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—— (E)-3-(4-fluorophenyl)-N-(4-methyl-1,3-thiazol-2-yl)-N-phenylbut-2-enamide —— C20H17FN2OS
(E)-3-(4-fluorophenyl)-N-(4-methyl-1,3-thiazol-2-yl)-N-phenylbut-2-enamide
—— ethyl 4-[[(Z)-3-(2-methoxyphenyl)prop-2-enyl]amino]piperidine-1-carboxylate —— C18H26N2O3
ethyl 4-[[(Z)-3-(2-methoxyphenyl)prop-2-enyl]amino]piperidine-1-carboxylate
—— (E)-2-cyano-N-[(3S)-2,3-dihydro-1-benzofuran-3-yl]-3-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]prop-2-enamide —— C21H23N3O3
(E)-2-cyano-N-[(3S)-2,3-dihydro-1-benzofuran-3-yl]-3-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]prop-2-enamide
—— (E)-N-cyclopropyl-2-methyl-N-[(1R)-1-naphthalen-2-ylethyl]pent-2-enamide —— C21H25NO
(E)-N-cyclopropyl-2-methyl-N-[(1R)-1-naphthalen-2-ylethyl]pent-2-enamide
—— (E)-N-[3-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-3-oxopropyl]-2-methylpent-2-enamide —— C18H24N2O3
(E)-N-[3-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-3-oxopropyl]-2-methylpent-2-enamide
—— (E)-2-methyl-N-[[(2S,3S)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methyl]-3-phenylprop-2-en-1-amine —— C19H25N3O
(E)-2-methyl-N-[[(2S,3S)-2-(1-methylpyrazol-4-yl)oxolan-3-yl]methyl]-3-phenylprop-2-en-1-amine
—— ethyl 6-fluoro-7-(4-methylpiperazin-1-yl)-4-oxo-1H-[1,3]thiazeto[3,2-a]quinoline-3-carboxylate —— C18H20FN3O3S
ethyl 6-fluoro-7-(4-methylpiperazin-1-yl)-4-oxo-1H-[1,3]thiazeto[3,2-a]quinoline-3-carboxylate
—— (E)-2-methyl-N-[[(8S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-8-yl]methyl]-3-phenylprop-2-en-1-amine —— C19H25N3
(E)-2-methyl-N-[[(8S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-8-yl]methyl]-3-phenylprop-2-en-1-amine
—— (E)-2-methyl-N-[[(8R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-8-yl]methyl]-3-phenylprop-2-en-1-amine —— C19H25N3
(E)-2-methyl-N-[[(8R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-8-yl]methyl]-3-phenylprop-2-en-1-amine
—— (E)-N-cyclopropyl-2-methyl-N-[(1S)-1-naphthalen-2-ylethyl]pent-2-enamide —— C21H25NO
(E)-N-cyclopropyl-2-methyl-N-[(1S)-1-naphthalen-2-ylethyl]pent-2-enamide
—— (E)-2-(1H-indole-3-carbonyl)-3-(1-methylbenzotriazol-5-yl)prop-2-enenitrile —— C19H13N5O
(E)-2-(1H-indole-3-carbonyl)-3-(1-methylbenzotriazol-5-yl)prop-2-enenitrile
—— ethyl 2-[[(5S,7S)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H24BrF3N4O3S
ethyl 2-[[(5S,7S)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(5R,7R)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H24BrF3N4O3S
ethyl 2-[[(5R,7R)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(5R,7S)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H24BrF3N4O3S
ethyl 2-[[(5R,7S)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 4-[5-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-7-oxo-6-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-3-yl]benzoate —— C27H32N4O5S3
ethyl 4-[5-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-7-oxo-6-[[(2S)-oxolan-2-yl]methyl]-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-3-yl]benzoate
—— ethyl 2-[[(5S,7R)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H24BrF3N4O3S
ethyl 2-[[(5S,7R)-5-(4-bromophenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl N-[(Z,3S,4S)-6-[tert-butyl(dimethyl)silyl]oxy-2,4-dimethyl-5-methylsulfanylhex-5-en-3-yl]carbamate —— C18H37NO3SSi
ethyl N-[(Z,3S,4S)-6-[tert-butyl(dimethyl)silyl]oxy-2,4-dimethyl-5-methylsulfanylhex-5-en-3-yl]carbamate
—— Ethyl 4,4,5,5,5-pentafluoro-2-(naphthalen-1-ylmethyl)-3-oxopentanoate —— C18H15F5O3
Ethyl 4,4,5,5,5-pentafluoro-2-(naphthalen-1-ylmethyl)-3-oxopentanoate
—— Ethyl 5-(4,6-diphenylpyridin-2-yl)oxypentanoate —— C24H25NO3
Ethyl 5-(4,6-diphenylpyridin-2-yl)oxypentanoate
—— E-1-azabicyclo[2.2.2]oct-3-yl α-(1-bromo-1-propen-3-yl)-α-hydroxy-α-phenylacetate —— C18H22BrNO3
E-1-azabicyclo[2.2.2]oct-3-yl α-(1-bromo-1-propen-3-yl)-α-hydroxy-α-phenylacetate
—— ethyl 4-[5-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-7-oxo-6-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-3-yl]benzoate —— C27H32N4O5S3
ethyl 4-[5-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-7-oxo-6-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-3-yl]benzoate
—— ethyl 4-(4-methylphenyl)-2-[[(1R)-2,2,2-trichloro-1-(naphthalene-1-carbonylamino)ethyl]amino]thiophene-3-carboxylate —— C27H23Cl3N2O3S
ethyl 4-(4-methylphenyl)-2-[[(1R)-2,2,2-trichloro-1-(naphthalene-1-carbonylamino)ethyl]amino]thiophene-3-carboxylate
—— Ethyl 3-amino-4-(2-phenyl-2-prop-2-enoxycarbonyloxyethyl)benzoate —— C21H23NO5
Ethyl 3-amino-4-(2-phenyl-2-prop-2-enoxycarbonyloxyethyl)benzoate
—— Ethyl 1-(2,4-Difluorobenzyl)-5-hydroxycarbamoyl-1H-pyrrolo[2,3-c]pyridine-2-carboxylate —— C18H15F2N3O4
Ethyl 1-(2,4-Difluorobenzyl)-5-hydroxycarbamoyl-1H-pyrrolo[2,3-c]pyridine-2-carboxylate
—— (E)-1-(4-chlorophenyl)-3-(3,5-ditert-butyl-4-hydroxyphenyl)prop-2-en-1-one —— C23H27ClO2
(E)-1-(4-chlorophenyl)-3-(3,5-ditert-butyl-4-hydroxyphenyl)prop-2-en-1-one
—— ethyl N-[(2R,3R)-2,3-bis(4-methoxyphenyl)cyclopropyl]-N-nitrosocarbamate —— C20H22N2O5
ethyl N-[(2R,3R)-2,3-bis(4-methoxyphenyl)cyclopropyl]-N-nitrosocarbamate
—— ethyl (3R,4S)-2-(benzenesulfonyl)-4-(methoxymethoxy)-3,5-dimethylhexanoate —— C18H28O6S
ethyl (3R,4S)-2-(benzenesulfonyl)-4-(methoxymethoxy)-3,5-dimethylhexanoate
—— (E)-3-(3-bromo-4-fluorophenyl)-N-isoquinolin-5-ylprop-2-enamide —— C18H12BrFN2O
(E)-3-(3-bromo-4-fluorophenyl)-N-isoquinolin-5-ylprop-2-enamide
—— ethyl 2-[[(2S)-2-(dibenzylamino)-4-hydroxybutyl]amino]acetate —— C22H30N2O3
ethyl 2-[[(2S)-2-(dibenzylamino)-4-hydroxybutyl]amino]acetate
—— ethyl 4-phenyl-2-[[(1R)-2,2,2-trichloro-1-(naphthalene-1-carbonylamino)ethyl]amino]thiophene-3-carboxylate —— C26H21Cl3N2O3S
ethyl 4-phenyl-2-[[(1R)-2,2,2-trichloro-1-(naphthalene-1-carbonylamino)ethyl]amino]thiophene-3-carboxylate
—— ethyl 4-[[(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate —— C29H28FN3O5S
ethyl 4-[[(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate
—— [(E,4S,5S)-4-[tert-butyl(dimethyl)silyl]oxyundec-2-en-6-yn-5-yl] 2-chloroacetate —— C19H33ClO3Si
[(E,4S,5S)-4-[tert-butyl(dimethyl)silyl]oxyundec-2-en-6-yn-5-yl] 2-chloroacetate
—— Ethyl 10-hydroxy-5-methoxy-1,9,10-trimethyl-3,4-dihydropyrrolo[3,2-b]carbazole-2-carboxylate —— C21H24N2O4
Ethyl 10-hydroxy-5-methoxy-1,9,10-trimethyl-3,4-dihydropyrrolo[3,2-b]carbazole-2-carboxylate
—— ethyl 4-[[(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate —— C29H28FN3O5S
ethyl 4-[[(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate
—— ethyl 4-(1-methoxycarbonyl-2H-pyridin-3-yl)-2,6-dimethyl-5-nitro-1,4-dihydropyridine-3-carboxylate —— C17H21N3O6
ethyl 4-(1-methoxycarbonyl-2H-pyridin-3-yl)-2,6-dimethyl-5-nitro-1,4-dihydropyridine-3-carboxylate
—— (E)-Methyl 3-bromo-3-(2-bromophenyl)-2-(formylamino)acrylate —— C11H9Br2NO3
(E)-Methyl 3-bromo-3-(2-bromophenyl)-2-(formylamino)acrylate
—— Ethyl 7,9-bis(propanoylsulfanyl)nonanoate —— C17H30O4S2
Ethyl 7,9-bis(propanoylsulfanyl)nonanoate
—— ethyl 2-[[(2R)-2-[[4-methyl-5-[[(4-methyl-3-nitrobenzoyl)amino]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H30N6O6S2
ethyl 2-[[(2R)-2-[[4-methyl-5-[[(4-methyl-3-nitrobenzoyl)amino]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[[5-[[(3-fluorobenzoyl)amino]methyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C31H32FN5O4S2
ethyl 2-[[(2S)-2-[[5-[[(3-fluorobenzoyl)amino]methyl]-4-(2-phenylethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[[5-[[(2-chloro-6-fluorobenzoyl)amino]methyl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C24H25ClFN5O4S2
ethyl 2-[[(2S)-2-[[5-[[(2-chloro-6-fluorobenzoyl)amino]methyl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[[5-[(furan-2-carbonylamino)methyl]-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C28H29N5O6S2
ethyl 2-[[(2S)-2-[[5-[(furan-2-carbonylamino)methyl]-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl (3S)-1-[5-methyl-4-oxo-3-[2-oxo-2-[3-(trifluoromethyl)anilino]ethyl]thieno[2,3-d]pyrimidine-6-carbonyl]piperidine-3-carboxylate —— C25H25F3N4O5S
ethyl (3S)-1-[5-methyl-4-oxo-3-[2-oxo-2-[3-(trifluoromethyl)anilino]ethyl]thieno[2,3-d]pyrimidine-6-carbonyl]piperidine-3-carboxylate
—— (E)-N,N,N',N'-tetraphenylethene-1,2-diamine —— C26H22N2
(E)-N,N,N',N'-tetraphenylethene-1,2-diamine
—— ethyl 2-[[(2R)-2-[[4-benzyl-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C28H29N5O5S2
ethyl 2-[[(2R)-2-[[4-benzyl-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 4-[3-[(4-methoxybenzoyl)amino]-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzoyl]piperazine-1-carboxylate —— C33H37N5O6
ethyl 4-[3-[(4-methoxybenzoyl)amino]-4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]benzoyl]piperazine-1-carboxylate
—— ethyl 2-[[(2S)-2-[[4-methyl-5-[[(4-methyl-3-nitrobenzoyl)amino]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H30N6O6S2
ethyl 2-[[(2S)-2-[[4-methyl-5-[[(4-methyl-3-nitrobenzoyl)amino]methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[[5-[[[2-(4-chlorophenoxy)acetyl]amino]methyl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C25H28ClN5O5S2
ethyl 2-[[(2S)-2-[[5-[[[2-(4-chlorophenoxy)acetyl]amino]methyl]-4-methyl-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[[4-methyl-5-[(thiophene-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H27N5O4S3
ethyl 2-[[(2R)-2-[[4-methyl-5-[(thiophene-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[[4-butyl-5-[(thiophene-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C25H31N5O4S3
ethyl 2-[[(2S)-2-[[4-butyl-5-[(thiophene-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 4-[4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-3-(thiophene-2-carbonylamino)benzoyl]piperazine-1-carboxylate —— C30H33N5O5S
ethyl 4-[4-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-3-(thiophene-2-carbonylamino)benzoyl]piperazine-1-carboxylate