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中文名称 英文名称 CAS号 化学式 结构式图片
—— Ethyl 4-[[5-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2,2-diphenylpentyl]amino]-4-oxobutanoate —— C34H41ClN2O4
Ethyl 4-[[5-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2,2-diphenylpentyl]amino]-4-oxobutanoate
—— ethyl (2E,4E)-5-[1-[(2R,4S,5R)-4-hydroxy-5-[[[[(2S)-1-methoxy-1-oxopropan-2-yl]amino]-phenoxyphosphoryl]oxymethyl]oxolan-2-yl]-2,4-dioxopyrimidin-5-yl]penta-2,4-dienoate —— C26H32N3O11P
ethyl (2E,4E)-5-[1-[(2R,4S,5R)-4-hydroxy-5-[[[[(2S)-1-methoxy-1-oxopropan-2-yl]amino]-phenoxyphosphoryl]oxymethyl]oxolan-2-yl]-2,4-dioxopyrimidin-5-yl]penta-2,4-dienoate
—— Ethyl 2-[[2-[[3-[3-(4-carbamimidoylphenyl)propanoyl]-1-methylindole-5-carbonyl]-propylamino]acetyl]amino]acetate;hydrochloride —— C29H36ClN5O5
Ethyl 2-[[2-[[3-[3-(4-carbamimidoylphenyl)propanoyl]-1-methylindole-5-carbonyl]-propylamino]acetyl]amino]acetate;hydrochloride
—— ethyl 1-[7-[(4-chlorophenyl)methyl]-2-(cyclopropylamino)-6-oxo-7,13-dihydrobenzimidazolo[1,2-d][1,4]benzodiazepin-11-yl]piperidine-3-carboxylate —— C33H34ClN5O3
ethyl 1-[7-[(4-chlorophenyl)methyl]-2-(cyclopropylamino)-6-oxo-7,13-dihydrobenzimidazolo[1,2-d][1,4]benzodiazepin-11-yl]piperidine-3-carboxylate
—— (E)-4-(4-hydroxy-3-nitrophenyl)-4-oxobut-2-enoic acid —— C10H7NO6
(E)-4-(4-hydroxy-3-nitrophenyl)-4-oxobut-2-enoic acid
—— ethyl 4-[2-[(E)-2-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]ethenyl]-4-oxoquinazolin-3-yl]benzoate —— C27H25ClN4O5S
ethyl 4-[2-[(E)-2-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]ethenyl]-4-oxoquinazolin-3-yl]benzoate
—— ethyl (2Z,5R)-3-oxo-5-phenyl-7-(trifluoromethyl)-2-[(3,4,5-trimethoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H23F3N2O6S
ethyl (2Z,5R)-3-oxo-5-phenyl-7-(trifluoromethyl)-2-[(3,4,5-trimethoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-[[(S)-[2-[4-[(E)-2-carboxyethenyl]phenyl]sulfonyloxynaphthalen-1-yl]-phenylmethyl]sulfamoyl]phenyl]prop-2-enoic acid —— C35H27NO9S2
(E)-3-[4-[[(S)-[2-[4-[(E)-2-carboxyethenyl]phenyl]sulfonyloxynaphthalen-1-yl]-phenylmethyl]sulfamoyl]phenyl]prop-2-enoic acid
—— Ethyl 2-diethoxyphosphoryl-2-[[2-[2-methoxy-4-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]phenoxy]acetyl]amino]acetate —— C22H28F3N4O8P
Ethyl 2-diethoxyphosphoryl-2-[[2-[2-methoxy-4-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]phenoxy]acetyl]amino]acetate
—— ethyl (6S)-2-[[(E)-[2-[3-(diethylsulfamoyl)phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C32H35N3O6S2
ethyl (6S)-2-[[(E)-[2-[3-(diethylsulfamoyl)phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(2R)-1-[2-[2-(2-chlorophenyl)quinoline-4-carbonyl]hydrazinyl]-3-methyl-1-oxobutan-2-yl]-2-phenylethenesulfonamide —— C29H27ClN4O4S
(E)-N-[(2R)-1-[2-[2-(2-chlorophenyl)quinoline-4-carbonyl]hydrazinyl]-3-methyl-1-oxobutan-2-yl]-2-phenylethenesulfonamide
—— ethyl (1S)-5-(3-bromophenyl)sulfonyl-3-oxo-2-[(1-pyridin-4-ylpiperidin-4-yl)methyl]cyclohexane-1-carboxylate —— C26H31BrN2O5S
ethyl (1S)-5-(3-bromophenyl)sulfonyl-3-oxo-2-[(1-pyridin-4-ylpiperidin-4-yl)methyl]cyclohexane-1-carboxylate
—— ethyl (6R)-2-[[(E)-[2-[3-(diethylsulfamoyl)phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C32H35N3O6S2
ethyl (6R)-2-[[(E)-[2-[3-(diethylsulfamoyl)phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-[[2-[[3-[3-(4-carbamimidoylphenyl)propanoyl]-1-methylindole-5-carbonyl]-propylamino]acetyl]amino]acetate —— C29H35N5O5
Ethyl 2-[[2-[[3-[3-(4-carbamimidoylphenyl)propanoyl]-1-methylindole-5-carbonyl]-propylamino]acetyl]amino]acetate
—— (E)-N-[(2S)-1-[2-[2-(2-chlorophenyl)quinoline-4-carbonyl]hydrazinyl]-3-methyl-1-oxobutan-2-yl]-2-phenylethenesulfonamide —— C29H27ClN4O4S
(E)-N-[(2S)-1-[2-[2-(2-chlorophenyl)quinoline-4-carbonyl]hydrazinyl]-3-methyl-1-oxobutan-2-yl]-2-phenylethenesulfonamide
—— ethyl (6S)-2-[[(E)-[2-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C35H33N3O7S2
ethyl (6S)-2-[[(E)-[2-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-[3-(2,3-dihydroindol-1-ylsulfonyl)-4,5-dimethoxyphenyl]-N-[(2R)-2-phenyl-2-(2-phenyl-1H-indol-3-yl)ethyl]prop-2-enamide —— C41H37N3O5S
(E)-3-[3-(2,3-dihydroindol-1-ylsulfonyl)-4,5-dimethoxyphenyl]-N-[(2R)-2-phenyl-2-(2-phenyl-1H-indol-3-yl)ethyl]prop-2-enamide
—— (E)-3-[3-[8-(4-methoxyphenyl)octoxy]-6-(quinolin-7-ylsulfanylmethyl)pyridin-2-yl]prop-2-enoic acid —— C33H36N2O4S
(E)-3-[3-[8-(4-methoxyphenyl)octoxy]-6-(quinolin-7-ylsulfanylmethyl)pyridin-2-yl]prop-2-enoic acid
—— ethyl (6R)-2-[[(E)-[2-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C35H33N3O7S2
ethyl (6R)-2-[[(E)-[2-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-[3-(2,3-dihydroindol-1-ylsulfonyl)-4,5-dimethoxyphenyl]-N-[(2S)-2-phenyl-2-(2-phenyl-1H-indol-3-yl)ethyl]prop-2-enamide —— C41H37N3O5S
(E)-3-[3-(2,3-dihydroindol-1-ylsulfonyl)-4,5-dimethoxyphenyl]-N-[(2S)-2-phenyl-2-(2-phenyl-1H-indol-3-yl)ethyl]prop-2-enamide
—— Et-DL-Phe(4-F)-DL-N(Me)Val-DL-N(Me)Tyr(3-tBu)-NHMe —— C32H47FN4O4
Et-DL-Phe(4-F)-DL-N(Me)Val-DL-N(Me)Tyr(3-tBu)-NHMe
—— ethyl 2-(1,3-diethoxypropan-2-ylcarbamoyl)-4-[[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]amino]-1H-imidazole-5-carboxylate —— C26H36N4O9
ethyl 2-(1,3-diethoxypropan-2-ylcarbamoyl)-4-[[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]amino]-1H-imidazole-5-carboxylate
—— ethyl (4S)-6-[[(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C29H29ClN4O5
ethyl (4S)-6-[[(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[(4E)-4-[[5-[(2-chlorophenyl)sulfamoyl]-2-piperidin-1-ylanilino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C36H33ClN4O6S
ethyl 4-[(4E)-4-[[5-[(2-chlorophenyl)sulfamoyl]-2-piperidin-1-ylanilino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— [(E)-3-[(6R,7R)-2-carboxy-7-[(2-naphthalen-2-ylsulfanylacetyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]prop-2-enyl]-(3-hydroxypropyl)-dimethylazanium —— C27H32N3O5S2+
[(E)-3-[(6R,7R)-2-carboxy-7-[(2-naphthalen-2-ylsulfanylacetyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]prop-2-enyl]-(3-hydroxypropyl)-dimethylazanium
—— (E)-3-[4-chloro-1-(2-chloro-4-phenylbenzyl)-2-methylimidazol-5-yl]-N-((4-methylbenzene)sulfonyl)-2-propenamide —— C27H23Cl2N3O3S
(E)-3-[4-chloro-1-(2-chloro-4-phenylbenzyl)-2-methylimidazol-5-yl]-N-((4-methylbenzene)sulfonyl)-2-propenamide
—— (E)-3-[4-[4-[4-[(E)-2-carboxyethenyl]phenyl]-2-(2,3,5-trichlorophenyl)-1H-imidazol-5-yl]phenyl]prop-2-enoic acid —— C27H17Cl3N2O4
(E)-3-[4-[4-[4-[(E)-2-carboxyethenyl]phenyl]-2-(2,3,5-trichlorophenyl)-1H-imidazol-5-yl]phenyl]prop-2-enoic acid
—— (E)-(6R,7R)-3-[3-[(3-Hydroxy-propyl)-dimethyl-ammonio]-propenyl]-7-[2-(naphthalen-2-ylsulfanyl)-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate 253301-63-2 C27H31N3O5S2
(E)-(6R,7R)-3-[3-[(3-Hydroxy-propyl)-dimethyl-ammonio]-propenyl]-7-[2-(naphthalen-2-ylsulfanyl)-acetylamino]-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylate
—— (E)-2-fluoro-3-[3-[(Z)-N'-hydroxycarbamimidoyl]phenyl]-N-[4-(2-sulfamoylphenyl)-2-(trifluoromethyl)phenyl]but-2-enamide —— C24H20F4N4O4S
(E)-2-fluoro-3-[3-[(Z)-N'-hydroxycarbamimidoyl]phenyl]-N-[4-(2-sulfamoylphenyl)-2-(trifluoromethyl)phenyl]but-2-enamide
—— Ethyl 3-[[3-ethoxy-2-(octanoylamino)-3-oxopropyl]disulfanyl]-2-(heptylamino)propanoate —— C25H48N2O5S2
Ethyl 3-[[3-ethoxy-2-(octanoylamino)-3-oxopropyl]disulfanyl]-2-(heptylamino)propanoate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (3S)-2-(5-bromo-2-ethoxyphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C24H24BrN3O6S
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (3S)-2-(5-bromo-2-ethoxyphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— ethyl (1S)-1'-[(2R)-2-[(2-amino-2-methylpropanoyl)amino]-5-phenylpentanoyl]spiro[1,2-dihydroindene-3,4'-piperidine]-1-carboxylate;hydrochloride —— C31H42ClN3O4
ethyl (1S)-1'-[(2R)-2-[(2-amino-2-methylpropanoyl)amino]-5-phenylpentanoyl]spiro[1,2-dihydroindene-3,4'-piperidine]-1-carboxylate;hydrochloride
—— ethyl (4R)-6-[[(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C29H29ClN4O5
ethyl (4R)-6-[[(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate —— C23H26ClN3O7S2
ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate
—— ethyl 4-[[3,5-bis(trifluoromethyl)phenyl]methyl-methoxycarbonylamino]-6-ethyl-2-methyl-3,4-dihydro-2H-quinoline-1-carboxylate —— C26H28F6N2O4
ethyl 4-[[3,5-bis(trifluoromethyl)phenyl]methyl-methoxycarbonylamino]-6-ethyl-2-methyl-3,4-dihydro-2H-quinoline-1-carboxylate
—— ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate —— C23H26ClN3O7S2
ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4-cyclopropylthiophene-3-carboxylate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (3R)-2-(5-bromo-2-ethoxyphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxylate —— C24H24BrN3O6S
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (3R)-2-(5-bromo-2-ethoxyphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxylate
—— (E)-3-[4-[[2-(furan-2-ylsulfonyl-(2-methylpropyl)amino)-5-(trifluoromethyl)phenoxy]methyl]phenyl]prop-2-enoic acid —— C25H24F3NO6S
(E)-3-[4-[[2-(furan-2-ylsulfonyl-(2-methylpropyl)amino)-5-(trifluoromethyl)phenoxy]methyl]phenyl]prop-2-enoic acid
—— ethyl (4R)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H24ClFN4O5
ethyl (4R)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 3-[4-[2-[(3,6-dipropyl-9H-fluoren-9-yl)oxy]ethyl]phenyl]-2-ethoxypropanoate —— C34H42O4
ethyl 3-[4-[2-[(3,6-dipropyl-9H-fluoren-9-yl)oxy]ethyl]phenyl]-2-ethoxypropanoate
—— (E)-4-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-4-oxobut-2-enoic acid —— C22H39N9O6
(E)-4-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-4-oxobut-2-enoic acid
—— ethyl 4-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]-2-methylpropyl]phenoxy]benzoate —— C28H33NO6
ethyl 4-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]-2-methylpropyl]phenoxy]benzoate
—— ethyl (4S)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H24ClFN4O5
ethyl (4S)-6-[[(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— Ethyl 4-[[2-(naphthalene-2-carbonylamino)-3-phenylpropanoyl]amino]-5-phenylpent-2-ynoate —— C33H30N2O4
Ethyl 4-[[2-(naphthalene-2-carbonylamino)-3-phenylpropanoyl]amino]-5-phenylpent-2-ynoate
—— ethyl (3S)-1-[(2S)-2-[(2-amino-2-methylpropanoyl)amino]-3-(1H-indol-3-yl)propanoyl]-3-benzylpiperidine-3-carboxylate —— C30H38N4O4
ethyl (3S)-1-[(2S)-2-[(2-amino-2-methylpropanoyl)amino]-3-(1H-indol-3-yl)propanoyl]-3-benzylpiperidine-3-carboxylate
—— Ethyl 2-[(5-chloro-1-benzofuran-2-carbonyl)amino]-2-[1-methyl-5-(4-morpholin-4-ylphenyl)imidazol-2-yl]acetate —— C27H27ClN4O5
Ethyl 2-[(5-chloro-1-benzofuran-2-carbonyl)amino]-2-[1-methyl-5-(4-morpholin-4-ylphenyl)imidazol-2-yl]acetate
—— (E)-7-[(1R,2R,3R,5S)-6,6-dimethyl-3-[[(5-pyrrol-1-ylsulfonylthiophene-2-carbonyl)amino]methyl]-2-bicyclo[3.1.1]heptanyl]hept-5-enoic acid —— C26H34N2O5S2
(E)-7-[(1R,2R,3R,5S)-6,6-dimethyl-3-[[(5-pyrrol-1-ylsulfonylthiophene-2-carbonyl)amino]methyl]-2-bicyclo[3.1.1]heptanyl]hept-5-enoic acid
—— [(E)-[4-[(8S,11R,13S,14S,17S)-17-azido-17-hydroxy-13-methyl-3-oxo-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-11-yl]phenyl]methylideneamino] ethylsulfanylformate —— C28H32N4O4S
[(E)-[4-[(8S,11R,13S,14S,17S)-17-azido-17-hydroxy-13-methyl-3-oxo-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-11-yl]phenyl]methylideneamino] ethylsulfanylformate
—— (E)-1-[(1R)-1-(2,3-dihydro-1-benzofuran-5-yl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-3-[6-[2-(dimethylamino)ethoxy]pyridin-3-yl]prop-2-en-1-one —— C31H32N4O3
(E)-1-[(1R)-1-(2,3-dihydro-1-benzofuran-5-yl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-3-[6-[2-(dimethylamino)ethoxy]pyridin-3-yl]prop-2-en-1-one
—— ethyl 2-ethoxy-3-[4-[2-[(2-phenyl-9H-fluoren-9-yl)oxy]ethyl]phenyl]propanoate —— C34H34O4
ethyl 2-ethoxy-3-[4-[2-[(2-phenyl-9H-fluoren-9-yl)oxy]ethyl]phenyl]propanoate