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—— (E)-3-[3-(1-benzofuran-2-yl)-1-benzylpyrazol-4-yl]-2-cyanoprop-2-enamide —— C22H16N4O2
(E)-3-[3-(1-benzofuran-2-yl)-1-benzylpyrazol-4-yl]-2-cyanoprop-2-enamide
—— ethyl 1-[(6-nitro-4H-1,3-benzodioxin-8-yl)methyl]piperidine-4-carboxylate —— C17H22N2O6
ethyl 1-[(6-nitro-4H-1,3-benzodioxin-8-yl)methyl]piperidine-4-carboxylate
—— (E)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C20H22N4O
(E)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-N-benzyl-2-cyano-3-hydroxy-4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)oxybut-2-enamide —— C24H18N4O3S
(E)-N-benzyl-2-cyano-3-hydroxy-4-(5-phenylthieno[2,3-d]pyrimidin-4-yl)oxybut-2-enamide
—— Ethyl 4-[[2-[furan-2-ylmethyl(methyl)amino]acetyl]amino]benzoate —— C17H20N2O4
Ethyl 4-[[2-[furan-2-ylmethyl(methyl)amino]acetyl]amino]benzoate
—— ethyl 2-[(E)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]ethenyl]-5-nitropyridine-3-carboxylate —— C21H19FN4O4
ethyl 2-[(E)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]ethenyl]-5-nitropyridine-3-carboxylate
—— (E)-2-cyano-3-(3-fluoro-4-methoxyphenyl)-N-[(1R,2R)-2-methylcyclohexyl]prop-2-enamide —— C18H21FN2O2
(E)-2-cyano-3-(3-fluoro-4-methoxyphenyl)-N-[(1R,2R)-2-methylcyclohexyl]prop-2-enamide
—— (E)-2-cyano-3-(3-fluoro-4-methoxyphenyl)-N-(2-methylphenyl)prop-2-enamide —— C18H15FN2O2
(E)-2-cyano-3-(3-fluoro-4-methoxyphenyl)-N-(2-methylphenyl)prop-2-enamide
—— (E)-3-[1-benzyl-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrazol-4-yl]-2-cyanoprop-2-enoate —— C23H18N3O4-
(E)-3-[1-benzyl-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyrazol-4-yl]-2-cyanoprop-2-enoate
—— (E)-N-benzyl-2-cyano-4-(4,5-dichloro-6-oxopyridazin-1-yl)-3-hydroxybut-2-enamide —— C16H12Cl2N4O3
(E)-N-benzyl-2-cyano-4-(4,5-dichloro-6-oxopyridazin-1-yl)-3-hydroxybut-2-enamide
—— Ethyl 2-[[2-[furan-2-ylmethyl(methyl)amino]acetyl]amino]-5-methyl-4-phenylthiophene-3-carboxylate —— C22H24N2O4S
Ethyl 2-[[2-[furan-2-ylmethyl(methyl)amino]acetyl]amino]-5-methyl-4-phenylthiophene-3-carboxylate
—— ethyl (4S)-6-[[[(1R)-1-(3,4-difluorophenyl)ethyl]-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H23F2N3O3
ethyl (4S)-6-[[[(1R)-1-(3,4-difluorophenyl)ethyl]-methylamino]methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl N-[4-[[(3R)-3-carbamoyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-2-oxochromen-7-yl]carbamate —— C23H23N3O5
ethyl N-[4-[[(3R)-3-carbamoyl-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-2-oxochromen-7-yl]carbamate
—— ethyl (3S)-1-[2-[prop-2-enyl(thiophen-2-ylmethyl)amino]acetyl]piperidine-3-carboxylate —— C18H26N2O3S
ethyl (3S)-1-[2-[prop-2-enyl(thiophen-2-ylmethyl)amino]acetyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[prop-2-enyl(thiophen-2-ylmethyl)amino]acetyl]piperidine-3-carboxylate —— C18H26N2O3S
ethyl (3R)-1-[2-[prop-2-enyl(thiophen-2-ylmethyl)amino]acetyl]piperidine-3-carboxylate
—— (E)-N-benzyl-4-(4-chloro-3-methylphenoxy)-2-cyano-3-hydroxybut-2-enamide —— C19H17ClN2O3
(E)-N-benzyl-4-(4-chloro-3-methylphenoxy)-2-cyano-3-hydroxybut-2-enamide
—— ethyl 2-[[2-[(3R)-3-carbamoyl-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]amino]-5-ethylthiophene-3-carboxylate —— C21H25N3O4S
ethyl 2-[[2-[(3R)-3-carbamoyl-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]amino]-5-ethylthiophene-3-carboxylate
—— ethyl 2-[[2-[(3R)-3-carbamoyl-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]amino]-4-(2-methylpropyl)thiophene-3-carboxylate —— C23H29N3O4S
ethyl 2-[[2-[(3R)-3-carbamoyl-3,4-dihydro-1H-isoquinolin-2-yl]acetyl]amino]-4-(2-methylpropyl)thiophene-3-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(2,5-dimethoxyphenyl)prop-2-enamide —— C20H21N3O3
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(2,5-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C19H16F3N3O
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-quinoxalin-2-ylprop-2-enoate —— C17H14N4O3
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-quinoxalin-2-ylprop-2-enoate
—— (E)-N-[(1R,5R)-8-azabicyclo[3.2.1]octan-3-yl]but-2-enamide —— C11H18N2O
(E)-N-[(1R,5R)-8-azabicyclo[3.2.1]octan-3-yl]but-2-enamide
—— (E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide —— C26H22N6O
(E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-[5-chloro-1-[(2-chlorophenyl)methyl]-3-methylpyrazol-4-yl]prop-2-enoate —— C20H18Cl2N4O3
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-[5-chloro-1-[(2-chlorophenyl)methyl]-3-methylpyrazol-4-yl]prop-2-enoate
—— Ethyl 1-[[3-(2,5-dimethylphenyl)-2-sulfanylideneimidazol-1-yl]methyl]piperidin-1-ium-4-carboxylate —— C20H28N3O2S+
Ethyl 1-[[3-(2,5-dimethylphenyl)-2-sulfanylideneimidazol-1-yl]methyl]piperidin-1-ium-4-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide —— C26H22N6O
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(1R,5R)-8-azabicyclo[3.2.1]octan-3-yl]-N-methylbut-2-enamide —— C12H20N2O
(E)-N-[(1R,5R)-8-azabicyclo[3.2.1]octan-3-yl]-N-methylbut-2-enamide
—— (E)-N-[(1S,5S)-8-azabicyclo[3.2.1]octan-3-yl]but-2-enamide —— C11H18N2O
(E)-N-[(1S,5S)-8-azabicyclo[3.2.1]octan-3-yl]but-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate —— C20H20N4O3
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoate
—— ethyl 5-[[(1S)-1-(1H-benzimidazol-2-yl)ethyl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C19H22N4O3
ethyl 5-[[(1S)-1-(1H-benzimidazol-2-yl)ethyl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide —— C20H21N3O3
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide
—— (E)-4-[(5-anilino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-benzyl-2-cyano-3-hydroxybut-2-enamide —— C20H17N5O2S2
(E)-4-[(5-anilino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-benzyl-2-cyano-3-hydroxybut-2-enamide
—— (E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C19H16F3N3O
(E)-N-[(1S)-1-(1H-benzimidazol-2-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)prop-2-enoate —— C20H19ClN4O3
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (Z)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)prop-2-enoate
—— ethyl (E)-3-[4-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]phenyl]prop-2-enoate —— C20H25NO3
ethyl (E)-3-[4-[[2-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]phenyl]prop-2-enoate
—— ethyl 5-[[(1R)-1-(1H-benzimidazol-2-yl)ethyl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C19H22N4O3
ethyl 5-[[(1R)-1-(1H-benzimidazol-2-yl)ethyl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 1-[(2R)-2-[3-(4-fluorophenyl)propanoyloxy]propanoyl]piperidine-4-carboxylate —— C20H26FNO5
ethyl 1-[(2R)-2-[3-(4-fluorophenyl)propanoyloxy]propanoyl]piperidine-4-carboxylate
—— ethyl (4S)-6-[[(3S)-3-benzamidobutanoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H27N3O6
ethyl (4S)-6-[[(3S)-3-benzamidobutanoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 1-[(2S)-2-[3-(4-fluorophenyl)propanoyloxy]propanoyl]piperidine-4-carboxylate —— C20H26FNO5
ethyl 1-[(2S)-2-[3-(4-fluorophenyl)propanoyloxy]propanoyl]piperidine-4-carboxylate
—— ethyl (4S)-6-[[(3R)-3-benzamidobutanoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H27N3O6
ethyl (4S)-6-[[(3R)-3-benzamidobutanoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(3S)-3-benzamidobutanoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H27N3O6
ethyl (4R)-6-[[(3S)-3-benzamidobutanoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 1-[(2R)-2-[4-[(2,5-dioxopyrrolidin-1-yl)methyl]benzoyl]oxypropanoyl]piperidine-4-carboxylate —— C23H28N2O7
ethyl 1-[(2R)-2-[4-[(2,5-dioxopyrrolidin-1-yl)methyl]benzoyl]oxypropanoyl]piperidine-4-carboxylate
—— ethyl (4S)-6-[[4-[(2,5-dioxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H25N3O7
ethyl (4S)-6-[[4-[(2,5-dioxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 1-[(2S)-2-[3-(2-ethoxyphenyl)propanoyloxy]propanoyl]piperidine-4-carboxylate —— C22H31NO6
ethyl 1-[(2S)-2-[3-(2-ethoxyphenyl)propanoyloxy]propanoyl]piperidine-4-carboxylate
—— (E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(3,4-dichlorophenyl)prop-2-enamide —— C18H15Cl2N3O
(E)-N-[(1R)-1-(1H-benzimidazol-2-yl)ethyl]-3-(3,4-dichlorophenyl)prop-2-enamide
—— ethyl (4S)-2-oxo-6-[3-(2-oxo-1,3-benzoxazol-3-yl)propanoyloxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H23N3O7
ethyl (4S)-2-oxo-6-[3-(2-oxo-1,3-benzoxazol-3-yl)propanoyloxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-2-oxo-6-[3-(2-oxo-1,3-benzoxazol-3-yl)propanoyloxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H23N3O7
ethyl (4R)-2-oxo-6-[3-(2-oxo-1,3-benzoxazol-3-yl)propanoyloxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (E)-3-[4-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]phenyl]prop-2-enoate —— C20H25NO3
ethyl (E)-3-[4-[[2-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]acetyl]amino]phenyl]prop-2-enoate
—— ethyl N-[4-[[4-(dimethylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate —— C18H21N3O5S
ethyl N-[4-[[4-(dimethylsulfamoyl)phenyl]carbamoyl]phenyl]carbamate
—— ethyl (4R)-6-[[4-[(2,5-dioxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H25N3O7
ethyl (4R)-6-[[4-[(2,5-dioxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate