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中文名称 英文名称 CAS号 化学式 结构式图片
—— [6-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C21H33N5O
[6-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— [6-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C21H33N5O
[6-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 6-benzyl-N-[(2S)-butan-2-yl]-10-methyl-2-oxo-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide —— C23H24N4O2
6-benzyl-N-[(2S)-butan-2-yl]-10-methyl-2-oxo-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide
—— 6-[3-(hydroxymethyl)phenyl]-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C22H29N3O2
6-[3-(hydroxymethyl)phenyl]-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— 6-(trifluoromethyl)-3-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one —— C12H10F6N2O3
6-(trifluoromethyl)-3-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one
—— 6-[3-(hydroxymethyl)phenyl]-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C22H29N3O2
6-[3-(hydroxymethyl)phenyl]-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— 6-[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]-N,N-dimethylpyrazine-2-carboxamide —— C21H27N5O2
6-[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]-N,N-dimethylpyrazine-2-carboxamide
—— 6-[(3S)-1-cyclopentylpiperidin-3-yl]-3-propan-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C16H25N5S
6-[(3S)-1-cyclopentylpiperidin-3-yl]-3-propan-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-benzyl-5-[(2R)-2-ethylpiperidine-1-carbonyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one —— C25H26N4O2
6-benzyl-5-[(2R)-2-ethylpiperidine-1-carbonyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one
—— 6-(trifluoromethyl)-3-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one —— C12H10F6N2O3
6-(trifluoromethyl)-3-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one
—— 6-[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]-N,N-dimethylpyrazine-2-carboxamide —— C21H27N5O2
6-[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl]-N,N-dimethylpyrazine-2-carboxamide
—— (6R,9R)-9-(2-chlorophenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H17ClN4O
(6R,9R)-9-(2-chlorophenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(2-chlorophenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H17ClN4O
(6R,9S)-9-(2-chlorophenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(4-ethoxy-3-methoxyphenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6S,9S)-9-(4-ethoxy-3-methoxyphenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-benzyl-5-[(2S)-2-ethylpiperidine-1-carbonyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one —— C25H26N4O2
6-benzyl-5-[(2S)-2-ethylpiperidine-1-carbonyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaen-2-one
—— (6S)-2,6-diamino-4-(1-methyl-3-phenylpyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C20H20N6
(6S)-2,6-diamino-4-(1-methyl-3-phenylpyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— (6S,9R)-9-(4-ethoxy-3-methoxyphenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O3
(6S,9R)-9-(4-ethoxy-3-methoxyphenyl)-6-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6-methoxy-1H-indol-2-yl)-(4-methylpiperazin-4-ium-1-yl)methanone —— C15H20N3O2+
(6-methoxy-1H-indol-2-yl)-(4-methylpiperazin-4-ium-1-yl)methanone
—— 6-ethyl 3-methyl 2-(2-(4-fluorophenyl)acetamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate —— C20H21FN2O5S
6-ethyl 3-methyl 2-(2-(4-fluorophenyl)acetamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate
—— 6-ethanoyl-2-[2-(4-fluorophenyl)ethanoylamino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide —— C18H18FN3O3S
6-ethanoyl-2-[2-(4-fluorophenyl)ethanoylamino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide
—— 6-Ethyl-2-[[2-(4-fluorophenyl)acetyl]amino]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-6-ium-3-carboxamide —— C18H21FN3O2S+
6-Ethyl-2-[[2-(4-fluorophenyl)acetyl]amino]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-6-ium-3-carboxamide
—— (6S)-2-[[2-(4-fluorophenyl)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H19FN2O2S
(6S)-2-[[2-(4-fluorophenyl)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-Acetyl-2-(2-(2,4-dimethylphenyl)acetamido)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxamide —— C20H23N3O3S
6-Acetyl-2-(2-(2,4-dimethylphenyl)acetamido)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxamide
—— (6R)-2,6-diamino-4-(1-methyl-3-phenylpyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C20H20N6
(6R)-2,6-diamino-4-(1-methyl-3-phenylpyrazol-4-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— (6S)-2-[[2-(2,4-dimethylphenyl)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C20H24N2O2S
(6S)-2-[[2-(2,4-dimethylphenyl)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-2-[[2-(2,4-dimethylphenyl)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C20H24N2O2S
(6R)-2-[[2-(2,4-dimethylphenyl)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-bromo-2-tert-butyl-8-propan-2-ylquinoline-4-carboxylic acid —— C17H20BrNO2
6-bromo-2-tert-butyl-8-propan-2-ylquinoline-4-carboxylic acid
—— 6-methyl-5-[[(2R)-2-(3-phenylpropyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C19H25N3O3
6-methyl-5-[[(2R)-2-(3-phenylpropyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-methyl-5-[[(2S)-2-(3-phenylpropyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C19H25N3O3
6-methyl-5-[[(2S)-2-(3-phenylpropyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-[(2R)-1-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-2-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C13H19N7S
6-[(2R)-1-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-2-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6R,9S)-6-(2-hydroxyphenyl)-9-(4-hydroxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H18N4O3
(6R,9S)-6-(2-hydroxyphenyl)-9-(4-hydroxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-[(2S)-1-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-2-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C13H19N7S
6-[(2S)-1-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-2-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6S,9S)-6-(2-hydroxyphenyl)-9-(4-hydroxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H18N4O3
(6S,9S)-6-(2-hydroxyphenyl)-9-(4-hydroxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-[(1S)-1-(3-methoxyphenoxy)ethyl]-3-propan-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C15H18N4O2S
6-[(1S)-1-(3-methoxyphenoxy)ethyl]-3-propan-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-cyclopentyl-2-methoxy-3-[[[(3R)-thiolan-3-yl]amino]methyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C18H25N3O2S
6-cyclopentyl-2-methoxy-3-[[[(3R)-thiolan-3-yl]amino]methyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— 6-[[(2S)-2-[[3-(trifluoromethyl)phenyl]methyl]morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C17H18F3N3O3
6-[[(2S)-2-[[3-(trifluoromethyl)phenyl]methyl]morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione
—— 6-[(3S)-3-(2,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile —— C20H21N3O3
6-[(3S)-3-(2,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile
—— 6-(3-methoxypropyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide —— C23H24N4O3
6-(3-methoxypropyl)-2-oxo-N-[(1S)-1-phenylethyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide
—— 6-benzyl-N-[(2S)-butan-2-yl]-2-oxo-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide —— C22H22N4O2
6-benzyl-N-[(2S)-butan-2-yl]-2-oxo-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide
—— (6S)-2,6-diamino-4-(4-fluoro-3-methoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C17H17FN4O
(6S)-2,6-diamino-4-(4-fluoro-3-methoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— 6-cyclopentyl-2-methoxy-3-[[[(3S)-thiolan-3-yl]amino]methyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C18H25N3O2S
6-cyclopentyl-2-methoxy-3-[[[(3S)-thiolan-3-yl]amino]methyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— 6-benzyl-N-[(2R)-butan-2-yl]-2-oxo-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide —— C22H22N4O2
6-benzyl-N-[(2R)-butan-2-yl]-2-oxo-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide
—— (6R,9R)-9-(2-fluorophenyl)-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H19FN4O2
(6R,9R)-9-(2-fluorophenyl)-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-cyano-N-ethyl-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C14H17N3O2
6-cyano-N-ethyl-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— 6-[(2S)-2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine —— C9H11F3N4O
6-[(2S)-2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
—— 6-(3-methoxypropyl)-2-oxo-N-[(1R)-1-phenylethyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide —— C23H24N4O3
6-(3-methoxypropyl)-2-oxo-N-[(1R)-1-phenylethyl]-1,6,8-triazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carboxamide
—— (6R,9S)-9-(2-fluorophenyl)-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H19FN4O2
(6R,9S)-9-(2-fluorophenyl)-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]-1H-indazole —— C14H14N4O
6-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]-1H-indazole
—— (6R)-6-methyl-2-[[2-[(6-methyl-5-oxo-4H-1,2,4-triazin-3-yl)sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C16H19N5O3S2
(6R)-6-methyl-2-[[2-[(6-methyl-5-oxo-4H-1,2,4-triazin-3-yl)sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-6-methyl-2-[[2-[(6-methyl-5-oxo-4H-1,2,4-triazin-3-yl)sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C16H19N5O3S2
(6S)-6-methyl-2-[[2-[(6-methyl-5-oxo-4H-1,2,4-triazin-3-yl)sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide