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—— ethyl 2-[[(4S)-4-(2-fluorophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H33FN2O4S
ethyl 2-[[(4S)-4-(2-fluorophenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (4S)-4-(2,5-dimethylphenyl)-2-oxo-6-[[5-(2-phenylethyl)-[1,2,4]triazino[5,6-b]indol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C33H32N6O3S
ethyl (4S)-4-(2,5-dimethylphenyl)-2-oxo-6-[[5-(2-phenylethyl)-[1,2,4]triazino[5,6-b]indol-3-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[[2-[(4R)-1-(4-fluorophenyl)-5-oxo-3-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-2-sulfanylideneimidazolidin-4-yl]acetyl]amino]benzoate —— C31H29FN4O5S
ethyl 4-[[2-[(4R)-1-(4-fluorophenyl)-5-oxo-3-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-2-sulfanylideneimidazolidin-4-yl]acetyl]amino]benzoate
—— ethyl 4-[(4R)-3-[(2-fluorophenyl)methyl]-5-oxo-4-[2-oxo-2-(4-propoxyanilino)ethyl]-2-sulfanylideneimidazolidin-1-yl]benzoate —— C30H30FN3O5S
ethyl 4-[(4R)-3-[(2-fluorophenyl)methyl]-5-oxo-4-[2-oxo-2-(4-propoxyanilino)ethyl]-2-sulfanylideneimidazolidin-1-yl]benzoate
—— ethyl 4-[(4S)-3-[3-(4-carbamoylpiperidin-1-yl)propyl]-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate —— C30H37N5O6S
ethyl 4-[(4S)-3-[3-(4-carbamoylpiperidin-1-yl)propyl]-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate
—— ethyl 4-[(4R)-4-[2-(4-fluoroanilino)-2-oxoethyl]-5-oxo-2-sulfanylidene-3-(thiophene-2-carbonylamino)imidazolidin-1-yl]benzoate —— C25H21FN4O5S2
ethyl 4-[(4R)-4-[2-(4-fluoroanilino)-2-oxoethyl]-5-oxo-2-sulfanylidene-3-(thiophene-2-carbonylamino)imidazolidin-1-yl]benzoate
—— ethyl 4-[(4S)-4-[2-(4-ethoxyanilino)-2-oxoethyl]-3-[(2-fluorophenyl)methyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate —— C29H28FN3O5S
ethyl 4-[(4S)-4-[2-(4-ethoxyanilino)-2-oxoethyl]-3-[(2-fluorophenyl)methyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate
—— Ethyl 1-[2-(aminomethyl)phenyl]-6-[4-(2-methylsulfonylphenyl)phenyl]-7-oxopyrazolo[4,3-d]pyrimidine-3-carboxylate —— C28H25N5O5S
Ethyl 1-[2-(aminomethyl)phenyl]-6-[4-(2-methylsulfonylphenyl)phenyl]-7-oxopyrazolo[4,3-d]pyrimidine-3-carboxylate
—— ethyl 2-[5-[[(2S)-2-[[5-(2-phenylethyl)-[1,2,4]triazino[5,6-b]indol-3-yl]sulfanyl]butanoyl]amino]-1,3,4-thiadiazol-2-yl]acetate —— C27H27N7O3S2
ethyl 2-[5-[[(2S)-2-[[5-(2-phenylethyl)-[1,2,4]triazino[5,6-b]indol-3-yl]sulfanyl]butanoyl]amino]-1,3,4-thiadiazol-2-yl]acetate
—— ethyl 4-[[2-[(4S)-1-benzyl-5-oxo-3-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-2-sulfanylideneimidazolidin-4-yl]acetyl]amino]benzoate —— C32H32N4O5S
ethyl 4-[[2-[(4S)-1-benzyl-5-oxo-3-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-2-sulfanylideneimidazolidin-4-yl]acetyl]amino]benzoate
—— ethyl 2-[5-[[(2R)-2-[[5-(2-phenylethyl)-[1,2,4]triazino[5,6-b]indol-3-yl]sulfanyl]butanoyl]amino]-1,3,4-thiadiazol-2-yl]acetate —— C27H27N7O3S2
ethyl 2-[5-[[(2R)-2-[[5-(2-phenylethyl)-[1,2,4]triazino[5,6-b]indol-3-yl]sulfanyl]butanoyl]amino]-1,3,4-thiadiazol-2-yl]acetate
—— ethyl 3-[4-[2-[[3,6-bis(2-phenylethyl)-9H-fluoren-9-yl]oxy]ethyl]phenyl]-2-ethoxypropanoate —— C44H46O4
ethyl 3-[4-[2-[[3,6-bis(2-phenylethyl)-9H-fluoren-9-yl]oxy]ethyl]phenyl]-2-ethoxypropanoate
—— ethyl 4-[acetyl-[2-[3,5-bis(trifluoromethyl)phenyl]acetyl]amino]-2-cyclopropyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinoline-1-carboxylate —— C28H25F9N2O4
ethyl 4-[acetyl-[2-[3,5-bis(trifluoromethyl)phenyl]acetyl]amino]-2-cyclopropyl-6-(trifluoromethyl)-3,4-dihydro-2H-quinoline-1-carboxylate
—— ethyl (Z)-3-[4-[[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]amino]phenyl]prop-2-enoate —— C23H25N3O4
ethyl (Z)-3-[4-[[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]amino]phenyl]prop-2-enoate
—— (E,Z)-1-{4-[5-(4,4,5,5,5-pentafluoropentylsulfinyl)-pentyloxy]phenyl}-1-(4-hydroxyphenyl)-2-phenyl-but-1-ene —— C32H35F5O3S
(E,Z)-1-{4-[5-(4,4,5,5,5-pentafluoropentylsulfinyl)-pentyloxy]phenyl}-1-(4-hydroxyphenyl)-2-phenyl-but-1-ene
—— ethyl 4-[[2-[(4R)-1-benzyl-5-oxo-3-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-2-sulfanylideneimidazolidin-4-yl]acetyl]amino]benzoate —— C32H32N4O5S
ethyl 4-[[2-[(4R)-1-benzyl-5-oxo-3-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]-2-sulfanylideneimidazolidin-4-yl]acetyl]amino]benzoate
—— ethyl 4-[(4R)-4-[2-(3-ethoxyanilino)-2-oxoethyl]-3-[(3-fluorobenzoyl)amino]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate —— C29H27FN4O6S
ethyl 4-[(4R)-4-[2-(3-ethoxyanilino)-2-oxoethyl]-3-[(3-fluorobenzoyl)amino]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate
—— ethyl 4-[[2-[(4R)-5-oxo-1-phenyl-2-sulfanylidene-3-[(2,3,4,5-tetrafluorophenyl)methyl]imidazolidin-4-yl]acetyl]amino]benzoate —— C27H21F4N3O4S
ethyl 4-[[2-[(4R)-5-oxo-1-phenyl-2-sulfanylidene-3-[(2,3,4,5-tetrafluorophenyl)methyl]imidazolidin-4-yl]acetyl]amino]benzoate
—— (E)-1-[4-[(Z)-3-phenylprop-2-enyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C21H23N3O
(E)-1-[4-[(Z)-3-phenylprop-2-enyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— ethyl 4-[[(Z)-3-(3-phenylmethoxyphenyl)prop-2-enoyl]amino]piperidine-1-carboxylate —— C24H28N2O4
ethyl 4-[[(Z)-3-(3-phenylmethoxyphenyl)prop-2-enoyl]amino]piperidine-1-carboxylate
—— ethyl 2-[2-[[(2S)-2-[[(Z)-3-phenylprop-2-enoyl]amino]propanoyl]amino]-1,3-thiazol-4-yl]acetate —— C19H21N3O4S
ethyl 2-[2-[[(2S)-2-[[(Z)-3-phenylprop-2-enoyl]amino]propanoyl]amino]-1,3-thiazol-4-yl]acetate
—— (E)-3-(4-bromophenyl)-N-methyl-2-thiophen-2-yl-N-(thiophen-3-ylmethyl)prop-2-enamide —— C19H16BrNOS2
(E)-3-(4-bromophenyl)-N-methyl-2-thiophen-2-yl-N-(thiophen-3-ylmethyl)prop-2-enamide
—— (E)-N-(1,3-benzodioxol-5-ylmethyl)-3-(4-fluorophenyl)-N-methyl-2-thiophen-2-ylprop-2-enamide —— C22H18FNO3S
(E)-N-(1,3-benzodioxol-5-ylmethyl)-3-(4-fluorophenyl)-N-methyl-2-thiophen-2-ylprop-2-enamide
—— ethyl (3S)-3-[[4,6-bis[3-(trifluoromethyl)anilino]-1,3,5-triazin-2-yl]amino]-3-(4-methylphenyl)propanoate —— C29H26F6N6O2
ethyl (3S)-3-[[4,6-bis[3-(trifluoromethyl)anilino]-1,3,5-triazin-2-yl]amino]-3-(4-methylphenyl)propanoate
—— ethyl 4-[(4S)-3-[2-(1-adamantyl)ethyl]-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate —— C33H39N3O5S
ethyl 4-[(4S)-3-[2-(1-adamantyl)ethyl]-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate
—— ethyl 4-[[2-[(4S)-5-oxo-1-phenyl-2-sulfanylidene-3-[(2,3,4,5-tetrafluorophenyl)methyl]imidazolidin-4-yl]acetyl]amino]benzoate —— C27H21F4N3O4S
ethyl 4-[[2-[(4S)-5-oxo-1-phenyl-2-sulfanylidene-3-[(2,3,4,5-tetrafluorophenyl)methyl]imidazolidin-4-yl]acetyl]amino]benzoate
—— ethyl 2-[[(Z)-3-[4-(cyclopropylcarbamoyl)phenyl]prop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C22H24N2O4S
ethyl 2-[[(Z)-3-[4-(cyclopropylcarbamoyl)phenyl]prop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl (Z)-3-[4-[[2-(4-nitroimidazol-1-yl)acetyl]amino]phenyl]prop-2-enoate —— C16H16N4O5
ethyl (Z)-3-[4-[[2-(4-nitroimidazol-1-yl)acetyl]amino]phenyl]prop-2-enoate
—— (E)-N-[2-[(5E)-5-[(2,4-dichlorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-3-pyridin-3-ylprop-2-enamide —— C20H15Cl2N3O3S
(E)-N-[2-[(5E)-5-[(2,4-dichlorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-3-pyridin-3-ylprop-2-enamide
—— (E)-3-(4-methoxyphenyl)-N-methyl-N-[(4-oxo-1H-quinazolin-2-yl)methyl]-2-thiophen-2-ylprop-2-enamide —— C24H21N3O3S
(E)-3-(4-methoxyphenyl)-N-methyl-N-[(4-oxo-1H-quinazolin-2-yl)methyl]-2-thiophen-2-ylprop-2-enamide
—— (E)-3-(4-bromophenyl)-1-piperidin-1-yl-2-thiophen-2-ylprop-2-en-1-one —— C18H18BrNOS
(E)-3-(4-bromophenyl)-1-piperidin-1-yl-2-thiophen-2-ylprop-2-en-1-one
—— ethyl 2-[[2-[2-methoxy-4-[(Z)-3-methoxy-3-oxoprop-1-enyl]phenoxy]acetyl]amino]thiophene-3-carboxylate —— C20H21NO7S
ethyl 2-[[2-[2-methoxy-4-[(Z)-3-methoxy-3-oxoprop-1-enyl]phenoxy]acetyl]amino]thiophene-3-carboxylate
—— Ethyl 1-[2-(aminomethyl)phenyl]-6-[4-(2-methylsulfonylphenyl)phenyl]-7-oxopyrazolo[4,3-d]pyrimidine-3-carboxylate;2,2,2-trifluoroacetic acid —— C30H26F3N5O7S
Ethyl 1-[2-(aminomethyl)phenyl]-6-[4-(2-methylsulfonylphenyl)phenyl]-7-oxopyrazolo[4,3-d]pyrimidine-3-carboxylate;2,2,2-trifluoroacetic acid
—— (E)-but-2-enedioic acid;N-[(2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-phenylpropan-2-yl]adamantane-1-carboxamide;hydrate —— C35H47N3O7
(E)-but-2-enedioic acid;N-[(2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-phenylpropan-2-yl]adamantane-1-carboxamide;hydrate
—— (E)-N-methyl-N-[(4-oxo-1H-quinazolin-2-yl)methyl]-3-phenyl-2-thiophen-2-ylprop-2-enamide —— C23H19N3O2S
(E)-N-methyl-N-[(4-oxo-1H-quinazolin-2-yl)methyl]-3-phenyl-2-thiophen-2-ylprop-2-enamide
—— ethyl (Z)-3-[4-[(4-methyl-6-methylsulfanyl-2-propan-2-ylpyrimidine-5-carbonyl)amino]phenyl]prop-2-enoate —— C21H25N3O3S
ethyl (Z)-3-[4-[(4-methyl-6-methylsulfanyl-2-propan-2-ylpyrimidine-5-carbonyl)amino]phenyl]prop-2-enoate
—— ethyl 4-[(4S)-4-[2-(3-ethoxyanilino)-2-oxoethyl]-3-[(3-fluorobenzoyl)amino]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate —— C29H27FN4O6S
ethyl 4-[(4S)-4-[2-(3-ethoxyanilino)-2-oxoethyl]-3-[(3-fluorobenzoyl)amino]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoate
—— ethyl (4S)-6-[[(Z)-3-[(2S)-5-methoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-enoyl]oxymethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H28N2O8
ethyl (4S)-6-[[(Z)-3-[(2S)-5-methoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-enoyl]oxymethyl]-4-(5-methylfuran-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2R)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-2-[[(Z)-3-(4-fluorophenyl)prop-2-enoyl]amino]acetate —— C24H23F2N3O3
ethyl (2R)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-2-[[(Z)-3-(4-fluorophenyl)prop-2-enoyl]amino]acetate
—— (E)-3-[4-[(2S,3S,4R,5R)-5-[(E)-N-[(3,4-difluorophenyl)methoxy]-C-methylcarbonimidoyl]-3-fluoro-4-hydroxyoxolan-2-yl]oxy-2-hydroxyphenyl]-N-(4,6-dihydroxy-1,3-benzodioxol-5-yl)-2-methylprop-2-enamide —— C30H27F3N2O10
(E)-3-[4-[(2S,3S,4R,5R)-5-[(E)-N-[(3,4-difluorophenyl)methoxy]-C-methylcarbonimidoyl]-3-fluoro-4-hydroxyoxolan-2-yl]oxy-2-hydroxyphenyl]-N-(4,6-dihydroxy-1,3-benzodioxol-5-yl)-2-methylprop-2-enamide
—— (E)-3-(4-phenylphenyl)-2-[5-(trifluoromethyl)pyridin-2-yl]prop-2-enenitrile —— C21H13F3N2
(E)-3-(4-phenylphenyl)-2-[5-(trifluoromethyl)pyridin-2-yl]prop-2-enenitrile
—— (E)-N-cyclopropyl-3-(3-phenylmethoxyphenyl)-2-thiophen-2-ylprop-2-enamide —— C23H21NO2S
(E)-N-cyclopropyl-3-(3-phenylmethoxyphenyl)-2-thiophen-2-ylprop-2-enamide
—— ethyl 4-[(4R)-4-[2-(4-fluoroanilino)-2-oxoethyl]-5-oxo-3-(pyridine-3-carbonylamino)-2-sulfanylideneimidazolidin-1-yl]benzoate —— C26H22FN5O5S
ethyl 4-[(4R)-4-[2-(4-fluoroanilino)-2-oxoethyl]-5-oxo-3-(pyridine-3-carbonylamino)-2-sulfanylideneimidazolidin-1-yl]benzoate
—— Ethyl 3-[4-[[6-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]-1-methylbenzimidazol-2-yl]methoxy]phenyl]-2-phenoxypropanoate —— C40H44N2O7
Ethyl 3-[4-[[6-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]-1-methylbenzimidazol-2-yl]methoxy]phenyl]-2-phenoxypropanoate
—— (E)-5-amino-N,5-dimethyl-N-[(2R)-1-[methyl-[(2R)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]hex-2-enamide;(Z)-but-2-enedioic acid —— C36H44N4O7
(E)-5-amino-N,5-dimethyl-N-[(2R)-1-[methyl-[(2R)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]hex-2-enamide;(Z)-but-2-enedioic acid
—— (E)-N-(1,3-benzodioxol-5-ylmethyl)-3-(4-methoxyphenyl)-N-methyl-2-thiophen-2-ylprop-2-enamide —— C23H21NO4S
(E)-N-(1,3-benzodioxol-5-ylmethyl)-3-(4-methoxyphenyl)-N-methyl-2-thiophen-2-ylprop-2-enamide
—— (E)-3-(3-methoxyphenyl)-2-phenyl-N-prop-2-enylprop-2-enamide —— C19H19NO2
(E)-3-(3-methoxyphenyl)-2-phenyl-N-prop-2-enylprop-2-enamide
—— ethyl 2-[(3S,5S)-5-[[4-[4-(N-hexadecoxycarbonylcarbamimidoyl)phenyl]phenoxy]methyl]-2-oxopyrrolidin-3-yl]acetate —— C39H57N3O6
ethyl 2-[(3S,5S)-5-[[4-[4-(N-hexadecoxycarbonylcarbamimidoyl)phenyl]phenoxy]methyl]-2-oxopyrrolidin-3-yl]acetate
—— ethyl (2S)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-2-[[(Z)-3-(4-fluorophenyl)prop-2-enoyl]amino]acetate —— C24H23F2N3O3
ethyl (2S)-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-2-[[(Z)-3-(4-fluorophenyl)prop-2-enoyl]amino]acetate
—— ethyl 2-(1-chloro-2-fluoroethyl)sulfanyl-6,7-difluoro-4-[(2R)-2-phenyl-2-(phenylmethoxycarbonylamino)acetyl]oxyquinoline-3-carboxylate —— C30H24ClF3N2O6S
ethyl 2-(1-chloro-2-fluoroethyl)sulfanyl-6,7-difluoro-4-[(2R)-2-phenyl-2-(phenylmethoxycarbonylamino)acetyl]oxyquinoline-3-carboxylate