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—— (E)-N-(4,6-difluoro-3-methylbenzo[d]thiazol-2(3H)-ylidene)-4-(piperidin-1-ylsulfonyl)benzamide —— C20H19F2N3O3S2
(E)-N-(4,6-difluoro-3-methylbenzo[d]thiazol-2(3H)-ylidene)-4-(piperidin-1-ylsulfonyl)benzamide
—— (E)-3-[3-chloro-4-(2-morpholin-4-ylethoxy)phenyl]-2-(1H-indole-3-carbonyl)prop-2-enenitrile —— C24H22ClN3O3
(E)-3-[3-chloro-4-(2-morpholin-4-ylethoxy)phenyl]-2-(1H-indole-3-carbonyl)prop-2-enenitrile
—— Ethyl 4-[[2-[1-[(2-methylphenyl)methyl]indol-3-yl]sulfanylacetyl]amino]benzoate —— C27H26N2O3S
Ethyl 4-[[2-[1-[(2-methylphenyl)methyl]indol-3-yl]sulfanylacetyl]amino]benzoate
—— (E)-3-(4-chlorophenyl)-4,4,4-trifluoro-N-[(2-hydroxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]but-2-enamide —— C22H21ClF3NO3
(E)-3-(4-chlorophenyl)-4,4,4-trifluoro-N-[(2-hydroxyphenyl)methyl]-N-[[(2R)-oxolan-2-yl]methyl]but-2-enamide
—— Ethyl 2-(6-ethyl-4-oxothieno[2,3-d]pyrimidin-3-yl)butanoate —— C14H18N2O3S
Ethyl 2-(6-ethyl-4-oxothieno[2,3-d]pyrimidin-3-yl)butanoate
—— (E)-N-(6-chloro-3-methylbenzo[d]thiazol-2(3H)-ylidene)-4-((3-methylpiperidin-1-yl)sulfonyl)benzamide —— C21H22ClN3O3S2
(E)-N-(6-chloro-3-methylbenzo[d]thiazol-2(3H)-ylidene)-4-((3-methylpiperidin-1-yl)sulfonyl)benzamide
—— (E)-3-pyridin-4-yl-N-[(1S)-1-(4-sulfamoylphenyl)ethyl]but-2-enamide —— C17H19N3O3S
(E)-3-pyridin-4-yl-N-[(1S)-1-(4-sulfamoylphenyl)ethyl]but-2-enamide
—— (E)-3-(4-chlorophenyl)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-4,4,4-trifluorobut-2-en-1-one —— C21H19ClF3NO3
(E)-3-(4-chlorophenyl)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-4,4,4-trifluorobut-2-en-1-one
—— (E)-2-(2,6-dichlorobenzoyl)-3-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)prop-2-enenitrile —— C20H15Cl2N3O
(E)-2-(2,6-dichlorobenzoyl)-3-(3-propan-2-ylimidazo[1,5-a]pyridin-1-yl)prop-2-enenitrile
—— ethyl (2S)-2-[[(E)-3-(4-chlorophenyl)-4,4,4-trifluorobut-2-enoyl]amino]propanoate —— C15H15ClF3NO3
ethyl (2S)-2-[[(E)-3-(4-chlorophenyl)-4,4,4-trifluorobut-2-enoyl]amino]propanoate
—— (E)-3-pyridin-4-yl-N-[(1R)-1-(4-sulfamoylphenyl)ethyl]but-2-enamide —— C17H19N3O3S
(E)-3-pyridin-4-yl-N-[(1R)-1-(4-sulfamoylphenyl)ethyl]but-2-enamide
—— (E)-3-(4-chlorophenyl)-4,4,4-trifluoro-N-[(2-hydroxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]but-2-enamide —— C22H21ClF3NO3
(E)-3-(4-chlorophenyl)-4,4,4-trifluoro-N-[(2-hydroxyphenyl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]but-2-enamide
—— ethyl 4-[(Z)-3-(3-cyanophenyl)-3-oxoprop-1-enyl]-1H-pyrazole-5-carboxylate —— C16H13N3O3
ethyl 4-[(Z)-3-(3-cyanophenyl)-3-oxoprop-1-enyl]-1H-pyrazole-5-carboxylate
—— ethyl 4-[(E)-2-cyano-2-(2,5-dichlorophenyl)sulfonylethenyl]-1H-pyrazole-5-carboxylate —— C15H11Cl2N3O4S
ethyl 4-[(E)-2-cyano-2-(2,5-dichlorophenyl)sulfonylethenyl]-1H-pyrazole-5-carboxylate
—— (E)-3-(4-chlorophenyl)-N-[2-(dimethylamino)-2-oxoethyl]-4,4,4-trifluoro-N-propylbut-2-enamide —— C17H20ClF3N2O2
(E)-3-(4-chlorophenyl)-N-[2-(dimethylamino)-2-oxoethyl]-4,4,4-trifluoro-N-propylbut-2-enamide
—— Ethyl 4-[(E)-2-cyano-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-3-oxoprop-1-enyl]-1H-pyrazole-5-carboxylate —— C18H16N4O5
Ethyl 4-[(E)-2-cyano-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-3-oxoprop-1-enyl]-1H-pyrazole-5-carboxylate
—— (E)-3-(4-chlorophenyl)-4,4,4-trifluoro-N-[4-[(S)-methylsulfinyl]phenyl]but-2-enamide —— C17H13ClF3NO2S
(E)-3-(4-chlorophenyl)-4,4,4-trifluoro-N-[4-[(S)-methylsulfinyl]phenyl]but-2-enamide
—— (E)-N-[(2-cyanophenyl)methylsulfonyl]-3-pyridin-4-ylbut-2-enamide —— C17H15N3O3S
(E)-N-[(2-cyanophenyl)methylsulfonyl]-3-pyridin-4-ylbut-2-enamide
—— (E)-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-pyridin-4-ylbut-2-en-1-one —— C15H20N2O2
(E)-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-pyridin-4-ylbut-2-en-1-one
—— (E)-3-(4-fluorophenyl)-N-[methyl(propyl)sulfamoyl]but-2-enamide —— C14H19FN2O3S
(E)-3-(4-fluorophenyl)-N-[methyl(propyl)sulfamoyl]but-2-enamide
—— (E)-3-(2-Bromo-4,6-dimethoxyphenyl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide —— C18H14BrClN2O3
(E)-3-(2-Bromo-4,6-dimethoxyphenyl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide
—— ethyl 4-[(Z)-3-(5-chlorothiophen-2-yl)-3-oxoprop-1-enyl]-1H-pyrazole-5-carboxylate —— C13H11ClN2O3S
ethyl 4-[(Z)-3-(5-chlorothiophen-2-yl)-3-oxoprop-1-enyl]-1H-pyrazole-5-carboxylate
—— (E)-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3-pyridin-4-ylbut-2-en-1-one —— C15H20N2O2
(E)-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3-pyridin-4-ylbut-2-en-1-one
—— (E)-3-(4-fluorophenyl)-N-[4-[2-(2-hydroxyethylamino)-2-oxoethyl]phenyl]but-2-enamide —— C20H21FN2O3
(E)-3-(4-fluorophenyl)-N-[4-[2-(2-hydroxyethylamino)-2-oxoethyl]phenyl]but-2-enamide
—— (E)-3-(3-fluorophenyl)-N-[(2S)-2-hydroxy-3-methoxypropyl]-N-methylbut-2-enamide —— C15H20FNO3
(E)-3-(3-fluorophenyl)-N-[(2S)-2-hydroxy-3-methoxypropyl]-N-methylbut-2-enamide
—— Ethyl 2-(2-{[4-(2,5-dimethylphenyl)-5-{[(3-methoxyphenyl)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}acetamido)-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate —— C31H33N5O5S2
Ethyl 2-(2-{[4-(2,5-dimethylphenyl)-5-{[(3-methoxyphenyl)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}acetamido)-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate
—— ethyl 4-[(E)-(4,5-dimethyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-trien-10-ylidene)methyl]-1H-pyrazole-5-carboxylate —— C18H18N4O3S
ethyl 4-[(E)-(4,5-dimethyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-trien-10-ylidene)methyl]-1H-pyrazole-5-carboxylate
—— ethyl 3'-(3-chlorophenyl)-3H,3'H-spiro[1,3-benzothiazole-2,2'-[1,3,4]thiadiazole]-5'-carboxylate —— C17H14ClN3O2S2
ethyl 3'-(3-chlorophenyl)-3H,3'H-spiro[1,3-benzothiazole-2,2'-[1,3,4]thiadiazole]-5'-carboxylate
—— ethyl (Z)-3-[4-[(4-carbamoyl-1,4-diazepane-1-carbonyl)amino]phenyl]prop-2-enoate —— C18H24N4O4
ethyl (Z)-3-[4-[(4-carbamoyl-1,4-diazepane-1-carbonyl)amino]phenyl]prop-2-enoate
—— Ethyl 2-{2-[(4-cyclohexyl-5-{[(3,4-dimethoxyphenyl)formamido]methyl}-4H-1,2,4-triazol-3-YL)sulfanyl]propanamido}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C32H41N5O6S2
Ethyl 2-{2-[(4-cyclohexyl-5-{[(3,4-dimethoxyphenyl)formamido]methyl}-4H-1,2,4-triazol-3-YL)sulfanyl]propanamido}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 6-bromo-5-methoxy-1-methyl-2-[(4-methylpiperidin-1-ium-1-yl)methyl]indole-3-carboxylate —— C20H28BrN2O3+
Ethyl 6-bromo-5-methoxy-1-methyl-2-[(4-methylpiperidin-1-ium-1-yl)methyl]indole-3-carboxylate
—— (E)-3-(3-chlorophenyl)-N-[3-(tetrazol-1-yl)phenyl]sulfonylbut-2-enamide —— C17H14ClN5O3S
(E)-3-(3-chlorophenyl)-N-[3-(tetrazol-1-yl)phenyl]sulfonylbut-2-enamide
—— Ethyl 4-[4-[[3-(2-methoxy-2-oxoethyl)-6-sulfamoyl-1,3-benzothiazol-2-ylidene]carbamoyl]phenyl]sulfonylpiperazine-1-carboxylate —— C24H27N5O9S3
Ethyl 4-[4-[[3-(2-methoxy-2-oxoethyl)-6-sulfamoyl-1,3-benzothiazol-2-ylidene]carbamoyl]phenyl]sulfonylpiperazine-1-carboxylate
—— Ethyl 3-[2-(4-acetamidobenzoyl)hydrazinyl]-2-propan-2-ylbut-3-enoate —— C18H25N3O4
Ethyl 3-[2-(4-acetamidobenzoyl)hydrazinyl]-2-propan-2-ylbut-3-enoate
—— (E)-3-[2-[(Z)-2-[4-(1,2,4-triazol-1-yl)phenyl]ethenyl]-1,3-thiazol-5-yl]prop-2-enoic acid —— C16H12N4O2S
(E)-3-[2-[(Z)-2-[4-(1,2,4-triazol-1-yl)phenyl]ethenyl]-1,3-thiazol-5-yl]prop-2-enoic acid
—— (E)-3-(4-fluorophenyl)-N-[4-(methanesulfonamido)phenyl]-2-methylprop-2-enamide —— C17H17FN2O3S
(E)-3-(4-fluorophenyl)-N-[4-(methanesulfonamido)phenyl]-2-methylprop-2-enamide
—— ethyl 5-[(Z)-2-chloro-2-(4-oxo-3H-quinazolin-2-yl)ethenyl]furan-2-carboxylate —— C17H13ClN2O4
ethyl 5-[(Z)-2-chloro-2-(4-oxo-3H-quinazolin-2-yl)ethenyl]furan-2-carboxylate
—— (E)-2-methyl-N-(2-phenylpyrimidin-5-yl)but-2-enamide —— C15H15N3O
(E)-2-methyl-N-(2-phenylpyrimidin-5-yl)but-2-enamide
—— (E)-3-(2,4-difluorophenyl)-N-[3-(methanesulfonamido)propyl]but-2-enamide —— C14H18F2N2O3S
(E)-3-(2,4-difluorophenyl)-N-[3-(methanesulfonamido)propyl]but-2-enamide
—— (E)-3-[2-[(Z)-2-(4-methyl-1,3-thiazol-5-yl)ethenyl]-1,3-thiazol-5-yl]prop-2-enoic acid —— C12H10N2O2S2
(E)-3-[2-[(Z)-2-(4-methyl-1,3-thiazol-5-yl)ethenyl]-1,3-thiazol-5-yl]prop-2-enoic acid
—— Ethyl 2-[2-[2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfonylacetyl]imino-1,3-benzothiazol-3-yl]acetate —— C19H23N3O6S2
Ethyl 2-[2-[2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfonylacetyl]imino-1,3-benzothiazol-3-yl]acetate
—— (E)-3-[2-(difluoromethoxy)phenyl]-N-(2-oxo-2-pyrrolidin-1-ylethyl)but-2-enamide —— C17H20F2N2O3
(E)-3-[2-(difluoromethoxy)phenyl]-N-(2-oxo-2-pyrrolidin-1-ylethyl)but-2-enamide
—— (E)-3-[2-[(Z)-2-[4-(methylcarbamoyl)phenyl]ethenyl]-1,3-thiazol-5-yl]prop-2-enoic acid —— C16H14N2O3S
(E)-3-[2-[(Z)-2-[4-(methylcarbamoyl)phenyl]ethenyl]-1,3-thiazol-5-yl]prop-2-enoic acid
—— (E)-1-[4-(ethoxymethyl)piperidin-1-yl]-3-(3-methoxyphenyl)but-2-en-1-one —— C19H27NO3
(E)-1-[4-(ethoxymethyl)piperidin-1-yl]-3-(3-methoxyphenyl)but-2-en-1-one
—— ethyl 6-ethyl-2-[[3-(trifluoromethyl)benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C20H21F3N2O3S
ethyl 6-ethyl-2-[[3-(trifluoromethyl)benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— (E)-3-(4-fluorophenyl)-2-methyl-N-(1H-pyrazol-4-yl)prop-2-enamide —— C13H12FN3O
(E)-3-(4-fluorophenyl)-2-methyl-N-(1H-pyrazol-4-yl)prop-2-enamide
—— (E)-3-(4-fluorophenyl)-2-methyl-1-[(2R)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]prop-2-en-1-one —— C19H23FN2O3
(E)-3-(4-fluorophenyl)-2-methyl-1-[(2R)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]prop-2-en-1-one
—— Ethyl 4-amino-2-oxo-3-phenyl-1,3-thiazole-5-carboxylate —— C12H12N2O3S
Ethyl 4-amino-2-oxo-3-phenyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[(Z)-2-(6-imidazol-1-ylpyridin-3-yl)ethenyl]-4-methyl-1,3-thiazole-5-carboxylate —— C17H16N4O2S
ethyl 2-[(Z)-2-(6-imidazol-1-ylpyridin-3-yl)ethenyl]-4-methyl-1,3-thiazole-5-carboxylate
—— Ethyl 5-phenyl-2-[(2-piperidin-1-ium-1-ylacetyl)amino]thiophene-3-carboxylate —— C20H25N2O3S+
Ethyl 5-phenyl-2-[(2-piperidin-1-ium-1-ylacetyl)amino]thiophene-3-carboxylate