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—— (E)-N-[4-[[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide —— C26H32N2O5S
(E)-N-[4-[[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide
—— ethyl N-[3-[methyl-[2-(4-methylanilino)-2-oxoethyl]carbamoyl]phenyl]carbamate —— C20H23N3O4
ethyl N-[3-[methyl-[2-(4-methylanilino)-2-oxoethyl]carbamoyl]phenyl]carbamate
—— ethyl (2R)-1-[2-[(3R)-5-(2-fluorophenyl)-3-(2-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C26H30FN3O4
ethyl (2R)-1-[2-[(3R)-5-(2-fluorophenyl)-3-(2-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl (2R)-1-[2-[(3R)-3,5-bis(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C27H33N3O5
ethyl (2R)-1-[2-[(3R)-3,5-bis(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— (E)-N-[4-[[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide —— C26H32N2O5S
(E)-N-[4-[[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide
—— Ethyl 3-[[1-(furan-2-carbonyl)piperidine-4-carbonyl]amino]benzoate —— C20H22N2O5
Ethyl 3-[[1-(furan-2-carbonyl)piperidine-4-carbonyl]amino]benzoate
—— ethyl (3S)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(3,4-dimethylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C27H32ClN3O3
ethyl (3S)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(3,4-dimethylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(3,4-dimethylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C27H32ClN3O3
ethyl (3R)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(3,4-dimethylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C25H27ClFN3O3
ethyl (3R)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (2S)-1-[2-[(3R)-3,5-bis(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C27H33N3O5
ethyl (2S)-1-[2-[(3R)-3,5-bis(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl 4-cyclopropyl-2-[[2-[[(1S)-1-(3,4-difluorophenyl)ethyl]amino]acetyl]amino]thiophene-3-carboxylate —— C20H22F2N2O3S
ethyl 4-cyclopropyl-2-[[2-[[(1S)-1-(3,4-difluorophenyl)ethyl]amino]acetyl]amino]thiophene-3-carboxylate
—— ethyl (2S)-1-[2-[(3R)-5-(2-fluorophenyl)-3-(2-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C26H30FN3O4
ethyl (2S)-1-[2-[(3R)-5-(2-fluorophenyl)-3-(2-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl (3S)-1-[2-[(3R)-3-(2-fluorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C25H27F2N3O3
ethyl (3S)-1-[2-[(3R)-3-(2-fluorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (2S)-1-[2-[(3R)-3-(2-methoxyphenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C27H33N3O5
ethyl (2S)-1-[2-[(3R)-3-(2-methoxyphenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl N-[3-[(5-chlorothiophen-2-yl)methyl-methylcarbamoyl]phenyl]carbamate —— C16H17ClN2O3S
ethyl N-[3-[(5-chlorothiophen-2-yl)methyl-methylcarbamoyl]phenyl]carbamate
—— ethyl (3R)-1-[2-[(3R)-3-(2-fluorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C25H27F2N3O3
ethyl (3R)-1-[2-[(3R)-3-(2-fluorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (2S)-1-[2-[(3R)-3-(4-chlorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C26H30ClN3O4
ethyl (2S)-1-[2-[(3R)-3-(4-chlorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl (3R)-1-[2-[(3R)-3-(2-fluorophenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C26H30FN3O4
ethyl (3R)-1-[2-[(3R)-3-(2-fluorophenyl)-5-(3-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl 5-amino-4-cyano-3-[[[(1S)-1-(3,4-difluorophenyl)ethyl]amino]methyl]thiophene-2-carboxylate —— C17H17F2N3O2S
ethyl 5-amino-4-cyano-3-[[[(1S)-1-(3,4-difluorophenyl)ethyl]amino]methyl]thiophene-2-carboxylate
—— (E)-N-[4-[[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(3-chlorophenyl)prop-2-enamide —— C24H27ClN2O3S
(E)-N-[4-[[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-(3-chlorophenyl)prop-2-enamide
—— (E)-N-[4-[[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-phenylprop-2-enamide —— C24H28N2O3S
(E)-N-[4-[[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]sulfamoyl]phenyl]-3-phenylprop-2-enamide
—— ethyl (2S)-1-[2-[(3R)-5-(2,4-dimethoxyphenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C28H35N3O5
ethyl (2S)-1-[2-[(3R)-5-(2,4-dimethoxyphenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl 2-[[[(1S)-1-(3,4-difluorophenyl)ethyl]amino]methyl]-4-methylquinoline-3-carboxylate —— C22H22F2N2O2
ethyl 2-[[[(1S)-1-(3,4-difluorophenyl)ethyl]amino]methyl]-4-methylquinoline-3-carboxylate
—— ethyl (2R)-1-[2-[(3R)-3-(4-chlorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate —— C26H30ClN3O4
ethyl (2R)-1-[2-[(3R)-3-(4-chlorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-2-carboxylate
—— ethyl 4-cyclopropyl-2-[[2-[[(1R)-1-(3,4-difluorophenyl)ethyl]amino]acetyl]amino]thiophene-3-carboxylate —— C20H22F2N2O3S
ethyl 4-cyclopropyl-2-[[2-[[(1R)-1-(3,4-difluorophenyl)ethyl]amino]acetyl]amino]thiophene-3-carboxylate
—— ethyl (3S)-1-[2-[(3R)-5-(2-chlorophenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C25H28ClN3O3
ethyl (3S)-1-[2-[(3R)-5-(2-chlorophenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C25H27ClFN3O3
ethyl (3S)-1-[2-[(3R)-3-(2-chlorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[(3R)-5-(2-chlorophenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate —— C25H28ClN3O3
ethyl (3R)-1-[2-[(3R)-5-(2-chlorophenyl)-3-phenyl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]piperidine-3-carboxylate
—— (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide —— C22H23ClN2O4
(E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide
—— ethyl (2S)-1-[2-[2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetyl]oxyacetyl]piperidine-2-carboxylate —— C19H22N2O5S2
ethyl (2S)-1-[2-[2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (2E)-1-ethyl-2-[(2Z)-2-(3-ethyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)ethylidene]-3-(2-phenylethyl)benzimidazole-5-carboxylate —— C27H29N3O3S2
ethyl (2E)-1-ethyl-2-[(2Z)-2-(3-ethyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)ethylidene]-3-(2-phenylethyl)benzimidazole-5-carboxylate
—— ethyl (2R)-1-[2-[2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetyl]oxyacetyl]piperidine-2-carboxylate —— C19H22N2O5S2
ethyl (2R)-1-[2-[2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetyl]oxyacetyl]piperidine-2-carboxylate
—— (E)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C20H19N3O6
(E)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— (E)-N-[(5-chlorothiophen-2-yl)methyl]-3-(3-fluoro-4-methoxyphenyl)-N-methylprop-2-enamide —— C16H15ClFNO2S
(E)-N-[(5-chlorothiophen-2-yl)methyl]-3-(3-fluoro-4-methoxyphenyl)-N-methylprop-2-enamide
—— ethyl 2-[[(3R)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carbonyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C20H22FN3O4S
ethyl 2-[[(3R)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carbonyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— (E)-3-(2-chloro-6-fluorophenyl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide —— C19H18ClFN2O2
(E)-3-(2-chloro-6-fluorophenyl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide
—— Ethyl 1-[1-(furan-2-carbonyl)piperidine-4-carbonyl]piperidine-4-carboxylate —— C19H26N2O5
Ethyl 1-[1-(furan-2-carbonyl)piperidine-4-carbonyl]piperidine-4-carboxylate
—— Ethyl 2-({[1-(furan-2-ylcarbonyl)piperidin-4-yl]carbonyl}amino)benzoate —— C20H22N2O5
Ethyl 2-({[1-(furan-2-ylcarbonyl)piperidin-4-yl]carbonyl}amino)benzoate
—— (E)-3-(4-ethylphenyl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide —— C21H24N2O2
(E)-3-(4-ethylphenyl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide
—— ethyl 2-[[(3S)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carbonyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C20H22FN3O4S
ethyl 2-[[(3S)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carbonyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 1-[(2S)-2-(4-bromo-1H-pyrrole-2-carbonyl)oxypropanoyl]piperidine-4-carboxylate —— C16H21BrN2O5
ethyl 1-[(2S)-2-(4-bromo-1H-pyrrole-2-carbonyl)oxypropanoyl]piperidine-4-carboxylate
—— Ethyl 2,5-dimethyl-1-[2-[methyl-[2-(4-methylanilino)-2-oxoethyl]amino]-2-oxoethyl]pyrrole-3-carboxylate —— C21H27N3O4
Ethyl 2,5-dimethyl-1-[2-[methyl-[2-(4-methylanilino)-2-oxoethyl]amino]-2-oxoethyl]pyrrole-3-carboxylate
—— (E)-3-(2-methoxy-5-methylphenyl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide —— C21H24N2O3
(E)-3-(2-methoxy-5-methylphenyl)-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide
—— ethyl 3-[[(3S)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carbonyl]amino]benzoate —— C22H23FN2O4
ethyl 3-[[(3S)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidine-3-carbonyl]amino]benzoate
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[(S)-furan-2-yl(phenyl)methyl]prop-2-enamide —— C23H22ClNO4
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[(S)-furan-2-yl(phenyl)methyl]prop-2-enamide
—— ethyl N-[3-[[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]carbamoyl]phenyl]carbamate —— C23H25N5O3
ethyl N-[3-[[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]carbamoyl]phenyl]carbamate
—— (E)-2-(4-fluorobenzoyl)-3-(3-fluoro-4-methoxyphenyl)prop-2-enenitrile —— C17H11F2NO2
(E)-2-(4-fluorobenzoyl)-3-(3-fluoro-4-methoxyphenyl)prop-2-enenitrile
—— ethyl N-[4-[[[(2S)-2-(2-fluorophenoxy)propanoyl]amino]carbamoyl]phenyl]carbamate —— C19H20FN3O5
ethyl N-[4-[[[(2S)-2-(2-fluorophenoxy)propanoyl]amino]carbamoyl]phenyl]carbamate
—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[(R)-furan-2-yl(phenyl)methyl]prop-2-enamide —— C23H20N2O4
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-[(R)-furan-2-yl(phenyl)methyl]prop-2-enamide
—— ethyl N-[2-[ethyl-[2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanyl)acetyl]amino]acetyl]carbamate —— C15H19N5O4S
ethyl N-[2-[ethyl-[2-([1,2,4]triazolo[4,3-a]pyridin-3-ylsulfanyl)acetyl]amino]acetyl]carbamate