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—— ethyl (3S)-3-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate —— C16H27NO3
ethyl (3S)-3-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]-4-oxopentanoate
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one —— C23H35N5O2+2
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one —— C24H35N5O+2
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one
—— ethyl (2E,5S)-2-[[5-bromo-2-[(2-chloro-6-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H22BrCl2FN2O4S
ethyl (2E,5S)-2-[[5-bromo-2-[(2-chloro-6-fluorophenyl)methoxy]phenyl]methylidene]-5-(4-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-(adamantane-1-carbonyloxy)-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H36N2O6S
ethyl (2Z,5S)-2-[[4-(adamantane-1-carbonyloxy)-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2R)-5-(2-chlorophenyl)-2-cyano-3-oxopentanoate —— C14H14ClNO3
ethyl (2R)-5-(2-chlorophenyl)-2-cyano-3-oxopentanoate
—— ethyl (2Z,5R)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H26F3N3O8S
ethyl (2Z,5R)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-[4-[(2,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-[(2-methoxynaphthalen-1-yl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C36H30Cl2N2O6S
ethyl (2E,5S)-5-[4-[(2,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-[(2-methoxynaphthalen-1-yl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[3-ethoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H26F3N3O7S
ethyl (2E,5S)-2-[[3-ethoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24F3N3O7S
ethyl (2Z,5R)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2S)-4-(2-chlorophenoxy)-2-cyano-3-oxobutanoate —— C13H12ClNO4
ethyl (2S)-4-(2-chlorophenoxy)-2-cyano-3-oxobutanoate
—— ethyl (2E,5S)-7-methyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H35N5O5S
ethyl (2E,5S)-7-methyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2R)-2-[(5E)-5-[[4-[2-(4-fluoroanilino)-2-oxoethoxy]phenyl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C23H21FN2O6S
ethyl (2R)-2-[(5E)-5-[[4-[2-(4-fluoroanilino)-2-oxoethoxy]phenyl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— ethyl (2S)-5-(4-chlorophenyl)-2-cyano-3-oxopentanoate —— C14H14ClNO3
ethyl (2S)-5-(4-chlorophenyl)-2-cyano-3-oxopentanoate
—— ethyl (2R)-4-(4-chlorophenoxy)-2-cyano-3-oxobutanoate —— C13H12ClNO4
ethyl (2R)-4-(4-chlorophenoxy)-2-cyano-3-oxobutanoate
—— ethyl (2E,5R)-5-(4-methoxyphenyl)-7-methyl-2-[[1-[(4-nitrophenyl)methyl]indol-2-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H28N4O6S
ethyl (2E,5R)-5-(4-methoxyphenyl)-7-methyl-2-[[1-[(4-nitrophenyl)methyl]indol-2-yl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(4-chlorophenyl)-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31ClN5O5S+
ethyl (2E,5R)-5-(4-chlorophenyl)-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2S)-5-(3-chlorophenyl)-2-cyano-3-oxopentanoate —— C14H14ClNO3
ethyl (2S)-5-(3-chlorophenyl)-2-cyano-3-oxopentanoate
—— ethyl (2S)-5-(2-chlorophenyl)-2-cyano-3-oxopentanoate —— C14H14ClNO3
ethyl (2S)-5-(2-chlorophenyl)-2-cyano-3-oxopentanoate
—— Ethyl 2-[[4-amino-5-(methoxymethyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C8H14N4O3S
Ethyl 2-[[4-amino-5-(methoxymethyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl (2R)-5-(4-chlorophenyl)-2-cyano-3-oxopentanoate —— C14H14ClNO3
ethyl (2R)-5-(4-chlorophenyl)-2-cyano-3-oxopentanoate
—— (E)-1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(3-nitrophenyl)prop-2-en-1-one —— C20H20N2O4
(E)-1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(3-nitrophenyl)prop-2-en-1-one
—— ethyl N'-[(Z)-benzylideneamino]-N-[3-phenyl-4,5-bis(phenylimino)-1,3-thiazolidin-2-ylidene]carbamimidothioate —— C31H26N6S2
ethyl N'-[(Z)-benzylideneamino]-N-[3-phenyl-4,5-bis(phenylimino)-1,3-thiazolidin-2-ylidene]carbamimidothioate
—— (E)-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-1-[(2R)-2-phenylpyrrolidin-1-yl]prop-2-en-1-one —— C26H28N2O4
(E)-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-1-[(2R)-2-phenylpyrrolidin-1-yl]prop-2-en-1-one
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide —— C20H17ClFNO2
(E)-3-(6-chloro-2H-chromen-3-yl)-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide
—— ethyl 6-(4-methylphenylamino)-3,4-diphenylpyrido[2',3':4,5]thieno[2,3-c]pyridazine-7-carboxylate —— C31H24N4O2S
ethyl 6-(4-methylphenylamino)-3,4-diphenylpyrido[2',3':4,5]thieno[2,3-c]pyridazine-7-carboxylate
—— ethyl (2E,5S)-7-methyl-2-[(5-nitro-2-piperidin-1-ylphenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26N4O5S2
ethyl (2E,5S)-7-methyl-2-[(5-nitro-2-piperidin-1-ylphenyl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-7-methyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5-(3,4,5-trimethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H35N5O8S
ethyl (2E,5S)-7-methyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5-(3,4,5-trimethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3-methoxyphenyl)-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34N5O6S+
ethyl (2E,5S)-5-(3-methoxyphenyl)-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(4-fluorophenyl)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H29FN5O5S+
ethyl (2E,5R)-5-(4-fluorophenyl)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H33N5O7S
ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H31N4O6S+
ethyl (2E,5S)-5-(1,3-benzodioxol-5-yl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E)-5-(3-methoxyphenyl)-7-methyl-2-{[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H30N4O5S
ethyl (2E)-5-(3-methoxyphenyl)-7-methyl-2-{[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2-bromo-4,5-dimethoxyphenyl)-2-[(2-hydroxy-3-nitrophenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H22BrN3O8S
ethyl (2E,5S)-5-(2-bromo-4,5-dimethoxyphenyl)-2-[(2-hydroxy-3-nitrophenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H34N5O7S+
ethyl (2E,5S)-5-(2,5-dimethoxyphenyl)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[(5-nitro-2-piperidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H32N4O7S
ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-7-methyl-2-[(5-nitro-2-piperidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 5-(2,4-dimethoxyphenyl)-7-methyl-2-{[5-(4-methyl-1-piperazinyl)-2-furyl]methylene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H32N4O6S
ethyl 5-(2,4-dimethoxyphenyl)-7-methyl-2-{[5-(4-methyl-1-piperazinyl)-2-furyl]methylene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(3-methoxyphenyl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H35N4O5S+
ethyl (2E,5R)-5-(3-methoxyphenyl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[5-(2-methoxycarbonylphenyl)furan-2-yl]methylidene]-7-methyl-3-oxo-5-(3,4,5-trimethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O9S
ethyl (2E,5S)-2-[[5-(2-methoxycarbonylphenyl)furan-2-yl]methylidene]-7-methyl-3-oxo-5-(3,4,5-trimethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 5-methyl-3-(5-nitrofuran-2-yl)-1-(4-nitrophenyl)pyrazole-4-carboxylate —— C17H14N4O7
Ethyl 5-methyl-3-(5-nitrofuran-2-yl)-1-(4-nitrophenyl)pyrazole-4-carboxylate
—— ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H35N4O6S+
ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H31N5O7S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(2-methoxyphenyl)-2-[[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H34N4O5S
ethyl (2E,5R)-5-(2-methoxyphenyl)-2-[[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(4-ethoxyphenyl)-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H32N4O7S
ethyl (2E,5S)-5-(4-ethoxyphenyl)-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(2-methoxy-5-methylphenyl)-1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]prop-2-en-1-one —— C22H25NO3
(E)-3-(2-methoxy-5-methylphenyl)-1-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]prop-2-en-1-one
—— ethyl (2S)-2-cyano-4-(4-methoxyphenoxy)-3-oxobutanoate —— C14H15NO5
ethyl (2S)-2-cyano-4-(4-methoxyphenoxy)-3-oxobutanoate
—— ethyl 2-[4-[bis[(5S)-1-methyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-yl]methyl]-2-chloro-6-methoxyphenoxy]acetate —— C22H23ClN4O8S2
ethyl 2-[4-[bis[(5S)-1-methyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-yl]methyl]-2-chloro-6-methoxyphenoxy]acetate
—— (E)-N-[(E)-(3-chloro-4,5-dimethoxyphenyl)methylideneamino]-3-methyl-1,3-benzothiazol-2-imine —— C17H16ClN3O2S
(E)-N-[(E)-(3-chloro-4,5-dimethoxyphenyl)methylideneamino]-3-methyl-1,3-benzothiazol-2-imine
—— ethyl (2R)-2-cyano-5-(3-methylphenoxy)-3-oxopentanoate —— C15H17NO4
ethyl (2R)-2-cyano-5-(3-methylphenoxy)-3-oxopentanoate
—— (E)-N-[(E)-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)methylideneamino]-3-methyl-1,3-benzothiazol-2-imine —— C14H10ClN5S2
(E)-N-[(E)-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)methylideneamino]-3-methyl-1,3-benzothiazol-2-imine