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—— (E)-N-[2-[4-oxo-5-[[3-(trifluoromethyl)phenyl]methyl]pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide —— C19H18F3N5O2
(E)-N-[2-[4-oxo-5-[[3-(trifluoromethyl)phenyl]methyl]pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(1-benzofuran-2-yl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C22H16N2O5
(E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(1-benzofuran-2-yl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[(5R)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]prop-2-enamide —— C20H18N2O5
(E)-3-(1,3-benzodioxol-5-yl)-N-[[(5R)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]prop-2-enamide
—— (E)-N-[2-[5-[(4-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C26H26FN5O5
(E)-N-[2-[5-[(4-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[[5-(1,3-benzodioxol-5-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C22H20N2O6
(E)-N-[[5-(1,3-benzodioxol-5-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[2-[5-[(2-methylphenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide —— C19H21N5O2
(E)-N-[2-[5-[(2-methylphenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide
—— (E)-N-[2-[5-[(2-methylphenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-phenylprop-2-enamide —— C24H23N5O2
(E)-N-[2-[5-[(2-methylphenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-phenylprop-2-enamide
—— (E)-N-[[(5R)-3-(1,3-benzodioxol-5-yl)-2-oxo-1,3-oxazolidin-5-yl]methyl]but-2-enamide —— C15H16N2O5
(E)-N-[[(5R)-3-(1,3-benzodioxol-5-yl)-2-oxo-1,3-oxazolidin-5-yl]methyl]but-2-enamide
—— (E)-N-[[5-(2,4-difluorophenyl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C22H20F2N2O5
(E)-N-[[5-(2,4-difluorophenyl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[2-[5-[(2-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-phenylprop-2-enamide —— C23H20FN5O2
(E)-N-[2-[5-[(2-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-phenylprop-2-enamide
—— (E)-N-[[5-(2,4-difluorophenyl)-1,2-oxazol-3-yl]methyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C21H18F2N2O4
(E)-N-[[5-(2,4-difluorophenyl)-1,2-oxazol-3-yl]methyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-1-[4-(5,7-dimethyl-1,3-benzothiazol-2-yl)piperazin-1-yl]prop-2-en-1-one —— C24H27N3O3S
(E)-3-(3,4-dimethoxyphenyl)-1-[4-(5,7-dimethyl-1,3-benzothiazol-2-yl)piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C20H15FN2O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C22H22N2O5
(E)-3-(3,4-dimethoxyphenyl)-N-[[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-N-[[(5R)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]but-2-enamide —— C14H16N2O3
(E)-N-[[(5R)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]but-2-enamide
—— (E)-N-[[5-(1-benzofuran-2-yl)-1,2-oxazol-3-yl]methyl]-3-phenylprop-2-enamide —— C21H16N2O3
(E)-N-[[5-(1-benzofuran-2-yl)-1,2-oxazol-3-yl]methyl]-3-phenylprop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]prop-2-enamide —— C19H18N2O4S
(E)-3-(3,4-dimethoxyphenyl)-N-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]prop-2-enamide
—— (E)-N-[[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C22H21FN2O5
(E)-N-[[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[[5-(1-benzofuran-2-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C24H22N2O6
(E)-N-[[5-(1-benzofuran-2-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]prop-2-enamide —— C21H20N2O4
(E)-3-(3,4-dimethoxyphenyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]prop-2-enamide
—— (E)-N-[[(5S)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]-3-phenylprop-2-enamide —— C19H18N2O3
(E)-N-[[(5S)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]-3-phenylprop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C22H22N2O5
(E)-3-(3,4-dimethoxyphenyl)-N-[[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-N-[[(5S)-3-(1,3-benzodioxol-5-yl)-2-oxo-1,3-oxazolidin-5-yl]methyl]but-2-enamide —— C15H16N2O5
(E)-N-[[(5S)-3-(1,3-benzodioxol-5-yl)-2-oxo-1,3-oxazolidin-5-yl]methyl]but-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[5-(3,4-dimethoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C23H24N2O6
(E)-3-(3,4-dimethoxyphenyl)-N-[[5-(3,4-dimethoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-N-[[5-(1,3-benzodioxol-5-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C23H22N2O7
(E)-N-[[5-(1,3-benzodioxol-5-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C20H15ClN2O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]prop-2-enamide —— C18H14N2O4S
(E)-3-(1,3-benzodioxol-5-yl)-N-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]prop-2-enamide
—— (E)-N-[[(3R)-1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]methyl]but-2-enamide —— C16H19FN2O2
(E)-N-[[(3R)-1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]methyl]but-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(1,3-benzodioxol-5-yl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C21H16N2O6
(E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(1,3-benzodioxol-5-yl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-[4-oxo-5-[[3-(trifluoromethyl)phenyl]methyl]pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]prop-2-enamide —— C25H20F3N5O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-[4-oxo-5-[[3-(trifluoromethyl)phenyl]methyl]pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]prop-2-enamide
—— (E)-N-[[(3S)-1-(1,3-benzodioxol-5-yl)-5-oxopyrrolidin-3-yl]methyl]-3-(4-methoxyphenyl)prop-2-enamide —— C22H22N2O5
(E)-N-[[(3S)-1-(1,3-benzodioxol-5-yl)-5-oxopyrrolidin-3-yl]methyl]-3-(4-methoxyphenyl)prop-2-enamide
—— (E)-N-[2-[5-[(3-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C26H26FN5O5
(E)-N-[2-[5-[(3-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-[6-methylsulfanyl-4-(propylamino)pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]prop-2-enamide —— C21H24N6O3S
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-[6-methylsulfanyl-4-(propylamino)pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-[6-methylsulfanyl-4-(propan-2-ylamino)pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]prop-2-enamide —— C21H24N6O3S
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-[6-methylsulfanyl-4-(propan-2-ylamino)pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]prop-2-enamide
—— (E)-N-[2-[5-[(3-methylphenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide —— C19H21N5O2
(E)-N-[2-[5-[(3-methylphenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide
—— EtSO2-D-Phg-Oic-NHBn(4-amidino) —— C27H35N5O4S
EtSO2-D-Phg-Oic-NHBn(4-amidino)
—— (E)-3-[5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl]-1-[(1R)-1-(2-methylpyrimidin-5-yl)-1H-phthalazin-2-yl]prop-2-en-1-one —— C29H28N8O3
(E)-3-[5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl]-1-[(1R)-1-(2-methylpyrimidin-5-yl)-1H-phthalazin-2-yl]prop-2-en-1-one
—— (E)-N-[2-[5-[(3-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide —— C18H18FN5O2
(E)-N-[2-[5-[(3-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]but-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C21H18N2O5
(E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-N-[2-[5-[(3-chlorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C26H26ClN5O5
(E)-N-[2-[5-[(3-chlorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C20H20N2O5S
(E)-N-[(5-thiophen-2-yl-1,2-oxazol-3-yl)methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C20H20N2O6
(E)-N-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— ethyl 3-[[(3R)-3-hydroxy-3-(hydroxymethyl)pyrrolidine-1-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C17H20N2O5S
ethyl 3-[[(3R)-3-hydroxy-3-(hydroxymethyl)pyrrolidine-1-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— (E)-N-[[5-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1,2-oxazol-3-yl]methyl]-3-phenylprop-2-enamide —— C22H20N2O3
(E)-N-[[5-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1,2-oxazol-3-yl]methyl]-3-phenylprop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C21H18N2O5
(E)-3-(1,3-benzodioxol-5-yl)-N-[[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide —— C21H19FN2O4
(E)-3-(3,4-dimethoxyphenyl)-N-[[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-(5-benzyl-4-oxopyrazolo[3,4-d]pyrimidin-1-yl)ethyl]prop-2-enamide —— C24H21N5O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-(5-benzyl-4-oxopyrazolo[3,4-d]pyrimidin-1-yl)ethyl]prop-2-enamide
—— (E)-N-[[(3S)-1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]methyl]but-2-enamide —— C16H19FN2O2
(E)-N-[[(3S)-1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]methyl]but-2-enamide
—— (E)-N-[2-[5-[(2-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C26H26FN5O5
(E)-N-[2-[5-[(2-fluorophenyl)methyl]-4-oxopyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N-[[(5S)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]but-2-enamide —— C14H16N2O3
(E)-N-[[(5S)-2-oxo-3-phenyl-1,3-oxazolidin-5-yl]methyl]but-2-enamide