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中文名称 英文名称 CAS号 化学式 结构式图片
—— (E)-1-[4-[(2R)-oxolane-2-carbonyl]piperazin-1-yl]-3-(5-phenylthiophen-2-yl)prop-2-en-1-one —— C22H24N2O3S
(E)-1-[4-[(2R)-oxolane-2-carbonyl]piperazin-1-yl]-3-(5-phenylthiophen-2-yl)prop-2-en-1-one
—— ethyl (Z)-3-(1-benzyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enoate —— C20H19N3O2
ethyl (Z)-3-(1-benzyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enoate
—— (E)-N-[3-[2-[2-(cyclopropylamino)-2-oxoacetyl]hydrazinyl]-3-oxopropyl]-3-phenylprop-2-enamide —— C17H20N4O4
(E)-N-[3-[2-[2-(cyclopropylamino)-2-oxoacetyl]hydrazinyl]-3-oxopropyl]-3-phenylprop-2-enamide
—— (E)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]-N-[2-(dimethylamino)-2-oxoethyl]prop-2-enamide —— C24H26N4O2
(E)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]-N-[2-(dimethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-N-[2-(dimethylamino)-2-oxoethyl]prop-2-enamide —— C20H23N3O4
(E)-3-[1-(1,3-benzodioxol-5-yl)-2,5-dimethylpyrrol-3-yl]-N-[2-(dimethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-(dimethylamino)-2-oxoethyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide —— C16H16N6O2
(E)-N-[2-(dimethylamino)-2-oxoethyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide
—— (E)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[2-(dimethylamino)-2-oxoethyl]prop-2-enamide —— C25H28N4O2
(E)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[2-(dimethylamino)-2-oxoethyl]prop-2-enamide
—— ethyl (5E)-2-anilino-4-oxo-5-[[2-(pyridin-2-ylmethoxy)phenyl]methylidene]furan-3-carboxylate —— C26H22N2O5
ethyl (5E)-2-anilino-4-oxo-5-[[2-(pyridin-2-ylmethoxy)phenyl]methylidene]furan-3-carboxylate
—— ethyl (2Z,5S)-2-[[4-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)oxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H37N7O7S
ethyl (2Z,5S)-2-[[4-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)oxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 3,5-dimethyl-4-[(Z)-3-[2-(pyridin-2-ylmethoxy)phenyl]prop-2-enoyl]-1H-pyrrole-2-carboxylate —— C24H24N2O4
ethyl 3,5-dimethyl-4-[(Z)-3-[2-(pyridin-2-ylmethoxy)phenyl]prop-2-enoyl]-1H-pyrrole-2-carboxylate
—— ethyl (2E,5R)-2-[(3,5-ditert-butyl-4-hydroxyphenyl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H38N2O5S
ethyl (2E,5R)-2-[(3,5-ditert-butyl-4-hydroxyphenyl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[3-ethoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H28F3N3O8S
ethyl (2E,5R)-2-[[3-ethoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[[5-(4-chlorophenyl)furan-2-yl]methyl]prop-2-enamide —— C22H19ClN2O4
(E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[[5-(4-chlorophenyl)furan-2-yl]methyl]prop-2-enamide
—— ethyl (2E,5R)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-2-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H27Cl2N3O4S
ethyl (2E,5R)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-2-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one —— C25H36N4O+2
(E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one
—— ethyl (2E,5S)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-2-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H27Cl2N3O4S
ethyl (2E,5S)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-2-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E)-2-[4-oxo-3-[(2R)-1-oxo-1-(2,4,6-trimethylanilino)propan-2-yl]-1,3-thiazolidin-2-ylidene]acetate —— C19H24N2O4S
ethyl (2E)-2-[4-oxo-3-[(2R)-1-oxo-1-(2,4,6-trimethylanilino)propan-2-yl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2Z,5S)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H24F3N3O7S
ethyl (2Z,5S)-2-[[3-methoxy-4-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-1-[4-(2-pyrrolidin-1-ylethyl)piperazin-1-yl]prop-2-en-1-one —— C25H34N4O
(E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-1-[4-(2-pyrrolidin-1-ylethyl)piperazin-1-yl]prop-2-en-1-one
—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[[4-(dimethylamino)phenyl]methyl]-N-methylprop-2-enamide —— C22H27N3O4
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[[4-(dimethylamino)phenyl]methyl]-N-methylprop-2-enamide
—— ethyl 2-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-9H-purin-9-yl)acetate —— C11H14N4O4
ethyl 2-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-9H-purin-9-yl)acetate
—— ethyl (2E,5R)-5-(3-methoxyphenyl)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28N4O6S
ethyl (2E,5R)-5-(3-methoxyphenyl)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[4-[(2-chloro-6-fluorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H30ClFN2O6S
ethyl (2Z,5R)-2-[[4-[(2-chloro-6-fluorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H28ClFN2O6S
ethyl (2Z,5S)-2-[[4-[(2-chloro-6-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[[3-[(4-chlorophenyl)methoxy]-4-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29ClN2O6S
ethyl (2E,5R)-2-[[3-[(4-chlorophenyl)methoxy]-4-methoxyphenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-5-(4-chlorophenyl)-2-[[3,5-dibromo-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H22Br2ClFN2O4S
ethyl (2Z,5R)-5-(4-chlorophenyl)-2-[[3,5-dibromo-4-[(4-fluorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one —— C26H38N4O+2
(E)-3-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]-1-[4-(2-pyrrolidin-1-ium-1-ylethyl)piperazin-4-ium-1-yl]prop-2-en-1-one
—— Ethyl 2-[[4-amino-5-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C9H16N4O3S
Ethyl 2-[[4-amino-5-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— ethyl (2Z,5R)-2-[[4-[(2-chloro-6-fluorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H28ClFN2O5S
ethyl (2Z,5R)-2-[[4-[(2-chloro-6-fluorophenyl)methoxy]-3-ethoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-ethyl-N-[(3-fluoro-4-methoxyphenyl)methyl]prop-2-enamide —— C22H21ClFNO3
(E)-3-(6-chloro-2H-chromen-3-yl)-N-ethyl-N-[(3-fluoro-4-methoxyphenyl)methyl]prop-2-enamide
—— ethyl (2E,5R)-5-(2-ethoxy-3-methoxyphenyl)-7-methyl-3-oxo-2-[(E)-3-phenylprop-2-enylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28N2O5S
ethyl (2E,5R)-5-(2-ethoxy-3-methoxyphenyl)-7-methyl-3-oxo-2-[(E)-3-phenylprop-2-enylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide —— C20H21FN2O4
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide
—— (E)-N-[[4-(dimethylamino)phenyl]methyl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methylprop-2-enamide —— C23H28N4O2
(E)-N-[[4-(dimethylamino)phenyl]methyl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methylprop-2-enamide
—— ethyl (2Z,5R)-2-[[4-(3-bromobenzoyl)oxy-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25BrN2O6S
ethyl (2Z,5R)-2-[[4-(3-bromobenzoyl)oxy-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[4-(2-iodobenzoyl)oxy-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H25IN2O6S
ethyl (2Z,5S)-2-[[4-(2-iodobenzoyl)oxy-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E)-2-[4-oxo-3-[(2S)-1-oxo-1-(2,4,6-trimethylanilino)propan-2-yl]-1,3-thiazolidin-2-ylidene]acetate —— C19H24N2O4S
ethyl (2E)-2-[4-oxo-3-[(2S)-1-oxo-1-(2,4,6-trimethylanilino)propan-2-yl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (5Z)-5-[(2-fluorophenyl)methylidene]-3-methyl-4-oxo-6,7-dihydro-1H-indole-2-carboxylate —— C19H18FNO3
ethyl (5Z)-5-[(2-fluorophenyl)methylidene]-3-methyl-4-oxo-6,7-dihydro-1H-indole-2-carboxylate
—— ethyl (2Z,5R)-2-[[4-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)oxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H37N7O7S
ethyl (2Z,5R)-2-[[4-[(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)oxy]-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-7-phenyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H26N4O6S2
ethyl (2E,5R)-2-[(2-morpholin-4-yl-5-nitrophenyl)methylidene]-3-oxo-7-phenyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(4-fluorophenyl)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H25FN4O5S
ethyl (2E,5S)-5-(4-fluorophenyl)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide —— C19H19FN2O3
(E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide
—— ethyl (2E,5R)-5-(4-methoxyphenyl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H33N4O5S+
ethyl (2E,5R)-5-(4-methoxyphenyl)-2-[[5-(4-methylpiperazin-4-ium-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3-ethoxy-4-methoxyphenyl)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H32N4O7S
ethyl (2E,5S)-5-(3-ethoxy-4-methoxyphenyl)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[[5-bromo-2-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H23BrF3N3O7S
ethyl (2Z,5S)-2-[[5-bromo-2-[2-nitro-4-(trifluoromethyl)phenoxy]phenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H26N4O5S
ethyl (2E,5S)-7-methyl-2-[(5-nitro-2-pyrrolidin-1-ylphenyl)methylidene]-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(3-methoxyphenyl)-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H33N5O6S
ethyl (2E,5S)-5-(3-methoxyphenyl)-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H30N5O5S+
ethyl (2E,5R)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2-methoxyphenyl)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32N5O6S+
ethyl (2E,5S)-5-(2-methoxyphenyl)-7-methyl-2-[[2-(4-methylpiperazin-4-ium-1-yl)-5-nitrophenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 5-amino-4-cyano-3-[[5-[(Z)-2-(5-methylfuran-2-yl)ethenyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]thiophene-2-carboxylate —— C18H17N5O3S2
ethyl 5-amino-4-cyano-3-[[5-[(Z)-2-(5-methylfuran-2-yl)ethenyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]thiophene-2-carboxylate
—— ethyl (2E,5S)-5-(4-methoxyphenyl)-7-methyl-2-[(5-nitro-2-piperidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H30N4O6S
ethyl (2E,5S)-5-(4-methoxyphenyl)-7-methyl-2-[(5-nitro-2-piperidin-1-ylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate