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中文名称 英文名称 CAS号 化学式 结构式图片
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(5S)-1,5-dimethyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide —— C18H18N4O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[(5S)-1,5-dimethyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(5R)-1,5-dimethyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide —— C18H18N4O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[(5R)-1,5-dimethyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(4S)-1-methyl-6-oxo-4-phenyl-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide —— C24H24N4O4
(E)-3-(3,4-dimethoxyphenyl)-N-[(4S)-1-methyl-6-oxo-4-phenyl-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(4S)-4-(furan-2-yl)-1-methyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide —— C21H18N4O5
(E)-3-(1,3-benzodioxol-5-yl)-N-[(4S)-4-(furan-2-yl)-1-methyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(4R)-1-methyl-6-oxo-4-thiophen-2-yl-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide —— C21H18N4O4S
(E)-3-(1,3-benzodioxol-5-yl)-N-[(4R)-1-methyl-6-oxo-4-thiophen-2-yl-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]prop-2-enamide
—— (E)-1-[4-[5-(5-methyl-1,2,4-oxadiazol-3-yl)pyridin-2-yl]piperazin-1-yl]-3-phenylprop-2-en-1-one —— C21H21N5O2
(E)-1-[4-[5-(5-methyl-1,2,4-oxadiazol-3-yl)pyridin-2-yl]piperazin-1-yl]-3-phenylprop-2-en-1-one
—— (E)-N-[(5R)-1,5-dimethyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]-3-phenylprop-2-enamide —— C17H18N4O2
(E)-N-[(5R)-1,5-dimethyl-6-oxo-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-3-yl]-3-phenylprop-2-enamide
—— ethyl 4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethoxy]benzoate —— C17H23NO4
ethyl 4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethoxy]benzoate
—— ethyl 4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethoxy]benzoate —— C17H23NO4
ethyl 4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethoxy]benzoate
—— (E)-N-(1,2,3,5,6,10b-hexahydropyrrolo[2,1-a]isoquinolin-9-yl)-3-(2-nitrophenyl)prop-2-enamide —— C21H21N3O3
(E)-N-(1,2,3,5,6,10b-hexahydropyrrolo[2,1-a]isoquinolin-9-yl)-3-(2-nitrophenyl)prop-2-enamide
—— E-2-Amino-5-[2,4-difluorophenyl]-5-[3,4-dimethoxyphenyl]-4-pentenoic acid —— C19H19F2NO4
E-2-Amino-5-[2,4-difluorophenyl]-5-[3,4-dimethoxyphenyl]-4-pentenoic acid
—— ethyl (3Z)-3-[(5-methoxy-1H-indol-3-yl)methylidene]-2-oxo-1H-indole-5-carboxylate —— C21H18N2O4
ethyl (3Z)-3-[(5-methoxy-1H-indol-3-yl)methylidene]-2-oxo-1H-indole-5-carboxylate
—— (E)-N-[2-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide —— C21H24N4O3S
(E)-N-[2-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide
—— (E)-N-[2-[2-(2-methoxyethylamino)-2-oxoethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide —— C19H22N4O3S
(E)-N-[2-[2-(2-methoxyethylamino)-2-oxoethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide
—— (E)-N-[5-cyclopropyl-2-(6-methyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C22H23N5O4
(E)-N-[5-cyclopropyl-2-(6-methyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]prop-2-enamide —— C22H24N4O5S
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]prop-2-enamide
—— (E)-1-[(3S)-3-(5-methyl-1,3,4-thiadiazol-2-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one —— C17H19N3OS
(E)-1-[(3S)-3-(5-methyl-1,3,4-thiadiazol-2-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one
—— (E)-3-phenyl-1-[(3R)-3-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]prop-2-en-1-one —— C20H19N3O2S
(E)-3-phenyl-1-[(3R)-3-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]prop-2-en-1-one
—— (E)-N-[2-[2-[(4-methoxyphenyl)methylamino]-2-oxoethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide —— C24H24N4O3S
(E)-N-[2-[2-[(4-methoxyphenyl)methylamino]-2-oxoethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide
—— (E)-1-[4-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one —— C18H21N3OS
(E)-1-[4-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one
—— (E)-1-[(3R)-3-(5-methyl-1,3,4-thiadiazol-2-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one —— C17H19N3OS
(E)-1-[(3R)-3-(5-methyl-1,3,4-thiadiazol-2-yl)piperidin-1-yl]-3-phenylprop-2-en-1-one
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]prop-2-enamide —— C22H24N4O5S
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]prop-2-enamide
—— (E)-3-(1H-indol-6-yl)-2-methyl-1-(3,4,5-trimethoxyphenyl)prop-2-en-1-one —— C21H21NO4
(E)-3-(1H-indol-6-yl)-2-methyl-1-(3,4,5-trimethoxyphenyl)prop-2-en-1-one
—— (E)-1-[(3S)-3-[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one —— C23H21N3O4
(E)-1-[(3S)-3-[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[5-cyclopropyl-2-(4-oxo-6-propan-2-yl-1H-pyrimidin-2-yl)pyrazol-3-yl]prop-2-enamide —— C23H23N5O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[5-cyclopropyl-2-(4-oxo-6-propan-2-yl-1H-pyrimidin-2-yl)pyrazol-3-yl]prop-2-enamide
—— (E)-N-[5-cyclopropyl-2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-phenylprop-2-enamide —— C21H21N5O2
(E)-N-[5-cyclopropyl-2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-phenylprop-2-enamide
—— Ethyl 2-amino-3-(1-octanoylindol-3-yl)propanoate —— C21H30N2O3
Ethyl 2-amino-3-(1-octanoylindol-3-yl)propanoate
—— (E)-N-[2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide —— C21H24N4O3S
(E)-N-[2-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3-phenylprop-2-enamide
—— (E)-1-[(3R)-3-[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one —— C23H21N3O4
(E)-1-[(3R)-3-[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one
—— (E)-N-[5-cyclopropyl-2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C23H25N5O4
(E)-N-[5-cyclopropyl-2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[5-cyclopropyl-2-(6-methyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-phenylprop-2-enamide —— C20H19N5O2
(E)-N-[5-cyclopropyl-2-(6-methyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-phenylprop-2-enamide
—— (E)-3-phenyl-N-[3-(4-pyrimidin-2-ylpiperazin-1-yl)sulfonylpropyl]prop-2-enamide —— C20H25N5O3S
(E)-3-phenyl-N-[3-(4-pyrimidin-2-ylpiperazin-1-yl)sulfonylpropyl]prop-2-enamide
—— (E)-N-[5-cyclopropyl-2-(4-oxo-6-propan-2-yl-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C24H27N5O4
(E)-N-[5-cyclopropyl-2-(4-oxo-6-propan-2-yl-1H-pyrimidin-2-yl)pyrazol-3-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)-5-(furan-2-yl)pyrazol-3-yl]-3-phenylprop-2-enamide —— C22H19N5O3
(E)-N-[2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)-5-(furan-2-yl)pyrazol-3-yl]-3-phenylprop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[5-cyclopropyl-2-(6-methyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]prop-2-enamide —— C21H19N5O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[5-cyclopropyl-2-(6-methyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[2-(4-methylpiperazin-1-yl)-1,3-benzothiazol-6-yl]prop-2-enamide —— C23H26N4O3S
(E)-3-(3,4-dimethoxyphenyl)-N-[2-(4-methylpiperazin-1-yl)-1,3-benzothiazol-6-yl]prop-2-enamide
—— ethyl (2E)-2-[4-(3-cyclopentyloxy-4-methoxyphenyl)pyrrolidin-2-ylidene]acetate —— C20H27NO4
ethyl (2E)-2-[4-(3-cyclopentyloxy-4-methoxyphenyl)pyrrolidin-2-ylidene]acetate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)-5-(furan-2-yl)pyrazol-3-yl]prop-2-enamide —— C23H19N5O5
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)-5-(furan-2-yl)pyrazol-3-yl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[5-cyclopropyl-2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]prop-2-enamide —— C22H21N5O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[5-cyclopropyl-2-(5,6-dimethyl-4-oxo-1H-pyrimidin-2-yl)pyrazol-3-yl]prop-2-enamide
—— (E)-3-phenyl-1-[4-[(1-phenyltetrazol-5-yl)methyl]piperazin-1-yl]prop-2-en-1-one —— C21H22N6O
(E)-3-phenyl-1-[4-[(1-phenyltetrazol-5-yl)methyl]piperazin-1-yl]prop-2-en-1-one
—— ethyl 4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethoxy]benzoate —— C17H23NO4
ethyl 4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethoxy]benzoate
—— (E)-2-[2-Methyl-3-(4-trifluoromethyl-phenyl)-acryloylamino]-nicotinic acid —— C17H13F3N2O3
(E)-2-[2-Methyl-3-(4-trifluoromethyl-phenyl)-acryloylamino]-nicotinic acid
—— (E)-3-(1,3-benzodioxol-5-yl)-1-[4-[[1-(4-fluorophenyl)tetrazol-5-yl]methyl]piperazin-1-yl]prop-2-en-1-one —— C22H21FN6O3
(E)-3-(1,3-benzodioxol-5-yl)-1-[4-[[1-(4-fluorophenyl)tetrazol-5-yl]methyl]piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(1,3-benzodioxol-5-yl)-1-[4-[[1-(3-fluorophenyl)tetrazol-5-yl]methyl]piperazin-1-yl]prop-2-en-1-one —— C22H21FN6O3
(E)-3-(1,3-benzodioxol-5-yl)-1-[4-[[1-(3-fluorophenyl)tetrazol-5-yl]methyl]piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[5-(2-methylpyrazol-3-yl)-1,3,4-oxadiazol-2-yl]prop-2-enamide —— C16H13N5O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[5-(2-methylpyrazol-3-yl)-1,3,4-oxadiazol-2-yl]prop-2-enamide
—— ethyl (1R,4R)-5-acetyl-4-(benzo[3,4-d]1,3-dioxolan-5-yl)-3,5-thiazolidinecarboxylate 248249-47-0 C15H17NO5S
ethyl (1R,4R)-5-acetyl-4-(benzo[3,4-d]1,3-dioxolan-5-yl)-3,5-thiazolidinecarboxylate
—— Ethyl 4-(5,6-dihydro-[1,3]thiazolo[2,3-b][1,3]benzodiazepin-3-yl)benzoate —— C20H18N2O2S
Ethyl 4-(5,6-dihydro-[1,3]thiazolo[2,3-b][1,3]benzodiazepin-3-yl)benzoate
—— ethyl 4-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethoxy]benzoate —— C18H25NO4
ethyl 4-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethoxy]benzoate
—— ethyl 7-nitro-2-oxo-6-phenyl-1H-quinoline-3-carboxylate —— C18H14N2O5
ethyl 7-nitro-2-oxo-6-phenyl-1H-quinoline-3-carboxylate
—— (E)-1-[4-[[1-(3-fluorophenyl)tetrazol-5-yl]methyl]piperazin-1-yl]-3-phenylprop-2-en-1-one —— C21H21FN6O
(E)-1-[4-[[1-(3-fluorophenyl)tetrazol-5-yl]methyl]piperazin-1-yl]-3-phenylprop-2-en-1-one