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—— (E,2S)-2-cyano-5-(2-methyl-1,3-thiazol-4-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide —— C16H21N3O3S
(E,2S)-2-cyano-5-(2-methyl-1,3-thiazol-4-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide
—— (E,2R)-2-cyano-5-(4-fluorophenyl)-N-(3-methoxyphenyl)-3-oxopent-4-enamide —— C19H15FN2O3
(E,2R)-2-cyano-5-(4-fluorophenyl)-N-(3-methoxyphenyl)-3-oxopent-4-enamide
—— (E,2R)-5-(4-chlorophenyl)-2-cyano-N-(3-methoxyphenyl)-3-oxopent-4-enamide —— C19H15ClN2O3
(E,2R)-5-(4-chlorophenyl)-2-cyano-N-(3-methoxyphenyl)-3-oxopent-4-enamide
—— (E,2R)-2-cyano-5-(5-methylfuran-2-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide —— C17H22N2O4
(E,2R)-2-cyano-5-(5-methylfuran-2-yl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide
—— (E,2R)-2-cyano-N-(3-methoxyphenyl)-3-oxo-5-quinolin-8-ylpent-4-enamide —— C22H17N3O3
(E,2R)-2-cyano-N-(3-methoxyphenyl)-3-oxo-5-quinolin-8-ylpent-4-enamide
—— ethyl (3S)-1-[2-[6-(4-methoxyphenyl)-4-oxothieno[3,2-d]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate —— C23H25N3O5S
ethyl (3S)-1-[2-[6-(4-methoxyphenyl)-4-oxothieno[3,2-d]pyrimidin-3-yl]acetyl]piperidine-3-carboxylate
—— (E,2R)-2-cyano-5-(4-fluorophenyl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide —— C18H21FN2O3
(E,2R)-2-cyano-5-(4-fluorophenyl)-3-oxo-N-(3-propan-2-yloxypropyl)pent-4-enamide
—— (E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(4-methylphenyl)prop-2-enamide —— C25H22N2O3
(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(4-methylphenyl)prop-2-enamide
—— (E,2R)-2-cyano-3-oxo-N-(3-propan-2-yloxypropyl)-5-quinolin-8-ylpent-4-enamide —— C21H23N3O3
(E,2R)-2-cyano-3-oxo-N-(3-propan-2-yloxypropyl)-5-quinolin-8-ylpent-4-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-methyl-N-[[4-(trifluoromethyl)phenyl]methyl]prop-2-enamide —— C19H16F3NO3
(E)-3-(1,3-benzodioxol-5-yl)-N-methyl-N-[[4-(trifluoromethyl)phenyl]methyl]prop-2-enamide
—— ethyl (4R)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H28N2O6
ethyl (4R)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-(furan-2-ylmethyl)-N-[2-(2-methoxyanilino)-2-oxoethyl]-3-(3-methylthiophen-2-yl)prop-2-enamide —— C22H22N2O4S
(E)-N-(furan-2-ylmethyl)-N-[2-(2-methoxyanilino)-2-oxoethyl]-3-(3-methylthiophen-2-yl)prop-2-enamide
—— (E)-N-[2-(2,6-dimethylanilino)-2-oxoethyl]-N-methyl-3-(4-nitrophenyl)prop-2-enamide —— C20H21N3O4
(E)-N-[2-(2,6-dimethylanilino)-2-oxoethyl]-N-methyl-3-(4-nitrophenyl)prop-2-enamide
—— (E)-N-methyl-3-(2-nitrophenyl)-N-[[4-(trifluoromethyl)phenyl]methyl]prop-2-enamide —— C18H15F3N2O3
(E)-N-methyl-3-(2-nitrophenyl)-N-[[4-(trifluoromethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(4-methylquinolin-8-yl)prop-2-enamide —— C28H23N3O3
(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(4-methylquinolin-8-yl)prop-2-enamide
—— ethyl 2-[[2-[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C20H25NO5S
ethyl 2-[[2-[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl (4S)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H28N2O6
ethyl (4S)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(2-methoxy-4-nitrophenyl)prop-2-enamide —— C25H21N3O6
(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(2-methoxy-4-nitrophenyl)prop-2-enamide
—— ethyl (4R)-6-[[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H28N2O6
ethyl (4R)-6-[[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[[2-[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C20H25NO5S
ethyl 2-[[2-[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[3-[(Z)-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]iminomethyl]indol-1-yl]acetate —— C22H21N3O4
ethyl 2-[3-[(Z)-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]iminomethyl]indol-1-yl]acetate
—— ethyl (4R)-6-[[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H26N2O5
ethyl (4R)-6-[[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H26N2O5
ethyl (4R)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[[2-[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5-ethylthiophene-3-carboxylate —— C19H25NO5S
ethyl 2-[[2-[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5-ethylthiophene-3-carboxylate
—— ethyl (4S)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H26N2O5
ethyl (4S)-6-[[(1R,2R,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H26N2O5
ethyl (4S)-6-[[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-2-oxo-6-[3-(4-oxo-1,2,3-benzotriazin-3-yl)propanoyloxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H23N5O6
ethyl (4S)-2-oxo-6-[3-(4-oxo-1,2,3-benzotriazin-3-yl)propanoyloxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[3-[(Z)-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]iminomethyl]-2-methylindol-1-yl]acetate —— C23H23N3O4
ethyl 2-[3-[(Z)-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]iminomethyl]-2-methylindol-1-yl]acetate
—— ethyl (4R)-4-(4-methoxyphenyl)-2-oxo-6-[[2-(2-phenyl-1,3-oxazol-4-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H25N3O7
ethyl (4R)-4-(4-methoxyphenyl)-2-oxo-6-[[2-(2-phenyl-1,3-oxazol-4-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-methoxyphenyl)-2-oxo-6-[[2-(2-phenyl-1,3-oxazol-4-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H25N3O7
ethyl (4S)-4-(4-methoxyphenyl)-2-oxo-6-[[2-(2-phenyl-1,3-oxazol-4-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(1S)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]prop-2-enamide —— C19H23NO3
(E)-3-(1,3-benzodioxol-5-yl)-N-[(1S)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]prop-2-enamide
—— ethyl 2-[[2-[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5-ethylthiophene-3-carboxylate —— C19H25NO5S
ethyl 2-[[2-[(1R,2S,4R)-bicyclo[2.2.1]heptane-2-carbonyl]oxyacetyl]amino]-5-ethylthiophene-3-carboxylate
—— ethyl 1-[2-oxo-2-[(3S)-3-phenyl-2,3-dihydro-1,4-benzoxazin-4-yl]ethyl]piperidin-1-ium-4-carboxylate —— C24H29N2O4+
ethyl 1-[2-oxo-2-[(3S)-3-phenyl-2,3-dihydro-1,4-benzoxazin-4-yl]ethyl]piperidin-1-ium-4-carboxylate
—— ethyl 2-[[(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]prop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C27H26N2O5S
ethyl 2-[[(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]prop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(1R)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]prop-2-enamide —— C19H23NO3
(E)-3-(1,3-benzodioxol-5-yl)-N-[(1R)-1-[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]prop-2-enamide
—— (E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(4-methoxyphenyl)prop-2-enamide —— C25H22N2O4
(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(4-methoxyphenyl)prop-2-enamide
—— ethyl 2-chloro-5-[5-[(Z)-[(1R,2R,6R,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]iminomethyl]furan-2-yl]benzoate —— C25H21ClN2O5
ethyl 2-chloro-5-[5-[(Z)-[(1R,2R,6R,7R,8S,10S)-3,5-dioxo-4-azatetracyclo[5.3.2.02,6.08,10]dodec-11-en-4-yl]iminomethyl]furan-2-yl]benzoate
—— ethyl (4R)-6-[[(2S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrrolidin-1-yl]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H31N3O5
ethyl (4R)-6-[[(2S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrrolidin-1-yl]methyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-[2-(difluoromethoxy)-3-methoxyphenyl]-N-[3-(3-methylphenoxy)propyl]prop-2-enamide —— C21H23F2NO4
(E)-3-[2-(difluoromethoxy)-3-methoxyphenyl]-N-[3-(3-methylphenoxy)propyl]prop-2-enamide
—— (E)-N-(4-bromophenyl)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]prop-2-enamide —— C24H19BrN2O3
(E)-N-(4-bromophenyl)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]prop-2-enamide
—— ethyl 1-[2-oxo-2-[(3R)-3-phenyl-2,3-dihydro-1,4-benzoxazin-4-yl]ethyl]piperidin-1-ium-4-carboxylate —— C24H29N2O4+
ethyl 1-[2-oxo-2-[(3R)-3-phenyl-2,3-dihydro-1,4-benzoxazin-4-yl]ethyl]piperidin-1-ium-4-carboxylate
—— ethyl 2-[[2-[(2S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrrolidin-1-yl]acetyl]amino]benzoate —— C24H28N2O5
ethyl 2-[[2-[(2S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrrolidin-1-yl]acetyl]amino]benzoate
—— (E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]prop-2-enoic acid —— C18H15NO4
(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]prop-2-enoic acid
—— ethyl 5-(4-chlorophenyl)-3-[[(2R)-oxolane-2-carbonyl]amino]thiophene-2-carboxylate —— C18H18ClNO4S
ethyl 5-(4-chlorophenyl)-3-[[(2R)-oxolane-2-carbonyl]amino]thiophene-2-carboxylate
—— Ethyl 4-amino-3-nonoxybenzoate —— C18H29NO3
Ethyl 4-amino-3-nonoxybenzoate
—— (E)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(5-methyltetrazol-1-yl)-3-phenylprop-2-enamide —— C20H25N5O
(E)-N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-2-(5-methyltetrazol-1-yl)-3-phenylprop-2-enamide
—— (E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(1,3-thiazol-2-yl)prop-2-enamide —— C21H17N3O3S
(E)-3-[3-[(1R,2R,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]phenyl]-N-(1,3-thiazol-2-yl)prop-2-enamide
—— ethyl 2-[[2-[[(3R)-1,1-dioxothiolan-3-yl]-propylamino]acetyl]amino]-4-phenylthiophene-3-carboxylate —— C22H28N2O5S2
ethyl 2-[[2-[[(3R)-1,1-dioxothiolan-3-yl]-propylamino]acetyl]amino]-4-phenylthiophene-3-carboxylate
—— (E)-3-(1-benzyl-3-pyridin-3-ylpyrazol-4-yl)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]prop-2-en-1-one —— C28H28N6O
(E)-3-(1-benzyl-3-pyridin-3-ylpyrazol-4-yl)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]prop-2-en-1-one
—— ethyl 2-[[2-[(2R)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrrolidin-1-yl]acetyl]amino]benzoate —— C24H28N2O5
ethyl 2-[[2-[(2R)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrrolidin-1-yl]acetyl]amino]benzoate