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—— ethyl (3R)-1-[3-[[5-(3-chlorophenoxy)-2-(4-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H28ClFN4O5
ethyl (3R)-1-[3-[[5-(3-chlorophenoxy)-2-(4-fluorophenyl)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— (E)-1-(1,1-dioxo-1,2-thiazolidin-2-yl)-3-[3-(trifluoromethyl)phenyl]but-2-en-1-one —— C14H14F3NO3S
(E)-1-(1,1-dioxo-1,2-thiazolidin-2-yl)-3-[3-(trifluoromethyl)phenyl]but-2-en-1-one
—— ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-(3-propan-2-ylphenoxy)pyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C34H35FN4O5
ethyl (3R)-1-[4-[[2-(4-fluorophenyl)-3-oxo-5-(3-propan-2-ylphenoxy)pyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31FN4O5
ethyl (3S)-1-[4-[[2-(4-fluorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C31H29ClN4O5
ethyl (3S)-1-[4-[[2-(2-chlorophenyl)-3-oxo-5-phenoxypyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H38F3N5O3S
ethyl (3S)-1-[4-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[4-tert-butyl-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C35H45N5O4S
ethyl (3S)-1-[3-[[4-tert-butyl-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[2-(2-chlorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H31ClN4O5
ethyl (3R)-1-[4-[[2-(2-chlorophenyl)-5-(3-methylphenoxy)-3-oxopyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[(2-benzyl-3-oxo-5-phenoxypyridazin-4-yl)amino]benzoyl]piperidine-3-carboxylate —— C32H32N4O5
ethyl (3R)-1-[3-[(2-benzyl-3-oxo-5-phenoxypyridazin-4-yl)amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-(methoxymethyl)-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H41N5O5S
ethyl (3R)-1-[3-[[4-(methoxymethyl)-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C30H34F3N5O4S
ethyl (3R)-1-[5-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H41N5O4S
ethyl (3R)-1-[4-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C26H33F3N4O4S
ethyl (3S)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H41N5O4S
ethyl (3R)-1-[3-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H42N4O5S
ethyl (3S)-1-[4-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-phenyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C37H38F3N5O3S
ethyl (3S)-1-[4-[[4-phenyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C30H36ClN5O5S
ethyl (3R)-1-[5-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-tert-butyl-6-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C35H46N4O5S
ethyl (3R)-1-[3-[[4-tert-butyl-6-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H41N5O4S
ethyl (3S)-1-[4-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-tert-butyl-6-[cyclohexyl(methyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C29H42N4O4S
ethyl (3R)-1-[5-[[4-tert-butyl-6-[cyclohexyl(methyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-[[4-tert-butyl-6-[cyclohexyl(methyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C29H42N4O4S
ethyl (3S)-1-[5-[[4-tert-butyl-6-[cyclohexyl(methyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[4-[benzyl(methyl)amino]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C30H36N4O4S
ethyl (3S)-1-[3-[[4-[benzyl(methyl)amino]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H42N4O5S
ethyl (3R)-1-[3-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-[4-(2-fluorophenyl)piperazin-1-yl]-6-phenylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C36H38FN5O3S
ethyl (3S)-1-[4-[[4-[4-(2-fluorophenyl)piperazin-1-yl]-6-phenylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-[benzyl(methyl)amino]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C30H36N4O4S
ethyl (3R)-1-[3-[[4-[benzyl(methyl)amino]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C26H33F3N4O4S
ethyl (3R)-1-[5-[[4-[cyclohexyl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H42N4O5S
ethyl (3S)-1-[3-[[4-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C30H34F3N5O4S
ethyl (3S)-1-[5-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H39N5O4S
ethyl (3S)-1-[3-[[4-[4-(4-methoxyphenyl)piperazin-1-yl]-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-(4-benzylpiperazin-1-yl)-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C31H39N5O5S
ethyl (3R)-1-[5-[[4-(4-benzylpiperazin-1-yl)-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[4-(4-acetylpiperazin-1-yl)-6-ethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C28H37N5O4S
ethyl (3R)-1-[4-[[4-(4-acetylpiperazin-1-yl)-6-ethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H36F3N5O3S
ethyl (3S)-1-[4-[[4-methyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-(4-ethylpiperazin-1-yl)-6-phenylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H39N5O3S
ethyl (3R)-1-[3-[[4-(4-ethylpiperazin-1-yl)-6-phenylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H38F3N5O3S
ethyl (3R)-1-[4-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[4-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H38ClN5O4S
ethyl (3S)-1-[4-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[4-[[4-[4-(2-fluorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H38FN5O4S
ethyl (3R)-1-[4-[[4-[4-(2-fluorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-[[4-tert-butyl-6-(4-ethylpiperazin-1-yl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C28H41N5O4S
ethyl (3S)-1-[5-[[4-tert-butyl-6-(4-ethylpiperazin-1-yl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-tert-butyl-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C35H45N5O4S
ethyl (3R)-1-[3-[[4-tert-butyl-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[4-(4-benzylpiperazin-1-yl)-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H39N5O3S
ethyl (3R)-1-[3-[[4-(4-benzylpiperazin-1-yl)-6-methylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[3-[[5-(3-methylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate —— C32H32N4O5
ethyl (3R)-1-[3-[[5-(3-methylphenoxy)-3-oxo-2-phenylpyridazin-4-yl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[3-[[4-(methoxymethyl)-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H41N5O5S
ethyl (3S)-1-[3-[[4-(methoxymethyl)-6-[4-(4-methoxyphenyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— [(E,3S)-1-(benzenesulfonyl)-3-(methoxymethoxy)-4-methylpent-1-enyl]-trimethylsilane —— C17H28O4SSi
[(E,3S)-1-(benzenesulfonyl)-3-(methoxymethoxy)-4-methylpent-1-enyl]-trimethylsilane
—— ethyl (3S)-1-[4-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C32H38ClN5O3S
ethyl (3S)-1-[4-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-5,6-dimethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-tert-butyl-6-(4-ethylpiperazin-1-yl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C28H41N5O4S
ethyl (3R)-1-[5-[[4-tert-butyl-6-(4-ethylpiperazin-1-yl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3R)-1-[5-[[4-(4-acetylpiperazin-1-yl)-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C26H35N5O6S
ethyl (3R)-1-[5-[[4-(4-acetylpiperazin-1-yl)-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-[5-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate —— C30H36ClN5O5S
ethyl (3S)-1-[5-[[4-[4-(2-chlorophenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carbonyl]piperidine-3-carboxylate
—— (E)-3-[3-[3-(dimethylamino)-2-hydroxypropoxy]-4-methoxyphenyl]-1-pyridin-4-ylprop-2-en-1-one —— C20H24N2O4
(E)-3-[3-[3-(dimethylamino)-2-hydroxypropoxy]-4-methoxyphenyl]-1-pyridin-4-ylprop-2-en-1-one
—— ethyl (3S)-1-[3-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C33H38F3N5O3S
ethyl (3S)-1-[3-[[4,5-dimethyl-6-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate
—— Ethyl 2-[6-(4-tert-butyl-1,3-oxazol-2-yl)naphthalen-2-yl]oxyacetate —— C21H23NO4
Ethyl 2-[6-(4-tert-butyl-1,3-oxazol-2-yl)naphthalen-2-yl]oxyacetate
—— ethyl (3S)-1-[4-[[4-(4-acetylpiperazin-1-yl)-6-ethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate —— C28H37N5O4S
ethyl (3S)-1-[4-[[4-(4-acetylpiperazin-1-yl)-6-ethylpyrimidin-2-yl]sulfanylmethyl]benzoyl]piperidine-3-carboxylate