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—— (E)-3-[1-(furan-2-ylmethyl)-2,5-dimethylpyrrol-3-yl]-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide —— C24H27N3O3
(E)-3-[1-(furan-2-ylmethyl)-2,5-dimethylpyrrol-3-yl]-N-methyl-N-[2-(4-methylanilino)-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-[2-(4-ethoxybenzoyl)hydrazinyl]-2-oxoethyl]-3-phenylprop-2-enamide —— C20H21N3O4
(E)-N-[2-[2-(4-ethoxybenzoyl)hydrazinyl]-2-oxoethyl]-3-phenylprop-2-enamide
—— ethyl N-[2-[ethyl-[2-(5-fluoro-2-nitrophenoxy)acetyl]amino]acetyl]carbamate —— C15H18FN3O7
ethyl N-[2-[ethyl-[2-(5-fluoro-2-nitrophenoxy)acetyl]amino]acetyl]carbamate
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide —— C21H22FN3O2
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide —— C22H22FN3O
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[2-(2-fluorophenyl)ethyl]prop-2-enamide
—— (E)-N-[2-[(2-fluorophenyl)methylsulfanyl]ethyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide —— C21H18FN5OS
(E)-N-[2-[(2-fluorophenyl)methylsulfanyl]ethyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide
—— (E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[2-(2-methoxyphenyl)ethyl]prop-2-enamide —— C20H22N2O4
(E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[2-(2-methoxyphenyl)ethyl]prop-2-enamide
—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[2-(methylamino)-2-oxoethyl]prop-2-enamide —— C15H19N3O5
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[2-(methylamino)-2-oxoethyl]prop-2-enamide
—— (E)-N-(2,5-diethoxyphenyl)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide —— C23H27N3O4
(E)-N-(2,5-diethoxyphenyl)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide
—— (E)-1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-en-1-one —— C22H29N3O2
(E)-1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-en-1-one
—— (E)-1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one —— C23H29N3O
(E)-1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (E)-1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one —— C23H29N3O
(E)-1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (E)-1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-en-1-one —— C21H23N5O
(E)-1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-en-1-one
—— (E)-1-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one —— C23H29N3O
(E)-1-[(4aS,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one
—— ethyl 4-[[5-[(Z)-2-(4-acetamido-3-methyl-1,2-oxazol-5-yl)ethenyl]thiophen-2-yl]sulfonylamino]benzoate —— C21H21N3O6S2
ethyl 4-[[5-[(Z)-2-(4-acetamido-3-methyl-1,2-oxazol-5-yl)ethenyl]thiophen-2-yl]sulfonylamino]benzoate
—— (E)-1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one —— C23H29N3O
(E)-1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one
—— ethyl 3-[[5-[(Z)-2-(4-acetamido-3-methyl-1,2-oxazol-5-yl)ethenyl]thiophen-2-yl]sulfonylamino]benzoate —— C21H21N3O6S2
ethyl 3-[[5-[(Z)-2-(4-acetamido-3-methyl-1,2-oxazol-5-yl)ethenyl]thiophen-2-yl]sulfonylamino]benzoate
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide —— C18H22N4O2
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-(ethylamino)-2-oxoethyl]-3-[1-[(4-methylphenyl)methyl]-3-phenylpyrazol-4-yl]prop-2-enamide —— C24H26N4O2
(E)-N-[2-(ethylamino)-2-oxoethyl]-3-[1-[(4-methylphenyl)methyl]-3-phenylpyrazol-4-yl]prop-2-enamide
—— (E)-N-[(3S)-1-benzylpyrrolidin-1-ium-3-yl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide —— C24H29N4O2+
(E)-N-[(3S)-1-benzylpyrrolidin-1-ium-3-yl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide
—— (E)-3-[1-[(2-chlorophenyl)methyl]-3-phenylpyrazol-4-yl]-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide —— C23H23ClN4O2
(E)-3-[1-[(2-chlorophenyl)methyl]-3-phenylpyrazol-4-yl]-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide —— C25H28N4O2
(E)-3-[1-benzyl-3-(4-ethylphenyl)pyrazol-4-yl]-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one —— C23H29N3O
(E)-1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-en-1-one
—— (E)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide —— C24H26N4O2
(E)-3-[1-benzyl-3-(4-methylphenyl)pyrazol-4-yl]-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-(ethylamino)-2-oxoethyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide —— C16H16N6O2
(E)-N-[2-(ethylamino)-2-oxoethyl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide
—— (E)-1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-en-1-one —— C21H23N5O
(E)-1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-en-1-one
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methyl-N-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]prop-2-enamide —— C21H29N5O3
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methyl-N-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]prop-2-enamide
—— (E)-N-[(3R)-1-benzylpyrrolidin-3-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide —— C25H28N4O
(E)-N-[(3R)-1-benzylpyrrolidin-3-yl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-en-1-one —— C21H23N5O
(E)-1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-en-1-one
—— (E)-N-[(3R)-1-benzylpyrrolidin-1-ium-3-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide —— C23H23N6O+
(E)-N-[(3R)-1-benzylpyrrolidin-1-ium-3-yl]-3-([1,2,4]triazolo[3,4-a]phthalazin-3-yl)prop-2-enamide
—— (E)-N-[(3R)-1-benzylpyrrolidin-3-yl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide —— C24H28N4O2
(E)-N-[(3R)-1-benzylpyrrolidin-3-yl]-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]prop-2-enamide
—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[(2-methylphenyl)methyl]prop-2-enamide —— C20H22N2O4
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[(2-methylphenyl)methyl]prop-2-enamide
—— (E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methyl-N-[2-(4-methylpiperazin-4-ium-1-yl)-2-oxoethyl]prop-2-enamide —— C21H30N5O3+
(E)-3-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-methyl-N-[2-(4-methylpiperazin-4-ium-1-yl)-2-oxoethyl]prop-2-enamide
—— (E)-3-(1-benzyl-3-phenylpyrazol-4-yl)-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide —— C23H24N4O2
(E)-3-(1-benzyl-3-phenylpyrazol-4-yl)-N-[2-(ethylamino)-2-oxoethyl]prop-2-enamide
—— (E)-N-(2-acetamidoethyl)-3-[4-(2-amino-2-oxoethoxy)phenyl]prop-2-enamide —— C15H19N3O4
(E)-N-(2-acetamidoethyl)-3-[4-(2-amino-2-oxoethoxy)phenyl]prop-2-enamide
—— (E)-3-(6-chloro-2H-chromen-3-yl)-N-methyl-N-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]prop-2-enamide —— C20H24ClN3O3
(E)-3-(6-chloro-2H-chromen-3-yl)-N-methyl-N-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]prop-2-enamide
—— ethyl (2E)-2-[3-(2-imidazo[1,5-a]pyridin-3-ylsulfanylethyl)-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C16H17N3O3S2
ethyl (2E)-2-[3-(2-imidazo[1,5-a]pyridin-3-ylsulfanylethyl)-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-methyl-N-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]prop-2-enamide —— C21H26ClN5O2
(E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-methyl-N-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]prop-2-enamide
—— Ethyl 4-amino-2-[2-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]amino]-2-oxoethyl]sulfanylpyrimidine-5-carboxylate —— C19H19N5O4S
Ethyl 4-amino-2-[2-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]amino]-2-oxoethyl]sulfanylpyrimidine-5-carboxylate
—— (E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide —— C25H27N3O2
(E)-3-(2,5-dimethyl-1-phenylpyrrol-3-yl)-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide
—— (E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide —— C21H23N3O4
(E)-3-[4-(2-amino-2-oxoethoxy)phenyl]-N-[2-(2-ethylanilino)-2-oxoethyl]prop-2-enamide
—— ethyl (2E)-2-[4-oxo-3-[2-[[5-oxo-4-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C19H22N4O4S2
ethyl (2E)-2-[4-oxo-3-[2-[[5-oxo-4-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— Ethyl 6-[(2-chloroquinolin-3-yl)methylsulfanyl]-5-cyano-2-methylpyridine-3-carboxylate —— C20H16ClN3O2S
Ethyl 6-[(2-chloroquinolin-3-yl)methylsulfanyl]-5-cyano-2-methylpyridine-3-carboxylate
—— ethyl 6-[[5-(2-methylpropylsulfanyl)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H20N4O3S3
ethyl 6-[[5-(2-methylpropylsulfanyl)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[3-[(E)-[3-methyl-2-(2-methylphenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]phenoxy]acetate —— C22H22N2O4S
ethyl 2-[3-[(E)-[3-methyl-2-(2-methylphenyl)imino-4-oxo-1,3-thiazolidin-5-ylidene]methyl]phenoxy]acetate
—— ethyl (2E)-2-[3-[2-[[(10bR)-1,10b-dihydropyrazolo[1,5-c]quinazolin-5-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C19H20N4O3S2
ethyl (2E)-2-[3-[2-[[(10bR)-1,10b-dihydropyrazolo[1,5-c]quinazolin-5-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[3-[2-[1-(4-methoxyphenyl)tetrazol-5-yl]sulfanylethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C17H19N5O4S2
ethyl (2E)-2-[3-[2-[1-(4-methoxyphenyl)tetrazol-5-yl]sulfanylethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[3-[2-[[5-(3-methoxyphenyl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C24H24N4O4S2
ethyl (2E)-2-[3-[2-[[5-(3-methoxyphenyl)-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[3-[2-[[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C18H17N3O6S2
ethyl (2E)-2-[3-[2-[[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2E)-2-[3-[2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C18H19F2N5O4S2
ethyl (2E)-2-[3-[2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]sulfanyl]ethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate