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—— (E)-N-[[(2S)-1-benzylpiperidin-2-yl]methyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide —— C26H33N3O2
(E)-N-[[(2S)-1-benzylpiperidin-2-yl]methyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide
—— (E)-N-[(R)-cyano-(2,3-dichlorophenyl)methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C22H18Cl2N4O
(E)-N-[(R)-cyano-(2,3-dichlorophenyl)methyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(2R)-1-(1,1-dioxo-1,4-thiazinan-4-yl)-1-oxopropan-2-yl]-3-(3-phenylphenyl)prop-2-enamide —— C22H24N2O4S
(E)-N-[(2R)-1-(1,1-dioxo-1,4-thiazinan-4-yl)-1-oxopropan-2-yl]-3-(3-phenylphenyl)prop-2-enamide
—— (E)-N-[2-[(2R)-1-cyanopropan-2-yl]sulfanylphenyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C24H24N4OS
(E)-N-[2-[(2R)-1-cyanopropan-2-yl]sulfanylphenyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-3-(4-morpholin-4-ylphenyl)-N-[(1R)-1-[3-(2-oxopyrrolidin-1-yl)phenyl]ethyl]prop-2-enamide —— C25H29N3O3
(E)-3-(4-morpholin-4-ylphenyl)-N-[(1R)-1-[3-(2-oxopyrrolidin-1-yl)phenyl]ethyl]prop-2-enamide
—— (E)-N-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide —— C21H30N2O4S
(E)-N-butyl-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide
—— (E)-N-[(2S)-1-(2,4-dimethylphenyl)propan-2-yl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C23H29NO4
(E)-N-[(2S)-1-(2,4-dimethylphenyl)propan-2-yl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[2-[(2S)-1-cyanopropan-2-yl]sulfanylphenyl]-3-(3-methoxy-4-propoxyphenyl)prop-2-enamide —— C23H26N2O3S
(E)-N-[2-[(2S)-1-cyanopropan-2-yl]sulfanylphenyl]-3-(3-methoxy-4-propoxyphenyl)prop-2-enamide
—— (E)-N-[(2R)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide —— C25H30FN3O3
(E)-N-[(2R)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide
—— (E)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C27H27N3O3S
(E)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— (E)-N-[(2R)-1-(2,4-dimethylphenyl)propan-2-yl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C23H29NO4
(E)-N-[(2R)-1-(2,4-dimethylphenyl)propan-2-yl]-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[(S)-cyano-(2,3-dichlorophenyl)methyl]-3-[2-(difluoromethoxy)phenyl]prop-2-enamide —— C18H12Cl2F2N2O2
(E)-N-[(S)-cyano-(2,3-dichlorophenyl)methyl]-3-[2-(difluoromethoxy)phenyl]prop-2-enamide
—— ethyl 2-[2-[[(2S)-3-(2,4-dichlorophenyl)-2-methylpropanoyl]amino]-1,3-thiazol-4-yl]acetate —— C17H18Cl2N2O3S
ethyl 2-[2-[[(2S)-3-(2,4-dichlorophenyl)-2-methylpropanoyl]amino]-1,3-thiazol-4-yl]acetate
—— (E)-3-[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylsulfonylethyl)prop-2-enamide —— C17H24N2O4S2
(E)-3-[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylsulfonylethyl)prop-2-enamide
—— (E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[4-(difluoromethoxy)-3-ethoxyphenyl]prop-2-enamide —— C25H26F2N2O4
(E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[4-(difluoromethoxy)-3-ethoxyphenyl]prop-2-enamide
—— (E)-N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-methylprop-2-enamide —— C22H28N2O3S
(E)-N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-methylprop-2-enamide
—— (E)-N-[(3-methoxyphenyl)methyl]-3-(4-morpholin-4-ylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C26H32N2O4
(E)-N-[(3-methoxyphenyl)methyl]-3-(4-morpholin-4-ylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(S)-(2-methoxyphenyl)-phenylmethyl]prop-2-enamide —— C24H21NO4
(E)-3-(1,3-benzodioxol-5-yl)-N-[(S)-(2-methoxyphenyl)-phenylmethyl]prop-2-enamide
—— (E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide —— C23H21F3N2O2
(E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide
—— (E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enamide —— C26H30N2O4
(E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enamide
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[[(2R)-oxan-2-yl]methyl]-N-propylprop-2-enamide —— C23H31N3O2
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[[(2R)-oxan-2-yl]methyl]-N-propylprop-2-enamide
—— ethyl (2S)-2-[(3,6-dichloropyridine-2-carbonyl)amino]-2-methyloctanoate —— C17H24Cl2N2O3
ethyl (2S)-2-[(3,6-dichloropyridine-2-carbonyl)amino]-2-methyloctanoate
—— (E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C27H27N3O3S
(E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[2-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— ethyl (2R)-2-benzyl-3-[(3-cyanophenyl)methylsulfonylamino]propanoate —— C20H22N2O4S
ethyl (2R)-2-benzyl-3-[(3-cyanophenyl)methylsulfonylamino]propanoate
—— ethyl (1S,2S,4R,5R,6R)-3,8-dioxatricyclo[3.2.1.02,4]octane-6-carboxylate —— C9H12O4
ethyl (1S,2S,4R,5R,6R)-3,8-dioxatricyclo[3.2.1.02,4]octane-6-carboxylate
—— ethyl 3-[[(1S,2S)-2-(4-chlorophenyl)cyclopropanecarbonyl]-(pyridin-3-ylmethyl)amino]propanoate —— C21H23ClN2O3
ethyl 3-[[(1S,2S)-2-(4-chlorophenyl)cyclopropanecarbonyl]-(pyridin-3-ylmethyl)amino]propanoate
—— (E)-N-[(1S)-1-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C23H24N2O4S
(E)-N-[(1S)-1-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— ethyl 3-[[(1R,2R)-2-(4-chlorophenyl)cyclopropanecarbonyl]-(pyridin-3-ylmethyl)amino]propanoate —— C21H23ClN2O3
ethyl 3-[[(1R,2R)-2-(4-chlorophenyl)cyclopropanecarbonyl]-(pyridin-3-ylmethyl)amino]propanoate
—— (E)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide —— C24H26N2O4
(E)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide
—— (E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-[(2-thiophen-2-ylacetyl)amino]phenyl]prop-2-enamide —— C26H26N2O4S
(E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-[(2-thiophen-2-ylacetyl)amino]phenyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]prop-2-enamide —— C23H22N2O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]prop-2-enamide
—— ethyl (2S)-2-benzyl-3-[(3-cyanophenyl)methylsulfonylamino]propanoate —— C20H22N2O4S
ethyl (2S)-2-benzyl-3-[(3-cyanophenyl)methylsulfonylamino]propanoate
—— ethyl (2R)-2-benzyl-3-[[1-(3-methoxyphenyl)cyclopentanecarbonyl]amino]propanoate —— C25H31NO4
ethyl (2R)-2-benzyl-3-[[1-(3-methoxyphenyl)cyclopentanecarbonyl]amino]propanoate
—— (E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide —— C26H31ClFN3O3
(E)-N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide
—— (E)-N-[(1R)-1-(3,4-diethoxyphenyl)-2-methylpropyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide —— C27H36N2O4
(E)-N-[(1R)-1-(3,4-diethoxyphenyl)-2-methylpropyl]-3-(4-morpholin-4-ylphenyl)prop-2-enamide
—— ethyl 2-[2-[[(2R)-3-(2,4-dichlorophenyl)-2-methylpropanoyl]amino]-1,3-thiazol-4-yl]acetate —— C17H18Cl2N2O3S
ethyl 2-[2-[[(2R)-3-(2,4-dichlorophenyl)-2-methylpropanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 5-[bis(4-methoxyphenyl)methylamino]-2-[3-[(E)-5-[[2-[[3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]-4-[(2-methylpropan-2-yl)oxy]-4-oxobutanoyl]amino]pent-3-enoyl]oxytetradecanoylamino]-5-oxopentanoate —— C62H89N5O14
ethyl 5-[bis(4-methoxyphenyl)methylamino]-2-[3-[(E)-5-[[2-[[3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]-4-[(2-methylpropan-2-yl)oxy]-4-oxobutanoyl]amino]pent-3-enoyl]oxytetradecanoylamino]-5-oxopentanoate
—— (E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide —— C24H26N2O4
(E)-N-[2-[[2-[(1R)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide —— C23H21F3N2O2
(E)-N-[2-[[2-[(1S)-cyclopent-2-en-1-yl]acetyl]amino]phenyl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide
—— ethyl (3R)-1-[2-[[2-fluoro-4-(4-methylphenyl)benzoyl]-methylamino]acetyl]piperidine-3-carboxylate —— C25H29FN2O4
ethyl (3R)-1-[2-[[2-fluoro-4-(4-methylphenyl)benzoyl]-methylamino]acetyl]piperidine-3-carboxylate
—— ethyl 2-[[2-[[5-[[(Z)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]amino]-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]amino]acetate —— C18H18N4O6S2
ethyl 2-[[2-[[5-[[(Z)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]amino]-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]amino]acetate
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-fluoro-2-[[(2R)-oxolan-2-yl]methoxy]phenyl]prop-2-enamide —— C25H26FN3O3
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-fluoro-2-[[(2R)-oxolan-2-yl]methoxy]phenyl]prop-2-enamide
—— (E)-N-(2-acetamido-5-chlorophenyl)-3-[2-[(2S)-butan-2-yl]oxyphenyl]prop-2-enamide —— C21H23ClN2O3
(E)-N-(2-acetamido-5-chlorophenyl)-3-[2-[(2S)-butan-2-yl]oxyphenyl]prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[(1R)-1-(4-phenyl-1,3-thiazol-2-yl)ethyl]prop-2-enamide —— C23H22F2N2O3S
(E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-[(1R)-1-(4-phenyl-1,3-thiazol-2-yl)ethyl]prop-2-enamide
—— (E)-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylsulfonylethyl)prop-2-enamide —— C17H24N2O4S2
(E)-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]-N-(2-thiomorpholin-4-ylsulfonylethyl)prop-2-enamide
—— (E)-N-[(1R)-1-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C23H24N2O4S
(E)-N-[(1R)-1-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(R)-(2-methoxyphenyl)-phenylmethyl]prop-2-enamide —— C24H21NO4
(E)-3-(1,3-benzodioxol-5-yl)-N-[(R)-(2-methoxyphenyl)-phenylmethyl]prop-2-enamide
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-fluoro-2-[[(2S)-oxolan-2-yl]methoxy]phenyl]prop-2-enamide —— C25H26FN3O3
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[5-fluoro-2-[[(2S)-oxolan-2-yl]methoxy]phenyl]prop-2-enamide
—— (E)-1-[(2R)-2-(2,4-dichloro-5-fluorophenyl)morpholin-4-yl]-3-(3,4-dimethoxyphenyl)prop-2-en-1-one —— C21H20Cl2FNO4
(E)-1-[(2R)-2-(2,4-dichloro-5-fluorophenyl)morpholin-4-yl]-3-(3,4-dimethoxyphenyl)prop-2-en-1-one
—— (E)-1-[(2R)-2-(2,4-dichloro-5-fluorophenyl)morpholin-4-yl]-3-(4-nitrophenyl)prop-2-en-1-one —— C19H15Cl2FN2O4
(E)-1-[(2R)-2-(2,4-dichloro-5-fluorophenyl)morpholin-4-yl]-3-(4-nitrophenyl)prop-2-en-1-one