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—— ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H33N3O3S
ethyl (5R)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3S)-1-[4-[(2-phenoxyacetyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O6S
ethyl (3S)-1-[4-[(2-phenoxyacetyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (4S)-2-oxo-6-[[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H27N3O6
ethyl (4S)-2-oxo-6-[[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H28FN3O3S
ethyl (5R)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2-fluorophenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3S)-1-[4-[(3-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O6S
ethyl (3S)-1-[4-[(3-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(2,2-dimethylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C27H37N3O5S
ethyl (3R)-1-[4-(2,2-dimethylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-(cyclopentanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C28H37N3O5S
ethyl (3S)-1-[4-(cyclopentanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl 2,5-dimethyl-4-[2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylacetyl]-1H-pyrrole-3-carboxylate —— C19H21N5O3S
ethyl 2,5-dimethyl-4-[2-[1-(4-methylphenyl)tetrazol-5-yl]sulfanylacetyl]-1H-pyrrole-3-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H33N3O3S
ethyl (5S)-3-[2-[[(1S,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3S)-1-[4-[(2,2-dichloroacetyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C24H29Cl2N3O5S
ethyl (3S)-1-[4-[(2,2-dichloroacetyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H33N3O3S
ethyl (5S)-3-[2-[[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(2,4-dimethylphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3R)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-(3-phenylpropanoylamino)phenyl]piperidine-3-carboxylate —— C31H37N3O5S
ethyl (3R)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-(3-phenylpropanoylamino)phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(1,3-benzodioxole-5-carbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H33N3O7S
ethyl (3R)-1-[4-(1,3-benzodioxole-5-carbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(4-chlorophenoxy)acetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H34ClN3O6S
ethyl (3S)-1-[4-[[2-(4-chlorophenoxy)acetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate —— C31H37N3O6S
ethyl (3R)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-(3-phenylpropanoylamino)phenyl]piperidine-3-carboxylate —— C31H37N3O5S
ethyl (3S)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-(3-phenylpropanoylamino)phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate —— C31H37N3O6S
ethyl (3S)-1-[2-[[(1R)-1-phenylethyl]sulfamoyl]-4-[(2-phenylmethoxyacetyl)amino]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(cyclopropanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C26H33N3O5S
ethyl (3R)-1-[4-(cyclopropanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (4R)-2-oxo-6-[[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H27N3O6
ethyl (4R)-2-oxo-6-[[3-[(2-oxopyrrolidin-1-yl)methyl]benzoyl]oxymethyl]-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (3S)-1-[4-[(2-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O6S
ethyl (3S)-1-[4-[(2-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (2R)-1-[2-[3-(3-fluoro-4-methylphenyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-2-carboxylate —— C25H26FN3O4S
ethyl (2R)-1-[2-[3-(3-fluoro-4-methylphenyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-2-carboxylate
—— ethyl 4-methyl-2-[[(3S)-1-(phenylcarbamoyl)piperidine-3-carbonyl]oxymethyl]quinoline-3-carboxylate —— C27H29N3O5
ethyl 4-methyl-2-[[(3S)-1-(phenylcarbamoyl)piperidine-3-carbonyl]oxymethyl]quinoline-3-carboxylate
—— ethyl (3R)-1-[4-(3-cyclopentylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H41N3O5S
ethyl (3R)-1-[4-(3-cyclopentylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(cyclopentanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C28H37N3O5S
ethyl (3R)-1-[4-(cyclopentanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[(2-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O6S
ethyl (3R)-1-[4-[(2-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— (E)-N-[(1S)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methyl-3-(2-nitrophenyl)prop-2-enamide —— C19H17N3O3S
(E)-N-[(1S)-1-(1,3-benzothiazol-2-yl)ethyl]-N-methyl-3-(2-nitrophenyl)prop-2-enamide
—— ethyl (3S)-1-[4-(2-methylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C26H35N3O5S
ethyl (3S)-1-[4-(2-methylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[(3-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H35N3O6S
ethyl (3R)-1-[4-[(3-methoxybenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-(3-cyclopentylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H41N3O5S
ethyl (3S)-1-[4-(3-cyclopentylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(4-methoxyphenyl)acetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C31H37N3O6S
ethyl (3S)-1-[4-[[2-(4-methoxyphenyl)acetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(cyclobutanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C27H35N3O5S
ethyl (3R)-1-[4-(cyclobutanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (2S)-1-[2-[3-(3-fluoro-4-methylphenyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-2-carboxylate —— C25H26FN3O4S
ethyl (2S)-1-[2-[3-(3-fluoro-4-methylphenyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]piperidine-2-carboxylate
—— (E)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-3-thiophen-2-ylprop-2-enamide —— C17H16ClNO3S
(E)-N-[(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl]-3-thiophen-2-ylprop-2-enamide
—— ethyl (3S)-1-[4-(cyclopropanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C26H33N3O5S
ethyl (3S)-1-[4-(cyclopropanecarbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl 1-[2-[(3S)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]oxyacetyl]piperidine-4-carboxylate —— C19H23NO7
ethyl 1-[2-[(3S)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]oxyacetyl]piperidine-4-carboxylate
—— ethyl (3R)-1-[4-[[(2R)-2-chloro-2-phenylacetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H34ClN3O5S
ethyl (3R)-1-[4-[[(2R)-2-chloro-2-phenylacetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[(3-bromobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32BrN3O5S
ethyl (3S)-1-[4-[(3-bromobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[(2-fluorobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32FN3O5S
ethyl (3S)-1-[4-[(2-fluorobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[(4-bromobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C29H32BrN3O5S
ethyl (3R)-1-[4-[(4-bromobenzoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-(2-methylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C26H35N3O5S
ethyl (3R)-1-[4-(2-methylpropanoylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[(2R)-2-chloro-2-phenylacetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H34ClN3O5S
ethyl (3S)-1-[4-[[(2R)-2-chloro-2-phenylacetyl]amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[(3-chloro-2,2-dimethylpropanoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C27H36ClN3O5S
ethyl (3S)-1-[4-[(3-chloro-2,2-dimethylpropanoyl)amino]-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— (E)-3-(1,3-diphenylpyrazol-4-yl)-N-[3-(4-methylpiperazine-1,4-diium-1-yl)propyl]prop-2-enamide —— C26H33N5O+2
(E)-3-(1,3-diphenylpyrazol-4-yl)-N-[3-(4-methylpiperazine-1,4-diium-1-yl)propyl]prop-2-enamide
—— ethyl (3S)-1-[4-(1,3-benzodioxole-5-carbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate —— C30H33N3O7S
ethyl (3S)-1-[4-(1,3-benzodioxole-5-carbonylamino)-2-[[(1R)-1-phenylethyl]sulfamoyl]phenyl]piperidine-3-carboxylate
—— ethyl (2S)-1-[2-[4-chloro-2-(2-oxopyrrolidin-1-yl)benzoyl]oxyacetyl]piperidine-2-carboxylate —— C21H25ClN2O6
ethyl (2S)-1-[2-[4-chloro-2-(2-oxopyrrolidin-1-yl)benzoyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (4S)-6-[[(3S)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]oxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H22N2O7
ethyl (4S)-6-[[(3S)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]oxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[(3S)-1,1-dioxothiolane-3-carbonyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H20N2O7S
ethyl (4S)-6-[[(3S)-1,1-dioxothiolane-3-carbonyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(3R)-1,1-dioxothiolane-3-carbonyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H20N2O7S
ethyl (4R)-6-[[(3R)-1,1-dioxothiolane-3-carbonyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[(3R)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]oxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H22N2O7
ethyl (4S)-6-[[(3R)-2,3-dihydro-1,4-benzodioxine-3-carbonyl]oxymethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[[(2R)-2-[(3R)-1,1-dioxothiolane-3-carbonyl]oxypropanoyl]amino]-4-phenylthiophene-3-carboxylate —— C21H23NO7S2
ethyl 2-[[(2R)-2-[(3R)-1,1-dioxothiolane-3-carbonyl]oxypropanoyl]amino]-4-phenylthiophene-3-carboxylate