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—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(2-chlorophenyl)-N-methylprop-2-enamide —— C18H16Cl2N2O2
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(2-chlorophenyl)-N-methylprop-2-enamide
—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methyl-3-(3-methylphenyl)prop-2-enamide —— C19H19ClN2O2
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methyl-3-(3-methylphenyl)prop-2-enamide
—— (E)-3-(5-bromothiophen-2-yl)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methylprop-2-enamide —— C16H14BrClN2O2S
(E)-3-(5-bromothiophen-2-yl)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methylprop-2-enamide
—— (E)-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-[(1R)-1-(4-fluorophenyl)ethyl]prop-2-enamide —— C18H15ClFN3O
(E)-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-[(1R)-1-(4-fluorophenyl)ethyl]prop-2-enamide
—— (E)-N-[(1R)-1-(4-fluorophenyl)ethyl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide —— C18H15F4NO
(E)-N-[(1R)-1-(4-fluorophenyl)ethyl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide
—— ethyl (2S)-2-[[(2R,3S)-2-amino-3-hydroxybutanoyl]amino]-3-(4-hydroxyphenyl)propanoate —— C15H22N2O5
ethyl (2S)-2-[[(2R,3S)-2-amino-3-hydroxybutanoyl]amino]-3-(4-hydroxyphenyl)propanoate
—— (E)-3-(1,3-benzothiazol-2-yl)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methylprop-2-enamide —— C19H16ClN3O2S
(E)-3-(1,3-benzothiazol-2-yl)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methylprop-2-enamide
—— (E)-3-(3-chloro-4-fluorophenyl)-N-[(1R)-1-(4-fluorophenyl)ethyl]prop-2-enamide —— C17H14ClF2NO
(E)-3-(3-chloro-4-fluorophenyl)-N-[(1R)-1-(4-fluorophenyl)ethyl]prop-2-enamide
—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methyl-3-[4-(trifluoromethoxy)phenyl]prop-2-enamide —— C19H16ClF3N2O3
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-N-methyl-3-[4-(trifluoromethoxy)phenyl]prop-2-enamide
—— ethyl (2R)-2-[[(2S,3S)-2-amino-3-hydroxybutanoyl]amino]-3-(4-hydroxyphenyl)propanoate —— C15H22N2O5
ethyl (2R)-2-[[(2S,3S)-2-amino-3-hydroxybutanoyl]amino]-3-(4-hydroxyphenyl)propanoate
—— Ethyl 4-[(6-phenylthieno[2,3-d]pyrimidin-4-yl)hydrazinylidene]piperidine-1-carboxylate —— C20H21N5O2S
Ethyl 4-[(6-phenylthieno[2,3-d]pyrimidin-4-yl)hydrazinylidene]piperidine-1-carboxylate
—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(3-chloro-4-methylphenyl)-N-methylprop-2-enamide —— C19H18Cl2N2O2
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(3-chloro-4-methylphenyl)-N-methylprop-2-enamide
—— ethyl 4-[[(3R)-1-thiophen-2-ylsulfonylpiperidine-3-carbonyl]amino]piperidine-1-carboxylate —— C18H27N3O5S2
ethyl 4-[[(3R)-1-thiophen-2-ylsulfonylpiperidine-3-carbonyl]amino]piperidine-1-carboxylate
—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-methylprop-2-enamide —— C19H16Cl2N4O2
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-methylprop-2-enamide
—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-methylprop-2-enamide —— C21H20ClN3O4
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-methylprop-2-enamide
—— (E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(2,3-dimethoxyphenyl)-N-methylprop-2-enamide —— C20H21ClN2O4
(E)-N-[2-(2-chloroanilino)-2-oxoethyl]-3-(2,3-dimethoxyphenyl)-N-methylprop-2-enamide
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[(1R)-1-(4-fluorophenyl)ethyl]prop-2-enamide —— C19H19ClFNO3
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[(1R)-1-(4-fluorophenyl)ethyl]prop-2-enamide
—— (E)-3-(4-cyanophenyl)-N-methyl-N-[2-(4-morpholin-4-ylanilino)-2-oxoethyl]prop-2-enamide —— C23H24N4O3
(E)-3-(4-cyanophenyl)-N-methyl-N-[2-(4-morpholin-4-ylanilino)-2-oxoethyl]prop-2-enamide
—— (E)-3-(2,3-dimethoxyphenyl)-N-[(2-fluorophenyl)methyl]-N-methylprop-2-enamide —— C19H20FNO3
(E)-3-(2,3-dimethoxyphenyl)-N-[(2-fluorophenyl)methyl]-N-methylprop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(2-fluorophenyl)methyl]-N-methylprop-2-enamide —— C18H16FNO3
(E)-3-(1,3-benzodioxol-5-yl)-N-[(2-fluorophenyl)methyl]-N-methylprop-2-enamide
—— ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O3S
ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5E)-2-anilino-5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methylidene]-4-oxofuran-3-carboxylate —— C22H20BrNO6
ethyl (5E)-2-anilino-5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methylidene]-4-oxofuran-3-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H28FN3O3S
ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2S)-1-[2-[2-(2-methylindol-1-yl)acetyl]oxyacetyl]piperidine-2-carboxylate —— C21H26N2O5
ethyl (2S)-1-[2-[2-(2-methylindol-1-yl)acetyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (5Z)-2-anilino-5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methylidene]-4-oxofuran-3-carboxylate —— C22H20BrNO6
ethyl (5Z)-2-anilino-5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methylidene]-4-oxofuran-3-carboxylate
—— ethyl (3R)-1-[2-[1-(4-methoxyphenyl)tetrazol-5-yl]sulfanylacetyl]piperidine-3-carboxylate —— C18H23N5O4S
ethyl (3R)-1-[2-[1-(4-methoxyphenyl)tetrazol-5-yl]sulfanylacetyl]piperidine-3-carboxylate
—— ethyl (2R)-1-[2-[2-(2-methylindol-1-yl)acetyl]oxyacetyl]piperidine-2-carboxylate —— C21H26N2O5
ethyl (2R)-1-[2-[2-(2-methylindol-1-yl)acetyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (1S,2S,3R,6R,7R,9S)-2-(benzenesulfonyl)-5-oxo-4-oxatricyclo[4.2.1.03,7]nonane-9-carboxylate —— C17H18O6S
ethyl (1S,2S,3R,6R,7R,9S)-2-(benzenesulfonyl)-5-oxo-4-oxatricyclo[4.2.1.03,7]nonane-9-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-methyl-N-[2-(4-morpholin-4-ylanilino)-2-oxoethyl]prop-2-enamide —— C23H27N3O4
(E)-3-(4-methoxyphenyl)-N-methyl-N-[2-(4-morpholin-4-ylanilino)-2-oxoethyl]prop-2-enamide
—— ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H28FN3O3S
ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(2-fluorophenyl)methyl]-N-methylprop-2-enamide —— C19H20FNO3
(E)-3-(3,4-dimethoxyphenyl)-N-[(2-fluorophenyl)methyl]-N-methylprop-2-enamide
—— ethyl (1S,2S,3R,6R,7R,9R)-2-(benzenesulfonyl)-5-oxo-4-oxatricyclo[4.2.1.03,7]nonane-9-carboxylate —— C17H18O6S
ethyl (1S,2S,3R,6R,7R,9R)-2-(benzenesulfonyl)-5-oxo-4-oxatricyclo[4.2.1.03,7]nonane-9-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O3S
ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2,4-dimethyl-5-[(2S)-2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylpropanoyl]-1H-pyrrole-3-carboxylate —— C20H23N5O3S
ethyl 2,4-dimethyl-5-[(2S)-2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylpropanoyl]-1H-pyrrole-3-carboxylate
—— ethyl (3R)-1-[4-[(3-chlorobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32ClN3O5S
ethyl (3R)-1-[4-[(3-chlorobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— Ethyl 5-amino-4-cyano-3-[[1-(4-methylphenyl)tetrazol-5-yl]sulfanylmethyl]thiophene-2-carboxylate —— C17H16N6O2S2
Ethyl 5-amino-4-cyano-3-[[1-(4-methylphenyl)tetrazol-5-yl]sulfanylmethyl]thiophene-2-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[5-[(3R)-1,1-dioxothiolan-3-yl]-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methylquinoline-3-carboxylate —— C21H24N4O4S2
ethyl 2-[[5-[(3R)-1,1-dioxothiolan-3-yl]-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methylquinoline-3-carboxylate
—— ethyl (2S)-1-[2-[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxyacetyl]piperidine-2-carboxylate —— C22H28N2O6
ethyl (2S)-1-[2-[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O3S
ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3S)-1-[4-[(2-methylbenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O5S
ethyl (3S)-1-[4-[(2-methylbenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (2R)-1-[2-[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxyacetyl]piperidine-2-carboxylate —— C22H28N2O6
ethyl (2R)-1-[2-[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H33N3O3S
ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3R)-1-[4-[(3-bromobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32BrN3O5S
ethyl (3R)-1-[4-[(3-bromobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[(2-methylbenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O5S
ethyl (3R)-1-[4-[(2-methylbenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O3S
ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H28FN3O3S
ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate