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—— ethyl 3-[[(2S,4S,5S)-5-amino-4-hydroxy-6-phenyl-2-propan-2-ylhexanoyl]amino]propanoate —— C20H32N2O4
ethyl 3-[[(2S,4S,5S)-5-amino-4-hydroxy-6-phenyl-2-propan-2-ylhexanoyl]amino]propanoate
—— Ethyl 2-[4-[4-(4-chlorophenyl)-1,3-oxazol-2-yl]phenoxy]acetate —— C19H16ClNO4
Ethyl 2-[4-[4-(4-chlorophenyl)-1,3-oxazol-2-yl]phenoxy]acetate
—— (E)-3-(3-chlorophenyl)-N-[(4,5-dimethyl-1,2,4-triazol-3-yl)methyl]-N-methylpent-2-enamide —— C17H21ClN4O
(E)-3-(3-chlorophenyl)-N-[(4,5-dimethyl-1,2,4-triazol-3-yl)methyl]-N-methylpent-2-enamide
—— (E)-3-(3-chlorophenyl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]pent-2-enamide —— C16H22ClNO3S
(E)-3-(3-chlorophenyl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]pent-2-enamide
—— (E)-3-(3-chlorophenyl)-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]pent-2-enamide —— C16H22ClNO3S
(E)-3-(3-chlorophenyl)-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]pent-2-enamide
—— ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-(3-propan-2-ylphenoxy)pyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C34H35FN4O5
ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-(3-propan-2-ylphenoxy)pyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (2S)-2-[(4-ethylphenyl)carbamothioylamino]-3-phenylpropanoate —— C20H24N2O2S
ethyl (2S)-2-[(4-ethylphenyl)carbamothioylamino]-3-phenylpropanoate
—— ethyl (3R)-1-[4-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C33H34N4O5
ethyl (3R)-1-[4-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[5-(3-methylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H32N4O5
ethyl (3S)-1-[3-[[5-(3-methylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[5-(4-fluorophenoxy)-2-(4-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H28F2N4O5
ethyl (3R)-1-[3-[[5-(4-fluorophenoxy)-2-(4-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[2-(4-fluorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31FN4O5
ethyl (3R)-1-[3-[[2-(4-fluorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— (E)-N-methylsulfonyl-3-[3-(trifluoromethyl)phenyl]but-2-enamide —— C12H12F3NO3S
(E)-N-methylsulfonyl-3-[3-(trifluoromethyl)phenyl]but-2-enamide
—— ethyl (3S)-1-[4-[[5-(2,3-dihydro-1H-inden-5-yloxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C35H36N4O6
ethyl (3S)-1-[4-[[5-(2,3-dihydro-1H-inden-5-yloxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[5-(2,3-dimethylphenoxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C34H36N4O6
ethyl (3S)-1-[3-[[5-(2,3-dimethylphenoxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[5-(1,3-benzodioxol-5-yloxy)-2-(3,4-dichlorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H28Cl2N4O7
ethyl (3S)-1-[3-[[5-(1,3-benzodioxol-5-yloxy)-2-(3,4-dichlorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (4R)-1-[[3-(4-benzylpiperidine-1-carbonyl)phenyl]methyl]-4-(3,4-dichlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C35H36Cl2N2O4
ethyl (4R)-1-[[3-(4-benzylpiperidine-1-carbonyl)phenyl]methyl]-4-(3,4-dichlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— ethyl (3R)-1-[3-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C33H34N4O5
ethyl (3R)-1-[3-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H29ClN4O5
ethyl (3R)-1-[3-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(2-chlorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31ClN4O5
ethyl (3S)-1-[4-[[2-(2-chlorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H29FN4O5
ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[5-(4-chloro-3-methylphenoxy)-2-(3-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H30ClFN4O5
ethyl (3R)-1-[3-[[5-(4-chloro-3-methylphenoxy)-2-(3-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H29ClN4O5
ethyl (3S)-1-[3-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C33H34N4O5
ethyl (3S)-1-[3-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[5-(2,3-dihydro-1H-inden-5-yloxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C35H36N4O6
ethyl (3R)-1-[4-[[5-(2,3-dihydro-1H-inden-5-yloxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[2-(4-fluorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31FN4O5
ethyl (3S)-1-[3-[[2-(4-fluorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (6S)-3-methyl-2-oxo-6-(3-phenoxyphenyl)-4-[[3-(trifluoromethyl)phenoxy]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C28H25F3N2O5
ethyl (6S)-3-methyl-2-oxo-6-(3-phenoxyphenyl)-4-[[3-(trifluoromethyl)phenoxy]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3S)-1-[4-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C33H34N4O5
ethyl (3S)-1-[4-[[5-(2,3-dimethylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(3,4-dichlorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H30Cl2N4O5
ethyl (3S)-1-[4-[[2-(3,4-dichlorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[5-(4-chloro-3-methylphenoxy)-2-(3-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H30ClFN4O5
ethyl (3S)-1-[3-[[5-(4-chloro-3-methylphenoxy)-2-(3-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(4-chlorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31ClN4O6
ethyl (3S)-1-[4-[[2-(4-chlorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (4S)-1-[[3-(4-benzylpiperidine-1-carbonyl)phenyl]methyl]-4-(3,4-dichlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate —— C35H36Cl2N2O4
ethyl (4S)-1-[[3-(4-benzylpiperidine-1-carbonyl)phenyl]methyl]-4-(3,4-dichlorophenyl)-6-methyl-2-oxo-3,4-dihydropyridine-5-carboxylate
—— (E)-N-[(4-hydroxyoxan-4-yl)methyl]-3-[3-(trifluoromethyl)phenyl]but-2-enamide —— C17H20F3NO3
(E)-N-[(4-hydroxyoxan-4-yl)methyl]-3-[3-(trifluoromethyl)phenyl]but-2-enamide
—— ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31FN4O6
ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— (E)-N-methylsulfonyl-3-[2-(trifluoromethyl)phenyl]but-2-enamide —— C12H12F3NO3S
(E)-N-methylsulfonyl-3-[2-(trifluoromethyl)phenyl]but-2-enamide
—— ethyl (3R)-1-[3-[[5-(1,3-benzodioxol-5-yloxy)-2-(3,4-dichlorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H28Cl2N4O7
ethyl (3R)-1-[3-[[5-(1,3-benzodioxol-5-yloxy)-2-(3,4-dichlorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[(2-benzyl-3-oxo-5-phenoxypyridazin-4-yl)amino]benzoyl]piperidine-3-carboxylate —— C32H32N4O5
ethyl (3S)-1-[3-[(2-benzyl-3-oxo-5-phenoxypyridazin-4-yl)amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31FN4O5
ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H29ClN4O5
ethyl (3R)-1-[4-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H42N4O5S
ethyl (3R)-1-[4-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (6R)-3-methyl-2-oxo-6-(3-phenoxyphenyl)-4-[[3-(trifluoromethyl)phenoxy]methyl]-1,6-dihydropyrimidine-5-carboxylate —— C28H25F3N2O5
ethyl (6R)-3-methyl-2-oxo-6-(3-phenoxyphenyl)-4-[[3-(trifluoromethyl)phenoxy]methyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (3R)-1-[4-[[2-(3,4-dichlorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H30Cl2N4O5
ethyl (3R)-1-[4-[[2-(3,4-dichlorophenyl)-5-(4-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(3,4-dichlorophenyl)-5-(2,3-dihydro-1H-inden-5-yloxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C34H32Cl2N4O5
ethyl (3S)-1-[4-[[2-(3,4-dichlorophenyl)-5-(2,3-dihydro-1H-inden-5-yloxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H38F3N5O3S
ethyl (3R)-1-[3-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-[4-(2-fluorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H38FN5O4S
ethyl (3S)-1-[4-[[4-[4-(2-fluorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H29FN4O5
ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31FN4O6
ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(4-chlorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31ClN4O6
ethyl (3R)-1-[4-[[2-(4-chlorophenyl)-5-(4-methoxyphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[5-(3-chlorophenoxy)-2-(4-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H28ClFN4O5
ethyl (3S)-1-[3-[[5-(3-chlorophenoxy)-2-(4-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(3,4-dichlorophenyl)-5-(2,3-dihydro-1H-inden-5-yloxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C34H32Cl2N4O5
ethyl (3R)-1-[4-[[2-(3,4-dichlorophenyl)-5-(2,3-dihydro-1H-inden-5-yloxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[5-(2,3-dimethylphenoxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C34H36N4O6
ethyl (3R)-1-[3-[[5-(2,3-dimethylphenoxy)-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate