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—— (E)-N-[2-(2-amino-2-oxoethyl)phenyl]-3-[3-ethoxy-4-(2-phenoxyethoxy)phenyl]prop-2-enamide —— C27H28N2O5
(E)-N-[2-(2-amino-2-oxoethyl)phenyl]-3-[3-ethoxy-4-(2-phenoxyethoxy)phenyl]prop-2-enamide
—— ethyl (4S)-2-oxo-4-phenyl-6-[[(2S)-1-pyrimidin-2-ylpiperidine-2-carbonyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H27N5O5
ethyl (4S)-2-oxo-4-phenyl-6-[[(2S)-1-pyrimidin-2-ylpiperidine-2-carbonyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-methoxyphenyl)-2-oxo-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H22N4O6
ethyl (4S)-4-(4-methoxyphenyl)-2-oxo-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H29N3O5
ethyl (4S)-6-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-2-oxo-4-phenyl-6-[[(2R)-1-pyrimidin-2-ylpiperidine-2-carbonyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H27N5O5
ethyl (4S)-2-oxo-4-phenyl-6-[[(2R)-1-pyrimidin-2-ylpiperidine-2-carbonyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(E)-[(E)-3-(1-benzyltriazol-4-yl)prop-2-enylidene]amino]urea —— C13H14N6O
[(E)-[(E)-3-(1-benzyltriazol-4-yl)prop-2-enylidene]amino]urea
—— ethyl (4R)-6-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H29N3O5
ethyl (4R)-6-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-methoxyphenyl)-2-oxo-6-[[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H30N4O4
ethyl (4S)-4-(4-methoxyphenyl)-2-oxo-6-[[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(2-imidazol-1-ylphenyl)prop-2-enamide —— C20H16ClN3O3
(E)-3-(5-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(2-imidazol-1-ylphenyl)prop-2-enamide
—— (E)-3-[5-(4-fluorophenyl)thiophen-2-yl]-N-[(6-pyrrolidin-1-ylpyridin-3-yl)methyl]prop-2-enamide —— C23H22FN3OS
(E)-3-[5-(4-fluorophenyl)thiophen-2-yl]-N-[(6-pyrrolidin-1-ylpyridin-3-yl)methyl]prop-2-enamide
—— ethyl 6-[4-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]piperazin-1-yl]pyridine-3-carboxylate —— C22H27N3O3S
ethyl 6-[4-[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl 6-[4-[(4S)-3-benzoyl-1,3-thiazolidine-4-carbonyl]piperazin-1-yl]pyridine-3-carboxylate —— C23H26N4O4S
ethyl 6-[4-[(4S)-3-benzoyl-1,3-thiazolidine-4-carbonyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl 6-[4-[(Z)-2-cyano-3-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]prop-2-enoyl]piperazin-1-yl]pyridine-3-carboxylate —— C26H33N5O4
ethyl 6-[4-[(Z)-2-cyano-3-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]prop-2-enoyl]piperazin-1-yl]pyridine-3-carboxylate
—— (E)-3-[3-ethoxy-4-(2-phenoxyethoxy)phenyl]-N-[(6-pyrrolidin-1-ylpyridin-3-yl)methyl]prop-2-enamide —— C29H33N3O4
(E)-3-[3-ethoxy-4-(2-phenoxyethoxy)phenyl]-N-[(6-pyrrolidin-1-ylpyridin-3-yl)methyl]prop-2-enamide
—— ethyl (4S)-6-[[4-(3,4-difluorobenzoyl)piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H26F2N4O4
ethyl (4S)-6-[[4-(3,4-difluorobenzoyl)piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 6-[4-[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]piperazin-1-yl]pyridine-3-carboxylate —— C22H27N3O3S
ethyl 6-[4-[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl 6-[4-[(3R)-3-acetamido-3-(4-chlorophenyl)propanoyl]piperazin-1-yl]pyridine-3-carboxylate —— C23H27ClN4O4
ethyl 6-[4-[(3R)-3-acetamido-3-(4-chlorophenyl)propanoyl]piperazin-1-yl]pyridine-3-carboxylate
—— (E)-3-[3-ethoxy-4-(2-phenoxyethoxy)phenyl]-N-(3-pyrazol-1-ylpropyl)prop-2-enamide —— C25H29N3O4
(E)-3-[3-ethoxy-4-(2-phenoxyethoxy)phenyl]-N-(3-pyrazol-1-ylpropyl)prop-2-enamide
—— ethyl 6-[4-[(3R)-2-(furan-2-carbonyl)-3,4-dihydro-1H-isoquinoline-3-carbonyl]piperazin-1-yl]pyridine-3-carboxylate —— C27H28N4O5
ethyl 6-[4-[(3R)-2-(furan-2-carbonyl)-3,4-dihydro-1H-isoquinoline-3-carbonyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl (3R)-1-[(2R)-1-methoxy-1-oxopropan-2-yl]piperidine-3-carboxylate —— C12H21NO4
ethyl (3R)-1-[(2R)-1-methoxy-1-oxopropan-2-yl]piperidine-3-carboxylate
—— ethyl 6-[4-[(Z)-2-cyano-3-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]prop-2-enoyl]piperazin-1-yl]pyridine-3-carboxylate —— C26H33N5O4
ethyl 6-[4-[(Z)-2-cyano-3-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]prop-2-enoyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl 6-[4-[(3S)-2-(furan-2-carbonyl)-3,4-dihydro-1H-isoquinoline-3-carbonyl]piperazin-1-yl]pyridine-3-carboxylate —— C27H28N4O5
ethyl 6-[4-[(3S)-2-(furan-2-carbonyl)-3,4-dihydro-1H-isoquinoline-3-carbonyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl (3S)-1-[(2R)-2-[4-[[4-(trifluoromethoxy)phenyl]methyl]piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C23H32F3N3O4
ethyl (3S)-1-[(2R)-2-[4-[[4-(trifluoromethoxy)phenyl]methyl]piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[(2R)-2-[4-[[4-(trifluoromethoxy)phenyl]methyl]piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C23H32F3N3O4
ethyl (3R)-1-[(2R)-2-[4-[[4-(trifluoromethoxy)phenyl]methyl]piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— ethyl 6-[4-[(4R)-3-benzoyl-1,3-thiazolidine-4-carbonyl]piperazin-1-yl]pyridine-3-carboxylate —— C23H26N4O4S
ethyl 6-[4-[(4R)-3-benzoyl-1,3-thiazolidine-4-carbonyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl (3R)-1-[(2R)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C22H29F2N3O4
ethyl (3R)-1-[(2R)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— ethyl 6-[4-[(3S)-3-acetamido-3-(4-chlorophenyl)propanoyl]piperazin-1-yl]pyridine-3-carboxylate —— C23H27ClN4O4
ethyl 6-[4-[(3S)-3-acetamido-3-(4-chlorophenyl)propanoyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl (3S)-1-[(2R)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C22H29F2N3O4
ethyl (3S)-1-[(2R)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— ethyl (2R)-1-[2-[cyclopropyl-[(4-methylphenyl)methyl]amino]acetyl]piperidine-2-carboxylate —— C21H30N2O3
ethyl (2R)-1-[2-[cyclopropyl-[(4-methylphenyl)methyl]amino]acetyl]piperidine-2-carboxylate
—— ethyl (3S)-1-[(2S)-2-[4-[[4-(trifluoromethoxy)phenyl]methyl]piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C23H32F3N3O4
ethyl (3S)-1-[(2S)-2-[4-[[4-(trifluoromethoxy)phenyl]methyl]piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— ethyl (2S)-1-[2-[cyclopropyl-[(4-methylphenyl)methyl]amino]acetyl]piperidine-2-carboxylate —— C21H30N2O3
ethyl (2S)-1-[2-[cyclopropyl-[(4-methylphenyl)methyl]amino]acetyl]piperidine-2-carboxylate
—— ethyl (4R)-6-[[4-(3,4-difluorobenzoyl)piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H26F2N4O4
ethyl (4R)-6-[[4-(3,4-difluorobenzoyl)piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (3S)-1-[(2S)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C22H29F2N3O4
ethyl (3S)-1-[(2S)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[(2S)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate —— C22H29F2N3O4
ethyl (3R)-1-[(2S)-2-[4-(3,4-difluorobenzoyl)piperazin-1-yl]propanoyl]piperidine-3-carboxylate
—— [(E)-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)methylideneamino]urea —— C12H16ClN3O3
[(E)-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)methylideneamino]urea
—— [(E)-1-(4-bromophenyl)propylideneamino]urea —— C10H12BrN3O
[(E)-1-(4-bromophenyl)propylideneamino]urea
—— ethyl 2-[[(2R)-2-(2-cyanophenoxy)propanoyl]amino]-4-phenyl-1,3-thiazole-5-carboxylate —— C22H19N3O4S
ethyl 2-[[(2R)-2-(2-cyanophenoxy)propanoyl]amino]-4-phenyl-1,3-thiazole-5-carboxylate
—— [(E)-1,1-diphenylpropan-2-ylideneamino]urea —— C16H17N3O
[(E)-1,1-diphenylpropan-2-ylideneamino]urea
—— ethyl (3S)-1-[(2R)-1-[[(2S)-2-cyano-3-methylbutan-2-yl]amino]-1-oxopropan-2-yl]piperidine-3-carboxylate —— C17H29N3O3
ethyl (3S)-1-[(2R)-1-[[(2S)-2-cyano-3-methylbutan-2-yl]amino]-1-oxopropan-2-yl]piperidine-3-carboxylate
—— ethyl (1R,6S)-4-[(Z)-2-[4-(dimethylamino)phenyl]ethenyl]-2-oxo-6-phenylcyclohex-3-ene-1-carboxylate —— C25H27NO3
ethyl (1R,6S)-4-[(Z)-2-[4-(dimethylamino)phenyl]ethenyl]-2-oxo-6-phenylcyclohex-3-ene-1-carboxylate
—— ethyl (3R)-1-[(2R)-1-[[(2S)-2-cyano-3-methylbutan-2-yl]amino]-1-oxopropan-2-yl]piperidine-3-carboxylate —— C17H29N3O3
ethyl (3R)-1-[(2R)-1-[[(2S)-2-cyano-3-methylbutan-2-yl]amino]-1-oxopropan-2-yl]piperidine-3-carboxylate
—— ethyl (1S,6S)-4-[(Z)-2-[4-(dimethylamino)phenyl]ethenyl]-2-oxo-6-phenylcyclohex-3-ene-1-carboxylate —— C25H27NO3
ethyl (1S,6S)-4-[(Z)-2-[4-(dimethylamino)phenyl]ethenyl]-2-oxo-6-phenylcyclohex-3-ene-1-carboxylate
—— (E)-1-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine —— C11H13ClN6O2S
(E)-1-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine
—— (E)-1-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine —— C13H10ClFN6
(E)-1-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine
—— (E)-1-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine —— C11H15ClN6
(E)-1-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-(1,2,4-triazol-4-yl)methanimine
—— (E)-N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C17H23NO2
(E)-N-[(1S)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— (E)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C24H27N3O3
(E)-N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl 2-[[(3R)-1-(1,3-benzodioxol-5-yl)-5-oxopyrrolidine-3-carbonyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate —— C23H20N2O7S
ethyl 2-[[(3R)-1-(1,3-benzodioxol-5-yl)-5-oxopyrrolidine-3-carbonyl]amino]-4-(furan-2-yl)thiophene-3-carboxylate
—— (E)-N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C17H23NO2
(E)-N-[(1R)-1-[(1S,2R,4S)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— (E)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C24H27N3O3
(E)-N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide