10-diazatetracyclo[5.5.2.02,6.08,12]tetradec-13-ene-13-carboxylate —— C33H33BrN2O8
ethyl (2S,6R,8S,12R)-7-bromo-4,10-bis(4-ethoxyphenyl)-1,14-dimethyl-3,5,9,11-tetraoxo-4,10-diazatetracyclo[5.5.2.02,6.08,12]tetradec-13-ene-13-carboxylate
—— ethyl 4-[(3R)-3-[N-(4-fluorophenyl)-N'-methylcarbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate —— C21H20FN3O4S
ethyl 4-[(3R)-3-[N-(4-fluorophenyl)-N'-methylcarbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl 4-[(3S)-2,5-dioxo-3-[2-phenylethyl-[[3-(trifluoromethyl)phenyl]carbamothioyl]amino]pyrrolidin-1-yl]benzoate —— C29H26F3N3O4S
ethyl 4-[(3S)-2,5-dioxo-3-[2-phenylethyl-[[3-(trifluoromethyl)phenyl]carbamothioyl]amino]pyrrolidin-1-yl]benzoate
—— (E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C24H28N4O3S2
(E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl 4-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-fluorophenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate —— C30H30FN3O6S
ethyl 4-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-fluorophenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate
—— (E)-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide —— C22H29N3O4S
(E)-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-(4-ethoxy-3-methoxyphenyl)prop-2-enamide
—— ethyl 4-[(3S)-3-[benzylcarbamothioyl(2-phenylethyl)amino]-2,5-dioxopyrrolidin-1-yl]benzoate —— C29H29N3O4S
ethyl 4-[(3S)-3-[benzylcarbamothioyl(2-phenylethyl)amino]-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl (2E,5S)-2-[(1,5-dimethylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H24N4O4S
ethyl (2E,5S)-2-[(1,5-dimethylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-naphthalen-1-ylprop-2-enamide —— C23H25N3O2S
(E)-N-[4-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-naphthalen-1-ylprop-2-enamide
—— ethyl 4-[(3R)-3-[N-(3-fluorophenyl)-N'-methylcarbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate —— C21H20FN3O4S
ethyl 4-[(3R)-3-[N-(3-fluorophenyl)-N'-methylcarbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl 4-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-methoxyphenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate —— C31H33N3O7S
ethyl 4-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-methoxyphenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl 4-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-methoxyphenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate —— C31H33N3O7S
ethyl 4-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-methoxyphenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate
—— ethyl 5-[butyl-[(3S)-1,1-dioxothiolan-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C18H28N2O5S
ethyl 5-[butyl-[(3S)-1,1-dioxothiolan-3-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-3-(5-nitrofuran-2-yl)-N-[4-[[(E)-3-(5-nitrofuran-2-yl)prop-2-enylidene]amino]-6-phenyl-1,3,5-triazin-2-yl]prop-2-en-1-imine —— C23H15N7O6
(E)-3-(5-nitrofuran-2-yl)-N-[4-[[(E)-3-(5-nitrofuran-2-yl)prop-2-enylidene]amino]-6-phenyl-1,3,5-triazin-2-yl]prop-2-en-1-imine
—— ethyl (2E,5S,6R,8aR)-5-[4-(2-ethoxy-2-oxoethoxy)-3-methoxyphenyl]-7-methyl-2-(naphthalen-1-ylmethylidene)-3-oxo-6,8a-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H32N2O7S
ethyl (2E,5S,6R,8aR)-5-[4-(2-ethoxy-2-oxoethoxy)-3-methoxyphenyl]-7-methyl-2-(naphthalen-1-ylmethylidene)-3-oxo-6,8a-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-2-[(1,5-dimethylpyrazol-4-yl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H26N4O5S
ethyl (2E,5R)-5-(3,4-dimethoxyphenyl)-2-[(1,5-dimethylpyrazol-4-yl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-naphthalen-1-ylprop-2-enamide —— C23H25N3O2S
(E)-N-[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-naphthalen-1-ylprop-2-enamide
—— ethyl (2R,3Z)-3-[(4-bromophenyl)hydrazinylidene]-2-methyl-4,5-dioxo-1-phenylpyrrolidine-2-carboxylate —— C20H18BrN3O4
ethyl (2R,3Z)-3-[(4-bromophenyl)hydrazinylidene]-2-methyl-4,5-dioxo-1-phenylpyrrolidine-2-carboxylate
—— ethyl (2E,5R)-2-[[4-[(2-cyanophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C42H33N3O6S
ethyl (2E,5R)-2-[[4-[(2-cyanophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(2-methoxynaphthalen-1-yl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl N-[2-[(4-bromobenzoyl)-ethylamino]acetyl]carbamate —— C14H17BrN2O4
ethyl N-[2-[(4-bromobenzoyl)-ethylamino]acetyl]carbamate
—— ethyl 4-[(3R)-3-[N'-(1,3-benzodioxol-5-ylmethyl)-N-(4-chlorophenyl)carbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate —— C28H24ClN3O6S
ethyl 4-[(3R)-3-[N'-(1,3-benzodioxol-5-ylmethyl)-N-(4-chlorophenyl)carbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate
—— (E)-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C24H28N4O3S2
(E)-N-[4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl 4-[(3R)-3-[N-(2-methoxyphenyl)-N'-methylcarbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate —— C22H23N3O5S
ethyl 4-[(3R)-3-[N-(2-methoxyphenyl)-N'-methylcarbamimidoyl]sulfanyl-2,5-dioxopyrrolidin-1-yl]benzoate
—— (E)-N-[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C24H28N4O3S2
(E)-N-[4-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-1,3-thiazol-2-yl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl (2E,5R)-5-(2-bromo-4,5-dimethoxyphenyl)-2-[(5-chloro-2-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H22BrClN2O6S
ethyl (2E,5R)-5-(2-bromo-4,5-dimethoxyphenyl)-2-[(5-chloro-2-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-fluorophenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate —— C30H30FN3O6S
ethyl 4-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-[(4-fluorophenyl)carbamothioyl]amino]-2,5-dioxopyrrolidin-1-yl]benzoate