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—— (E)-N-[(3,5-dimethoxyphenyl)methyl]-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enamide —— C25H29N3O3
(E)-N-[(3,5-dimethoxyphenyl)methyl]-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enamide
—— ethyl 2-[[(3S)-1-(1,3-benzodioxol-5-yl)-5-oxopyrrolidine-3-carbonyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate —— C23H20N2O7S
ethyl 2-[[(3S)-1-(1,3-benzodioxol-5-yl)-5-oxopyrrolidine-3-carbonyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate
—— (E)-3-(1-butyl-5-chloro-3-methylpyrazol-4-yl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C21H28ClN3O3
(E)-3-(1-butyl-5-chloro-3-methylpyrazol-4-yl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— ethyl (5R,6S,7S)-2-ethylsulfanyl-7-hydroxy-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate —— C24H24N4O6S
ethyl (5R,6S,7S)-2-ethylsulfanyl-7-hydroxy-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate
—— (E)-N-cyclopropyl-3-thiophen-2-yl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide —— C19H18F3NOS
(E)-N-cyclopropyl-3-thiophen-2-yl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-cyclopropyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide —— C23H21F3N2O2
(E)-3-[4-(cyanomethoxy)phenyl]-N-cyclopropyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide
—— (E)-N-[(1S)-1-(3-chlorophenyl)ethyl]-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]-N-methylprop-2-enamide —— C23H23ClN2O4S
(E)-N-[(1S)-1-(3-chlorophenyl)ethyl]-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]-N-methylprop-2-enamide
—— (E)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-3-(2-ethoxyphenyl)prop-2-enamide —— C21H25NO4
(E)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-3-(2-ethoxyphenyl)prop-2-enamide
—— ethyl (5R,6R,7S)-7-hydroxy-2-methylsulfanyl-5-(4-nitrophenyl)-4-oxo-7-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate —— C23H22N4O6S
ethyl (5R,6R,7S)-7-hydroxy-2-methylsulfanyl-5-(4-nitrophenyl)-4-oxo-7-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C21H22ClNO5
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-cyclopropyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide —— C23H21F3N2O2
(E)-3-[4-(cyanomethoxy)phenyl]-N-cyclopropyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide
—— ethyl (5S,6S,7S)-2-ethylsulfanyl-7-hydroxy-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate —— C24H24N4O6S
ethyl (5S,6S,7S)-2-ethylsulfanyl-7-hydroxy-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate
—— (E)-3-(1-butyl-5-chloro-3-methylpyrazol-4-yl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C21H28ClN3O3
(E)-3-(1-butyl-5-chloro-3-methylpyrazol-4-yl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-N-[(R)-(4-fluorophenyl)-phenylmethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C20H17FN2OS
(E)-N-[(R)-(4-fluorophenyl)-phenylmethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C21H22ClNO5
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— ethyl (5S,6S,7S)-7-hydroxy-2-methylsulfanyl-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate —— C23H22N4O6S
ethyl (5S,6S,7S)-7-hydroxy-2-methylsulfanyl-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate
—— (E)-N-cyclopropyl-3-thiophen-2-yl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide —— C19H18F3NOS
(E)-N-cyclopropyl-3-thiophen-2-yl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]prop-2-enamide
—— (E)-N-[(1R)-1-(3-chlorophenyl)ethyl]-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]-N-methylprop-2-enamide —— C23H23ClN2O4S
(E)-N-[(1R)-1-(3-chlorophenyl)ethyl]-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]-N-methylprop-2-enamide
—— (E)-N-[(S)-(4-fluorophenyl)-phenylmethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C20H17FN2OS
(E)-N-[(S)-(4-fluorophenyl)-phenylmethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— ethyl (5R,6S,7S)-7-hydroxy-2-methylsulfanyl-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate —— C23H22N4O6S
ethyl (5R,6S,7S)-7-hydroxy-2-methylsulfanyl-5-(4-nitrophenyl)-4-oxo-7-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate
—— ethyl (5R,6R,7S)-2-ethylsulfanyl-7-hydroxy-5-(4-nitrophenyl)-4-oxo-7-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate —— C24H24N4O6S
ethyl (5R,6R,7S)-2-ethylsulfanyl-7-hydroxy-5-(4-nitrophenyl)-4-oxo-7-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carboxylate
—— (E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(3-nitrophenyl)prop-2-enamide —— C20H19ClN2O3
(E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(3-nitrophenyl)prop-2-enamide
—— (E)-N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(3-nitrophenyl)prop-2-enamide —— C20H19ClN2O3
(E)-N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(3-nitrophenyl)prop-2-enamide
—— (E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-[4-(1,1-dioxo-1,2-thiazolidin-2-yl)phenyl]prop-2-enamide —— C23H25ClN2O3S
(E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-[4-(1,1-dioxo-1,2-thiazolidin-2-yl)phenyl]prop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(S)-(4-fluorophenyl)-phenylmethyl]prop-2-enamide —— C24H20FNO3
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(S)-(4-fluorophenyl)-phenylmethyl]prop-2-enamide
—— (E)-N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(2-nitrophenyl)prop-2-enamide —— C20H19ClN2O3
(E)-N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(2-nitrophenyl)prop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(R)-(4-fluorophenyl)-phenylmethyl]prop-2-enamide —— C24H20FNO3
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(R)-(4-fluorophenyl)-phenylmethyl]prop-2-enamide
—— (E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(2-nitrophenyl)prop-2-enamide —— C20H19ClN2O3
(E)-N-[(1R)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-(2-nitrophenyl)prop-2-enamide
—— (E)-N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-[4-(1,1-dioxo-1,2-thiazolidin-2-yl)phenyl]prop-2-enamide —— C23H25ClN2O3S
(E)-N-[(1S)-1-(4-chlorophenyl)ethyl]-N-cyclopropyl-3-[4-(1,1-dioxo-1,2-thiazolidin-2-yl)phenyl]prop-2-enamide
—— (E)-N-[(R)-(4-fluorophenyl)-phenylmethyl]-3-(2-methoxyphenyl)prop-2-enamide —— C23H20FNO2
(E)-N-[(R)-(4-fluorophenyl)-phenylmethyl]-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C22H25F2NO5
(E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-3-(3,4-diethoxyphenyl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C23H29NO5
(E)-3-(3,4-diethoxyphenyl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-N-[(1S)-1-(3-chlorophenyl)ethyl]-3-[4-(methanesulfonamido)phenyl]-N-methylprop-2-enamide —— C19H21ClN2O3S
(E)-N-[(1S)-1-(3-chlorophenyl)ethyl]-3-[4-(methanesulfonamido)phenyl]-N-methylprop-2-enamide
—— (E)-3-(5-bromothiophen-2-yl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C17H18BrNO3S
(E)-3-(5-bromothiophen-2-yl)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-N-[(S)-(4-fluorophenyl)-phenylmethyl]-3-(2-methoxyphenyl)prop-2-enamide —— C23H20FNO2
(E)-N-[(S)-(4-fluorophenyl)-phenylmethyl]-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-3-(5-bromothiophen-2-yl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C17H18BrNO3S
(E)-3-(5-bromothiophen-2-yl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-3-(3,4-diethoxyphenyl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C23H29NO5
(E)-3-(3,4-diethoxyphenyl)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-N-[(1R)-1-(3-chlorophenyl)ethyl]-3-[4-(methanesulfonamido)phenyl]-N-methylprop-2-enamide —— C19H21ClN2O3S
(E)-N-[(1R)-1-(3-chlorophenyl)ethyl]-3-[4-(methanesulfonamido)phenyl]-N-methylprop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide —— C22H25F2NO5
(E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-N-[(1S)-1-(3-chlorophenyl)ethyl]-N-methyl-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C22H23ClN2O2
(E)-N-[(1S)-1-(3-chlorophenyl)ethyl]-N-methyl-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-N-ethyl-N-[(1R)-1-(3-methoxyphenyl)ethyl]-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enamide —— C24H29NO4
(E)-N-ethyl-N-[(1R)-1-(3-methoxyphenyl)ethyl]-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enamide
—— (E)-N-[(1R)-1-(3-chlorophenyl)ethyl]-N-methyl-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C22H23ClN2O2
(E)-N-[(1R)-1-(3-chlorophenyl)ethyl]-N-methyl-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-N-cyclopropyl-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]prop-2-enamide —— C29H32N2O4
(E)-N-cyclopropyl-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]prop-2-enamide
—— (E)-N-[(1S)-1-(3-chlorophenyl)propyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide —— C20H23ClN2O4S
(E)-N-[(1S)-1-(3-chlorophenyl)propyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide
—— (E)-N-[(1R)-1-(3-chlorophenyl)propyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide —— C20H23ClN2O4S
(E)-N-[(1R)-1-(3-chlorophenyl)propyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide
—— (E)-3-(2-bromophenyl)-N-[(1S)-1-(4-cyanophenyl)ethyl]-N-ethylprop-2-enamide —— C20H19BrN2O
(E)-3-(2-bromophenyl)-N-[(1S)-1-(4-cyanophenyl)ethyl]-N-ethylprop-2-enamide
—— (E)-N-cyclopropyl-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]prop-2-enamide —— C29H32N2O4
(E)-N-cyclopropyl-3-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methoxy]-3-methoxyphenyl]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]prop-2-enamide
—— (E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(1S)-1-(3-chlorophenyl)ethyl]-N-methylprop-2-enamide —— C23H22ClN3O2S
(E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(1S)-1-(3-chlorophenyl)ethyl]-N-methylprop-2-enamide
—— (E)-3-(2-bromophenyl)-N-[(1R)-1-(4-cyanophenyl)ethyl]-N-ethylprop-2-enamide —— C20H19BrN2O
(E)-3-(2-bromophenyl)-N-[(1R)-1-(4-cyanophenyl)ethyl]-N-ethylprop-2-enamide
—— (E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-(2,4-dimethylphenyl)-N-ethylprop-2-enamide —— C24H24FN3O2S
(E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-(2,4-dimethylphenyl)-N-ethylprop-2-enamide