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—— ethyl 2-[[(2S)-2-[1-[2-[(3,4-dimethylbenzoyl)amino]ethyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C32H35N3O4S2
ethyl 2-[[(2S)-2-[1-[2-[(3,4-dimethylbenzoyl)amino]ethyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-(2-benzamidoethyl)indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C30H31N3O4S2
ethyl 2-[[(2R)-2-[1-(2-benzamidoethyl)indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-[(2,5-dimethylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C30H32N2O3S2
ethyl 2-[[(2R)-2-[1-[(2,5-dimethylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-[(2,5-dimethylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C31H34N2O3S2
ethyl 2-[[(2R)-2-[1-[(2,5-dimethylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-[(3-methylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H32N2O3S2
ethyl 2-[[(2R)-2-[1-[(3-methylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[1-[(2,5-dimethylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C30H32N2O3S2
ethyl 2-[[(2S)-2-[1-[(2,5-dimethylphenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C31H35N5O6S2
ethyl 2-[[(2S)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-[(4-fluorophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H29FN2O3S2
ethyl 2-[[(2R)-2-[1-[(4-fluorophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 3-carbamoyl-2-[[4-[(3R)-3-methylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate —— C24H30N4O6S2
ethyl 3-carbamoyl-2-[[4-[(3R)-3-methylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate
—— ethyl 2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C27H37N3O6S2
ethyl 2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C28H39N3O5S2
ethyl 2-[[4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[(2S)-2-[1-[(4-fluorophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H29FN2O3S2
ethyl 2-[[(2S)-2-[1-[(4-fluorophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 6-benzyl-2-[[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H35N3O6S2
ethyl 6-benzyl-2-[[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[4-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-ethyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C25H33N3O6S2
ethyl 2-[[4-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-ethyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H29BrN2O3S2
ethyl 2-[[(2R)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[4-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C27H37N3O6S2
ethyl 2-[[4-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C28H39N3O5S2
ethyl 2-[[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[(2S)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C28H27BrN2O3S2
ethyl 2-[[(2S)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 5,5,7,7-tetramethyl-2-[[4-[(2S)-2-methylpiperidin-1-yl]sulfonylbenzoyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C27H37N3O5S2
ethyl 5,5,7,7-tetramethyl-2-[[4-[(2S)-2-methylpiperidin-1-yl]sulfonylbenzoyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[(2R)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C29H31N5O5S2
ethyl 2-[[(2R)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C26H35N3O6S2
ethyl 2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 5-(1,3-benzodioxol-5-ylmethyl)-2-[[4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-4-methylthiophene-3-carboxylate —— C30H34N2O7S2
ethyl 5-(1,3-benzodioxol-5-ylmethyl)-2-[[4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-4-methylthiophene-3-carboxylate
—— ethyl 2-[[(2S)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H29BrN2O3S2
ethyl 2-[[(2S)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C28H27BrN2O3S2
ethyl 2-[[(2R)-2-[1-[(4-bromophenyl)methyl]indol-3-yl]sulfanylpropanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— Ethyl 4-[3-(3-methyl-4-oxopyrrolo[2,3-d]pyrimidin-7-yl)propylamino]benzoate —— C19H22N4O3
Ethyl 4-[3-(3-methyl-4-oxopyrrolo[2,3-d]pyrimidin-7-yl)propylamino]benzoate
—— ethyl 2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-ethyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C25H33N3O6S2
ethyl 2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-ethyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 6-benzyl-2-[[4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C31H37N3O5S2
ethyl 6-benzyl-2-[[4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate —— C27H37N3O6S2
ethyl 2-[[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylate
—— ethyl 4-[[(1S)-6,7-dimethoxy-2-(2-oxochromene-3-carbonyl)-3,4-dihydro-1H-isoquinolin-1-yl]methoxy]benzoate —— C31H29NO8
ethyl 4-[[(1S)-6,7-dimethoxy-2-(2-oxochromene-3-carbonyl)-3,4-dihydro-1H-isoquinolin-1-yl]methoxy]benzoate
—— Ethyl 2-[(2,2-dimethyl-3-nitrooxypropanoyl)amino]-3-propanoylsulfanylpropanoate —— C13H22N2O7S
Ethyl 2-[(2,2-dimethyl-3-nitrooxypropanoyl)amino]-3-propanoylsulfanylpropanoate
—— (E)-N-[1-[1-(2-hydroxyethyl)-3,4-dihydro-2H-quinolin-6-yl]ethyl]-3-phenylprop-2-enamide —— C22H26N2O2
(E)-N-[1-[1-(2-hydroxyethyl)-3,4-dihydro-2H-quinolin-6-yl]ethyl]-3-phenylprop-2-enamide
—— ethyl 2-[[(2R)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C31H35N5O6S2
ethyl 2-[[(2R)-2-[[4-(4-ethoxyphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— Ethyl 6,6-diphenyl-1,2,7,7a-tetrahydroindazole-3-carboxylate —— C22H22N2O2
Ethyl 6,6-diphenyl-1,2,7,7a-tetrahydroindazole-3-carboxylate
—— [Ethyl-(4-methyl-1-nitroacridin-9-yl)amino] propanoate —— C19H19N3O4
[Ethyl-(4-methyl-1-nitroacridin-9-yl)amino] propanoate
—— ethyl 2-[[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C26H35N3O6S2
ethyl 2-[[4-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 6-benzyl-2-[[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C31H37N3O5S2
ethyl 6-benzyl-2-[[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 3-carbamoyl-2-[[4-[(3S)-3-methylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate —— C24H30N4O6S2
ethyl 3-carbamoyl-2-[[4-[(3S)-3-methylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate
—— ethyl (2E,5R)-5-(4-chlorophenyl)-7-methyl-2-[[3-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H27ClN2O4S
ethyl (2E,5R)-5-(4-chlorophenyl)-7-methyl-2-[[3-(naphthalen-1-ylmethoxy)phenyl]methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(2S)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C29H31N5O5S2
ethyl 2-[[(2S)-2-[[4-(2,3-dimethylphenyl)-5-[(furan-2-carbonylamino)methyl]-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 5-(1,3-benzodioxol-5-ylmethyl)-2-[[4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-4-methylthiophene-3-carboxylate —— C30H34N2O7S2
ethyl 5-(1,3-benzodioxol-5-ylmethyl)-2-[[4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-4-methylthiophene-3-carboxylate
—— ethyl 4-[[(1R)-6,7-dimethoxy-2-(2-oxochromene-3-carbonyl)-3,4-dihydro-1H-isoquinolin-1-yl]methoxy]benzoate —— C31H29NO8
ethyl 4-[[(1R)-6,7-dimethoxy-2-(2-oxochromene-3-carbonyl)-3,4-dihydro-1H-isoquinolin-1-yl]methoxy]benzoate
—— ethyl 2-[[(2S)-2-[[5-[[(2-methoxybenzoyl)amino]methyl]-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C31H33N5O6S2
ethyl 2-[[(2S)-2-[[5-[[(2-methoxybenzoyl)amino]methyl]-4-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 6-benzyl-2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C30H35N3O6S2
ethyl 6-benzyl-2-[[4-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 2-[4-[(E)-[[4-[(E)-[4-(2-ethoxy-2-oxoethoxy)-3-methoxyphenyl]methylideneamino]-1,2,4-triazol-3-yl]hydrazinylidene]methyl]-2-methoxyphenoxy]acetate —— C26H30N6O8
ethyl 2-[4-[(E)-[[4-[(E)-[4-(2-ethoxy-2-oxoethoxy)-3-methoxyphenyl]methylideneamino]-1,2,4-triazol-3-yl]hydrazinylidene]methyl]-2-methoxyphenoxy]acetate
—— (E)-3-[4-[2-(2,6,6-trimethylcyclohexen-1-yl)ethyl]-1-benzofuran-2-yl]prop-2-enoic acid —— C22H26O3
(E)-3-[4-[2-(2,6,6-trimethylcyclohexen-1-yl)ethyl]-1-benzofuran-2-yl]prop-2-enoic acid
—— ethyl 4-[[(5E)-5-(5-chloro-3-ethyl-1,3-benzothiazol-2-ylidene)-3-(4-fluorophenyl)-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate —— C27H21ClFN3O3S2
ethyl 4-[[(5E)-5-(5-chloro-3-ethyl-1,3-benzothiazol-2-ylidene)-3-(4-fluorophenyl)-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate
—— ethyl 4-(3,4-dihydro-1H-isoquinolin-2-ylcarbamoyloxy)benzoate —— C19H20N2O4
ethyl 4-(3,4-dihydro-1H-isoquinolin-2-ylcarbamoyloxy)benzoate
—— ethyl 4-[[(5E)-5-(5-chloro-3-ethyl-1,3-benzothiazol-2-ylidene)-4-oxo-3-(2-phenylethyl)-1,3-thiazolidin-2-ylidene]amino]benzoate —— C29H26ClN3O3S2
ethyl 4-[[(5E)-5-(5-chloro-3-ethyl-1,3-benzothiazol-2-ylidene)-4-oxo-3-(2-phenylethyl)-1,3-thiazolidin-2-ylidene]amino]benzoate
—— ethyl (2Z,5R)-2-[[5-(dimethylamino)furan-2-yl]methylidene]-5-(4-ethoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H29N3O5S
ethyl (2Z,5R)-2-[[5-(dimethylamino)furan-2-yl]methylidene]-5-(4-ethoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 6-benzyl-2-[[4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C31H37N3O5S2
ethyl 6-benzyl-2-[[4-[(3R,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate